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1. 发明申请

WO2007113322A2 SUBSTITUTED 5-HETARYLPYRIMIDINES 审中-公开
标题翻译：取代的5 HETARYLPYRIMIDINE
公开(公告)号：WO2007113322A2
公开(公告)日：2007-10-11
申请号：PCT/EP2007053332
申请日：2007-04-04
申请人： BASF AG , RHEINHEIMER JOACHIM , GROTE THOMAS , MUELLER BERND , ULMSCHNEIDER SARAH
发明人： RHEINHEIMER JOACHIM , GROTE THOMAS , MUELLER BERND , ULMSCHNEIDER SARAH
CPC分类号： C07D401/04 , A01N43/54
摘要： The invention relates to 5-hetaryl-4-pyrimidines of formula (I) and to their salts and plant protection agents which contain at least one compound of said type as an active component, wherein W represents oxygen, sulphur, a group S=O or S(=O) 2 ; R 1 represents optionally substituted C 1 -C 8 -alkyl, C 3 -C 8 -cycloalkyl, C 5 -C 10 -bicycloalkyl, C 2 -C 8 -alkenyl, C 4 -C 10 -alkadienyl, C 3 -C 6 -cycloalkenyl, C 2 -C 8 -alkynyl, phenyl, naphthyl, or a C-bound five- or six-membered saturated, partially unsaturated or aromatic heterocycle containing one, two, three or four heteroatoms from the groups O, N or S as ring members; R 2 represents halogen, cyano, hydroxy, mercapto, N 3 , C 1 -C 6 -alkyl, C 2 -C 8 -alkenyl, C 2 -C 8 -alkynyl, C 1 C 6 -halogenalkyl, C 1 C 6 -alkoxy, C 3 -C 8 -alkenyloxy, C 3 -C 8 -alkynyloxy, C 1 C 6 -halogenalkoxy, C 1 -C 6 -alkylthio, C 3 -C 8 -alkenylthio, C 3 -C 8 -alkynylthio, C 1 -C 6 -halogenalkylthio, or a radical of formulae C(=Z)OR 21 , C(=Z)NR 22 R 23 , C(=Z)NR 24 -NR 22 R 23 , C(=Z)R 25 , CR 26 R 27 -OR 28 , CR 26 R 27 -NR 22 R 23 , ON(=CR 29 R 30 ), O-C(=Z)R 25 , NR 22 R 23a , NR 31 (C(=Z)R 25 ), NR 31 (C(=Z)OR 21 ), NR 31 (C(=Z)-NR 22 R 23 ), NR 32a (N=CR 29 R 30 ), NR 32 NR 22 R 23 , NR 32 OR 21 , or C(=N-Z'-R 25 )SR 21 ; or a cyclic radical; R3 represents hydrogen, OH, halogen, cyano, NR 37 R 38 , C 1 -C--alkyl, C 1 -C 8 -alkoxy, C 1 -C 8 -alkylthio, C 1 -C 8 -alkylsulfinyl, C 1 -C--alkylsulfonyl, C 2 -C 8 -alkenyl or C 2 -C 8 -alkinyl, whereby the seven latter radicals can be partially or totally halogenated and/or optionally can support one, two or three substitutes, selected among nitro, cyano, OH, C 1 -C 2 -alkoxy, C 1 -C 4 -alkoxycarbonyl, amino, C 1 -C 4 -alkylamino and Di-C 1 -C 4 -alkylamino, Het represents a substituted C- or N-bound, 5-or 6-membered aromatic heterocycle which comprises 1, 2, 3 or 4 heteroatoms as ring members selected among nitrogen, oxygen and sulphur. The invention also relates to the use of 5-hetaryl-4-pyrimidines of formula (I) and there salts for combating plant pathogenic fungi.
摘要翻译：本发明涉及式（I）的包含至少一种这样的化合物作为有效成分的5-杂芳基-4-嘧啶和它们的盐和杀虫剂。其中W = O或S（= O）_{2 表示氧，硫，基团S; [R ^{1 表示任选subsitituiert.esç_{1 -C _{8 烷基，C _{3 -C _{8 环烷基，C _{5 -C _{10 双环，C _{2 -C _{8 - 烯基，C _{4 -C _{10 链二烯基，C _{3 -C _{6 环烯基，C _{2 -C _{8 是炔基，苯基，萘基或C-连接的五元或六元饱和，部分不饱和或芳族的含有一个，两个，三个或四个杂原子的从杂环包含基团的O，N或S作为环成员; [R ^{2 表示卤素，氰基，羟基，巯基，N _{3 ，C _{1 -C _{6 烷基， ç_{2 -C _{8 烯基，C _{2 -C _{8 - 炔基，C _{1 C _{6 卤代烷基，C _{1 C _{6 烷氧基，C _{3 -C _{8 烯，C _{3 -C _{8 炔氧基，C _{1 C _{6 卤代烷氧基，C _{1 -C _{6 烷硫基，C _{3 -C _{8 烯，C _{3 -C _{8 炔硫基，C _{1 -C _{6 卤代烷硫基，或一个基团，式C（= Z） OR ^{21 ，C（= Z）NR ^{22 - [R ^{23 ，C（= Z）NR ^{24 -NR ^{22 - [R ^{23 ，C（= Z）R ^{25 ，CR ^{26 - [R ^{27 -OR ^{28 ，CR ^{26 - [R ^{27 -NR ^{22 - [R ^{23 ， ON（= CR ^{29 - [R ^{30 ），OC（= Z）R ^{25 ，NR ^{22 - [R ^{图23A ，NR ^{31 （C（= Z）R ^{25 ），NR ^{31 （C（= Z）OR 21 ）NR ^{31 （ C（= Z）-NR ^{22 - [R ^{23 ），NR ^{32A （N = CR ^{29 - [R ^{30 ），NR ^{32 NR ^{22 - [R ^{23 ，NR ^{32 OR ^{21 ，或C（= N-Z'-R ^{25 ）SR ^{21 ; 或环状基团; R 3是氢，OH，卤素，氰基，NR ^{37 - [R ^{38 ，C _{1 -C - 烷基，C _{1 -C _{8 烷氧基，C _{1 -C _{8 烷硫基，C _{1 -C _{8 烷基亚磺酰基，C _{1 -C - 烷基磺酰基，C _{2 -C _{8 链烯基或C _{2 -C _{8 炔基，其中所述7最后提到的基团可以部分或完全卤化和/或选自硝基一个，两个或三个取代基，氰基，OH，C _{1 -C _{2 烷氧基，C _{1 -C _{4 烷氧基羰基，氨基，C _{1 -C _{4 烷基氨基和二C _{1 -C _{4可携带>烷基氨基，}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}

2. 发明申请

WO2007110418A3 SUBSTITUTED 5-HETARYL-4-AMINOPYRIMIDINES 审中-公开
标题翻译：取代的5-杂芳基-4-氨基嘧啶
公开(公告)号：WO2007110418A3
公开(公告)日：2008-11-20
申请号：PCT/EP2007052888
申请日：2007-03-26
申请人： BASF SE , RHEINHEIMER JOACHIM , GROTE THOMAS , MUELLER BERND , GRAMMENOS WASSILIOS , ULMSCHNEIDER SARAH , RENNER JENS , STIERL REINHARD
发明人： RHEINHEIMER JOACHIM , GROTE THOMAS , MUELLER BERND , GRAMMENOS WASSILIOS , ULMSCHNEIDER SARAH , RENNER JENS , STIERL REINHARD
IPC分类号： A01N43/54 , A01N43/56 , A01N43/653 , A01N43/76 , A01N43/78 , A01N43/80 , A01P3/00 , A01P5/00 , A01P7/00 , A61K31/506 , C07D401/04 , C07D403/04 , C07D405/04 , C07D409/04 , C07D413/04 , C07D417/04
CPC分类号： A01N43/54
摘要： The present invention relates to the use of 5-hetaryl-4-aminopyrimidines of the formula I and of their salts for controlling phytopathogenic fungi. The invention also relates to novel 5-hetaryl-4-aminopyrimidines and to plant protection compositions which contain at least one such compound as active component. Het represents an optionally substituted 5- or 6-membered aromatic heterocycle which has 1, 2, 3 or 4 hetero atoms as ring members which are selected among nitrogen, oxygen and sulphur, where the 5- or 6-membered heteroaromatic radical can have 1, 2, 3 or 4 identical or different substituents L; R 1 , R 2 represent inter alia hydrogen, C 1 -C 8 -alkyl, C 3 -C 8 -cycloalkyl, C 5 -C 10 -bicycloalkyl, C 2 -C 8 -alkenyl, C 4 -C 10 -alkadienyl, C 3 -C 6 -cycloalkenyl, C 2 -C 8 -alkynyl, phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which has one, two, three or four hetero atoms from the series O, N or S as ring members; or together form a ring; R 3 represents, inter alia, hydrogen, OH, halogen, cyano, NR 31 R 32 , C 1 -C 8 -alkyl, C 1 -C 8 -alkoxy, C 1 -C 8 -alkylthio, C 1 -C 8 -alkylsulphinyl, C 1 -C 8 -alkyl-sulphonyl, C 2 -C 8 -alkenyl or C 2 -C 8 -alkynyl; and R 4 represents halogen, cyano, hydroxy, mercapto, N 3 , C 1 -C 6 -alkyl, C 2 -C 8 -alkenyl, C 2 -C 8 -alkynyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkoxy, C 3 -C 8 -alkenyloxy, C 3 -C 8 -alkynyloxy, C 1 -C 6 -haloalkoxy, C 1 -C 6 -alkylthio, C 3 -C 8 -alkenylthio, C 3 -C 8 -alkynylthio, C 1 -C 6 -haloalkylthio, or represents a radical of the formulae C(=Z)OR 41 , C(=Z)NR 42 R 43 , C(=Z)NR 44 -NR 42 R 43 , C(=Z)R 45 , CR 46 R 47 -OR 48 , CR 46 R 47 -NR 42 R 43 , ON(=CR 49 R 50 ), O-C(=Z)R 45 , NR 42 R 43a , NR 51 (C(=Z)R 45 ), NR 51 (C(=Z)OR 41 ), NR 51 (C(=Z)-NR 42 R 43 ), NR 52a (N=CR 49 R 50 ), NR 52 NR 42 R 43 , NR 52 OR 41 , or C(=N-X-R 45 )SR 41 .
摘要翻译：本发明涉及使用5-杂芳基-4-氨基嘧啶式I及其盐用于防治植物破坏性真菌。本发明还涉及新的5-杂芳基-4-氨基嘧啶和含有至少一个这样的化合物作为有效成分的杀虫剂。 Het代表任选substituerten 5-或6-元芳族杂环，其具有1,2，3或4个氮，氧和选定的作为环成员的硫杂原子，其中所述5元或6元杂芳族残基1，2，3 可以包括或4个相同或不同的取代基L，R ^{1 ，R ^{2 除其他外，氢，C _{1 -C _{8 烷基，C _{3 -C _{8 环烷基，C _{5 -C _{10 二环烷基， ç_{2 -C _{8 烯基，C _{4 -C _{10 链二烯基，C _{3 -C _{6 环烯基，C _{2 -C _{8 炔基，苯基，萘基或五 - 或六元饱和的，部分含有一个，具有从所述组的两个，三个或四个杂原子的不饱和或芳族杂环O，N或S作为环成员; 或一起形成一个环; [R ^{3 除其他外，氢，OH，卤素，氰基，NR ^{31 - [R ^{32 ，C _{1 -C 8 烷基，C _{1 -C _{8 烷氧基，C _{1 -C _{8 烷硫基，C _{1 -C _{8 烷基亚磺酰基，C _{1 -C _{8 烷基磺酰基，C 2 -C _{8 链烯基或C _{2 -C _{8 装置-Alkiny，且R ^{4 表示卤素，氰基，羟基，巯基，N _{3 ，C _{1 -C _{6 烷基，C _{2 -C _{8 烯基，C _{2 -C _{8 炔基，C _{1 -C 6 卤代烷基，C _{1 -C _{6 烷氧基，C _{3 -C _{8 烯，C _{3 -C _{8 炔氧基，C _{1 -C _{6 卤代烷氧基，C 1 -C _{6 烷硫基，C _{3 -C _{8 烯，C _{3 -C _{8 炔硫基，C _{1 -C _{6 卤代烷硫基，或一个基团，式C（= Z）或^{41 ，C（= Z）NR ^{42 ř ^{43 ，C（= Z）NR ^{44 -NR ^{42 - [R ^{43 ，C（= Z）R 45 ，CR ^{46 - [R ^{47 为-OR ^{48 ，CR ^{46 - [R ^{47 -NR ^{42 - [R ^{43 ，ON（= CR ^{49 - [R ^{50 ），OC（ = Z）R ^{45 ，NR ^{42 - [R ^{43A ，NR ^{51 （C（= Z）R ^{45 ），NR ^{51 （C（= Z）OR ^{41 ），NR ^{51 （C（= Z） - NR ^{42 - [R ^{43 ），NR ^{52A （N = CR ^{49 - [R ^{50 ），NR ^{52 NR ^{42 - [R ^{43 ，NR ^{52 或^{41 ，或 C（= NXR ^{45 ）SR ^{41 是。}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}

3. 发明申请

WO2007116011A3 SUBSTITUTED TRIAZOLOPYRIMIDINES, METHOD FOR THE PRODUCTION THEREOF, USE THEREOF FOR CONTROLLING HARMFUL FUNGI, AND SUBSTANCES CONTAINING THE SAME 审中-公开
标题翻译：取代的三唑并嘧啶类化合物，其制备方法及其用于控制受损蘑菇的用途以及含有该化合物的培养基
公开(公告)号：WO2007116011A3
公开(公告)日：2007-12-21
申请号：PCT/EP2007053355
申请日：2007-04-05
申请人： BASF AG , DIETZ JOCHEN , GROTE THOMAS , GRAMMENOS WASSILIOS , MUELLER BERND , LOHMANN JAN KLAAS , RENNER JENS , ULMSCHNEIDER SARAH
发明人： DIETZ JOCHEN , GROTE THOMAS , GRAMMENOS WASSILIOS , MUELLER BERND , LOHMANN JAN KLAAS , RENNER JENS , ULMSCHNEIDER SARAH
IPC分类号： C07D487/04 , A01N43/90
CPC分类号： C07D487/04
摘要： Disclosed are compounds of formula (I), wherein X, Y, and Z are defined as indicated in the description, methods and intermediate products for producing said compounds, substances containing the same, and the use thereof for controlling plant pathogenic fungi.
摘要翻译：其中X，Y和Z如所述定义的式（I）化合物，用于制备这些化合物的方法和中间体，含有它们的试剂及其用于防治植物病原性有害真菌的用途。

4. 发明申请

WO2008012234A2 AZOLYLMETHYLOXIRANES, USE THEREOF FOR CONTROLLING PLANT PATHOGENIC FUNGI, AND AGENTS CONTAINING THE SAME 审中-公开
标题翻译： Azolylmethyloxiranes，及其用于防治病原真菌植物及代理人含
公开(公告)号：WO2008012234A2
公开(公告)日：2008-01-31
申请号：PCT/EP2007057353
申请日：2007-07-17
申请人： BASF AG , DIETZ JOCHEN , GROTE THOMAS , MUELLER BERND , LOHMANN JAN KLAAS , RENNER JENS , ULMSCHNEIDER SARAH , GLAETTLI ALICE
发明人： DIETZ JOCHEN , GROTE THOMAS , MUELLER BERND , LOHMANN JAN KLAAS , RENNER JENS , ULMSCHNEIDER SARAH , GLAETTLI ALICE
IPC分类号： C07D405/14 , A01N43/707 , C07D409/14
CPC分类号： C07D405/14 , A01N43/653 , C07D409/14
摘要： The invention relates to azolylmethyloxiranes of general formula (I), wherein A or B is benzodioxolyl which is optionally substituted by between one and five of the following substituents, halogen, CN, NO 2 , amino, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 1 -C 4 halogenalkyl, C 1 -C 4 halogenalkoxy, C 1 -C 4 alkylamino, C 1 -C 4 dialkylamino, thio or C 1 -C 4 alkylthio, and the respective other substituent A or B is phenyl or 5-membered or 6-membered heteroaryl, said substituents being optionally substituted by between one and three of the following substituents, halogen, CN, NO 2 , amino, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 1 -C 4 halogenalkyl, C 1 -C 4 halogenalkoxy, C 1 -C 4 alkylamino, C 1 -C 4 dialkylamino, thio or C 1 -C 4 alkylthio. The invention also relates to the plant-tolerant acid addition salts or metal salts of said compounds, to the use of the compounds of formula (I) for controlling plant-pathogenic fungi, and to agents containing the same.
摘要翻译：本发明涉及通式（I），其中A或B是苯并二的azolylmethyloxirane其任选地被一个取代以下substi- tuenten卤素，CN，NO _{2 ，氨基，C <五 SUB> 1 -C _{4 烷基，C _{1 -C _{4 烷氧基，C _{1 -C _{4 - 卤代烷基，C _{1 -C 4卤代烷，C _{1 -C _{4 烷基氨基， ç_{1 -C _{4 二烷基氨基，硫代，或C _{1 -C _{4 是烷硫基，被取代的，和各其他取代基A或B为苯基或5元或6元杂芳基，所述取代基任选地被1-3个下列取代基取代：卤素，CN，NO _{2 ，氨基，C 1 -C _{4 烷基，C _{1 -C _{4 烷氧基，C _{1 -C _{4 卤代烷基，C _{1 -C _{4 - 卤代烷氧基，C _{1 -C _{4 - 烷基氨基，C _{1 -C _{4 二烷基氨基，巯基或C _{1 -C _{4 - 烷硫基，被取代的，和它们的植物耐受的酸加成盐或金属盐，使用式（I）的用于控制植物病原真菌包含它们的化合物和试剂。}}}}}}}}}}}}}}}}}}}}}}}}}}}

5. 发明申请

WO2006114405A2 USE OF 5-ALKYL-6-PHENYLALKYL-7-AMINO-AZOLOPYRIMIDINES, NOVEL AZOLOPYRIMIDINES, METHODS FOR THE PRODUCTION THEREOF, AND AGENTS CONTAINING THE SAME 审中-公开
标题翻译：使用5-烷基-6-苯基 - 7-氨基AZOLOPYRIMIDINEN，NEW azolopyrimidines，METHOD用于生产和AGENTS CONTAINING THE SAME
公开(公告)号：WO2006114405A2
公开(公告)日：2006-11-02
申请号：PCT/EP2006061786
申请日：2006-04-24
申请人： BASF AG , DIETZ JOCHEN , GRAMMENOS WASSILIOS , GROTE THOMAS , HUENGER UDO , LOHMANN JAN KLAAS , MUELLER BERND , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA
发明人： DIETZ JOCHEN , GRAMMENOS WASSILIOS , GROTE THOMAS , HUENGER UDO , LOHMANN JAN KLAAS , MUELLER BERND , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA
IPC分类号： A01N43/90
CPC分类号： A01N43/90 , C07D487/04
摘要： The invention relates to the use of 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines of formula I for controlling phytopathogenic fungi. The variables in formula I have the following designations: Y represents alkylene, alkenylene or alkinylene, optionally substituted by alkyl groups; R 1 represents halogen, cyano, nitro, hydroxy, mercapto, alkyl, halogenalkyl, alkenyl, cycloalkyl, cycloalkenyl, alkoxy, halogenalkoxy, alkenyloxy, alkinyloxy, alkylthio, NR A R B , alkylcarbonyl, phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group O, N or S; R A , R B represent hydrogen, alkyl and alkylcarbonyl; n represents 0, 1, 2, 3 or 4; R 2 represents alkyl, alkenyl, cycloalkyl, alkoxyalkyl and alkylthioalkyl; R 3 represents hydrogen, halogen, cyano, NR A R B , hydroxy, mercapto, alkyl, halogenalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, phenyl, phenoxy, phenylthio, benzyloxy, benzylthio, or alkyl-S(O) m- ; m represents 0, 1 or 2; A represents N and C-R a ; and R a represents hydrogen and alkyl. The carbon atoms in Y, R 1 , R 2 , R 3 and Ra can be substituted according to the description. The invention also relates to novel 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines, to methods for producing said compounds, and to agents containing the same.
摘要翻译：式的5-烷基-6-苯基-7-氨基azolopyrimidinen的使用I：其中各变量具有以下含义：Y是任选被烷基取代的亚烷基，亚烯基或亚炔基; [R ^{1 为卤素，氰基，硝基，羟基，巯基，烷基，卤代烷基，链烯基，环烷基，环烯基，烷氧基，卤代烷氧基，烯氧基，炔氧基，烷硫基，NR ^{一 - [R 乙，烷基羰基，苯基，萘基或五 - 或六元饱和环，其包含选自一至四个杂原子的部分不饱和或罗马杂环O，N或S; [R ^{一，R ^{乙是氢，烷基和烷基羰基; n是零，1，2，3或4; [R ^{2 烷基，烯基，环烷基，烷氧基烷基和烷硫基烷基; [R ^{3 为氢，卤素，氰基，NR ^{一 - [R ^{乙，羟基，巯基，烷基，卤代烷基，环烷基，烷氧基，烷硫基，环烷氧基，环烷硫基，羧基，甲酰基，烷基羰基，烷氧基羰基，烯氧基羰基，炔氧基羰基，苯基，苯氧基，苯硫基，苄氧基，苄硫基，烷基-S（O）_{米 - ; m是0，1或2; A N和C-R ^{一; [R ^{一氢和烷基; 其中Y中的碳原子，R ^{1 ，R ^{2 ，R ^{3 和R a可以按照该描述被取代; 防治植物病原性有害真菌; 新5-烷基-6-苯基-7- aminoazolopyrimidines，处理用于制备这些化合物和含有它们的组合物。}}}}}}}}}}}}}}

6. 发明申请

WO2005087771A3 5,6-DIALKYL-7-AMINO-TRIAZOLOPYRIMIDINES, METHOD FOR THEIR PRODUCTION, THEIR USE FOR CONTROLLING PATHOGENIC FUNGI AND AGENTS CONTAINING SAID COMPOUNDS 审中-公开
标题翻译： 5,6-二烷基 - 7-氨基三唑，方法用于生产和它们用于防治有害真菌及代理人含
公开(公告)号：WO2005087771A3
公开(公告)日：2005-12-01
申请号：PCT/EP2005002425
申请日：2005-03-08
申请人： BASF AG , TORMO I BLASCO JORDI , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , WAGNER OLIVER , NIEDENBRUECK MATTHIAS , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
发明人： TORMO I BLASCO JORDI , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , WAGNER OLIVER , NIEDENBRUECK MATTHIAS , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
IPC分类号： C07D487/04
CPC分类号： C07D487/04
摘要： The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R represents alkyl or alkoxyalkyl; R represents alkyl, R and/or R being substituted according to the description. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.
摘要翻译：式（I）的5,6-二烷基 - 7-氨基 - 三唑并嘧啶，其中取代基具有以下含义：R t <1>是烷基或烷氧基烷基，R <2>是烷基，其中R <1>和/或R <2> 可以如上所述被替换; 这些化合物的制备方法，含有它们的试剂及其用于防治植物病原性有害真菌的用途。

7. 发明申请

WO2005080396A2 AZOLOPYRIMIDINE COMPOUNDS AND USE THEREOF FOR COMBATING PARASITIC FUNGI 审中-公开
标题翻译： AZOLOPYRIMIDINE化合物及其在破坏性蘑菇中的应用
公开(公告)号：WO2005080396A2
公开(公告)日：2005-09-01
申请号：PCT/EP2005001965
申请日：2005-02-24
申请人： BASF AG , SCHWOEGLER ANJA , GEWEHR MARKUS , MUELLER BERND , GROTE THOMAS , GRAMMENOS WASSILIOS , TORMO I BLASCO JORDI , RHEINHEIMER JOACHIM , BLETTNER CARSTEN , SCHAEFER PETER , SCHIEWECK FRANK , WAGNER OLIVER , STIERL REINHARD , SCHOEFL ULRICH , STRATHMANN SIEGFRIED , SCHERER MARIA
发明人： SCHWOEGLER ANJA , GEWEHR MARKUS , MUELLER BERND , GROTE THOMAS , GRAMMENOS WASSILIOS , TORMO I BLASCO JORDI , RHEINHEIMER JOACHIM , BLETTNER CARSTEN , SCHAEFER PETER , SCHIEWECK FRANK , WAGNER OLIVER , STIERL REINHARD , SCHOEFL ULRICH , STRATHMANN SIEGFRIED , SCHERER MARIA
IPC分类号： A01N43/90 , C07D487/04 , C07D487/00
CPC分类号： C07D487/04
摘要： The invention relates to azolopyrimidine compounds of general formula (I), wherein A represents N or C-R ; X and Y, independent of one another, represent a chemical compound or oxygen, sulphur or a group N-R ; the variables R , R , R , R , R , R and R have the meanings cited in the claims and the description. The invention also relates to tautomers of compounds of formula (I) and to the agriculturally compatible salts of compounds (I) and of the tautomers thereof. The invention further relates to the use of azolopyrimidine compounds of general formula (I), to the tautomers thereof and to the agriculturally compatible salts thereof which are used to combat phytopathogenic fungi, and to a method for combating phytopathogenic fungi and means for combating fungi, said means containing at least one compound of general formula (I), a tautomer of formula (I) and/or an agriculturally compatible salt thereof or the tautomer thereof and at least one liquid or solid carrier medium.
摘要翻译：本发明涉及通式（I）的唑基嘧啶化合物，其中A是N或C-R 6; X，Y彼此独立地代表化学键或氧，硫或基团N-R 7; 其中变量R <1>，R <2>，R <3>，R <4>，R <5> - [R <6>和R <7>具有权利要求书所给出的含义和描述中，互变异构体式（I）化合物和化合物I及其互变异构体的农业上可接受的盐。本发明还涉及使用通式（I）的唑并嘧啶化合物，它们的互变异构体以及它们用于防治植物致病真菌（=有害真菌），以及用于防治植物病原性有害真菌的方法和用于防治有害真菌的手段农业上可接受的盐，含至少一种通式（I）的化合物，（I）的互变异构体和/或其农业上可接受的盐或其互变异构体以及至少一种液体或固体载体。

8. 发明申请

WO03008417A9 SUBSTITUTED 6-(2-TOLYL)-TRIAZOLOPYRIMIDINES AS FUNGICIDES 审中-公开
标题翻译：取代的6-（2-甲苯基） - 三唑并嘧啶作为杀真菌剂
公开(公告)号：WO03008417A9
公开(公告)日：2003-10-30
申请号：PCT/EP0207578
申请日：2002-07-08
申请人： BASF AG , TORMO I BLASCO JORDI , SAUTER HUBERT , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHAEFER PETER , SCHIEWECK FRANK , RACK MICHAEL , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD
发明人： TORMO I BLASCO JORDI , SAUTER HUBERT , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHAEFER PETER , SCHIEWECK FRANK , RACK MICHAEL , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD
IPC分类号： A01N43/90 , C07D487/04
CPC分类号： C07D487/04 , A01N43/90
摘要： Substituted 6-(2-tolyl)-triazolopyrimidines of formula (I) in which R and R independently denote hydrogen or alkyl, alkenyl, alkynyl, or alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R and R radicals may be unsubstituted or substituted as defined in the description, or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; R is halogen, cyano, alkyl, alkoxy, haloalkyl, or C(=O)A, wherein A is hydrogen, hydroxy, alkyl, amino, or mono- or dialkyl-amino; n is an integer from 1 to 4; and X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.
摘要翻译：式（I）的取代的6-（2-甲苯基） - 三唑并嘧啶，其中R 1和R 2独立地表示氢或烷基，烯基，炔基或链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5-或6-元杂环基，或者含有1-4个氮原子或1-3个氮原子的5-或6-元杂芳基，硫或氧原子，或者其中R 1和R 2基团可以如说明书中所定义的那样未被取代或被取代，或者R 1和R 2与中间的氮原子一起表示5或6 - 含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的可被取代的 - 元杂环; R 3是卤素，氰基，烷基，烷氧基，卤代烷基或C（= O）A，其中A是氢，羟基，烷基，氨基或单或二烷基氨基; n是1至4的整数; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基; 它们的制备方法，含有它们的组合物以及它们用于防治植物病原性真菌的用途。

9. 发明申请

WO02074753A3 5-PHENYLPYRIMIDINE, METHODS AND INTERMEDIATE PRODUCTS FOR THE PRODUCTION THEREOF AND USE OF THE SAME FOR CONTROLLING PATHOGENIC FUNGI 审中-公开
标题翻译： 5苯基嘧啶，流程和中间产物及其及其用途用于防治有害真菌
公开(公告)号：WO02074753A3
公开(公告)日：2002-12-27
申请号：PCT/EP0202739
申请日：2002-03-13
申请人： BASF AG , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHAEFER PETER , SCHIEWECK FRANK , SAUTER HUBERT , GEWEHR MARKUS , MUELLER BERND , TORMO I BLASCO JORDI , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD
发明人： GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHAEFER PETER , SCHIEWECK FRANK , SAUTER HUBERT , GEWEHR MARKUS , MUELLER BERND , TORMO I BLASCO JORDI , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD
IPC分类号： A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/64 , A01N43/647 , A01N43/653 , A01N43/713 , A01N43/90 , C07D239/42 , C07D401/14 , C07D403/04 , C07D471/04 , C07D473/06 , C07D487/04 , C07D521/00 , C07D473/00
CPC分类号： C07D239/42 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/647 , A01N43/653 , A01N43/713 , A01N43/90 , C07D231/12 , C07D233/56 , C07D249/08 , C07D403/04 , C07D473/06 , C07D487/04
摘要： The invention relates to 5-phenylpyrimidine of formula (I) wherein the substituents have the following designations: R represents a five to ten-membered saturated, partially unsaturated or aromatic monocyclic or bicyclic heterocycle which contains between one and four heteroatoms from the group 0, N or S, and which can be substituted as defined in the description; R represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R and R represent hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl; together with the nitrogen atom to which they are bonded, R and R can also form a five or six-membered ring which can be split by a heteroatom and can carry at least one substituent; R and R represent hydrogen, halogen, alkyl, halogenalkyl or alkoxy; R and R represent hydrogen, halogen, alkyl or halogenalkyl; and R represents hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, halogenalkoxy or alkoxycarbonyl. The invention also relates to methods and intermediate products for producing said compounds and the use of the same for controlling pathogenic fungi.
摘要翻译：式（I）其中取代基具有以下Begende含义的5-苯基嘧啶，R <1> 5〜10元饱和，部分不饱和或芳族单环或双环杂环，选自下组0含有一至四个杂原子，N或如说明书中所定义的可被取代的S，R <2>为氢，卤素，氰基，烷基，卤代烷基或烷氧基; [R <3>，R <4>是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，R <3>和R <4>可与氮原子一起他们连接，形成可以被杂原子中断并且可以携带一个或多个取代基的五元或六元环; [R <5> - [R <6>是氢，卤素，烷基，卤代烷基或烷氧基; [R <7> - [R <8>是氢，卤素，烷基或卤代烷基; [R <9>是氢，卤素，烷基，烷氧基，环烷氧基，卤代烷氧基或烷氧基羰，卤代烷氧基或烷氧羰，涉及用于制备这些化合物和它们在防治有害真菌中的用途的方法和中间体。

10. 发明申请

WO0248146A2 USE OF SUBSTITUTED IMIDAZOAZINES, NOVEL IMIDAZOAZINES, METHODS FOR THE PRODUCTION THEREOF, AND AGENTS CONTAINING THESE COMPOUNDS 审中-公开
标题翻译： USE取代IMIDAZOAZINEN，新imidazoazines，制造方法，和代理人含
公开(公告)号：WO0248146A2
公开(公告)日：2002-06-20
申请号：PCT/EP0114577
申请日：2001-12-12
申请人： BASF AG , CULLMANN OLIVER , GEWEHR MARKUS , GRAMMENOS WASSILIOS , TORMO I BLASCO JORDI , MUELLER BERND , SAUTER HUBERT , GYPSER ANDREAS , GROTE THOMAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHIEWECK FRANK , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD
发明人： CULLMANN OLIVER , GEWEHR MARKUS , GRAMMENOS WASSILIOS , TORMO I BLASCO JORDI , MUELLER BERND , SAUTER HUBERT , GYPSER ANDREAS , GROTE THOMAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHIEWECK FRANK , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD
IPC分类号： A01N43/90 , C07D471/04 , C07D487/04
CPC分类号： C07D471/04 , A01N43/90 , C07D487/04
摘要： The invention relates to the use of substituted imidazoazines of formula (I), in which the variables have the following meanings: R represents alkyl, phenyl, phenylalkyl, naphthyl, anthracenyl, cycloalkyl, 5-membered or 6-membered hetaryl or 5-membered or 6-membered heterocyclyl, containing one to three N atoms and/or one O atom or S atom or one or two O atoms and/or S atoms, or condensed 8-membered to 12-membered hetaryl or condensed 8-membered to 12-membered heterocyclyl, containing one to four N atoms and/or one O atom or S atom or one or two O atoms and/or S atoms, whereby R can be unsubstituted or can be substituted as cited in the description; R and R represent hydrogen, alkyl, alkenyl, alkynyl, alkyl halide, alkenyl halide, alkynyl halide, trialkyl silylalkyl, phenyl, phenylalkyl or R and R , together with the bridging N atom, form a 5-membered or 6-membered heterocyclic or heteroaromatic ring, which can be interrupted by one to three N atoms and/or one O atom or S atom or by one or two O atoms and/or S atoms, and which can be substituted; A and B represent N or CR ; R , R and R represent hydrogen, halogen, cyano, nitro, hydroxy, alkyl, alkyl halide, cycloalkyl, alkoxy, alkoxy halide, alkylthio, amino, alkyl amino, dialkylamino, alkenyl, alkenyloxy, alkynyl or alkynyloxy. The inventive compounds are used for controlling phytopathogenic harmful fungi. The invention further relates to agents containing the inventive compounds, to novel imidazoazines, and to methods for the production thereof.
摘要翻译：使用式（I）的取代的Imidazoazinen的，其中各变量具有以下含义：R t <1>是烷基，苯基，苯基烷基，萘基，蒽基，环烷基，5-或6-员杂芳基或5-或6-元杂环基含有1至3个N原子和/或一个O或S原子或一个或两个O和/或S原子，或稠合8-12 gliederiges杂芳基或稠合的8-12 gliederiges杂环基，含有一至四个N原子和/或一个O或S原子或一个或两个O和/或O原子，其中R是未取代的<1>或作为可在本说明书中被取代; [R <2>，R <3>是氢，烷基，烯基，炔基，卤代烷基，卤代烯基，卤代炔基，三烷基甲硅烷基，苯基，苯基烷基或R <2>，R <3>连同桥接氮原子的5-或6- 形成 - 元杂环基或可被一至三个N原子和/或一个O或S原子或一个或两个O和/或S原子被中断杂芳族环; A，B，N或CR <4>; [R <4>，R <5> - [R <6>为氢，卤素，氰基，硝基，羟基，烷基，卤代烷基，环烷基，烷氧基，卤代烷氧基，烷硫基，氨基，烷基氨基，二烷基氨基，烯基，烯氧基，炔氧基或炔氧基; 防治植物病原性有害真菌的，含有它们，它们的制备新imidazoazines和方法的组合物。

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