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标题翻译：（4,4-DIFLUOROBUT-3-ENYLTHIO） - 具有杀虫活性的杂环化合物或碳环化合物

公开(公告)号：WO1995024403A1

公开(公告)日：1995-09-14

申请号：PCT/GB1995000400

申请日：1995-02-27

申请人： ZENECA LIMITED , TURNBULL, Michael, Drysdale , BANSAL, Harjinder, Singh , SMITH, Alison, Mary , SALMON, Roger , FITZJOHN, Steven , GODFREY, Christopher, Richard, Ayles , HOTSON, Matthew, Brian , SILLARS, Nan, Catherine , DOWLING, Alan, John

发明人： ZENECA LIMITED

IPC分类号： C07D307/64

CPC分类号： C07D213/70 , A01N33/22 , A01N43/08 , A01N43/10 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/64 , A01N43/66 , A01N43/707 , A01N43/713 , A01N43/74 , A01N43/80 , A01N43/82 , C07C17/087 , C07C17/23 , C07C323/09 , C07D213/71 , C07D213/80 , C07D213/82 , C07D213/85 , C07D231/18 , C07D231/28 , C07D231/30 , C07D233/86 , C07D233/90 , C07D233/92 , C07D237/18 , C07D237/30 , C07D241/18 , C07D241/44 , C07D251/22 , C07D253/04 , C07D253/07 , C07D253/075 , C07D253/10 , C07D257/04 , C07D261/10 , C07D261/18 , C07D263/34 , C07D263/46 , C07D271/07 , C07D271/113 , C07D275/03 , C07D277/36 , C07D277/56 , C07D277/58 , C07D285/08 , C07D285/125 , C07D285/135 , C07D307/64 , C07D333/34 , C07D333/38 , C07D333/62 , C07D409/04 , C07D413/04 , C07D417/04 , C07D471/04 , C07C19/14 , C07C21/18

摘要： A compound of formula (I), or a salt thereof, wherein n is 0, 1 or 2; and R is a group of formulae (II) to (XXI), wherein: the S(O)nCH2CH2CH=CF2 group is at least one of R1 (when attached to a carbon atom), R2, R3, R4, R5 or R6; R1 (when attached to a carbon atom), R2, R3, R4, R5 and R6 are each independently hydrogen, optionally substituted alkyl, optionally substituted alkenyl, alkynyl, cycloalkyl, alkylcycloalkyl, alkoxy, alkenyloxy, alkynyloxy, hydroxyalkyl, alkoxyalkyl, optionally substituted aryl, optionally substituted arylalkyl, optionally substituted heteroaryl, optionally substituted heteroarylalkyl, optionally substituted aryloxy, optionally substituted arylalkoxy, optionally substituted aryloxyalkyl, optionally substituted heteroaryloxy, optionally substituted heteroarylalkoxy, optionally substituted heteroaryloxyalkyl, haloalkyl, haloalkenyl, haloalkynyl, haloalkoxy, haloalkenyloxy, haloalkynyloxy, halogen, hydroxy, cyano, nitro, -NR7R8, -NR7COR8, -NR7CSR8, -NR7SO2R8, -N(SO2R7)(SO2R8), -COR7, -CONR7R8, -alkylCONR7R8, CR7NR8, -COOR7, -OCOR7, -SR7, -SOR7, SO2R7, -alkylSR7, -alkylSOR7, -alkylSO2R7, -OSO2R7, -SO2NR7R8, -CSNR7R8, SiR7R8R9, -OCH2CO2R7, -OCH2CH2CO2R7, -CONR7SO2R8, -alkylCONR7SO2R8, -NHCONR7R8, -NHCSNR7R8, or an adjacent pair of R1, R2, R3, R4, R5 and R6 when taken together form a fused 5- or 6-membered carbocyclic or heterocyclic ring; R1 (when attached to a nitrogen atom) is hydrogen, optionally substituted alkyl, cycloalkyl, alkylcycloalkyl, hydroxyalkyl, alkoxyalkyl, optionally substituted aryl, optionally substituted arylalkyl, optionally substituted aryloxyalkyl, optionally substituted heteroaryl, optionally substituted heteroarylakyl, optionally substituted heteroaryloxyalkyl, haloalkyl, hydroxy, cyano, nitro, -NR7R8, -NR7COR8, NR7CSR8, -NR7COOR8, -NR7SO2R8, -N(SO2R7)(SO2R8), -COR7, -CONR7R8, -alkylCONR7R8, -CR7NR8, -COOR7, -OCOR7, -SOR7, -SO2R7, -alkylSR7, -alkylSOR7, -alkylSO2R7, -OSO2R7, -SO2NR7NR8, -SR7, -SOR7, -SO2R7, -CSNR7R8, -SiR7R8R7, -OCH2CO2R7, -OCH2CH2CO2R7, -CONR7SO2R8, -alkylCONR7SO2R8, -NHCOR7R8, or -NHCSR7R8; and R7, R8 and R9 are each independently hydrogen, optionally substituted alkyl, optionally substituted alkenyl, alkynyl, optionally substituted aryl or optionally substituted arylalkyl, haloalkyl, haloalkenyl, haloalkynyl, halogen, or hydroxy.

摘要翻译：式（I）化合物或其盐，其中n为0,1或2; 其中：S（O）nCH 2 CH 2 CH = CF 2基团是R 1（当连接到碳原子上），R 2，R 3，R 4，R 5或R 6中的至少一个时 ; R1（当连接到碳原子上）时，R 2，R 3，R 4，R 5和R 6各自独立地为氢，任选取代的烷基，任选取代的烯基，炔基，环烷基，烷基环烷基，烷氧基，烯氧基，炔氧基，羟烷基，烷氧基烷基，芳基，任选取代的芳基烷基，任选取代的杂芳基，任选取代的杂芳基烷基，任选取代的芳氧基，任选取代的芳基烷氧基，任选取代的芳氧基烷基，任选取代的杂芳氧基，任选取代的杂芳基烷氧基，任选取代的杂芳氧基烷基，卤代烷基，卤代烯基，卤代炔基，卤代烷氧基，卤素，羟基，氰基，硝基，-NR7R8，-NR7COR8，-NR7CSR8，-NR7SO2R8，-N（SO2R7）（SO2R8），-COR7，-CONR7R8， - 烷基CONR7R8，CR7NR8，-COOR7，-OCOR7，-SR7， SOR 7，SO 2 R 7， - 烷基R 7， - 烷基SOR 7， - 烷基SO 2 R 7，-OSO 2 R 7，-SO 2 NR 7 R 8，-CSNR 7 R 8，SiR 7 R 8 R 9，-OCH 2 CO 2 R 7，-OCH 2 CH 2 CO 2 R 7，-CONR 7 SO 2 R 8， - 烷基CONR 7 SO 2 R 8， NR7R8，-NHCSNR7R8或相邻的R1，R2，R3，R4，R5和R6组合在一起形成稠合的5元或6元碳环或杂环; R 1（当连接到氮原子时）是氢，任选取代的烷基，环烷基，烷基环烷基，羟烷基，烷氧基烷基，任选取代的芳基，任选取代的芳基烷基，任选取代的芳氧基烷基，任选取代的杂芳基，任选取代的杂芳基，任选取代的杂芳基烷基，卤代烷基，羟基，氰基，硝基，-NR7R8，-NR7COR8，NR7CSR8，-NR7COOR8，-NR7SO2R8，-N（SO2R7）（SO2R8），-COR7，-CONR7R8， - 烷基CONR7R8，-CR7NR8，-COOR7，-OCOR7，-SOR7， -SO 2 R 7， - 烷基R 7， - 烷基SOR 7， - 烷基SO 2 R 7，-OSO 2 R 7，-SO 2 NR 7 NR 8，-SR 7，-SOR 7，-SO 2 R 7，-CSNR 7 R 8，-SiR 7 R 8 R 7，-OCH 2 CO 2 R 7，-OCH 2 CH 2 CO 2 R 7，-CONR 7 SO 2 R 8， - 烷基CONR 7 SO 2 R 8，-NHCOR 7 R 8 - NHCSR7R8; 并且R 7，R 8和R 9各自独立地为氢，任选取代的烷基，任选取代的烯基，炔基，任选取代的芳基或任选取代的芳基烷基，卤代烷基，卤代烯基，卤代炔基，卤素或羟基。

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