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1. 发明授权

US08835427B2 Fungicidal heterocyclic compounds 有权
标题翻译：杀真菌杂环化合物
公开(公告)号：US08835427B2
公开(公告)日：2014-09-16
申请号：US13518943
申请日：2011-01-07
申请人： Andris Juris Liepa , Robert James Pasteris , Thomas Martin Stevenson
发明人： Andris Juris Liepa , Robert James Pasteris , Thomas Martin Stevenson
IPC分类号： C07D417/04 , C07D487/04 , A01N43/80 , A01N43/90
CPC分类号： C07D487/04 , A01N43/80 , A01N43/90 , C07D413/14 , C07D417/14
摘要： Disclosed are compounds of Formula 1 and Formula 1A including all stereoisomers, N-oxides, and salts thereof, wherein E, Y1, Y2, Y3, G, J, X1 and X2 are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 or Formula 1A and methods for controlling plant disease caused by a fungal pathogen comprising applying an effective amount of a compound or a composition of the invention.
摘要翻译：公开了式1和式1A的化合物，其包括所有立体异构体，N-氧化物及其盐，其中E，Y1，Y2，Y3，G，J，X1和X2如本公开所定义。还公开了含有式1或式1A化合物的组合物和用于控制由真菌病原体引起的植物病害的方法，包括施用有效量的本发明化合物或组合物。

2. 发明申请

US20120309752A1 FUNGICIDAL HETEROCYCLIC COMPOUNDS 有权
标题翻译：真菌杂环化合物
公开(公告)号：US20120309752A1
公开(公告)日：2012-12-06
申请号：US13518943
申请日：2011-01-07
申请人： Andris Juris Liepa , Robert James Pasteris , Thomas Martin Stevenson
发明人： Andris Juris Liepa , Robert James Pasteris , Thomas Martin Stevenson
IPC分类号： A01N43/80 , A01P3/00 , A01N43/90 , C07D417/14 , C07D487/04
CPC分类号： C07D487/04 , A01N43/80 , A01N43/90 , C07D413/14 , C07D417/14
摘要： Disclosed are compounds of Formula 1 and Formula 1A including all stereoisomers, N-oxides, and salts thereof, wherein E, Y1, Y2, Y3, G, J, X1 and X2 are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 or Formula 1A and methods for controlling plant disease caused by a fungal pathogen comprising applying an effective amount of a compound or a composition of the invention
摘要翻译：公开了式1和式1A的化合物，其包括所有立体异构体，N-氧化物及其盐，其中E，Y1，Y2，Y3，G，J，X1和X2如本公开所定义。还公开了含有式1或式1A化合物的组合物和用于控制由真菌病原体引起的植物病害的方法，包括施用有效量的本发明化合物或组合物

3. 发明申请

US20130030002A1 FUNGICIDAL OXIMES AND HYDRAZONES 失效
标题翻译：杀真菌毒素和水。
公开(公告)号：US20130030002A1
公开(公告)日：2013-01-31
申请号：US13640092
申请日：2011-04-15
申请人： Mary Ann Hanagan , Andris Juris Liepa , Eric Allen Marshall , Robert James Pasteris
发明人： Mary Ann Hanagan , Andris Juris Liepa , Eric Allen Marshall , Robert James Pasteris
IPC分类号： A01N43/78 , C07D417/06 , A01N43/40 , C07D417/14 , A01N43/58 , A01P3/00 , C07D401/06 , A01N43/56 , C07D277/30 , A01N43/54
CPC分类号： C07D417/04 , C07D403/14 , C07D407/14 , C07D409/14 , C07D413/14 , C07D417/14
摘要： Disclosed are compounds of Formula 1, including all stereoisomers, N-oxides, and salts thereof, wherein E, X, G, W2 and Z are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling plant disease caused by a fungal pathogen comprising applying an effective amount of a compound or a composition of the invention.Also disclosed are compounds of Formula 1A including all stereoisomers, N-oxides, and salts thereof, wherein E, X, G and Z1 are as defined in the disclosure. Also disclosed is the use of the compounds of Formula 1A as intermediates for preparing compounds of Formula 1.
摘要翻译：公开了式1的化合物，包括所有立体异构体，N-氧化物及其盐，其中E，X，G，W 2和Z如本公开所定义。还公开了含有式1化合物的组合物和用于控制由真菌病原体引起的植物病害的方法，包括施用有效量的本发明化合物或组合物。还公开了包括所有立体异构体，N-氧化物及其盐的式1A化合物，其中E，X，G和Z1如本公开所定义。还公开了式1A化合物作为制备式1化合物的中间体的用途。

4. 发明授权

US07754738B2 Pyrazole and pyrrole carboxamide insecticides 失效
标题翻译：吡唑和吡咯甲酰胺杀虫剂
公开(公告)号：US07754738B2
公开(公告)日：2010-07-13
申请号：US10514183
申请日：2003-06-10
申请人： George Philip Lahm , Robert James Pasteris , Thomas Martin Stevenson
发明人： George Philip Lahm , Robert James Pasteris , Thomas Martin Stevenson
IPC分类号： A01N43/40 , A61K31/44
CPC分类号： C07D401/04 , A01N43/40 , A01N43/56 , C07D401/14
摘要： This invention provides compounds of Formula (I), N-oxides and salts thereof wherein: A is O or S; B is a phenyl ring or a pyridine ring, each ring optionally substituted with 1 to 5 R; J is a pyrazole or a pyrrole heterocyclic ring system as defined herein; and; R1 is H; or C1-C6 alkyl, C2-C6 alkenyl, C2-C6 alkynyl or C3-C6 cycloalkyl each optionally substituted with one or more substituents selected from the group consisting of halogen, CN, NO2, hydroxy, C1-C4 alkoxy, C1-C4 alkylthio, C1-C4 alkylsulfinyl, C1-C4 alkylsulfonyl, C2-C4 alkoxycarbonyl, C1-C4 alkylamino, C2-C8 dialkylamino and C3-C6 cycloalkylamino. Also disclosed are methods for controlling at least one invertebrate pest comprising contacting the invertebrate pest or its environment with a biologically effective amount of at least one compound of Formula I, an N-oxide or a salt thereof (e.g., as a composition described herein). This invention also pertains to a composition comprising at least one compound of Formula I, an N-oxide or a salt thereof; and at least one additional component selected from the group consisting of a surfactant, a solid diluent and a liquid diluent.
摘要翻译：本发明提供式（I）的化合物，其N-氧化物及其盐，其中：A为O或S; B是苯环或吡啶环，每个环任选被1至5个R取代; J是如本文所定义的吡唑或吡咯杂环体系; 和; R1是H; 或C 1 -C 6烷基，C 2 -C 6烯基，C 2 -C 6炔基或C 3 -C 6环烷基，其各自任选被一个或多个选自卤素，CN，NO 2，羟基，C 1 -C 4烷氧基，C 1 -C 4 C 1 -C 4烷基亚磺酰基，C 1 -C 4烷基磺酰基，C 2 -C 4烷氧基羰基，C 1 -C 4烷基氨基，C 2 -C 8二烷基氨基和C 3 -C 6环烷基氨基。还公开了用于控制至少一种无脊椎害虫的方法，包括使无脊椎害虫或其环境与生物有效量的至少一种式I化合物，N-氧化物或其盐（例如，如本文所述的组合物）接触，。本发明还涉及包含至少一种式I化合物，N-氧化物或其盐的组合物; 和至少一种选自表面活性剂，固体稀释剂和液体稀释剂的另外的组分。

5. 发明授权

US08669277B2 Solid forms of an azocyclic amide 有权
标题翻译：固体形式的杂环酰胺
公开(公告)号：US08669277B2
公开(公告)日：2014-03-11
申请号：US13265138
申请日：2010-04-19
申请人： Matthew Richard Oberholzer , Robert James Pasteris , Rafael Shapiro
发明人： Matthew Richard Oberholzer , Robert James Pasteris , Rafael Shapiro
IPC分类号： A61K31/454 , C07D417/14
CPC分类号： C07D417/14 , A01N43/653 , A01N43/80 , A01N43/84 , A01N57/12 , A01N59/20
摘要： Disclosed are solid forms of 1-[4-[4-[5-(2,6-difluorophenyl)-4,5-dihydro-3-isoxazolyl]-2-thiazolyl]-1-piperidinyl]-2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethanone (Compound 1). Methods for the preparation of solid forms of Compound 1 and for the conversion of one solid form of Compound 1 into another are disclosed.Disclosed are fungicidal compositions comprising a fungicidally effective amount of a solid form of Compound 1 and at least one additional component selected from the group consisting of surfactants, solid diluents and liquid carriers. Compositions comprising a mixture of a solid form of Compound 1 and at least one other fungicide or insecticide are also disclosed.Also disclosed are methods for controlling plant diseases caused by fungal plant pathogens comprising applying to a plant or portion thereof, or to a plant seed, a fungicidally effective amount of a solid form of Compound 1.
摘要翻译：公开了1- [4- [4- [5-（2,6-二氟苯基）-4,5-二氢-3-异恶唑基] -2-噻唑基] -1-哌啶基] -2- [5- （三氟甲基）-1H-吡唑-1-基]乙酮（化合物1）。公开了制备化合物1的固体形式和将一种固体形式的化合物1转化成另一种的方法。公开了包含杀真菌有效量的固体形式的化合物1和至少一种选自表面活性剂，固体稀释剂和液体载体的另外的组分的杀真菌组合物。还公开了包含固体形式的化合物1和至少一种其它杀真菌剂或杀虫剂的混合物的组合物。还公开了用于控制由真菌植物病原体引起的植物疾病的方法，包括向植物或其部分或植物种子施用杀真菌有效量的化合物1的固体形式。

6. 发明申请

US20130045948A1 AZOCYCLIC INHIBITORS OF FATTY ACID AMIDE HYDROLASE 审中-公开
标题翻译：脂肪酸酰胺水解酶的AZOCYCLIC抑制剂
公开(公告)号：US20130045948A1
公开(公告)日：2013-02-21
申请号：US13515010
申请日：2010-12-10
申请人： Mei H. Dung , Robert James Pasteris
发明人： Mei H. Dung , Robert James Pasteris
IPC分类号： A61K31/454 , C07F7/10 , A61K31/695 , A61K31/4545 , A61P25/24 , A61K31/496 , A61P25/00 , A61P29/00 , A61P25/22 , C07D417/14 , A61K31/506
CPC分类号： C07D417/14
摘要： Disclosed are compounds of Formula 1, including all stereoisomers, N-oxides, and salts thereof, wherein A, W, X, G, R1, R2, R3, R4, m and n are as defined in the disclosure. Also disclosed are pharmaceutical compositions containing the compounds of Formula 1 and methods for treating a disease or condition mediated by fatty acid amide hydrolase activity comprising applying a therapeutically effective amount of a compound or a composition of the invention.
摘要翻译：公开了式1的化合物，包括所有立体异构体，N-氧化物及其盐，其中A，W，X，G，R 1，R 2，R 3，R 4，m和n如本公开所定义。还公开了含有式1化合物的药物组合物和用于治疗由脂肪酸酰胺水解酶活性介导的疾病或病症的方法，包括施用治疗有效量的本发明化合物或组合物。

7. 发明授权

US08349870B2 Fungicidal hetercyclic compounds 失效
标题翻译：杀真菌异环化合物
公开(公告)号：US08349870B2
公开(公告)日：2013-01-08
申请号：US12863875
申请日：2009-01-22
申请人： Balreddy Kamireddy , Robert James Pasteris , Mary Ann Hanagan
发明人： Balreddy Kamireddy , Robert James Pasteris , Mary Ann Hanagan
IPC分类号： A61K31/445 , C07D405/00
CPC分类号： C07D417/04 , C07D417/14
摘要： Disclosed are compounds of Formula 1, including all geometric and stereoisomers, N-oxides, and salts thereof, wherein E, R2, G, Z1, J and n are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling plant disease caused by a fungal pathogen comprising applying an effective amount of a compound or a composition of the invention.
摘要翻译：公开了式1的化合物，包括所有几何和立体异构体，N-氧化物及其盐，其中E，R 2，G，Z 1，J和n如本公开所定义。还公开了含有式1化合物的组合物和用于控制由真菌病原体引起的植物病害的方法，包括施用有效量的本发明化合物或组合物。

8. 发明申请

US20100292275A1 FUNGICIDAL HETEROCYCLIC COMPOUNDS 失效
标题翻译：真菌杂环化合物
公开(公告)号：US20100292275A1
公开(公告)日：2010-11-18
申请号：US12863875
申请日：2009-01-22
申请人： Balreddy Kamireddy , Robert James Pasteris , Mary Ann Hanagan
发明人： Balreddy Kamireddy , Robert James Pasteris , Mary Ann Hanagan
IPC分类号： A01N43/80 , C07D417/14 , A01P3/00
CPC分类号： C07D417/04 , C07D417/14
摘要： Disclosed are compounds of Formula 1, including all geometric and stereoisomers, N-oxides, and salts thereof, wherein E, R2, G, Z1, J and n are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling plant disease caused by a fungal pathogen comprising applying an effective amount of a compound or a composition of the invention.
摘要翻译：公开了式1的化合物，包括所有几何和立体异构体，N-氧化物及其盐，其中E，R 2，G，Z 1，J和n如本公开所定义。还公开了含有式1化合物的组合物和用于控制由真菌病原体引起的植物病害的方法，包括施用有效量的本发明化合物或组合物。

9. 发明授权

US08642634B2 Fungicidal azocyclic amides 有权
标题翻译：杀真菌唑环酰胺
公开(公告)号：US08642634B2
公开(公告)日：2014-02-04
申请号：US12303256
申请日：2007-07-27
申请人： Robert James Pasteris , Mary Ann Hanagan
发明人： Robert James Pasteris , Mary Ann Hanagan
IPC分类号： A61K31/422 , A61K31/427 , C07D263/10 , C07D277/10
CPC分类号： C07D495/10 , C07D211/62 , C07D263/14 , C07D401/06 , C07D401/14 , C07D413/04 , C07D417/04 , C07D417/14 , C07D498/10
摘要： Disclosed are compounds of Formulae 1, 1A, 1B and 1C including all geometric and stereoisomers, N-oxides, and salts thereof, wherein R1, R2, R4a1, R4a2, A, Aa, G, M, W, Z1, Z3, X, J, J1 and n are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling plant disease caused by a fungal pathogen comprising applying an effective amount of a compound or a composition of the invention.
摘要翻译：公开了具有所有几何和立体异构体，N-氧化物及其盐的式1A，1B和1C的化合物，其中R1，R2，R4a1，R4a2，A，Aa，G，M，W，Z1，Z3，X ，J，J1和n如本公开中所定义。还公开了含有式1化合物的组合物和用于控制由真菌病原体引起的植物病害的方法，包括施用有效量的本发明化合物或组合物。

10. 发明授权

US08618137B2 Fungicidal heterocyclic compounds 有权
标题翻译：杀真菌杂环化合物
公开(公告)号：US08618137B2
公开(公告)日：2013-12-31
申请号：US13127809
申请日：2009-12-02
申请人： Robert James Pasteris
发明人： Robert James Pasteris
IPC分类号： A01N43/40 , C07D401/14
CPC分类号： C07D417/04 , A01N43/78 , A01N43/80 , C07D413/04 , C07D413/14 , C07D417/14 , A01N2300/00
摘要： Disclosed are compounds of Formula 1, including all geometric and stereoisomers, tautomers, N-oxides, and salts thereof, wherein R1, R2, R3, R4, R5, A, W, X, G, Z, J and n are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling plant disease caused by a fungal pathogen comprising applying an effective amount of a compound or a composition of the invention.
摘要翻译：公开了式1的化合物，包括所有几何和立体异构体，互变异构体，N-氧化物及其盐，其中R 1，R 2，R 3，R 4，R 5，A，W，X，G，Z，J和n如在披露。还公开了含有式1化合物的组合物和用于控制由真菌病原体引起的植物病害的方法，包括施用有效量的本发明化合物或组合物。

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