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1. 发明申请

US20100280078A1 1-(Azolin-2-yl)amino-1,2-diphenylethane compounds for combating animal pests 有权
公开(公告)号：US20100280078A1
公开(公告)日：2010-11-04
申请号：US12667299
申请日：2008-07-02
申请人： Markus Kordes , Christopher Koradin , Ronan Le Vezouet , Ernst Baumann , Deborah L. Culbertson , Douglas D. Anspaugh , Hassan Oloumi-Sadeghi , Cecile Ebuenga
发明人： Markus Kordes , Christopher Koradin , Ronan Le Vezouet , Ernst Baumann , Deborah L. Culbertson , Douglas D. Anspaugh , Hassan Oloumi-Sadeghi , Cecile Ebuenga
IPC分类号： A01N43/78 , C07D277/18 , A61K31/426 , C07D417/12 , C07D417/14 , A61K31/427 , C07D263/28 , A01N43/76 , A61K31/421 , A61K31/4439 , A61P33/00 , A01P7/00 , A01P7/02 , A01P7/04 , A01P5/00
CPC分类号： C07D263/28 , A01N43/50 , A01N43/76 , A01N43/78 , A01N47/12 , A01N47/16 , C07D233/48 , C07D277/18 , C07D417/06 , C07D417/12
摘要： The present invention relates to 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and to their salts which are useful for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds. wherein A is a radical of formulae A.1 or A.2 wherein # denotes the bond to the remaining compound of formula I, X is selected from O, S and NRX, R1 is selected from the group consisting of —ORA, —NRB1RB2, C(═O)—RC, —C(═O)—ORD, —C(═O)—SRE, —C(═O)—NRB1RB2′, —C(═S)—RC′, —C(═S)—ORD′, —C(═S)—SRE′, —C(═S)—NRB1RB2, —C(═NR1a)—RC′, —C(═NR1b)—ORD′, —C(═NR1c)—SRE′, —C(═NR1d)—NRB1RB2, —S(═O)—RF, —S(═O)2—RG, —S(═O)2—NRB1RB2′, —P(═O)RH1RH2, —P(═S)RH1RH2, —B—C(═O)—RI, —B—O—C(═O)—RI, —B—S—C(═O)—RI, —B—N(RJ)—C(═O)—RK, —B—C(═S)—RK, —B—O—C(═S)—RK, —B—S—C(═S)—RK, —B—N(RJ)—C(═S)—RK, C1-C8-alkenyl, C1-C8-alkynyl, C3-C8-cycloalkyl, which is unsubstituted or may carry 1 to 4 substituents R1e, naphthyl, which is unsubstituted or may carry 1 to 4 substituents R1f, a saturated or partially unsaturated heterocycle, which is unsubstituted or may carry 1 to 4 substituents R1g, hetaryl, which is unsubstituted or may carry 1 to 4 substituents R1h, and C1-C6-alkyl, which carries a radical selected from the group consisting of —NR1iR1j, C1-C4-alkoxycarbonyl, C3-C8-cycloalkyl, aryl, aryloxy, arylthio, heterocyclyl, heterocyclyloxy and heterocyclylthio, R2, R3, R4, R5, R6 and R7 are each independently hydrogen, halogen, OH, SH, NH2, SO3H, COOH, cyano, nitro, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkylamino etc.

2. 发明授权

US08211924B2 1-(azolin-2-yl)amino-1,2-diphenylethane compounds for combating animal pests 有权
公开(公告)号：US08211924B2
公开(公告)日：2012-07-03
申请号：US12667299
申请日：2008-07-02
申请人： Markus Kordes , Christopher Koradin , Ronan Le Vezouet , Ernst Baumann , Deborah L. Culbertson , Douglas D. Anspaugh , Hassan Oloumi-Sadeghi , Cecille Ebuenga
发明人： Markus Kordes , Christopher Koradin , Ronan Le Vezouet , Ernst Baumann , Deborah L. Culbertson , Douglas D. Anspaugh , Hassan Oloumi-Sadeghi , Cecille Ebuenga
IPC分类号： A01N43/78 , A01N43/76 , A61K31/425 , A61K31/42 , C07D277/00 , C07D263/00
CPC分类号： C07D263/28 , A01N43/50 , A01N43/76 , A01N43/78 , A01N47/12 , A01N47/16 , C07D233/48 , C07D277/18 , C07D417/06 , C07D417/12
摘要： The present invention relates to 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and to their salts which are useful for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds. wherein A is a radical of formulae A.1 or A.2 wherein # denotes the bond to the remaining compound of formula I, X is selected from O, S and NRX, R1 is selected from the group consisting of —ORA, —NRB1RB2, —C(═O)—RC, —C(═O)—ORD, —C(═O)—SRE, —C(═O)—NRB1RB2′, —C(═S)—RC′, —C(═S)—ORD′, —C(═S)—SRE′, —C(═S)—NRB1RB2, —C(═NR1a)—RC′, —C(═NR1b)—ORD′, —C(═NR1c)—SRE′, —C(═NR1d)—NRB1RB2, —S(═O)—RF, —S(═O)2—RG, —S(═O)2—NRB1RB2′, —P(═O)RH1RH2, —P(═S)RH1RH2, —B—C(═O)—RI, —B—O—C(═O)—RI, —B—S—C(═O)—RI, —B—N(RJ)—C(═O)—RK, —B—C(═S)—RK, —B—O—C(═S)—RK, —B—S—C(═S)—RK, —B—N(RJ)—C(═S)—RK, C1-C8-alkenyl, C1-C8-alkynyl, C3-C8-cycloalkyl, which is unsubstituted or may carry 1 to 4 substituents R1e, naphthyl, which is unsubstituted or may carry 1 to 4 substituents R1f, a saturated or partially unsaturated heterocycle, which is unsubstituted or may carry 1 to 4 substituents R1g, hetaryl, which is unsubstituted or may carry 1 to 4 substituents R1h, and C1-C6-alkyl, which carries a radical selected from the group consisting of —NR1iR1j, C1-C4-alkoxycarbonyl, C3-C8-cycloalkyl, aryl, aryloxy, arylthio, heterocyclyl, heterocyclyloxy and heterocyclylthio, R2, R3, R4, R5, R6 and R7 are each independently hydrogen, halogen, OH, SH, NH2, SO3H, COOH, cyano, nitro, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkylamino etc.

3. 发明授权

US08173675B2 Substituted amino-thiourea compounds for combating animal pests 失效
标题翻译：用于对抗动物害虫的取代氨基 - 硫脲化合物
公开(公告)号：US08173675B2
公开(公告)日：2012-05-08
申请号：US12601017
申请日：2008-05-13
申请人： Christopher Koradin , Markus Kordes , Ernst Baumann , Ronan Le Vezouet , Deborah L. Culbertson
发明人： Christopher Koradin , Markus Kordes , Ernst Baumann , Ronan Le Vezouet , Deborah L. Culbertson
IPC分类号： A61K31/47 , C07D215/14
CPC分类号： A01N47/36 , A01N47/32 , C07C335/14 , C07C2602/08 , C07C2602/10 , C07D307/82 , C07D333/66
摘要： The invention relates to substituted amino-thiourea compounds of formula (I), to the enantiomers, diastereomers and salts thereof and to compositions comprising such compounds. The invention also relates to the use of the substituted amino-thiourea compounds, of their salts or of compositions comprising them for combating animal pests. Furthermore the invention relates also to methods of applying such compounds. The substituted amino-thiourea compounds are defined by the following formula (I): wherein A, B, R1, R2, R3, R4, R5.1, R5.2 and R6 are defined as in the description.
摘要翻译：本发明涉及式（I）的取代的氨基 - 硫脲化合物，其涉及其对映体，非对映异构体和盐以及包含这些化合物的组合物。本发明还涉及取代的氨基 - 硫脲化合物，其盐或包含它们的组合物用于对抗动物害虫的用途。此外，本发明还涉及应用这些化合物的方法。取代的氨基 - 硫脲化合物由下式（I）定义：其中A，B，R1，R2，R3，R4，R5.1，R5.2和R6如说明书所定义。

4. 发明申请

US20100298138A1 Aminoazoline and Urea Derivatives for Combating Animal Pests 审中-公开
标题翻译：用于防治动物害虫的氨基唑啉和尿素衍生物
公开(公告)号：US20100298138A1
公开(公告)日：2010-11-25
申请号：US12600852
申请日：2008-05-23
申请人： Christopher Koradin , Markus Kordes , Ernst Baumann , Ronan Le Vezouet , Deborah L. Culbertson
发明人： Christopher Koradin , Markus Kordes , Ernst Baumann , Ronan Le Vezouet , Deborah L. Culbertson
IPC分类号： A01C1/06 , A01P7/04 , A01P7/02 , A01P5/00 , A01N43/78 , A61K31/426 , C07D277/18 , A61P33/00 , C07C335/12 , A61K31/17 , A01N47/28 , C07C69/347 , C07C69/708 , C07D261/18 , A61K31/42 , A01N43/80 , C07D213/80 , A61K31/44 , A01N43/40 , C07C69/736 , A61K31/216 , C07C69/78 , C07D307/68 , A61K31/341 , A01N43/08
CPC分类号： C07D261/18 , A01N43/50 , A01N43/76 , A01N43/78 , A01N47/32 , C07C275/26 , C07C279/16 , C07C335/14 , C07C2602/08 , C07C2602/10 , C07D213/80 , C07D233/50 , C07D263/28 , C07D277/18 , C07D317/60
摘要： The present invention relates to the use of aminoazoline and urea derivatives for com-bating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds and to specific azoline and urea derivatives.
摘要翻译：本发明涉及氨基唑啉和脲衍生物在动物害虫中的应用。本发明还涉及通过使用这些化合物，种子和包含所述化合物的农业和兽用组合物以及特定的唑啉和脲衍生物来控制动物害虫的方法。

5. 发明申请

US20100167927A1 Substituted Amino-Thiourea Compounds For Combating Animal Pests 失效
标题翻译：用于抵抗动物害虫的替代氨基硫脲化合物
公开(公告)号：US20100167927A1
公开(公告)日：2010-07-01
申请号：US12601017
申请日：2008-05-13
申请人： Christopher Koradin , Markus Kordes , Ernst Baumann , Ronan Le Vezouet , Deborah L. Culbertson
发明人： Christopher Koradin , Markus Kordes , Ernst Baumann , Ronan Le Vezouet , Deborah L. Culbertson
IPC分类号： A01N25/26 , C07C335/12 , A01N47/32 , A61K31/17 , C07D307/82 , A61K31/343 , C07D333/66 , A61K31/381 , A61K31/222 , C07D311/68 , A61K31/353 , C07D335/06 , A61K31/382 , C07D209/40 , A61K31/404 , C07D215/46 , A61K31/47 , A61P33/00 , A01P7/02 , A01P7/04 , A01P5/00
CPC分类号： A01N47/36 , A01N47/32 , C07C335/14 , C07C2602/08 , C07C2602/10 , C07D307/82 , C07D333/66
摘要： The invention relates to substituted amino-thiourea compounds of formula (I), to the enantiomers, diastereomers and salts thereof and to compositions comprising such compounds. The invention also relates to the use of the substituted amino-thiourea compounds, of their salts or of compositions comprising them for combating animal pests. Furthermore the invention relates also to methods of applying such compounds. The substituted amino-thiourea compounds are defined by the following formula (I): wherein A, B, R1, R2, R3, R4, R5.1, R5.2 and R6 are defined as in the description.
摘要翻译：本发明涉及式（I）的取代的氨基 - 硫脲化合物，其涉及其对映体，非对映异构体和盐以及包含这些化合物的组合物。本发明还涉及取代的氨基 - 硫脲化合物，其盐或包含它们的组合物用于对抗动物害虫的用途。此外，本发明还涉及应用这些化合物的方法。取代的氨基 - 硫脲化合物由下式（I）定义：其中A，B，R1，R2，R3，R4，R5.1，R5.2和R6如说明书所定义。

6. 发明申请

US20100041700A1 Substituted 1-(Azolin-2-yl)-Amino-1,2-Heterocyclyl-Ethane Compounds For Combating Pests 审中-公开
标题翻译：取代的1-（唑啉-2-基） - 氨基-1,2-杂环基乙烷化合物用于防治害虫
公开(公告)号：US20100041700A1
公开(公告)日：2010-02-18
申请号：US12519985
申请日：2007-12-11
申请人： Markus Kordes , Ronan Le Vezouet , Christopher Koradin , Ernst Baumann , Deborah L. Culbertson
发明人： Markus Kordes , Ronan Le Vezouet , Christopher Koradin , Ernst Baumann , Deborah L. Culbertson
IPC分类号： A01N43/78 , C07D417/14 , A01N43/42 , A01P7/04 , A01P5/00
CPC分类号： C07D409/06 , A01N43/50 , A01N43/76 , A01N43/78 , C07D401/06 , C07D405/06 , C07D417/12 , C07D417/14
摘要： The present invention relates to 1-(Azolin-2-yl)-amino-1,2-heterocyclyl-ethane compounds, which are useful for combating insects, arachnids and nematodes. The present invention also relates to methods for combating animal pests and to compositions for combating animal pests. It has been found that animal pests can be combated by 1-(Azolin-2-yl)-amino-1,2-heterocyclyl-ethane compounds of the general formula (I): wherein A is a radical of the formulae A1 or A2: and wherein X is sulfur, oxygen or NR7, and HetA, HetB and R1 to R7 are defined as in the description.
摘要翻译：本发明涉及1-（唑啉-2-基） - 氨基-1,2-杂环基 - 乙烷化合物，其可用于防治昆虫，蜘蛛和线虫。本发明还涉及用于对抗动物害虫的方法和用于对抗动物害虫的组合物。已经发现可以通过通式（I）的1-（氮杂-2-基） - 氨基-1,2-杂环基 - 乙烷化合物来对抗动物害虫：其中A是式A1或A2的基团并且其中X是硫，氧或NR 7，并且HetA，HetB和R 1至R 7如描述中所定义。

7. 发明申请

US20080312085A1 Pesticidal Compositions 审中-公开
标题翻译：农药组合物
公开(公告)号：US20080312085A1
公开(公告)日：2008-12-18
申请号：US12158261
申请日：2006-12-11
申请人： Markus Kordes , Livio Tedeschi , Ronan Le Vezouet , Christopher Koradin , Deborah L. Culbertson
发明人： Markus Kordes , Livio Tedeschi , Ronan Le Vezouet , Christopher Koradin , Deborah L. Culbertson
IPC分类号： A01N43/78 , C07D417/12 , A01N43/40 , A01P7/04 , A01N43/42 , A01N43/836
CPC分类号： C07D417/12
摘要： The present invention relates to 1-(Azolin-2-yl)-amino-alkane compounds, which are useful for combating insects, arachnids and nematodes.The present invention also relates to a method for combating animal pests selected from insects, arachnids and nematodes, and to agricultural compositions for combating animal pests.It has been found that animal pests can be combated by 1-(Azolin-2-yl)-amino-alkane compounds of the general formula I: wherein A is a radical of the formulae A1 or A2: and wherein X is sulfur or oxygen and W, B and R1 to R6 are defined as in the description.
摘要翻译：本发明涉及1-（唑啉-2-基） - 氨基 - 烷烃化合物，其可用于防治昆虫，蜘蛛和线虫。本发明还涉及一种防治选自昆虫，蜘蛛和线虫的动物害虫的方法以及用于对抗动物害虫的农业组合物。已经发现，可以通过通式I的1-（氮杂-2-基） - 氨基 - 烷烃化合物与动物害虫相抗衡：其中A是式A1或A2的基团：其中X是硫或氧 W，B，R 1〜R 6如说明书所述。

8. 发明授权

US07989394B2 Substituted 1-(azolin-2-yl)-amino-2-aryl-1-hetaryl-ethane compounds 失效
标题翻译：取代的1-（吡唑-2-基） - 氨基-2-芳基-1-杂芳基 - 乙烷化合物
公开(公告)号：US07989394B2
公开(公告)日：2011-08-02
申请号：US12305419
申请日：2007-06-29
申请人： Markus Kordes , Delphine Breuninger , Ronan Le Vezouet , Christopher Koradin , Livio Tedeschi , Michael Puhl , Deborah L. Culbertson
发明人： Markus Kordes , Delphine Breuninger , Ronan Le Vezouet , Christopher Koradin , Livio Tedeschi , Michael Puhl , Deborah L. Culbertson
IPC分类号： A01N43/76 , A01N43/78 , C07D277/04 , C07D277/08
CPC分类号： C07D333/20 , C07D213/40 , C07D231/12 , C07D307/52 , C07D413/12 , C07D417/12
摘要： The present invention relates to 1-(azolin-2-yl)-amino-2-aryl-1-hetaryl-ethane compounds (I) and 1-(aminothiocarbonylamino)-2-aryl-1-hetaryl-ethane compounds (II) and their salts which are useful for combating animal pest, in particular insects, arachnids and nematodes. Furthermore, the present invention relates to a method for combating animal pests selected from insects, arachnids and nematodes, and to agricultural compositions for combating animal pests. Furthermore, the present invention relates to veterinary compositions for combating animal pests.
摘要翻译：本发明涉及1-（吡唑啉-2-基） - 氨基-2-芳基-1-杂芳基 - 乙烷化合物（I）和1-（氨基硫代羰基氨基）-2-芳基-1-杂芳基 - 乙烷化合物（II）和它们的盐可用于对抗动物害虫，特别是昆虫，蜘蛛和线虫。此外，本发明涉及一种防治选自昆虫，蜘蛛和线虫的动物害虫的方法以及用于对抗动物害虫的农业组合物。此外，本发明涉及用于对抗动物害虫的兽用组合物。

9. 发明申请

US20100167925A1 Substituted Azolin-2-yl-Amino Compounds 审中-公开
标题翻译：取代的唑啉-2-基氨基化合物
公开(公告)号：US20100167925A1
公开(公告)日：2010-07-01
申请号：US12376455
申请日：2007-08-06
申请人： Christopher Koradin , Markus Kordes , Ronan Le Vezouet , Deborah L. Culbertson , Douglas D. Anspaugh
发明人： Christopher Koradin , Markus Kordes , Ronan Le Vezouet , Deborah L. Culbertson , Douglas D. Anspaugh
IPC分类号： A01C1/06 , A01N43/78 , C07D417/02
CPC分类号： C07D417/12 , A01N43/50 , A01N43/76 , A01N43/78 , C07D277/18
摘要： The present invention relates to azolin-2-yl-amino compounds of formulae (I. a) and (1.b) and their salts which are useful for combating animal pest, in particular arthropod and nematodes. The present invention also relates to a method for combating such pests and for protecting crops against infestation or infection by such pests. Furthermore, the present invention relates to veterinary compositions for combating animal pests. Formula (I.a), formula (I.b) wherein n is 0 to 4; X is S, O or NR5; A is —C(R6a)(R6b)—, O, NR7, S, S(O) or S(O)2; B is a bond Or CH2; R1 is H, CN, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkylcarbonyl, C3-C6-cycloalkyl, phenyl, benzyl, etc.; R2a, R2b are H, CN, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkylcarbonyl, (C1-C6-alkyl)-thiocarbonyl, C(O)NRaRb, C(S)NRaRb, (SO2)NRaRb, phenyl, benzyl, 5 or 6 membered heterocyclic ring etc.; or R1 together with R2a is C3-C5-alkandiyl; or R1 together with R2 are C(O); R3a, R3b, R3c, R3d are H, halogen, CN, C1-C6-alkyl, C1-C6-alkylamino, C3-C6-cycloalkyl, phenyl, benzyl, etc.; R4a, R4b are H, halogen, C1-C6-alkyl, C2-C6-alkenyl, phenyl, benzyl, 5 or 6 membered hetaryl; or R4a together with Rb may also be ═O, ═NRC or ═CRdRe; or R2a together with R4a may form a bridging bivalent radical.
摘要翻译：本发明涉及用于对抗动物害虫，特别是节肢动物和线虫的式（Ⅰa）和（Ⅰb）的唑啉-2-基氨基化合物及其盐。本发明还涉及一种防治这种害虫并防止作物抵抗这种害虫侵染或感染的方法。此外，本发明涉及用于对抗动物害虫的兽用组合物。式（Ⅰa），式（Ⅰb）其中n为0-4; X是S，O或NR5; A是-C（R6a）（R6b） - ，O，NR7，S，S（O）或S（O） B是键或CH2; R1是H，CN，C1-C6-烷基，C2-C6-烯基，C1-C6-烷基羰基，C3-C6-环烷基，苯基，苄基等; R2a，R2b是H，CN，C1-C6-烷基，C2-C6-烯基，C1-C6-烷基羰基，（C1-C6-烷基） - 硫代羰基，C（O）NRaRb，C（S）NRaRb，（SO2 ）NRaRb，苯基，苄基，5或6元杂环等; 或R 1与R 2a一起为C 3 -C 5 - 烷二基; 或R 1与R 2一起为C（O）; R3a，R3b，R3c，R3d是H，卤素，CN，C1-C6-烷基，C1-C6-烷基氨基，C3-C6-环烷基，苯基，苄基等; R4a，R4b是H，卤素，C1-C6-烷基，C2-C6-烯基，苯基，苄基，5或6元杂芳基; 或R 4a与R b一起也可以是= O，= NRC或= CRdRe; 或R 2a与R 4a一起形成桥连二价基团。

10. 发明申请

US20100010058A1 Azoline Compounds for Combating Arthropod Pests 审中-公开
标题翻译：用于防治节肢动物害虫的唑啉化合物
公开(公告)号：US20100010058A1
公开(公告)日：2010-01-14
申请号：US12305267
申请日：2007-05-25
申请人： Christopher Koradin , Markus Kordes , Ronan Le Vezouet , Deborah L. Culbertson , Douglas D. Anspaugh , Henry Van Tuyl Cotter
发明人： Christopher Koradin , Markus Kordes , Ronan Le Vezouet , Deborah L. Culbertson , Douglas D. Anspaugh , Henry Van Tuyl Cotter
IPC分类号： A01N43/78 , C07D277/18 , A01P5/00 , A01P7/00
CPC分类号： C07D277/18
摘要： The present invention relates to azoline compounds and their salts which are useful for combating arthropod pests. The present invention also relates to a method for combating arthropod pests and to agricultural compositions for combating said pests. It has been found that these objectives can be achieved by azoline compounds of the general formulae Ia or Ib, wherein X is S, O or NR4; Ar is phenyl or a 5 or 6 membered heteroaromatic ring; R1 is H, C1-C6-alkyl, C2-C6-alkenyl, phenyl, a heteroaromatic ring etc.; R2a, R2b are H, CN, C1-C6-alkyl etc.; R1 together with R2a may also form a linear C2-C4-alkandiyl; R3a-d are H, halogen, C1-C6-alkyl etc.
摘要翻译：本发明涉及可用于防治节肢动物害虫的唑啉化合物及其盐。本发明还涉及一种防治节肢动物害虫的方法和用于对抗所述害虫的农业组合物。已经发现，这些目的可以通过通式Ia或Ib的唑啉化合物来实现，其中X是S，O或NR 4; Ar是苯基或5或6元杂芳环; R1是H，C1-C6-烷基，C2-C6-烯基，苯基，杂芳环等; R2a，R2b是H，CN，C1-C6-烷基等; R1与R2a一起也可以形成直链C 2 -C 4 - 烷二基; R3a-d为H，卤素，C1-C6烷基等。

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