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1. 发明授权

US5817863A Process and novel intermediates for preparing triazolinones 失效
标题翻译：制备三唑啉酮的方法和新型中间体
公开(公告)号：US5817863A
公开(公告)日：1998-10-06
申请号：US898981
申请日：1997-07-23
申请人： Heinz-Jurgen Wroblowsky
发明人： Heinz-Jurgen Wroblowsky
IPC分类号： C07C281/02 , C07C281/04 , C07D249/12
CPC分类号： C07C281/02 , C07C281/04 , C07D249/12
摘要： The present invention relates to a novel process for preparing triazolinones of the general formula (I) ##STR1## in which R.sup.1 represents halogenoalkyl, and R.sup.2 represents hydrogen, hydroxyl or amino, or represents alkyl, alkenyl, alkinyl, alkoxy, alkylamino, dialkylamino, cycloalkyl, cycloalkylalkyl, phenyl or phenylalkyl which are in each case optionally substituted, and also to novel intermediates for preparing these triazolinones and to processes for preparing the intermediates themselves.
摘要翻译：本发明涉及一种制备通式（I）的三唑啉酮的新方法，其中R1代表卤代烷基，R2代表氢，羟基或氨基，或代表烷基，烯基，炔基，烷氧基，烷基氨基在各种情况下任选被取代的二烷基氨基，环烷基，环烷基烷基，苯基或苯基烷基，以及制备这些三唑啉酮的新型中间体以及制备中间体本身的方法。

2. 发明授权

US4945165A Pest-combating agents based on pyrazole derivatives 失效
标题翻译：基于吡唑衍生物的抗虫剂
公开(公告)号：US4945165A
公开(公告)日：1990-07-31
申请号：US384188
申请日：1989-07-21
申请人： Uta Jensen-Korte , Reinhold Gehring , Otto Schallner , Jorg Stetter , Heinz-Jurgen Wroblowsky , Benedikt Becker , Bernhard Homeyer , Wolfgang Behrenz , Wilhelm Stendel , Peter Andrews
发明人： Uta Jensen-Korte , Reinhold Gehring , Otto Schallner , Jorg Stetter , Heinz-Jurgen Wroblowsky , Benedikt Becker , Bernhard Homeyer , Wolfgang Behrenz , Wilhelm Stendel , Peter Andrews
IPC分类号： A01N43/56 , A01N47/02 , C07D231/38 , C07D231/44 , C07D401/04
CPC分类号： C07D401/04 , A01N43/56 , A01N47/02 , C07D231/44
摘要： A 5-aminopyrazole of the formula (I) ##STR1## in which R.sup.2 represents CF.sub.3 or CCL.sub.2 F,R.sup.3 represents hydrogen or CH.sub.3and n represents the number 0 or 1.The 5-aminopyrazole of formula (I) is effective in combating insects, sense animals and nematodes.

3. 发明授权

US4771066A 4-haloalkylthio-5-amino-1-arylpyrazoles, composition containing them, and insecticidal and acaricidal method of using them 失效
标题翻译： 4-卤代烷硫基-5-氨基-1-芳基吡唑，含有它们的组合物，以及使用它们的杀虫和杀螨方法
公开(公告)号：US4771066A
公开(公告)日：1988-09-13
申请号：US13741
申请日：1987-02-12
申请人： Reinhold Gehring , Uta Jensen-Korte , Otto Schallner , Jorg Stetter , Heinz-Jurgen Wroblowsky , Benedikt Becker , Wolfgang Behrenz , Bernhard Homeyer , Wilhelm Stendel
发明人： Reinhold Gehring , Uta Jensen-Korte , Otto Schallner , Jorg Stetter , Heinz-Jurgen Wroblowsky , Benedikt Becker , Wolfgang Behrenz , Bernhard Homeyer , Wilhelm Stendel
IPC分类号： A01N43/56 , A01N47/02 , A61K31/415 , A61K31/44 , A61K31/4427 , A61P33/00 , C07D231/44 , C07D401/04
CPC分类号： C07D401/04 , A01N43/56 , A01N47/02 , C07D231/44
摘要： Insecticidally and acarididally active 1-arylpyrazoles of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl or halogen alkyl,R.sup.2 represents alkyl, alkenyl, alkinyl, cycloalkyl, halogenoalkyl, halogenoalkenyl, alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl, alkylsulphonylalkyl, optionally substituted aralkyl or optionally substituted aryl,R.sup.3 represents alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, alkoxyalkyl, alkylthioalkyl, cycloalkyl or optionally substituted aralkyl,R.sup.4 represents alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, alkoxyalkyl, alkylthioalkyl, cycloalkyl or optionally substituted aralkyl, and, in addition, also represents hydrogen in the case where R.sup.3 does not simultaneously represent unsubstituted alkyl, orR.sup.3 and R.sup.4, together with the nitrogen atom to which they are bound, represent a saturated heterocycle, which can optionally contain further heteroatoms,Ar represents in each case optionally substituted phenyl or pyridyl, andn represents a number 0, 1 or 2.
摘要翻译：具有式“IMAGE”的杀虫和杀螨活性1-芳基吡唑其中R1代表氢，烷基或卤素烷基，R2代表烷基，烯基，炔基，环烷基，卤代烷基，卤代烯基，烷氧基烷基，烷硫基烷基，烷基亚磺酰基烷基，烷基磺酰基烷基，任选取代的芳烷基或任选取代的芳基，R 3表示烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基烷基，烷硫基烷基，环烷基或任选取代的芳烷基，R 4表示烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基烷基，烷硫基烷基，环烷基或任选取代的芳烷基，此外，在R3不同时表示未取代的烷基的情况下也表示氢，或者R 3和R 4与它们所连接的氮原子一起代表饱和的杂环，其可以任选地含有另外的杂原子，Ar表示每个任选取代的苯基或吡啶基，n表示数字0，1或2。

4. 发明授权

US5892054A Process for the preparation of alkoxytriazolinones 失效
标题翻译：制备烷氧基三唑啉酮的方法
公开(公告)号：US5892054A
公开(公告)日：1999-04-06
申请号：US934501
申请日：1997-09-19
申请人： Heinz-Jurgen Wroblowsky , Klaus Konig
发明人： Heinz-Jurgen Wroblowsky , Klaus Konig
IPC分类号： C07C281/04 , C07C281/16 , C07D249/12
CPC分类号： C07D249/12 , C07C281/04
摘要： Alkoxytriazolinones of the formula (I), ##STR1## in which R.sup.1 and R.sup.2 independently of one another represent in each case optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkylalkyl, aryl or arylalkyl,(which can be used as intermediates for the preparation of herbicidal active compounds) are obtained in good yields and in high purity by reacting iminocarbonic diesters (II) with carbazinic esters (III) ##STR2## in which R.sup.2 and R.sup.3 in each case represent, for example, alkyl or aryl,at -20.degree. C. to +120.degree. C. (1st step) and subjecting the semicarbazide derivatives (IV) formed in this process with elimination of R.sup.2 -OH ##STR3## to a cyclizing condensation reaction in the presence of a base at 20.degree. C. to 150.degree. C. with elimination of R.sup.3 --OH, if appropriate (2nd step) and, finally, by reacting the resulting 5-alkoxytriazolinones of the formula (V) �=formula (I) where R.sup.1 =H! with an alkylating agent of the formula R.sup.1 --X (VI) �X, for example,=halogen or --OSO.sub.2 OR.sup.1 ! at 0.degree. C. to 150.degree. C., if appropriate in the presence of a base (3rd step: highly selective 4-alkylation).
摘要翻译：式（I）的烷氧基三唑啉酮，其中R 1和R 2彼此独立地表示，各自为任选取代的烷基，烯基，炔基，环烷基，环烷基烷基，芳基或芳基烷基（可用作中间体用于制备除草活性化合物）以良好的产率和高纯度通过使亚氨基碳酸二酯（II）与咔嗪酸酯（III）反应获得，其中R2和R3各自表示例如，烷基或芳基，在-20℃至+ 120℃（第一步），并将在该过程中形成的氨基脲衍生物（Ⅳ）与R 2 -OH反应生成环状在20℃至150℃存在下，在适当的情况下消除R3-OH（第二步），最后通过使得到的式（V）的5-烷氧基三唑啉酮[= 式（I）其中R1 = H]与式R1-X（VI）的烷基化剂[X，例如=卤素或 -OSO2OR1]在0℃至150℃，如果合适的话，在碱的存在下（第3步：高选择性4-烷基化）。

5. 发明授权

US4820725A 1-aryl-pyrazoles, pesticidal compositions and use 失效
标题翻译： 1-芳基吡唑，农药组合物和用途
公开(公告)号：US4820725A
公开(公告)日：1989-04-11
申请号：US893133
申请日：1986-08-04
申请人： Uta Jensen-Korte , Reinhold Gehring , Otto Schallner , Jorg Stetter , Heinz-Jurgen Wroblowsky , Benedikt Becker , Wilhelm Stendel , Berhard Homeyer , Wolfgang Behrenz
发明人： Uta Jensen-Korte , Reinhold Gehring , Otto Schallner , Jorg Stetter , Heinz-Jurgen Wroblowsky , Benedikt Becker , Wilhelm Stendel , Berhard Homeyer , Wolfgang Behrenz
IPC分类号： A01N25/04 , A01N43/40 , A01N43/56 , A01P7/02 , A01P7/04 , C07D231/18 , C07D401/04
CPC分类号： C07D401/04 , A01N43/56 , C07D231/18
摘要： 1-Aryl-pyrazole of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl or halogenoalkyl,R.sup.2 represents alkyl, halogenoalkyl or in each case optionally substituted aralkyl or aryl,R.sup.3 represents hydrogen or halogen,Ar represents optionally substituted phenyl or pyridyl, andn represents the number 0, 1 or 2,the 1-aryl-pyrazole being useful in agents for combating pests.
摘要翻译：其中R 1表示氢，烷基或卤代烷基，R 2表示烷基，卤代烷基或在各种情况下任选取代的芳烷基或芳基，R 3表示氢或卤素，Ar表示任意取代的苯基或吡啶基，并且n表示数字0,1或2，1-芳基 - 吡唑可用于防治害虫的试剂。

6. 发明授权

US4803215A 5-Heterocyclyl-1-aryl-pyrazoles, composition containing them, and method of using them to combat insects, acarids and nematodes 失效
标题翻译： 5-杂环基-1-芳基吡唑，含有它们的组合物及其用于对抗昆虫，螨虫和线虫的方法
公开(公告)号：US4803215A
公开(公告)日：1989-02-07
申请号：US942476
申请日：1986-12-16
申请人： Uta Jensen-Korte , Reinhold Gehring , Otto Schallner , Jorg Stetter , Heinz-Jurgen Wroblowsky , Benedikt Becker , Bernhard Homeyer , Wolfgang Behrenz , Wilhelm Stendel
发明人： Uta Jensen-Korte , Reinhold Gehring , Otto Schallner , Jorg Stetter , Heinz-Jurgen Wroblowsky , Benedikt Becker , Bernhard Homeyer , Wolfgang Behrenz , Wilhelm Stendel
IPC分类号： C07D231/44 , C07D401/14 , C07D403/04 , C07D521/00
CPC分类号： C07D231/12 , C07D231/44 , C07D233/56 , C07D249/08 , C07D401/14 , C07D403/04
摘要： Pesticidally active 5-heterocyclyl-1-aryl-pyrazoles of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl or haloalkyl,R.sup.2 represents alkyl, alkenyl, alkinyl, cycloalkyl, haloalkyl, haloalkenyl, optionally substituted aralkyl or optionally substituted aryl,Ar represents in each case optionally substituted phenyl or pyridyl,Het represents a heterocycle of the formula ##STR2## n represents a number 0, 1 or 2, whereR.sup.3 and R.sup.4, independently of one another, represent in each case hydrogen, alkyl or phenyl.Intermediates of the formulas ##STR3## are provided, the former also being pesticidal.
摘要翻译：式（Ia）的农药活性的5-杂环基-1-芳基 - 吡唑，其中R1代表氢，烷基或卤代烷基，R2代表烷基，烯基，炔基，环烷基，卤代烷基，卤代链烯基，任意取代的芳烷基或任意取代的芳基，Ar 在每种情况下表示任选取代的苯基或吡啶基，Het表示下式的杂环：其中R 3和R 4彼此独立地表示氢，烷基或苯基。提供了公式 + TR 的中间体，前者也是杀虫剂。

7. 发明授权

US6121204A Herbicidal or fungicidal sulphonylaminocarbonyltriazolinones with halogenated alk(en)oxy substituents 失效
标题翻译：具有卤代烷（en）氧取代基的除草或杀真菌磺酰氨基羰基三唑啉酮
公开(公告)号：US6121204A
公开(公告)日：2000-09-19
申请号：US894931
申请日：1997-12-08
申请人： Klaus-Helmut Muller , Rolf Kirsten , Ernst Rudolf F. Gesing , Joachim Kluth , Kurt Findeisen , Johannes R. Jansen , Klaus Konig , Hans-Jochem Riebel , Otto Schallner , Heinz-Jurgen Wroblowsky , Markus Dollinger , Hans-Joachim Santel , Klaus Stenzel
发明人： Klaus-Helmut Muller , Rolf Kirsten , Ernst Rudolf F. Gesing , Joachim Kluth , Kurt Findeisen , Johannes R. Jansen , Klaus Konig , Hans-Jochem Riebel , Otto Schallner , Heinz-Jurgen Wroblowsky , Markus Dollinger , Hans-Joachim Santel , Klaus Stenzel
IPC分类号： A01N47/38 , C07D249/08 , C07D249/12 , C07D249/14 , C07D405/12 , C07D409/12 , C07D417/12 , A01N43/653
CPC分类号： C07D249/08 , A01N47/38 , C07D249/12
摘要： The invention relates to novel sulphonylaminocarbonyltriazolinones having halogenoalkoxy substituents of the formula (I) ##STR1## in which R.sup.1 represents hydrogen, hydroxyl, amino, alkylideneamino or a respectively optionally substituted radical from the group consisting of alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkylamino, dialkylamino, alkanoylamino, cycloalkyl, cycloalkylalkyl, cycloalkylamino, aryl and arylalkyl,R.sup.2 represents respectively halogen-substituted alkyl or alkenyl, andR.sup.3 represents a respectively optionally substituted radical from the group consisting of alkyl, aralkyl, aryl and heteroaryl,and salts of compounds of the formula (I), and to processes and novel intermediates for preparing the compounds (I), and to their use as herbicides and/or fungicides.
摘要翻译： PCT No.PCT / EP96 / 00833 371 1997年12月8日第 102（e）日期1997年12月8日PCT 1996年3月1日PCT公布。出版物WO96 / 27590 日期1996年9月12日本发明涉及具有式（I）的卤代烷氧基取代基的新型磺酰基氨基羰基三唑啉酮，其中R1表示氢，羟基，氨基，亚烷基氨基或分别任选取代的基团，其由烷基，烯基，炔基，烷氧基，烯基氧基，烷基氨基，二烷基氨基，烷酰基氨基，环烷基，环烷基烷基，环烷基氨基，芳基和芳基烷基，R 2分别表示卤素取代的烷基或链烯基，R 3表示任选取代的由烷基，芳烷基，芳基和杂芳基组成的组中的基团，式（I）化合物的盐，以及用于制备化合物（I）的方法和新中间体，以及它们作为除草剂和/或杀真菌剂的用途。

8. 发明授权

US6054589A Process for preparing 2-chloro-benzimidazole derivatives 失效
标题翻译： 2-氯 - 苯并咪唑衍生物的制备方法
公开(公告)号：US6054589A
公开(公告)日：2000-04-25
申请号：US118954
申请日：1998-07-17
申请人： Michael Conrad , Lutz Assmann , Heinz-Jurgen Wroblowsky , Carl Casser , Dietmar Bielefeldt
发明人： Michael Conrad , Lutz Assmann , Heinz-Jurgen Wroblowsky , Carl Casser , Dietmar Bielefeldt
IPC分类号： B01J27/06 , B01J27/14 , C07B61/00 , C07D491/04 , C07D491/056 , C07D235/02
CPC分类号： C07D491/04
摘要： A novel process for the preparation of 2-chloro-benzimidazole derivatives of the formula ##STR1## in which A represents optionally halogenated alkylene having 1 or 2 carbon atoms,which process comprises reaction 1,3-dihydro-benzimidazol(ethi)ones of the formula ##STR2## in which X represents oxygen or sulphur,with phosphorus oxychloride.Novel 1,3-dihydro-benzimidazol(ethi)ones of the formula(II) and process for their preparation.
摘要翻译：一种用于制备下式的2-氯 - 苯并咪唑衍生物的新方法，其中A表示任选地具有1或2个碳原子的卤代亚烷基，该方法包括下式的反应1,3-二氢 - 苯并咪唑（ethi），其中 X表示氧或硫，与磷酰氯反应。新的式（II）的1,3-二氢 - 苯并咪唑（ethi）及其制备方法。

9. 发明授权

US5703260A Process for the preparation of alkoxytriazolinones 失效
标题翻译：制备烷氧基三唑啉酮的方法
公开(公告)号：US5703260A
公开(公告)日：1997-12-30
申请号：US714668
申请日：1996-09-16
申请人： Heinz-Jurgen Wroblowsky , Klaus Konig
发明人： Heinz-Jurgen Wroblowsky , Klaus Konig
IPC分类号： C07C281/06 , C07D249/12
CPC分类号： C07D249/12 , C07C281/06
摘要： Alkoxytriazolinones of the general formula (I), ##STR1## in which R.sup.1 represents hydrogen, or represents in each case optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkylalkyl, aryl or arylalkyl, and R.sup.2 represents in each case optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkylalkyl, ary or arylalkyl, (which can be used as intermediates for the preparation of herbicidal active compounds) are obtained in very good yields and in high purity by reacting imino(thio)carbonic esters (II) with alkoxyethyl carbazinates (III) ##STR2## in which Q represents O or S, R.sup.3 represents (for example) alkyl, aryl or aralkyl and R.sup.4 represents (for example) alkyl, at -20.degree. C. to +150.degree. C. (1st step) and subjecting the new semicarbazide derivatives (IV) ##STR3## which are formed with elimination of R.sup.3 --QH, if appropriate after intermediate isolation, to a cyclizing condensation reaction at 0.degree. C. to 200.degree. C., without the addition of a base, advantageously under reduced pressure, with the elimination of alkoxyethanols (2nd step).
摘要翻译：通式（I）的烷氧基三唑啉酮，其中R 1表示氢，或在每种情况下表示任选取代的烷基，烯基，炔基，环烷基，环烷基烷基，芳基或芳基烷基，和R 2表示在各种情况下任选取代的通过使亚氨基（硫代）碳酸酯（II）反应，以非常好的产率和高纯度获得烷基，链烯基，炔基，环烷基，环烷基烷基，芳基或芳烷基（可用作制备除草活性化合物的中间体）其中Q代表O或S，R3代表（例如）烷基，芳基或芳烷基，R4代表（例如）烷基，在-20℃至+ 150℃（第1步），在0℃〜200℃进行环化缩合反应，在中间分离后，如果合适，将R3-QH所形成的新的氨基脲衍生物（IV）没有添加基地，优势在减压下，剔除烷氧基乙醇（第二步）。

10. 发明授权

US5104439A Herbicidal agents based on pyrazole derivatives 失效
标题翻译：基于吡唑衍生物的除草剂
公开(公告)号：US5104439A
公开(公告)日：1992-04-14
申请号：US569493
申请日：1990-08-20
申请人： Otto Schallner , Reinhold Gehring , Erich Klauke , Jorg Stetter , Heinz-Jurgen Wroblowsky , Robert R. Schmidt , Hans-Joachim Santel
发明人： Otto Schallner , Reinhold Gehring , Erich Klauke , Jorg Stetter , Heinz-Jurgen Wroblowsky , Robert R. Schmidt , Hans-Joachim Santel
IPC分类号： A01N43/56 , A01N47/02 , A01N47/18 , A01N47/22 , A01N47/36 , A01N53/00 , A01N57/22 , A01N57/24 , C07C67/00 , C07C253/00 , C07C255/66 , C07C317/32 , C07C317/48 , C07C323/48 , C07D231/38 , C07D231/40 , C07F9/40 , C07F9/6509
CPC分类号： C07D231/38 , A01N43/56 , A01N47/02 , A01N47/18 , A01N47/22 , A01N47/36 , A01N53/00 , A01N57/22 , C07D231/40 , C07F9/4015 , C07F9/650935
摘要： Herbicidally active 5-amino-1-phenyl-pyrazoles, most of which are new, of the formula ##STR1##

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