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1. 发明申请

WO2007128744A2 TRIAZINE DERIVATIVES 审中-公开
标题翻译： TRIAZINE衍生物
公开(公告)号：WO2007128744A2
公开(公告)日：2007-11-15
申请号：PCT/EP2007054239
申请日：2007-05-02
申请人： CIBA SC HOLDING AG , EHLIS THOMAS , BORSOS ELEK
发明人： EHLIS THOMAS , BORSOS ELEK
IPC分类号： C07D251/52 , A61Q17/04 , C07D251/70
CPC分类号： C07D251/52 , C07D251/70
摘要： Disclosed are triazine derivatives of formula (1), wherein X 1 is a bivalent radical of formula (1a) -NR 9 -A-NR 9 -; (1b); or (1c) *-O-A-O-* A and A' independently from each other are unsubstituted or substituted, straight-chain or branched C 1 -C 12 alkylene, which is optionally interrupted by C 5 -C 12 cycloalkylene, N, O or S; C 5 -C 12 cycloalkylene; biphenylene; C 6 -C 10 arylene; or C 5 -C 10 arylene-(C 1 -C 12 alkylene); R 1 is a radical of formula (1d); (1e); (1f); (1g); or (1h); R 2 and R 3 independently from each other are hydrogen; C 1 -C 12 alkyl; OR 7 ; NR 7 R 8 ; C 6 -C 10 aryl; X 2 is O, or NH; W 1 is C 1 -C 20 alkyl; or a group Sp-Sil; Sp is a straight-chain or branched saturated or single or multiple unsaturated C 3 -C 12 hydrocarbon; Sil is a silane; an oligosiloxane; or a polysiloxane moiety; and R 4 , R 5 R 6 , R 7 , R 8 and R 9 independently from each other are hydrogen; C 1 -C 12 alkyl; or C 3 -C 12 cycloalkyl.
摘要翻译：公开了式（1）的三嗪衍生物，其中X 1是式（1a）的二价基团-NR 9 -A-NR 9 - ; （1B）; 或（1c）* -OAO- * A和A'彼此独立地是未取代或取代的直链或支链C 1 -C 12亚烷基，其是任选被C 5 -C 12亚环烷基，N，O或S中断; ç_{5 -C _{12 亚环烷基; 联苯; ç_{6 -C _{10 亚芳基; 或C 5 -C 10亚芳基 - （C 1 -C 12 - 亚烷基）; R 1是式（1d）的基团; （1E）; （1F）; （1G）; 或（1h）; R 2和R 3彼此独立地是氢; ç_{1 -C _{12 烷基; OR _{7 ; NR _{7 - [R _{8 ; ç_{6 -C _{10 芳基; X 2是O或NH; W 1是C 1 -C 20烷基; 或一组Sp-Sil; Sp是直链或支链饱和或单或多不饱和C 3 -C 12烃; 硅是硅烷; 低聚硅氧烷; 或聚硅氧烷部分; 和R 4，R 5 R 6，R 7，R 8和R 8，和 R 9彼此独立地是氢; ç_{1 -C _{12 烷基; 或C 3 -C 12环烷基。}}}}}}}}}}}}}

2. 发明申请

WO2004052837A3 AMINO SUBSTITUTED HYDROXYPHENYL BENZOPHENONE DERIVATIVES 审中-公开
标题翻译：氨基取代的羟苯基苯并噻吩酮衍生物
公开(公告)号：WO2004052837A3
公开(公告)日：2004-09-10
申请号：PCT/EP0350937
申请日：2003-12-03
申请人： CIBA SC HOLDING AG , HAASE JUERG , EHLIS THOMAS , BORSOS ELEK , MUELLER STEFAN
发明人： HAASE JUERG , EHLIS THOMAS , BORSOS ELEK , MUELLER STEFAN
IPC分类号： A61K8/42 , A61K8/44 , A61K8/49 , A61Q17/04 , C07C229/52 , C07C237/32 , C07C237/34 , C07C237/40 , C07C237/42 , C07D277/46 , C07D277/66 , C07D295/18 , C07D295/192 , C07D313/12 , A61K7/44
CPC分类号： C07D295/192 , A61K8/42 , A61K8/44 , A61K8/49 , A61K8/4973 , A61Q17/04 , C07C229/52 , C07C237/32 , C07C237/34 , C07C237/40 , C07C237/42 , C07D277/46 , C07D277/66 , C07D313/12
摘要： Described are amino substituted hydroxyphenyl benzophenone derivatives of formula (I), wherein R1, and R2 independently from each other are; C1,-C20alkyl; C2-C20alkenyl; C3-C10,cycloalkyl; C3-C10cycloalkenyl; or R1, and R2 together with the linking nitogen atom form a 5- or 6-membered heterocyclic ring; n1 is a number from 1 to 4; when n1=1, R3 is a saturated or unsaturated heterocyclic radical; hydroxy-C1-C5alkyl; cyclohexyl optionally substituted with one or more C1,-C5alkyl; phenyl optionally substituted with a heterocyclic radical, aminocarbonyl or C1-C5alkylcarboxy; wenn n1 is 2, R3 is an alkylene-, cycloalkylene- or alkenylene radical which is optionally substituted by a carbonyl- or carboxy group; o R3 together with A forms a bivalent radical of the formula (Ia), wherein n2 is a number from 1 to 3; when n1 is 3, R3 is an alkanetriyl radical; wenn n1 is 4, R3 is an alkanetetrayl radical; A is -O-; or -N(R5)-; and R5 is hydrogen; C1-C5alkyl; or hydroxy-C1-C5alkyl. The compounds are useful as UV filters in sunscreen applications.
摘要翻译：描述了式（I）的氨基取代的羟基苯基二苯甲酮衍生物，其中R1和R2彼此独立地为; C1，-C20alkyl; C2-C20alkenyl; C3-C10，环烷基; C3-C10cycloalkenyl; 或者R1和R2与连接氮原子一起形成5-或6-元杂环; n1是从1到4的数字; 当n1 = 1时，R3是饱和或不饱和的杂环基; 羟基C1-C5烷基; 任选被一个或多个C1-C5烷基取代的环己基; 任选被杂环基，氨基羰基或C 1 -C 5烷基羧基取代的苯基; n1是2，R3是任选被羰基或羧基取代的亚烷基 - ，亚环烷基 - 或亚烯基; R3与A一起形成式（Ia）的二价基团，其中n2是1至3的数; 当n1是3时，R3是链烷三基; 文n1为4，R3为链烷四基; A是-O-; 或-N（R 5） - ; 并且R5是氢; C1-C5烷基; 或羟基-C 1 -C 5烷基。该化合物在防晒应用中用作UV过滤剂。

3. 发明专利

JP2000063366A DIRESOLCINYL-ALKOXY AND ARYLOXY-S-TRIAZINE 失效
公开(公告)号：JP2000063366A
公开(公告)日：2000-02-29
申请号：JP10249099
申请日：1999-04-09
申请人： CIBA SC HOLDING AG
发明人： EHLIS THOMAS , BORSOS ELEK , LUTHER HELMUT , HERZOG BERND
IPC分类号： A61K8/00 , A61K8/49 , A61Q17/04 , C07D251/22 , C07D251/26 , C07D405/12 , C08K5/3492 , C09K3/00 , C09K15/30 , A61K7/00 , A61K7/42
摘要： PROBLEM TO BE SOLVED: To obtain the subject new compound which is a UV-A absorber and useful as light protecting agent in cosmetics, medicines and veterinary preparations as an ultraviolet screening agent. SOLUTION: This compound is represented by formula I [R1 is a 2-30C alkyl, a 2-30C alkenyl, a 5-12C cycloalkyl or the like; R2 to R4 are each H, hydroxyl, a 1-30C alkyl or alkenyl; R5 is H or a 1-5C alkyl], e.g. a compound of formula II. The compound of formula I is obtained by reacting, e.g. cyanuric chloride with a compound of the formula R1-OH in the presence of a solvent (e.g. acetone) to afford dichloroaryloxytriazine and reacting the compound with resorcinol by Friedel-Crafts reaction in the presence of a catalyst (e.g. aluminum chloride). The compound of formula I is useful for protecting organic materials, especially skins and hairs of human and animals which are sensitive to ultraviolet rays from ultraviolet irradiation.

4. 发明专利

BRPI0308369B1 Composição absorvedora de uv compreendendo um composto hidroxifeniltriazina e processo para a preparação do referido composto 未知
公开(公告)号：BRPI0308369B1
公开(公告)日：2015-05-26
申请号：BR0308369
申请日：2003-03-04
申请人： CIBA SC HOLDING AG
发明人： HAASE JÜRG , EHLIS THOMAS , BORSOS ELEK , HÜGLIN DIETMAR , HERZOG BERND
IPC分类号： C07D249/20 , A61K8/00 , A61K8/35 , A61K8/49 , A61Q5/02 , A61Q17/04 , C07D251/16 , C09K3/00

5. 发明专利

BR0316607B1 未知
公开(公告)号：BR0316607B1
公开(公告)日：2014-12-23
申请号：BR0316607
申请日：2003-12-03
申请人： CIBA SC HOLDING AG
发明人： BORSOS ELEK , HAASE JUERG , EHLIS THOMAS , MUELLER STEFAN
IPC分类号： A61K8/42 , A61K8/44 , A61K8/49 , A61Q17/04 , C07C229/52 , C07C237/32 , C07C237/34 , C07C237/40 , C07C237/42 , C07D277/46 , C07D277/66 , C07D295/18 , C07D295/192 , C07D313/12
摘要： Described are amino substituted hydroxyphenyl benzophenone derivatives of formula (I), wherein R 1 , and R 2 independently from each other are; C 1 -C 20 alkyl; C 2 -C 20 -alkenyl; C 3 -C 10 cycloalkyl; C 3 -C 10 cycloalkenyl; or R 1 , and R 2 together with the linking nitrogen atom form a 5- or 6-membered heterocyclic ring; n 1 is a number from 1 to 4; when n 1 =1, R 3 is a saturated or unsaturated heterocyclic radical; hydroxy-C 1 -C 5 alkyl; cyclohexyl optionally substituted with one or more C 1 -C 5 alkyl; phenyl optionally substituted with a heterocyclic radical, aminocarbonyl or C 1 -C 5 alkylcarboxy; when n 1 is 2, R 3 is an alkylene-, cycloalkylene- or alkenylene radical which is optionally substituted by a carbonyl- or carboxy group; o R 3 together with A forms a bivalent radical of the formula (Ia), wherein n 2 is a number from 1 to 3; when n 1 is 3, R 3 is an alkanetriyl radical; when n 1 is 4, R 3 is an alkanetetrayl radical; A is -O-; or -N(R 5 )-; and R 5 is hydrogen; C 1 -C 5 alkyl; or hydroxy-C 1 -C 5 alkyl. The compounds are useful as UV filters in sunscreen applications.

6. 发明专利

DE60320093D1 未知
公开(公告)号：DE60320093D1
公开(公告)日：2008-05-15
申请号：DE60320093
申请日：2003-03-04
申请人： CIBA SC HOLDING AG
发明人： HAASE JUERG , EHLIS THOMAS , BORSOS ELEK , HUEGLIN DIETMAR , HERZOG BERND
IPC分类号： A61Q17/04 , C07D249/20 , A61K8/00 , A61K8/35 , A61K8/49 , A61Q5/02 , C07D251/16 , C09K3/00
摘要： UV absorber compositions are described, comprising (a) from 1 to 99% by weight of a hydroxyphenyltriazine compound of formula (I) wherein R 1 , R 2 and R 3 are each independently of the others C 1 -C 18 alkyl; C 2 -C 10 ,alkenyl; or phenyl-C 1 -C 4 alkyl; R 4 is hydrogen; or C 1 -C 5 alkyl; and (b) from 99 to 1% by weight of a further UV absorber selected from the group of (b) hydroxyphenyltriazines that are different from component (a), (b 2 ) benzotriazoles, (b 3 ) dibenzoylmethane derivatives and (b 4 ) camphor derivatives. The compositions are suitable as UV filters in cosmetic compositions

7. 发明专利

BR0308369A 未知
公开(公告)号：BR0308369A
公开(公告)日：2005-01-11
申请号：BR0308369
申请日：2003-03-04
申请人： CIBA SC HOLDING AG
发明人： HAASE J RG , EHLIS THOMAS , BORSOS ELEK , GLIN DIETMAR H , HERZOG BERND
IPC分类号： C07D249/20 , A61K8/00 , A61K8/35 , A61K8/49 , A61Q5/02 , A61Q17/04 , C07D251/16 , C09K3/00 , A61K7/42
摘要： UV absorber compositions are described, comprising (a) from 1 to 99% by weight of a hydroxyphenyltriazine compound of formula (I) wherein R 1 , R 2 and R 3 are each independently of the others C 1 -C 18 alkyl; C 2 -C 10 ,alkenyl; or phenyl-C 1 -C 4 alkyl; R 4 is hydrogen; or C 1 -C 5 alkyl; and (b) from 99 to 1% by weight of a further UV absorber selected from the group of (b) hydroxyphenyltriazines that are different from component (a), (b 2 ) benzotriazoles, (b 3 ) dibenzoylmethane derivatives and (b 4 ) camphor derivatives. The compositions are suitable as UV filters in cosmetic compositions

8. 发明专利

AU2365399A Diresorcinyl-alkoxy- and -aryloxy-S-triazines 未知
公开(公告)号：AU2365399A
公开(公告)日：1999-10-21
申请号：AU2365399
申请日：1999-04-08
申请人： CIBA SC HOLDING AG
发明人： EHLIS THOMAS , BORSOS ELEK , LUTHER HELMUT , HERZOG BERND
IPC分类号： A61K8/00 , A61K8/49 , A61Q17/04 , C07D251/22 , C07D251/26 , C07D405/12 , C08K5/3492 , C09K3/00 , C09K15/30 , C07D251/24 , C07D311/58 , A61K7/42
摘要： 2,4-Diresorcinyl 6-(alkoxy or aryloxy)-1,3,5-triazines (I) are new. Also new are 2,4-dichlorotriazine intermediates (II). Diresorcinyl triazines of formula (I) are new. R1 = 2-20C alkyl, 2-30C alkenyl, 5-12C cycloalkyl (optionally substituted by one or more 1-5C alkyl), (1-5C)alkoxy-(1-12C) alkyl, 1-12C aminoalkyl (optionally N-substituted or N,N-disubstituted by 1-5C alkyl), -(CH2)n(O)mPh or a group of formula (a)-(c); R2-R4 - H, OH, 1-30C alkyl or 2-30C alkenyl; R5 = H or 1-5C alkyl; m = 0 or 1; n = 1-5. Independent claims are included for : (i) compounds (I) in micronized form, where 2-20C alkyl as a value for R1 is replaced by 1-7C alkyl; (ii) dichlorotriazine intermediates of formula (II), provided that R1 is 8-20C alkyl, -(CH2)n(O)mPh or a group of formula (a)-(c); and (iii) the preparation of (I).

9. 发明专利

AT390950T 未知
公开(公告)号：AT390950T
公开(公告)日：2008-04-15
申请号：AT03709744
申请日：2003-03-04
申请人： CIBA SC HOLDING AG
发明人： HAASE JUERG , EHLIS THOMAS , BORSOS ELEK , HUEGLIN DIETMAR , HERZOG BERND
IPC分类号： A61Q17/04 , C07D249/20 , A61K8/00 , A61K8/35 , A61K8/49 , A61Q5/02 , C07D251/16 , C09K3/00
摘要： UV absorber compositions are described, comprising (a) from 1 to 99% by weight of a hydroxyphenyltriazine compound of formula (I) wherein R 1 , R 2 and R 3 are each independently of the others C 1 -C 18 alkyl; C 2 -C 10 ,alkenyl; or phenyl-C 1 -C 4 alkyl; R 4 is hydrogen; or C 1 -C 5 alkyl; and (b) from 99 to 1% by weight of a further UV absorber selected from the group of (b) hydroxyphenyltriazines that are different from component (a), (b 2 ) benzotriazoles, (b 3 ) dibenzoylmethane derivatives and (b 4 ) camphor derivatives. The compositions are suitable as UV filters in cosmetic compositions

10. 发明专利

AU2003298343A1 AMINO SUBSTITUTED HYDROXYPHENYL BENZOPHENONE DERIVATIVES 未知
公开(公告)号：AU2003298343A1
公开(公告)日：2004-06-30
申请号：AU2003298343
申请日：2003-12-03
申请人： CIBA SC HOLDING AG
发明人： HAASE JURG , EHLIS THOMAS , BORSOS ELEK , MULLER STEFAN
IPC分类号： A61K8/42 , A61K8/44 , A61K8/49 , A61Q17/04 , C07C229/52 , C07C237/32 , C07C237/34 , C07C237/40 , C07C237/42 , C07D277/46 , C07D277/66 , C07D295/18 , C07D295/192 , C07D313/12
摘要： Described are amino substituted hydroxyphenyl benzophenone derivatives of formula (I), wherein R 1 , and R 2 independently from each other are; C 1 -C 20 alkyl; C 2 -C 20 -alkenyl; C 3 -C 10 cycloalkyl; C 3 -C 10 cycloalkenyl; or R 1 , and R 2 together with the linking nitrogen atom form a 5- or 6-membered heterocyclic ring; n 1 is a number from 1 to 4; when n 1 =1, R 3 is a saturated or unsaturated heterocyclic radical; hydroxy-C 1 -C 5 alkyl; cyclohexyl optionally substituted with one or more C 1 -C 5 alkyl; phenyl optionally substituted with a heterocyclic radical, aminocarbonyl or C 1 -C 5 alkylcarboxy; when n 1 is 2, R 3 is an alkylene-, cycloalkylene- or alkenylene radical which is optionally substituted by a carbonyl- or carboxy group; o R 3 together with A forms a bivalent radical of the formula (Ia), wherein n 2 is a number from 1 to 3; when n 1 is 3, R 3 is an alkanetriyl radical; when n 1 is 4, R 3 is an alkanetetrayl radical; A is -O-; or -N(R 5 )-; and R 5 is hydrogen; C 1 -C 5 alkyl; or hydroxy-C 1 -C 5 alkyl. The compounds are useful as UV filters in sunscreen applications.

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