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1. 发明申请

WO2013135606A1 METHOD FOR PRODUCING AN AQUEOUS SUSPENSION CONCENTRATE FORMULATION OF A PYRIPYROPENE INSECTICIDE 审中-公开
标题翻译：生产杀微生物剂的水悬浮浓缩液配方的方法
公开(公告)号：WO2013135606A1
公开(公告)日：2013-09-19
申请号：PCT/EP2013/054828
申请日：2013-03-11
申请人： BASF SE , BASF SCHWEIZ AG
发明人： KNIERIEM, Torsten , CHIODO, Tiziana , KORADIN, Christopher , WEBER, Tanja , WEISHAAR, Walter
IPC分类号： A01N43/90 , A01N53/00 , A01N25/04 , A01P7/04
CPC分类号： A01N53/00 , A01N25/08 , A01N43/90 , A01N25/04 , A01N2300/00
摘要： The present invention relates to a method for producing an aqueous suspension concentrate formulation and novel suspension concentrate formulations of the compound of formula I. The method comprises: a) providing an aqueous slurry of coarse particles of the compound of the formula I, where the compound of the formula I is at least partially present in its crystalline form B, which, in an X-ray powder diffractogram at 25°C and Cu-Kα radiation, shows at least three, preferably at least four, in particular at least 5 or at least 7 or at least 9 or all of the following reflexes, given as 2θ values:8.0± 0.2°, 9.5± 0.2°, 10.7± 0.2°, 11.0± 0.2°, 11.2± 0.2°,11.7± 0.2°, 14.2± 0.2°, 15.6± 0.2°, 6.5± 0.2°, 17.7± 0.2°, 21.5± 0.2°; b) comminuting the coarse particles in the slurry of the compound of formula I, which is at least partially present in its form B, in the presence of the at least one surfactant.
摘要翻译：本发明涉及一种制备水性悬浮液浓缩物制剂的方法和式I化合物的新型悬浮浓缩物制剂。该方法包括：a）提供式I化合物的粗颗粒的含水浆液，其中化合物式I的至少一部分至少部分以其结晶形式B存在，其在25℃的X射线粉末衍射图和Cu-Kalpha辐射中显示出至少三个，优选至少四个，特别是至少5个或至少7或至少9或全部以下反射，以2θ值给出：8.0±0.2°，9.5±0.2°，10.7±0.2°，11.0±0.2°，11.2±0.2°，11.7±0.2°，14.2 ±0.2°，15.6±0.2°，6.5±0.2°，17.7±0.2°，21.5±0.2°; b）在存在至少一种表面活性剂的情况下粉碎至少部分以其B形式存在的式I化合物的浆料中的粗颗粒。

2. 发明申请

WO2015169883A1 CRYSTALLINE FORM B OF AN ANTHRANILAMIDE INSECTICIDE AND CONVERSION OF FORM B INTO FORM A 审中-公开
标题翻译： ANTHRANILAMIDE INSECTICIDE的晶体形式B和形式B的转化形式A
公开(公告)号：WO2015169883A1
公开(公告)日：2015-11-12
申请号：PCT/EP2015/060018
申请日：2015-05-07
申请人： BASF SE
发明人： KÖRBER, Karsten , KORADIN, Christopher , ZIERKE, Thomas , CHIODO, Tiziana , VIERTELHAUS, Martin
IPC分类号： A01N43/56 , A01P7/04
CPC分类号： A01N43/56 , A01N25/12
摘要： The present invention relates to a crystalline form B of the anthranilamide insecticide 2-(3- chloro-2-pyridyl)-N-[2-methyl-4-chloro-6-[(diethyl-A4-sulfanylidene)carbamoyl]phenyl]-5- (trifluoromethyl)pyrazole-3-carboxamide (compound I) and to different processes for converting said crystalline form B into a crystalline form A of compound I.
摘要翻译：本发明涉及邻氨基苯甲酰胺杀虫剂2-（3-氯-2-吡啶基）-N- [2-甲基-4-氯-6 - [（二乙基亚苄基）氨基甲酰基]苯基] -5-（三氟甲基）吡唑-3-甲酰胺（化合物I），以及将所述结晶B转化为化合物I的结晶形式A的不同方法。

3. 发明申请

WO2009133178A1 VERFAHREN ZUR HERSTELLUNG VON 2-(AMINOMETHYLIDEN)-4,4-DIFLUOR-3-OXOBUTTERSÄUREESTERN 审中-公开
标题翻译：用于生产2-（氨基亚甲基）-4,4-二氟-3-氧代丁酸酯
公开(公告)号：WO2009133178A1
公开(公告)日：2009-11-05
申请号：PCT/EP2009/055283
申请日：2009-04-30
申请人： BASF SE , ZIERKE, Thomas , MAYWALD, Volker , RACK, Michael , SMIDT, Sebastian Peer , KEIL, Michael , WOLF, Bernd , KORADIN, Christopher
发明人： ZIERKE, Thomas , MAYWALD, Volker , RACK, Michael , SMIDT, Sebastian Peer , KEIL, Michael , WOLF, Bernd , KORADIN, Christopher
IPC分类号： C07C227/16 , C07C229/30 , C07D231/14
CPC分类号： C07D231/14 , C07C229/30 , C07D295/145
摘要： Die vorliegende Erfindung betrifft ein Verfahren zur Herstellung von difluormethylsubsti- tuierten Pyrazol4-ylcarbonsäuren und deren Ester, 2-(Aminomethyliden)-4,4-difluor-3- oxobuttersäureester der Formel (I), worin R 1 , R 2 und R 3 unabhängig voneinander für C 1 -C 6 -Alkyl, C 1 -C 6 -Haloalkyl, C 2 -C 6 -Alkenyl, C 3 -C 10 -Cycloalkyl oder Benzyl steht oder NR 2 R 3 für einen 5- bis 10-gliedrigen heterocyclischen Rest steht, ein Verfahren zur Herstellung von Verbindungen der Formel (I), bei dem man einen entsprechenden 3-Aminoacrylsäureester mit Difluoracetylfluorid umsetzt sowie die Verwendung von Verbindungen der Formel (I) in dem Verfahren zur Herstellung von difluormethylsubstituierten Pyrazol- 4-ylcarbonsäuren und deren Ester.
摘要翻译：本发明涉及一种用于difluormethylsubsti的制备 - 取代的吡唑基甲酸及其酯，2-（氨基亚甲基）的式（I）的-4,4-二氟-3-氧代丁酸乙酯，其特征在于R1，R2和R3各自独立地为C1 C6烷基，C1-C6卤代烷基，C2-C6链烯基，C3-C10环烷基或苄基或NR2R3表示5至10元杂环基团，为式I化合物的制备方法（I），该方法包括用二氟乙酰氟一个相应的3-氨基丙烯酸酯，以及用于制备吡唑difluormethylsubstituierten唑-4-基甲酸和它们的酯的使用过程中的式（I）的化合物的反应。

4. 发明申请

WO2009004032A1 1-(AZOLIN-2-YL)AMINO-1,2-DIPHENYLETHANE COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
标题翻译： 1-（AZOLIN-2-YL）氨基-1,2-二苯醚化合物，用于组合动物饲料
公开(公告)号：WO2009004032A1
公开(公告)日：2009-01-08
申请号：PCT/EP2008/058517
申请日：2008-07-02
申请人： BASF SE , KORDES, Markus , KORADIN, Christopher , LE VEZOUET, Ronan , BAUMANN, Ernst , CULBERTSON, Deborah L. , ANSPAUGH, Douglas D. , OLOUMI-SADEGHI, Hassan , EBUENGA, Cecile
发明人： KORDES, Markus , KORADIN, Christopher , LE VEZOUET, Ronan , BAUMANN, Ernst , CULBERTSON, Deborah L. , ANSPAUGH, Douglas D. , OLOUMI-SADEGHI, Hassan , EBUENGA, Cecile
IPC分类号： C07D233/48 , C07D263/28 , C07D277/18 , C07D417/12 , C07D417/06 , A01N43/50 , A01N43/76 , A01N43/78
CPC分类号： C07D263/28 , A01N43/50 , A01N43/76 , A01N43/78 , A01N47/12 , A01N47/16 , C07D233/48 , C07D277/18 , C07D417/06 , C07D417/12
摘要： The present invention relates to 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and to their salts which are useful for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds, wherein A is a radical of formulae A.1 or A.2 wherein # denotes the bond to the remaining compound of formula I, X is selected from O, S and NR x , R 1 is selected from the group consisting of -OR A , -NR B1 R B2 , -C(=O)-R C , -C(=O)-OR D , -C(=O)-SR E , -C(=O)-NR B1 R B2' , -C(=S)-R C' , -C(=S)-OR D' , -C(=S)-SR E' , -C(=S)-NR B1 R B2 , -C(=NR 1a )-R C' , -C(=NR 1b )-OR D' , -C(=NR 1c )-SR E' , -C(=NR 1d )-NR B1 R B2 , -S(=O)-R F , -S(=O) 2 -R G , -S(=O) 2 -NR B1 R B2' , -P(=O)R H1 R H2 , -P(=S)R H1 R H2 , -B-C(=O)-R I , -B-O-C(=O)-R I , -B-S-C(=O)-R I , -B-N(R J )-C(=O)-R K , -B-C(=S)-R K , -B-O-C(=S)-R K , -B-S-C(=S)-R K , -B-N(R J )-C(=S)-R K , C 1 -C 8 -alkenyl, C 1 -C 8 -alkynyl, C 3 -C 8 -cycloalkyl, which is unsubstituted or may carry 1 to 4 substituents R 1e , naphthyl, which is unsubstituted or may carry 1 to 4 substituents R 1f , a saturated or partially unsaturated heterocycle, which is unsubstituted or may carry 1 to 4 substituents R 1g , hetaryl, which is unsubstituted or may carry 1 to 4 substituents R 1h , and C 1 -C 6 -alkyl, which carries a radical selected from the group consisting of -NR 1i R 1j , C 1 -C 4 -alkoxycarbonyl, C 3 -C 8 -cycloalkyl, aryl, aryloxy, arylthio, heterocyclyl, heterocyclyloxy and heterocyclylthio, R 2 , R 3 , R 4 , R 5 , R 6 and R 7 are each independently hydrogen, halogen, OH, SH, NH 2 , SO 3 H, COOH, cyano, nitro, C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 1 -C 6 -alkylamino etc.
摘要翻译：本发明涉及式I的1-（吡唑-2-基）氨基-1,2-二苯基乙烷化合物及其盐，其可用于防治动物害虫。本发明还涉及通过使用这些化合物，种子和包含所述化合物的农业和兽医组合物来控制动物害虫的方法，其中A是式A.1或A.2的基团，其中＃表示与剩余的式I化合物，X选自O，S和NR x，R1选自-ORA，-NRB1RB2，-C（= O）-RC，-C（= O）-OR，-C （= O）-SRE，-C（= O）-NRB1RB2'，-C（= S）-RC'，-C（= S）-OR'，-C（= S）-SRE' =（NR1c）-SR'，-C（= NR1d）-NRB1RB2，-S（= O））-RF，-S（= O）2 -RG，-S（= O）2 -NRB 1 R B 2'，-P（= O）RH1RH 2，-P（= S）RH1RH 2，-BC（= O） -BOC（= O）-RI，-BSC（= O）-RI，-BN（RJ）-C（= O）-RK，-BC（= S）-RK，-BOC（= S）-RK， -BSC（= S）-RK，-BN（RJ）-C（= S）-RK，C1-C8-烯基，C1-C8-炔基，C3-C8-环烷基，其未被取代或可携带1至4 取代基R 1e，萘基，其是未取代的或可以携带1至4个取代基R 1f，饱和或部分不饱和的杂环，其为未制备的或可以携带1至4个未取代的或可以携带1至4个取代基R 1h的取代基R 1g，杂芳基，其中C 1 -C 6 - 烷基带有选自以下的基团：-NR 1 1 R 1，C 1 -C 4 - 烷氧基羰基， C 3 -C 8 - 环烷基，芳基，芳氧基，芳硫基，杂环基，杂环基氧基和杂环硫基，R 2，R 3，R 4，R 5，R 6和R 7各自独立地为氢，卤素，OH，SH，NH 2，SO 3 H，COOH，氰基，硝基， C 1 -C 6 - 烷基，C 1 -C 6 - 烷氧基，C 1 -C 6烷基氨基等

5. 发明申请

WO2022157323A1 METHOD FOR PREPARING AN ENANTIOMERICALLY ENRICHED FORM OF 3-(2-CHLOROTHIAZOL-5-YL)-8-METHYL-7-OXO-6-PHENYL-2,3-DIHYDROTHIAZOLO[3,2-A]PYRIMIDIN-4-IUM-5-OLATE 审中-公开
公开(公告)号：WO2022157323A1
公开(公告)日：2022-07-28
申请号：PCT/EP2022/051368
申请日：2022-01-21
申请人： BASF SE
发明人： KORADIN, Christopher , MCLAUGHLIN, Martin John , GOETZ, Roland , KADUSKAR, Rahul , SHINDE, Harish
IPC分类号： C07D495/04
摘要： The present invention relates to a method for preparing an enantiomerically enriched form of 3-(2-chlorothiazol-5-yl)-8-methyl-7-oxo-6-phenyl-2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium-5-olate.

6. 发明申请

WO2020152104A3 METHOD FOR PRODUCTION OF 4-CYANO BENZOIC ACID OR SALTS THEREOF 审中-公开
公开(公告)号：WO2020152104A3
公开(公告)日：2020-07-30
申请号：PCT/EP2020/051288
申请日：2020-01-20
申请人： BASF SE
发明人： GHISLIERI, Diego , WILLRODT, Christian , KORADIN, Christopher , SEEMAYER, Stefan , SCHACHTSCHABEL, Doreen , BALDENIUS, Kai-Uwe , GOETZ, Roland
IPC分类号： C12P13/00 , C12P7/40
摘要： The invention is directed to methods for the production of 4-cyano benzoic acid or salts thereof from terephthalonitrile using nitrilase as catalyst and compositions comprising 4-cyano benzoic acid.

7. 发明申请

WO2018197541A1 PROCESS FOR PREPARING OPTICALLY ACTIVE 2,3-DIHYDROTHIAZOLO[3,2-A]PYRIMIDIN-4-IUM COMPOUNDS 审中-公开
公开(公告)号：WO2018197541A1
公开(公告)日：2018-11-01
申请号：PCT/EP2018/060555
申请日：2018-04-25
申请人： BASF SE
发明人： SHINDE, Harish , KORADIN, Christopher , DICKHAUT, Joachim , GOETZ, Roland , RACK, Michael , KLAUBER, Eric , NARAYANAN, Sukunath , RAUT, Dhanyakumar
IPC分类号： C07D513/04 , C07D417/04 , C07D277/32 , A01N43/78
摘要： The present invention relates to a process for preparing optically active compounds of formula X and intermediates thereof, X wherein the variables of compound of formula X are as defined in the claims or the description.

8. 发明申请

WO2014154807A1 PROCESS FOR PREPARING SULFIMINES AND THEIR IN-SITU CONVERSION INTO N-(2-AMINO-BENZOYL)-SULFIMINES 审中-公开
标题翻译：制备硫化物的方法及其在N-（2-氨基苯甲酰基） - 硫脲中的原位转化
公开(公告)号：WO2014154807A1
公开(公告)日：2014-10-02
申请号：PCT/EP2014/056164
申请日：2014-03-27
申请人： BASF SE
发明人： FRASSETTO, Timo , JOCKERS, Harald , KORADIN, Christopher , ZIERKE, Thomas , KÖRBER, Karsten
IPC分类号： A01N43/56 , C07D401/04
CPC分类号： C07C381/10 , A01N37/28 , A01N43/56 , C07C2601/02 , C07D401/04 , C07D409/14
摘要： The present invention relates to a process for preparing a compound of the formulae (la) or (lb), or a mixture thereof, wherein R 1 and R 2 independently of one another are hydrogen, C 1 -C 10 -alkyl, C 1 -C 10 -haloalkyl, C 3 -C 10 -cycloalkyl, C 3 -C 10 -halocycloalkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -haloalkenyl or together represent an aliphatic chain, or the like; A- is HSO 4 - or 1/2 SO4 2- ; the process comprising the reaction of a sulfide of formula SR 1 R 2 with hydroxylamine- O-sulfonic acid of formula; wherein the reaction is carried out in an aqueous medium in the presence of a base. The present invention also relates to a process for preparing a compound of the formula (IV), wherein R 3 is halogen, cyano, C 1 -C 8 -alkyl, C 1 -C 8 -haloalkyl, C 3 -C 8 -cycloalkyl, C 3 -C 8 - halocycloalkyl, C 2 -C 8 -alkenyl, C 2 -C 8 -haloalkenyl, C 1 -C 8 -alkoxy, phenyl, or the like; R 4 is hydrogen, C 1 -C 10 -alkyl, C 1 -C 10 -haloalkyl, C 3 -C 8 -cycloalkyl, C 3 -C 8 -halocycloalkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -haloalkenyl, phenyl, or the like; p is 0, 1, 2, 3 or 4; the process comprising: (i) providing the compound of the formulae (la) or (lb), or a mixture thereof, (ii) reacting a compound of the formulae (la) or (lb), or a mixture thereof, obtained in step (i) with a compound of the formula (V) in the presence of a base,
摘要翻译：本发明涉及制备式（Ia）或（Ib）化合物或其混合物的方法，其中R 1和R 2彼此独立地是氢，C 1 -C 10 - 烷基，C 1 -C 10 - 卤代烷基， C 3 -C 10 - 环烷基，C 3 -C 10 - 卤代环烷基，C 2 -C 10 - 烯基，C 2 -C 10 - 卤代烯基或一起代表脂族链等; A-是HSO4-或1/2 SO42-; 该方法包括式SR 1 R 2的硫化物与式的羟胺-O-磺酸的反应; 其中反应在碱的存在下在水性介质中进行。本发明还涉及制备式（Ⅳ）化合物的方法，其中R 3为卤素，氰基，C 1 -C 8 - 烷基，C 1 -C 8 - 卤代烷基，C 3 -C 8 - 环烷基，C 3 -C 8 - 卤代环烷基， C 2 -C 8 - 烯基，C 2 -C 8 - 卤代烯基，C 1 -C 8 - 烷氧基，苯基等; R4是氢，C1-C10-烷基，C1-C10-卤代烷基，C3-C8-环烷基，C3-C8-卤代环烷基，C2-C10-烯基，C2-C10-卤代烯基，苯基等; p是0，1，2，3或4; 所述方法包括：（i）提供式（Ia）或（Ib）化合物或其混合物，（ii）使式（Ia）或（Ib）的化合物或其混合物与步骤（i）与式（Ⅴ）化合物在碱的存在下反应，

9. 发明申请

WO2008092851A3 PESTICIDAL COMPOSITIONS COMPRISING 3 -ACETYL-I- PHENYLPYRAZOLE COMPOUNDS 审中-公开
公开(公告)号：WO2008092851A3
公开(公告)日：2008-08-07
申请号：PCT/EP2008/051026
申请日：2008-01-29
申请人： BASF SE , KORADIN, Christopher , LANGEWALD, Jürgen , ANSPAUGH, Douglas D. , COTTER, Henry Van Tuyl
发明人： KORADIN, Christopher , LANGEWALD, Jürgen , ANSPAUGH, Douglas D. , COTTER, Henry Van Tuyl
IPC分类号： A01N43/56 , A01N47/02 , A01P7/04
摘要： The present invention relates to pesticidal compositionscomprising as active componentsat least one 3-acetyl-1-phenylpyrazole compound of the formula (I) or a salt thereof: wherein X is N or C-R 5 ; R 1 is C 1 -C 4 -alkyl or C 1 -C 4 -haloalkyl; R 2 is NR 6 R 7 or S(O) n R 8 ; R 3 is halogen, C 1 -C 4 -haloalkyl, C 1 -C 4 -haloalkoxy, SF 5 or S(O) p R 9 ; R 4 is hydrogen or halogen; R 5 is halogen; R 6 is hydrogen, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl,C(O)R 10 , S(O) q CF 3 ; R 7 is hydrogen or C 1 -C 4 -alkyl, or R 6 and R 7 are joined so as together form a C 4 - C 6 -alkylene moiety, wherein one CH 2 -group may be replaced by oxygen or a radical N-R 11 ; R 8 , R 9 , R 10 , R 11 are each independently hydrogen, C 1 -C 4 -alkylorC 1 -C 4 -haloalkyl; m, n, p and q are each independently 0, 1 or 2; and at least one further pesticidally active compound II, selected from A.1GABA-gated chloride channel antagonists; A.2Nicotinic acetylcholine receptor agonists/antagonists A.3Juvenile hormone mimics; A.4Compounds affecting the oxidative phosphorylation; A.5Inhibitors of the chitin biosynthesis; A.6Moulting disruptors; A.7Mitochondrial electron transport inhibitors;. A.8Voltage-dependent sodium channel blockers; A.9Inhibitors of the lipid synthesis; and A.10group of various compounds.

10. 发明申请

WO2008074686A1 SUBSTITUTED 1-(AZOLIN-2-YL)-AMINO-1,2-HETEROCYCLYL-ETHANE COMPOUNDS FOR COMBATING PESTS 审中-公开
标题翻译：取代的1-（亚氨基-2-YL） - 氨基-1,2-杂环化合物 - 乙炔化合物
公开(公告)号：WO2008074686A1
公开(公告)日：2008-06-26
申请号：PCT/EP2007/063654
申请日：2007-12-11
申请人： BASF SE , KORDES, Markus , VEZOUET, Ronan Le , KORADIN, Christopher , BAUMANN, Ernst , CULBERTSON, Deborah L.
发明人： KORDES, Markus , VEZOUET, Ronan Le , KORADIN, Christopher , BAUMANN, Ernst , CULBERTSON, Deborah L.
IPC分类号： C07D401/06 , C07D405/06 , C07D409/06 , C07D417/12 , C07D417/14 , A01N43/78
CPC分类号： C07D409/06 , A01N43/50 , A01N43/76 , A01N43/78 , C07D401/06 , C07D405/06 , C07D417/12 , C07D417/14
摘要： The present invention relates to 1-(Azolin-2-yl)-amino-1,2-heterocyclyl-ethane compounds, which are useful for combating insects, arachnids and nematodes. The present invention also relates to methods for combating animal pests and to compositions for combating animal pests. It has been found that animal pests can be combated by 1-(Azolin-2-yl)-amino-1,2- heterocyclyl-ethane compounds of the general formula (I): wherein A is a radical of the formulae A 1 or A 2 : and wherein X is sulfur, oxygen or NR 7 , and Het A , Het B and R 1 to R 7 are defined as in the description.
摘要翻译：本发明涉及1-（唑啉-2-基） - 氨基-1,2-杂环基 - 乙烷化合物，其可用于防治昆虫，蜘蛛和线虫。本发明还涉及用于对抗动物害虫的方法和用于对抗动物害虫的组合物。已经发现，可以通过通式（I）的1-（氮杂-2-基） - 氨基-1,2-杂环基 - 乙烷化合物来对抗动物害虫：其中A是式A

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