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1. 发明申请

WO2003048128A1 PYRIDYLOXYALKANOIC ACID AMIDE DERIVATIVES USEFUL AS FUNGICIDES 审中-公开
标题翻译：作为杀菌剂有用的吡咯烷酮酸酰胺衍生物
公开(公告)号：WO2003048128A1
公开(公告)日：2003-06-12
申请号：PCT/GB2002/005303
申请日：2002-11-25
申请人： SYNGENTA LIMITED , SYNGENTA PARTICIPATIONS AG , WHITTINGHAM, William, Guy , LAWSON, Kevin, Robert , WORTHINGTON, Paul, Anthony , RUSSELL, Charles, Adam , SALMON, Roger , MAY, Leslie, Francis , JORG, Mario , PACHLATKO, Johannes, Paul
发明人： WHITTINGHAM, William, Guy , LAWSON, Kevin, Robert , WORTHINGTON, Paul, Anthony , RUSSELL, Charles, Adam , SALMON, Roger , MAY, Leslie, Francis , JORG, Mario , PACHLATKO, Johannes, Paul
IPC分类号： C07D213/65
CPC分类号： C07D213/70 , A01N43/40 , C07D213/65 , C07D213/68 , C07D213/80 , C07D213/82 , C07D213/85
摘要： Fungicidal compounds of the general formula (I): wherein X and Y are independently H, halo, C 1-8 alkyl, C 3-6 cycloalkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 1-8 alkoxy, C 1-8 alkylthio, nitro, amino, mono- or di-(C 1-6 )alkylamino, mono- or di-(C 2-6 )alkenylamino, mono- or di-(C 2-6 )alkynylamino, formylamino, C 1-4 alkyl(formyl)amino, C 1-4 alkylcarbonylamino, C 1-4 alkyl(C 1-4 alkylcarbonyl)amino, cyano, formyl, C 1-4 alkylcarbonyl, C 1-4 alkoxycarbonyl, aminocarbonyl, mono- or di-(C 1-4 )alkylaminocarbonyl, carboxy, C 1-4 alkylcarbonyloxy, aryl(C 1-4 )alkylcarbonyloxy, C 1-4 alkylsulphinyl, C 1-4 alkylsulphonyl, C 1-4 alkylsulphonyloxy, aryl, heteroaryl, aryloxy, arylthio, heteroaryloxy or heteroarylthio wherein any of the foregoing alkyl, cycloalkyl, alkenyl, alkynyl, aryl, heteroaryl, groups or moieties are optionally substituted; R 1 is phenyl, cyano, C 1-4 alkyl, C 2-4 alkenyl or C 2-4 alkynyl in which the alkyl, alkenyl and alkynyl groups are optionally substituted on their terminal carbon atom with one, two or three halogen atoms, with a cyano group, with a C 1-4 alkylcarbonyl group, with a C 1-4 alkoxycarbonyl group or with a hydroxy group, or R 1 is alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl or alkylsulphonylalkyl in which the total number of carbon atoms is 2 or 3; R 2 is H, C 1-4 alkyl, C 1-4 alkoxymethyl or benzyloxymethyl in which the phenyl ring of the benzyl moiety is optionally substituted with C 1-4 alkoxy; R 3 and R 4 are independently H, C 1-3 alkyl, C 2-3 alkenyl or C 2-3 alkynyl provided that both are not H and that when both are other than H their combined total of carbon atoms does not exceed 4, or R 3 and R 4 join with the carbon atom to which they are attached to form a 3 or 4 membered carbocyclic ring optionally containing one O, S or N atom and optionally substituted with halo or C 1-4 alkyl; and R 5 is halo, C 1-4 alkyl or C 3-4 cycloalkyl in which the alkyl or cycloalkyl group is optionally substituted with halo, hydroxy, C 1-6 alkoxy, C 1-6 alkylthio, cyano, C 1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di(C 1-4 )alkylaminocarbonyloxy, or tri(C 1-4 )alkylsilyloxy. The compounds and compositions containing them are especially useful for combating fungal infections of plants.
摘要翻译：通式（I）的杀真菌化合物：其中X和Y独立地为H，卤素，C 1-8烷基，C 3-6环烷基，C 2-8链烯基，C 2-8 炔基，C> 1-8 <烷氧基，C 1-8烷基硫基，硝基，氨基，单 - 或二 - （C 1-6）烷基氨基，单 - 或二 - （C 2-6）链烯基氨基，单 - 或二 - （C 2-6）炔基氨基，甲酰氨基，C 1-4烷基（甲酰基）氨基，C 1-4烷基羰基氨基，C 1-4烷基（C 1 -4 <烷基羰基）氨基，氰基，甲酰基，C 1-4烷基羰基，C 1-4烷氧基羰基，氨基羰基，一或二 - （C 1-4）烷基氨基羰基，羧基， 4 <烷基羰基氧基，芳基（C 1-4）烷基羰基氧基，C 1-4烷基亚磺酰基，C 1-4烷基磺酰基，C 1-4烷基磺酰氧基，芳基，杂芳基，芳氧基，芳硫基，杂芳氧基或杂芳硫基其中任何前述烷基，环烷基，烯基，炔基，芳基，杂芳基，基团或部分任选被取代; R 1是苯基，氰基，C 1-4烷基，C 2-4链烯基或C 2-4炔基，其中烷基，烯基和炔基在其末端碳原子上任选被一个，两个或三个卤素原子取代，具有C 1-4烷基羰基，C 1-4烷氧基羰基或羟基的氰基，或者R 1是烷基烷基或烷基磺酰基烷基，其中总碳原子数为2或3的烷氧基烷基，烷硫基烷基，烷基亚磺酰基烷基或烷基磺酰基烷基 ; R 2是H，C 1-4烷基，C 1-4烷氧基甲基或苄氧基甲基，其中苄基部分的苯环任选被C 1-4烷氧基取代; R 3和R 4独立地是H，C 1-3烷基，C 2-3烯基或C 2-3炔基，条件是两者都不是H，当两者都不是H时，它们的总碳原子数不超过 4或R 3和R 4与它们所连接的碳原子一起形成任选含有一个O，S或N原子并任选被卤素或C 1-4烷基取代的3或4元碳环 ; 羟基，C 1-6烷氧基，C 1-6烷硫基，氰基，C 1-4烷基羰基氧基，氨基羰基氧基，C 1-4烷氧基，C 1-4烷氧基，，单或二（C 1-4）烷基氨基羰基氧基或三（C 1-4）烷基甲硅烷氧基。含有它们的化合物和组合物特别可用于防治植物的真菌感染。

2. 发明申请

WO02092801A2 METHODS AND COMPOSITIONS FOR MAKING EMAMECTIN 审中-公开
标题翻译：制备EMAMECTIN的方法和组合物
公开(公告)号：WO02092801A2
公开(公告)日：2002-11-21
申请号：PCT/EP0205363
申请日：2002-05-15
申请人： SYNGENTA PARTICIPATIONS AG , MOLNAR ISTVAN , LIGON JAMES MADISON , ZIRKLE ROSS ERIC , HAMMER PHILIP EUGENE , HILL DWIGHT STEVEN , PACHLATKO JOHANNES PAUL , BUCKEL THOMAS GUENTER
发明人： MOLNAR ISTVAN , LIGON JAMES MADISON , ZIRKLE ROSS ERIC , HAMMER PHILIP EUGENE , HILL DWIGHT STEVEN , PACHLATKO JOHANNES PAUL , BUCKEL THOMAS GUENTER
IPC分类号： C12N15/09 , C07K16/40 , C12N1/21 , C12N9/02 , C12N15/53 , C12P17/16 , C12P17/18 , C12P21/00 , C12N9/00
CPC分类号： C12N9/0077 , C12P17/181
摘要： Disclosed is a family of P450 monooxygenases, each member of which regioselectively oxidizes avermectin to 4"-keto-avermectin. The P450 monooxgenases find use in methods and formulations for making emamectin from avermectin. Also disclosed are methods for purifying the P450 monooxygenases of the invention, binding agents that specifically bind to the P450 monooxygenases of the invention, and genetically engineered cells that express the P450 monooxygenases of the invention. Also disclosed are ferrodoxins and ferredoxin reductases that are active with the P450 monooxygenases of the invention.
摘要翻译：公开了一种P450单加氧酶家族，其中每个成员区域选择性地将阿维菌素氧化为4“ - 除虫菌素，P450单加氧酶可用于制备来自阿维菌素的阿维菌素的方法和制剂，还公开了纯化本发明的P450单加氧酶的方法，特异性结合本发明的P450单加氧酶的结合剂，以及表达本发明的P450单加氧酶的遗传工程改造的细胞。还公开了与本发明的P450单加氧酶有活性的铁氧还蛋白和铁氧还蛋白还原酶。

3. 发明申请

WO2002092801A3 METHODS AND COMPOSITIONS FOR MAKING EMAMECTIN 审中-公开
公开(公告)号：WO2002092801A3
公开(公告)日：2002-11-21
申请号：PCT/EP2002/005363
申请日：2002-05-15
申请人： SYNGENTA PARTICIPATIONS AG , MOLNAR, Istvan , LIGON, James, Madison , ZIRKLE, Ross, Eric , HAMMER, Philip, Eugene , HILL, Dwight, Steven , PACHLATKO, Johannes, Paul , BUCKEL, Thomas, Günter
发明人： MOLNAR, Istvan , LIGON, James, Madison , ZIRKLE, Ross, Eric , HAMMER, Philip, Eugene , HILL, Dwight, Steven , PACHLATKO, Johannes, Paul , BUCKEL, Thomas, Günter
IPC分类号： C12P19/62
摘要： Disclosed is a family of P450 monooxygenases, each member of which regioselectively oxidizes avermectin to 4"-keto-avermectin. The P450 monooxgenases find use in methods and formulations for making emamectin from avermectin. Also disclosed are methods for purifying the P450 monooxygenases of the invention, binding agents that specifically bind to the P450 monooxygenases of the invention, and genetically engineered cells that express the P450 monooxygenases of the invention. Also disclosed are ferrodoxins and ferredoxin reductases that are active with the P450 monooxygenases of the invention.

4. 发明申请

WO1992011258A1 THIANGAZOLE, ITS PREPARATION, COMPOSITIONS AND USE THEREOF 审中-公开
标题翻译：泰坦尼亚唑，其制备，组合物及其用途
公开(公告)号：WO1992011258A1
公开(公告)日：1992-07-09
申请号：PCT/EP1991002336
申请日：1991-12-06
申请人： GESELLSCHAFT FÜR BIOTECHNOLOGISCHE FORSCHUNG MBH , CIBA-GEIGY AG , HÖFLE, Gerhard , BEDORF, Norbert , FORCHE, Edgar , GERTH, Klaus , IRSCHIK, Herbert , JANSEN, Rolf , KUNZE, Brigitte , REICHENBACH, Hans , SASSE, Florenz , STEINMETZ, Heinrich , TROWITZSCH-KIENAST, Wolfram , PACHLATKO, Johannes, Paul
发明人： GESELLSCHAFT FÜR BIOTECHNOLOGISCHE FORSCHUNG MBH , CIBA-GEIGY AG
IPC分类号： C07D417/14
CPC分类号： C07D417/14 , A01N43/78 , A01N63/02
摘要： The invention relates to compounds of general formula (I) especially the compound of formula (Ia) referred to as thiangazole their pharmaceutically acceptable acid addition salts, processes for their preparation and therapeutic compositions and compositions that can be used in crop-protection.
摘要翻译：本发明涉及通式（I）的化合物，特别是称为噻唑的药学上可接受的酸加成盐的式（Ia）化合物，其制备方法以及可用于作物保护的治疗组合物和组合物。

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