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    • 9. 发明申请
    • NOVEL PYRIMIDINYLOXY- AND PYRIMIDINYLAMINO-ETHYLPHENYL-DIOXOLANE DERIVATIVES
    • 新型吡咯烷酮和吡咯烷基氨基 - 乙基苯基二氧化物衍生物
    • WO1996017843A2
    • 1996-06-13
    • PCT/EP1995004795
    • 1995-12-06
    • SANDOZ LTD.SANDOZ-PATENT-GMBHSANDOZ-ERFINDUNGEN VERWALTUNGSGESELLSCHAFT M.B.H.LAMBERTH, ClemensSCHAUB, Fritz
    • SANDOZ LTD.SANDOZ-PATENT-GMBHSANDOZ-ERFINDUNGEN VERWALTUNGSGESELLSCHAFT M.B.H.
    • C07D405/12
    • C07D405/12A01N43/54C07C69/78C07D317/20C07D317/22C07D317/24C07D317/28C07D495/04
    • The invention discloses 2-[4-(2-(pyrimidin-4-yloxy- and -4-ylamino)-ethyl-phenyl]-dioxolanes of formula (I) wherein R1 is hydrogen, C1-4alkyl, C1-4haloalkyl or C3-6cycloalkyl, R2 is hydrogen, C1-10alkyl, C1-8alkoxy-C1-4alkyl, C3-8alkenyloxy-C1-4alkyl, C3-8haloalkenyloxy-C1-4alkyl, C3-8alkynyloxy-C1-4alkyl, C1-8haloalkoxy-C1-4alkyl, C1-8alkylthio-C1-4alkyl, aryl, aryloxy-C1-4alkyl, aryl-C1-4alkoxy-C1-4-alkyl, heteroaryloxy-C1-4alkyl, C1-4alkoxy-C1-4alkoxy-C1-4alkyl or aryl-C1-8alkyl, R3 and R4 independently are halogen, C1-4alkyl, C1-4alkoxy, C1-4alkoxy-C1-4alkyl, C1-4alkoxycarbonyl-C1-4alkyl, C1-4alkoxycarbonyl, cyano-C1-4alkyl, cyano, or -COOH, or R3 and R4 together form a bridge member selected from 1,4-butylene, 1,4-butadienylene, or -S-CH=CH-, each optionally substituted by one or two radicals selected from halogen or C1-4alkyl, and Z is NH or oxygen; the use of such compounds for the control of undesired acarinae, fungi, and insects, compositions for facilitating such use, and the preparation of the compounds of formula I.
    • 本发明公开了式(I)的2- [4-(2-(嘧啶-4-基氧基 - 和-4-基氨基) - 乙基 - 苯基] - 二氧杂环戊烷,其中R 1是氢,C 1-4烷基,C 1-4卤代烷基或C 3 -6-环烷基,R 2是氢,C 1-10烷基,C 1-8烷氧基-C 1-4烷基,C 3-8烯烃氧基-C 1-4烷基,C 3-8卤代烯氧基-C 1-4烷基,C 3-8炔氧基-C 1-4烷基,C 1-8卤代烷氧基-C 1-4烷基 ,C 1-8烷硫基-C 1-4烷基,芳基,芳氧基-C 1-4烷基,芳基-C 1-4烷氧基-C 1-4 - 烷基,杂芳氧基-C 1-4烷基,C 1-4烷氧基-C 1-4烷氧基-C 1-4烷基或芳基-C1 烷基,R 3和R 4独立地是卤素,C 1-4烷基,C 1-4烷氧基,C 1-4烷氧基-C 1-4烷基,C 1-4烷氧基羰基-C 1-4烷基,C 1-4烷氧基羰基,氰基-C 1-4烷基,氰基或-COOH, 或R 3和R 4一起形成选自1,4-亚丁基,1,4-丁二烯基或-S-CH = CH-的桥连体,每个任选被一个或两个选自卤素或C 1-4烷基的基团取代,Z 是NH或氧;使用这些化合物来控制不希望的螨虫,真菌和昆虫,用于促进这种使用的组合物,以及 制备式Ⅰ化合物。