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1. 发明专利

CA1281741C PHENYLBENZOYLUREAS 未知
公开(公告)号：CA1281741C
公开(公告)日：1991-03-19
申请号：CA489645
申请日：1985-08-29
申请人： EHRENFREUND JOSEF
发明人： EHRENFREUND JOSEF
IPC分类号： A01N47/34 , C07C67/00 , C07C239/00 , C07C275/54
摘要： Phenylbenzoylureas of the disclosure The invention relates to novel N-¢3-halo-4-(hexafluoropropoxy)-5-trifluoromethyl!phenyl-N'-benzoylureas of the formula wherein R1 is hydrogen or halogen and R2 and R3 are halogen, to a process and intermediate for the preparation of these compounds, and to compositions containing them for use in pest control, in particular for controlling insects and representatives of the order Acarina that attack plants and animals. The novel compounds exhibit in particular larvicidal activity.

2. 发明专利

CA1318680C PHENYLTHIOUREAS, PHENYLISOTHIOUREAS AND PHENYLCARBODIIMIDES, THEIR PREPARATION AND USE IN THE CONTROL OF PESTS 未知
公开(公告)号：CA1318680C
公开(公告)日：1993-06-01
申请号：CA575091
申请日：1988-08-18
申请人： EHRENFREUND JOSEF
发明人： EHRENFREUND JOSEF
IPC分类号： A01N47/30 , A01N47/32 , A01N47/40 , A01N47/42 , C07C67/00 , C07C241/00 , C07C267/00 , C07C325/00 , C07C331/28 , C07C335/16 , C07C335/32 , C07C335/36
摘要： Phenylthioureas, phenylisothioureas and phenylcarbodiimides, their preparation and use in the control of pests Novel substituted phenyl-thioureas, -isothioureas and -carbodiimides offormula I (I) in which R1 is C1-C8alkyl, C1-C8alkyl mono- or poly-substituted by halogen and/or by C1-C6alkoxy, C3-C8cycloalkyl, C3-C8cycloalkyl mono- or poly-substituted by C1-C3alkyl, or is C3-C8cycloalkyl-C1-C4alkyl; each of R2 and R3 is C1-C6alkyl, C5-C6cycloalkyl or C5-C6cycloalkenyl; each of R4 and R5 is hydrogen or C1-C4alkyl; each R6 is halogen, C1-C4alkyl, C1-C4-alkoxy, C1-C4haloalkyl, C1-C4haloalkoxy or a , or bridge in the 2,3-or 3,4-position: n is 0, 1 or 2; Z is -NH-CS-NH-, -N=C(SR7)-NH- or -N=C=N-, and R7 is C1-C10alkyl or C3-C5-alkenyl, and salts thereof with organic or inorganic acids, processes and intermediates for their manufacture, their use in the control of pests, and pesticidal compositions that contain at least one compound of formula I as active ingredient, are disclosed. The preferred field of use is the control of pests in and on animals and plants.

3. 发明申请

WO2007124907A3 HETEROCYCLYL-CARBOXYLIC ACID (BENZONORBORNENE-5-YL)AMIDE DERIVATIVES AS FUNGICIDES FOR AGROCHEMICAL USE 审中-公开
标题翻译：作为农药使用的间苯二酚 - 羧酸（苯并呋喃-5-基）酰胺衍生物
公开(公告)号：WO2007124907A3
公开(公告)日：2008-01-10
申请号：PCT/EP2007003653
申请日：2007-04-25
申请人： SYNGENTA PARTICIPATIONS AG , TOBLER HANS , CORSI CAMILLA , EHRENFREUND JOSEF , WALTER HARALD
发明人： TOBLER HANS , CORSI CAMILLA , EHRENFREUND JOSEF , WALTER HARALD
IPC分类号： C07D231/14 , A01N43/56
CPC分类号： C07D207/34 , C07C205/06 , C07C205/11 , C07C205/12 , C07C211/61 , C07C2602/42 , C07D231/14
摘要： The invention relates to fungicidally active compounds of formula (I): wherein Het, R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 8 and R 9 are as defined in claim 1, to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.
摘要翻译：本发明涉及式（I）的杀真菌活性化合物：其中Het，R 1，R 2，R 3，R 3， R 4，R 5，R 6，R 7，R 8和R 8， 9，如权利要求1中所定义，涉及这些化合物的制备，用于制备这些化合物的新型中间体，其包含至少一种新化合物作为活性成分的农药组合物，所提及的组合物以及在农业或园艺中使用活性成分或组合物来控制或预防植物病原微生物，优选真菌侵染植物。

4. 发明申请

WO2007124907A2 NOVEL MICROBIOCIDES 审中-公开
标题翻译：新型微生物
公开(公告)号：WO2007124907A2
公开(公告)日：2007-11-08
申请号：PCT/EP2007/003653
申请日：2007-04-25
申请人： SYNGENTA PARTICIPATIONS AG , TOBLER, Hans , CORSI, Camilla , EHRENFREUND, Josef , WALTER, Harald
发明人： TOBLER, Hans , CORSI, Camilla , EHRENFREUND, Josef , WALTER, Harald
CPC分类号： C07D207/34 , C07C205/06 , C07C205/11 , C07C205/12 , C07C211/61 , C07C2602/42 , C07D231/14
摘要： The invention relates to fungicidally active compounds of formula (I): wherein Het, R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 8 and R 9 are as defined in claim 1, to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.
摘要翻译：本发明涉及式（I）的杀真菌活性化合物：其中Het，R 1，R 2，R 3，R 3， R 4，R 5，R 6，R 7，R 8和R 8， 9，如权利要求1中所定义，涉及这些化合物的制备，用于制备这些化合物的新型中间体，其包含至少一种新化合物作为活性成分的农用化学组合物，提及的组合物以及在农业或园艺中使用活性成分或组合物来控制或预防植物病原微生物，优选真菌侵染植物的方法。

5. 发明申请

WO2006015866A1 METHOD FOR PROTECTING USEFUL PLANTS OR PLANT PROPAGATION MATERIAL 审中-公开
标题翻译：保护有用植物或植物传播材料的方法
公开(公告)号：WO2006015866A1
公开(公告)日：2006-02-16
申请号：PCT/EP2005/008752
申请日：2005-08-11
申请人： SYNGENTA PARTICIPATIONS AG , WALTER, Harald , ZEUN, Ronald , EHRENFREUND, Josef , TOBLER, Hans , CORSI, Camilla , LAMBERTH, Clemens
发明人： WALTER, Harald , ZEUN, Ronald , EHRENFREUND, Josef , TOBLER, Hans , CORSI, Camilla , LAMBERTH, Clemens
IPC分类号： A01N43/56
CPC分类号： A01N43/56
摘要： A method of controlling phytopathogenic diseases on useful plants or plant propagation material thereof, which comprises applying to said plant propagation material a fungicidally effective amount of a compound of formula (I) wherein R 1 is trifluoromethyl or difluoromethyl and R 2 is hydrogen or methyl, or a tautomer of such a compound, is particularly effective in controlling or preventing fungal diseases of crop plants.
摘要翻译：一种在有用植物或植物繁殖材料上控制植物病原性疾病的方法，其包括向所述植物繁殖材料施用杀真菌有效量的式（I）化合物，其中R

6. 发明申请

WO2004018438A3 MICROBIOCIDAL (E.G. FUNGICIDAL) 1,2,3-TRIAZOLE DERIVATIVES 审中-公开
标题翻译： MICROBIOCIDAL（E.G. Fungicidal）1,2,3-三唑衍生物
公开(公告)号：WO2004018438A3
公开(公告)日：2004-08-26
申请号：PCT/EP0309111
申请日：2003-08-18
申请人： SYNGENTA PARTICIPATIONS AG , EHRENFREUND JOSEF , TOBLER HANS , WALTER HARALD
发明人： EHRENFREUND JOSEF , TOBLER HANS , WALTER HARALD
IPC分类号： A01N43/647 , A01N55/00 , C07D249/04 , C07D333/36 , C07D401/12 , C07D405/12 , C07D409/12 , C07D409/14 , C07D411/12 , C07D413/12 , C07D417/12 , C07D487/08 , C07D493/08 , C07D495/08 , C07D209/94 , C07D307/00 , C07D403/12
CPC分类号： C07D401/12 , A01N43/647 , A01N55/00 , C07D249/04 , C07D333/36 , C07D405/12 , C07D409/12 , C07D409/14 , C07D411/12 , C07D413/12 , C07D417/12 , C07D487/08 , C07D493/08 , C07D495/08
摘要： A compound of formula (1):where A is an ortho-substituted ring selected from a number of specified rings; R is halogen, cyano, nitro, C 1-4 alkyl, C 1-4 haloalkyl, C 1-4 alkoxy or C 1-4 haloalkoxy or optionally substituted C 2-4 alkenyl, optionally substituted C 2-4 alkynyl or optionally substituted SO2(C 1-4)alkyl (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C 1-4 alkoxy); R is C 1-4 alkyl, C 1-4 haloalkyl, C 1-4 alkoxy(C 1-4)alkyl or C 1-4 alkyltbio(C 1-4)alkyl or [optionally substituted aryl](C 1-4)alkyl- or [optionally substituted aryl]oxy(C l-4)a1kyl(where the optionally substituted aryl moieties may each have up to 3 substituents, each independently selected from halogen and C 1-4 alkoxy); R 3 is hydrogen, CH2C =CR , CH2CR =C(H)R , CH=C=CH2 or COR or optionally substituted C 1-4 alkyl, optionally substituted C 1-4 alkoxy or optionally substituted (C I-4) alkylC(=O)O (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C 1-4 alkoxy, C 1-4 alkyl, C 1-2 haloalkoxy, bydroxy, cyano, carboxyl, methoxycarbonyl, ethoxycarbonyl, methylsulfonyl and ethylsulfonyl), The compound of Formula (I) have microbiocidal activity, in particular fungicidal activity.
摘要翻译：式（1）的化合物：其中A是选自多个指定环的邻位取代的环; R 1是卤素，氰基，硝基，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4卤代烷氧基或任选取代的C 2-4链烯基，任选取代的C 2-4炔基或任选取代的SO 2（C 1-4）烷基（其中任选取代的部分各自可具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 2是C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4）烷基或C 1-4烷基二（C 1-4）烷基或[任选取代的芳基]（C 1-4）烷基 - 或[任选取代的芳基]氧基（C 1-4）烷基（其中任选取代的芳基部分可各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 3是氢，CH 2 C = CR 4，CH 2 CR 4 = C（H）R 4，CH = C = CH 2或COR 5或任选取代的C 1-4烷基，任选取代的C 1- 4烷氧基或任选取代的（C 1-4）烷基C（= O）O（其中任选取代的部分各自可具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基，C 1-4烷基，C 1-2卤代烷氧基，二羟基，氰基，羧基，甲氧基羰基，乙氧基羰基，甲基磺酰基和乙基磺酰基）。式（I）化合物具有杀微生物活性，特别是杀真菌活性。

7. 发明申请

WO1995018123A1 PYRIDINE DERIVATIVES AS PESTICIDES 审中-公开
标题翻译：吡啶衍生物作为杀虫剂
公开(公告)号：WO1995018123A1
公开(公告)日：1995-07-06
申请号：PCT/EP1994004222
申请日：1994-12-19
申请人： CIBA-GEIGY AG , SZCZEPANSKI, Henry , KRISTINSSON, Haukur , MAIENFISCH, Peter , EHRENFREUND, Josef
发明人： CIBA-GEIGY AG
IPC分类号： C07D401/12
CPC分类号： C07D253/06 , A01N43/40 , A01N43/50 , A01N43/653 , C07D285/13 , C07D401/12
摘要： Compounds of formula (I) wherein n and Z are as defined in claim 1, and, where appropriate, tautomers thereof, in each case in free form, or in salt form, can be used as agrochemical active ingredients and can be prepared in a manner known per se.
摘要翻译：式（I）的化合物，其中n和Z如权利要求1中所定义，并且在适当的情况下，其互变异构体在每种情况下以游离形式或盐形式可用作农业化学活性成分，并且可以制备在本身已知的方式。

8. 发明申请

WO2009007098A8 ISOTHIAZOLE AND PYRAZOLE DERIVATIVES AS FUNGICIDES 审中-公开
公开(公告)号：WO2009007098A8
公开(公告)日：2009-01-15
申请号：PCT/EP2008/005589
申请日：2008-07-09
申请人： SYNGENTA PARTICIPATIONS AG , ACKERMANN, peter , BOBBIO, Carla , CORSI, Camilla , EHRENFREUND, Josef , MCGINLEY, Ann Monica , VERRAS, Andreas , RUUD, Titulaer
发明人： ACKERMANN, peter , BOBBIO, Carla , CORSI, Camilla , EHRENFREUND, Josef , MCGINLEY, Ann Monica , VERRAS, Andreas , RUUD, Titulaer
IPC分类号： C07D401/06 , C07D417/06 , C07D417/14 , A01N43/40 , A01N43/54
摘要： The present invention relates to compounds of Formula (I) wherein R 1 , R 2 , R 3 or R 4 are as defined in claim 1 or a salt or N-oxide thereof and their use in methods for the control and/or prevention of fungal infection, particularly in plants. The compounds claimed are isothiazole and pyrazole derivatives.

9. 发明申请

WO2007068417A3 PROCESS FOR THE PREPARATION OF AMINES 审中-公开
标题翻译：制备氨基酸的方法
公开(公告)号：WO2007068417A3
公开(公告)日：2007-10-04
申请号：PCT/EP2006011885
申请日：2006-12-11
申请人： SYNGENTA PARTICIPATIONS AG , TOBLER HANS , WALTER HARALD , CORSI CAMILLA , EHRENFREUND JOSEF , GIORDANO FANNY , ZELLER MARTIN
发明人： TOBLER HANS , WALTER HARALD , CORSI CAMILLA , EHRENFREUND JOSEF , GIORDANO FANNY , ZELLER MARTIN
IPC分类号： C07C209/28 , A01N45/02 , C07C211/31
CPC分类号： C07C209/62 , C07B2200/09 , C07C17/23 , C07C17/30 , C07C17/354 , C07C25/22 , C07C25/24 , C07C209/10 , C07C209/70 , C07C211/61 , C07C2603/66 , C07C23/10
摘要： The present invention relates to a novel a process for the preparation of the compound of the general formula (I), wherein R 1 and R 2 are independently H or C 1-6 alkyl, which comprises treating with a reducing agent either a compound of the general formula (II), wherein R 1 and R 2 have the meanings given for the compound of the formula (I), R 3 is H or C 1-4 alkyl and Ph is phenyl, or a compound of the general formula (III), wherein R 1 , R 2 , R 3 and Ph have the meanings given for the compound of the formula (II), the reducing agent being effective to cleave the benzyl moiety Ph-CH(R 3 )- from the benzylamino moiety PhCH(R 3 )NH- in the compound of the formula (II) or in the compound of the formula (III) to leave an amino group and, in addition, in the case of the compound of the formula (III), to reduce both the 2,3-double bond and the double bond joining the R 1 R 2 C- moiety to the 9-position of the benzonorbornene ring to single bonds. It also relates to processes for the preparation of the compounds (II) and (III) and their precursors and to the compounds (II) and (III) themselves and certain of their precursors, which are novel compounds. The compounds (I) are useful for the preparation of various fungicidal heterocyclyl-carboxylic acid benzonorbornen-5-yl-amides.
摘要翻译：本发明涉及一种制备通式（I）化合物的新方法，其中R 1和R 2独立地为H或C _{1 C-C部分到苯并降冰片烯环的9-位到单键。它还涉及制备化合物（II）和（III）及其前体以及化合物（II）和（III）本身及其某些新型化合物的前体的方法。化合物（I）可用于制备各种杀真菌性杂环基 - 羧酸苯并降冰片烯-5-基 - 酰胺。}

10. 发明申请

WO2007048556A1 HETEROCYCLIC AMIDE DERIVATIVES USEFUL AS MICROBIOCIDES 审中-公开
标题翻译：杂环酰胺衍生物作为微生物有用
公开(公告)号：WO2007048556A1
公开(公告)日：2007-05-03
申请号：PCT/EP2006/010185
申请日：2006-10-23
申请人： SYNGENTA PARTICIPATIONS AG , TOBLER, Hans , WALTER, Harald , EHRENFREUND, Josef , CORSI, Camilla
发明人： TOBLER, Hans , WALTER, Harald , EHRENFREUND, Josef , CORSI, Camilla
IPC分类号： C07D277/56 , C07D231/14 , C07D213/89 , C07D207/46 , C07D207/34 , C07C211/61 , C07C205/45 , C07C205/37 , C07C205/12 , C07C205/06 , A01N43/36 , A01N43/40 , A01N43/56 , A01N43/78
CPC分类号： C07C205/06 , A01N43/32 , A01N43/36 , A01N43/40 , A01N43/56 , A01N43/647 , A01N43/76 , A01N43/78 , C07C205/11 , C07C205/12 , C07C205/37 , C07C205/45 , C07C211/61 , C07C2603/66 , C07D207/34 , C07D207/46 , C07D213/89 , C07D231/14 , C07D249/04 , C07D263/34 , C07D277/56 , C07D327/06
摘要： The invention relates to a fungicidally active compound of formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by the groups R 6 , R 7 and R 8 ; R 1 is hydrogen, C 1-4 alkyl, C 1-4 haloalkyl, C 1-4 alkoxy, C 1-4 haloalkoxy, CH 2 C≡CR 9 , CH 2 CR 10 =CHR 11 , CH=C=CH 2 or COR 12 ; R 2 and R 3 are each, independently, hydrogen, halo, C 1-4 alkyl, C 1-4 alkoxy, C 1-4 haloalkyl or C 1-4 haloalkoxy; R 4 and R 5 are each independently selected from halo, cyano and nitro; or one of R 4 and R 5 is hydrogen and the other is selected from halo, cyano and nitro; R 6 , R 7 and R 8 are each, independently, hydrogen, halo, cyano, nitro, C 1-4 alkyl, C 1-4 haloalkyl, C 1-4 alkoxy(C 1-4 )alkyl, C 1-4 haloalkoxy(C 1-4 )alkyl or C 1-4 haloalkoxy, provided that at least one of R 6 , R 7 and R 8 is not hydrogen; R 9 , R 10 and R 11 are each, independently, hydrogen, halo, C 1-4 alkyl, C 1-4 haloalkyl or C 1-4 alkoxy(C 1-4 )alkyl; and R 12 is hydrogen, C 1-6 alkyl, C 1-6 haloalkyl, C 1-4 alkoxy(C 1-4 )alkyl, C 1-4 alkylthio(C 1-4 )- alkyl, C 1-4 alkoxy or aryl; to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.
摘要翻译：本发明涉及式（I）的杀真菌活性化合物：其中Het是含有一至三个杂原子的5-或6-元杂环，各自独立地选自氧，氮和硫，该环被基团R R＆lt; 6＆gt;，＆lt; 7＆gt;和＆lt; 8＆gt; R 1是氢，C 1-4 - 烷基，C 1-4 - 卤代烷基，C 1-4 - 烷氧基 C 1-4卤代烷氧基，CH 2 C = CR 9，CH 2 CR 10， CH = CHR 11，CH = C = CH 2或COR 12; R 2和R 3各自独立地为氢，卤素，C 1-4烷基，C 1-4烷基， C 1-4烷氧基，C 1-4卤代烷基或C 1-4卤代烷氧基; R 4和R 5各自独立地选自卤素，氰基和硝基; 或者R 4和R 5中的一个是氢，另一个选自卤素，氰基和硝基; R 6，R 7和R 8各自独立地为氢，卤素，氰基，硝基，C 1-4烷基， C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4 - ）烷基，C 1 -4个卤代烷氧基（C 1-4 - ）烷基或C 1-4 - 卤代烷氧基，条件是R 6 - R 7和R 8不是氢; R 9，R 10和R 11各自独立地为氢，卤素，C 1-4烷基 C 1-4卤代烷基或C 1-4烷氧基（C 1-4 - ）烷基; R 12是氢，C 1-6烷基，C 1-6卤代烷基，C 1-4烷基，烷氧基（C 1-4-4烷基）烷基，C 1-4烷硫基（C 1-4烷基） - 烷基，C 1〜 4烷氧基或芳基; 涉及这些化合物的制备，用于制备这些化合物的新型中间体，包括至少一种新化合物作为活性成分的农用化学组合物，所述组合物的制备以及使用活性成分或用于通过植物病原微生物，优选真菌控制或预防植物感染的农业或园艺成分。

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