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42. 发明专利

JPS52102259A PRODUCTION OF INDANE DERIVATIVES 失效
公开(公告)号：JPS52102259A
公开(公告)日：1977-08-27
申请号：JP10686575
申请日：1975-09-03
申请人： HOFFMANN LA ROCHE
发明人： ZORUTAN JIYOOJI HAAJIYOSU
IPC分类号： C07C225/12 , C07C49/513 , C07C49/557 , C07C49/613 , C07C49/653 , C07C49/753 , C07C61/13 , C07C62/18 , C07C62/24 , C07C62/26 , C07C62/38 , C07C67/00 , C07C225/00 , C07C233/12 , C07C301/00 , C07C303/28 , C07C309/65 , C07C317/00 , C07D317/26 , C07D317/30 , C07J1/00 , C07J75/00

43. 发明申请

US20150038705A1 METHODS OF USE COMPRISING A BIOCIDAL POLYAMINE 有权
标题翻译：使用生物聚氨酯的方法
公开(公告)号：US20150038705A1
公开(公告)日：2015-02-05
申请号：US14507431
申请日：2014-10-06
申请人： Curza Global, LLC , University of Utah Research Foundation
发明人： DUSTIN WILLIAMS , RYAN LOOPER , SUJEEVINI JEYAPALINA , TRAVIS HAUSSENER , PAUL R. SEBAHAR , HARI KANNA REDDY
IPC分类号： C07D333/20 , A01N33/04 , C07C211/11 , C07C211/14 , C07C217/54 , A01N33/10 , C07C225/12 , A01N37/06 , C07C237/34 , A01N37/18 , C07D317/58 , A01N43/30 , C07D295/135 , A01N43/84 , A01N43/10 , C07C211/09
CPC分类号： A01N43/84 , A01N33/00 , A01N33/02 , A01N33/04 , A01N33/10 , A01N37/06 , A01N37/18 , A01N37/20 , A01N37/30 , A01N43/10 , A01N43/30 , A01N43/40 , A01N47/12 , A61K31/135 , A61K31/137 , A61K31/166 , A61K31/325 , A61K31/357 , A61K31/381 , A61K31/4418 , A61K31/5375 , A61L12/14 , A61L12/147 , C07C211/01 , C07C211/09 , C07C211/11 , C07C211/14 , C07C211/27 , C07C217/54 , C07C217/58 , C07C225/12 , C07C233/78 , C07C237/34 , C07C271/20 , C07D213/38 , C07D213/64 , C07D295/135 , C07D317/46 , C07D317/58 , C07D333/20 , C09D5/1625
摘要： Compounds, compositions, and methods comprising a polyamine compound are described, which may be used to kill, disperse, treat, reduce biofilms, and/or inhibit or substantially prevent biofilm formation. In certain aspects, the present invention relates to compounds, compositions, and methods comprising polyamine compounds that have antimicrobial or dispersing activity against a variety of bacterial strains capable of forming biofilms.
摘要翻译：描述了包含多胺化合物的化合物，组合物和方法，其可用于杀死，分散，治疗，减少生物膜和/或抑制或基本上防止生物膜形成。在某些方面，本发明涉及包含对能够形成生物膜的各种细菌菌株具有抗微生物或分散活性的多胺化合物的化合物，组合物和方法。

44. 发明申请

US20110245493A1 DELIVERY OF DRUG AMINES THROUGH AN INHALATION ROUTE 审中-公开
标题翻译：通过吸入路线输送药物
公开(公告)号：US20110245493A1
公开(公告)日：2011-10-06
申请号：US13078525
申请日：2011-04-01
申请人： Joshua D. RABINOWITZ , Alejandro C. Zaffaroni
发明人： Joshua D. RABINOWITZ , Alejandro C. Zaffaroni
IPC分类号： C07D223/28 , C07D215/00 , C07D213/38 , C07D489/12 , C07C225/12 , C07D401/14 , C07D417/06 , C07D241/04 , C07D401/04 , G01N30/06
CPC分类号： A61K9/007 , A61K9/0073 , A61M11/001 , A61M11/041 , A61M15/00 , Y10S514/958
摘要： The present invention relates to the delivery of drug amines through an inhalation route. Specifically, it relates to aerosols containing drug amines that are used in inhalation therapy. In one aspect of the present invention, a method of delivering an amine drug in an aerosol form is provided. The method comprises: a) heating a coating, which includes an amine drug salt on a substrate contained in a device to a temperature sufficient to volatilize the amine drug from the coating, h) by said heating, forming an amine drug vapor, and c) during said heating, drawing air through said device, condensing said vapor to form aerosol particles containing less than 10% degradation products of the compound.
摘要翻译：本发明涉及通过吸入途径递送药物胺。具体地说，它涉及用于吸入治疗的含有药物胺的气溶胶。在本发明的一个方面，提供了以气雾剂形式递送胺药物的方法。该方法包括：a）将包含在装置中的基质上的胺药物盐的涂层加热到足以使胺药物从涂层挥发的温度，h）通过加热形成胺药物蒸气，和c ），通过所述装置吸入空气，冷凝所述蒸气以形成含有少于10％化合物降解产物的气溶胶颗粒。

45. 发明授权

US06867310B1 Arylation and vinylation of activated carbons 有权
标题翻译：活性炭的酰化和乙烯化
公开(公告)号：US06867310B1
公开(公告)日：2005-03-15
申请号：US09239024
申请日：1999-01-27
申请人： Stephen L. Buchwald , John P. Wolfe , Jens Ahman , Malisa Troutman , Michael Palucki , Ken Kamikawa , Andre Chieffi
发明人： Stephen L. Buchwald , John P. Wolfe , Jens Ahman , Malisa Troutman , Michael Palucki , Ken Kamikawa , Andre Chieffi
IPC分类号： C07C1/26 , C07C17/26 , C07C41/16 , C07C45/68 , C07C45/71 , C07C67/31 , C07C205/04 , C07C205/06 , C07C209/10 , C07C209/18 , C07C211/48 , C07C211/55 , C07C211/59 , C07C213/02 , C07C213/08 , C07C217/40 , C07C217/84 , C07C217/92 , C07C221/00 , C07C225/12 , C07C225/22 , C07C227/08 , C07C227/18 , C07C229/36 , C07C229/60 , C07C231/12 , C07C233/07 , C07C235/46 , C07C249/02 , C07C249/16 , C07C251/24 , C07C251/86 , C07C253/30 , C07C255/33 , C07C255/50 , C07C255/54 , C07C255/56 , C07C255/58 , C07D209/08 , C07D213/50 , C07D213/72 , C07D213/74 , C07D295/02 , C07D295/023 , C07D295/033 , C07D295/096 , C07D295/112 , C07D295/13 , C07D295/155 , C07D307/33 , C07D317/22 , C07D317/26 , C07D317/66 , C07D333/08 , C07D333/66 , C07D401/04 , C07F7/18 , C07F9/48 , C07F9/50 , C07F9/572 , C07F9/653 , C07F9/6547 , C07F9/6571 , C07F15/00 , C07D317/44
CPC分类号： C07D213/74 , C07C1/26 , C07C17/263 , C07C45/68 , C07C45/71 , C07C67/31 , C07C201/12 , C07C209/10 , C07C209/18 , C07C211/59 , C07C213/02 , C07C213/08 , C07C221/00 , C07C225/12 , C07C227/08 , C07C227/18 , C07C231/12 , C07C249/02 , C07C249/16 , C07C251/24 , C07C253/30 , C07C2601/02 , C07C2601/08 , C07C2601/16 , C07C2602/08 , C07C2602/10 , C07D209/08 , C07D213/50 , C07D213/72 , C07D295/023 , C07D295/033 , C07D295/096 , C07D295/112 , C07D295/13 , C07D295/155 , C07D307/33 , C07D317/22 , C07D317/26 , C07D317/66 , C07D333/08 , C07D333/66 , C07D401/04 , C07F7/1892 , C07F9/4875 , C07F9/5022 , C07F9/5027 , C07F9/5728 , C07F9/653 , C07F9/6547 , C07F9/65719 , C07F15/0066 , C07C25/18 , C07C49/657 , C07C49/755 , C07C49/215 , C07C49/245 , C07C49/782 , C07C49/683 , C07C49/213 , C07C49/84 , C07C49/255 , C07C47/575 , C07C49/67 , C07C69/92 , C07C211/48 , C07C211/55 , C07C217/40 , C07C217/84 , C07C217/92 , C07C225/22 , C07C229/36 , C07C229/60 , C07C233/07 , C07C235/46 , C07C251/86 , C07C255/33 , C07C255/50 , C07C255/54 , C07C255/56 , C07C255/58 , C07C205/04 , C07C205/06
摘要： The present invention provides transition-metal-catalyst-based methods for the arylation and vinylation of activated methyl, methylene, and methine carbons with aryl halides, vinyl halides, and the like. The methods of the invention provide several improvements over existing methods, including the ability to synthesize efficiently and under mild conditions α-aryl and α-vinyl products from a wide range of starting materials, including ketones, esters, hydrazones, and imines. Furthermore, the methods of the invention may be used in an asymmetric sense, i.e. to produce enantiomerically-enriched chiral α-aryl and α-vinyl products.
摘要翻译：本发明提供了基于过渡金属催化剂的方法，用于芳基卤化物，卤代乙烯等的活化的甲基，亚甲基和次甲基碳的芳基化和乙烯基化的方法。本发明的方法相对于现有方法提供了若干改进，包括在温和条件下有效合成α-芳基和α-乙烯基产物的能力，所述α-芳基和α-乙烯基产物包括酮，酯，腙和亚胺。此外，本发明的方法可以以不对称方式使用，即产生对映异构体富集的手性α-芳基和α-乙烯基产物。

46. 发明授权

US10301295B2 Herbicidal compounds 有权
公开(公告)号：US10301295B2
公开(公告)日：2019-05-28
申请号：US15520302
申请日：2015-10-13
申请人： Syngenta Participations AG
发明人： Shuji Hachisu , Alan Joseph Hennessy , Jeffrey Steven Wailes , Nigel James Willetts , Christopher John Mathews , Janice Black , Suzanna Jane Dale
IPC分类号： C07D413/12 , A01N35/06 , C07D333/34 , C07D295/195 , C07D263/58 , C07D261/18 , C07D239/42 , C07D231/16 , C07D213/81 , C07D213/75 , C07C335/26 , C07C335/16 , C07C311/29 , C07C311/16 , C07C311/03 , C07C275/64 , C07C275/28 , C07C275/24 , C07C255/58 , C07C251/38 , C07C225/12 , A01N47/36 , A01N47/34 , A01N47/30 , A01N47/28 , A01N43/84 , A01N43/76 , A01N43/56 , A01N43/40 , A01N43/10 , A01N41/06 , A01N37/50 , A01N37/34 , C07D401/12 , C07D403/12 , C07D213/74 , C07D213/76 , C07D213/78 , C07D213/84 , C07D233/96 , C07D239/28 , C07D261/04 , C07D261/14 , C07D213/61 , C07C275/54 , C07C225/18 , C07C255/57 , A01N37/44 , A01N41/10 , A01N43/54 , A01N43/80 , A01N47/38
摘要： The present invention relates to a compound of formula (I) wherein: wherein R1, R2, R3, R4, R5, R6, R7, R8, R9, R10, R11 and G are as defined herein; and wherein the compound of formula (I) is optionally present as an agrochemically acceptable salt thereof. These compounds are thought to be suitable for use as herbicides. The invention therefore also relates to a method of controlling weeds, especially grassy monocotyledonous weeds, in crops of useful plants, comprising applying a compound of formula (I), or a herbicidal composition comprising such a compound, to the plants or to the locus thereof.

47. 发明授权

US10196344B2 Glaucocalyxin a derivative and preparation method and application thereof 有权
公开(公告)号：US10196344B2
公开(公告)日：2019-02-05
申请号：US15561685
申请日：2015-12-17
申请人： SUZHOU PHARMAVAN CANCER RESEARCH CENTER CO., LTD.
发明人： Haimei Feng , Rensen Zhou , Xiang Chen , Yunhui Yu , Qian Liu , Yong Li , Shiping Deng , Chuangliang Jiang
IPC分类号： A61P35/00 , A61P37/00 , C07C221/00 , C07C225/12 , C07D207/00 , C07D233/60 , C07D473/18 , C07D295/116
摘要： Provided is a glaucocalyxin A derivative, or salt thereof, as represented by the formula (I), a method for preparation of said glaucocalyxin A derivative, and a use for said glaucocalyxin A derivative in preparing pharmaceuticals for fighting autoimmune diseases and tumors, e.g. difficult-to-treat diseases such as systemic lupus erythematosus, psoriasis and triple-negative breast cancer

48. 发明授权

US5731133A Process for the production of a chromogenically developed color photographic image using a compound capable of reacting with primary aromatic amines 失效
标题翻译：使用能够与伯芳香胺反应的化合物生产显色显影的彩色照相图像的方法
公开(公告)号：US5731133A
公开(公告)日：1998-03-24
申请号：US647640
申请日：1996-05-15
申请人： Thomas Hubsch , Arno Schmuck
发明人： Thomas Hubsch , Arno Schmuck
IPC分类号： G03C7/00 , C07C225/12 , C07C225/14 , C07C225/20 , C07C229/12 , C07C229/30 , C07C229/34 , C07C233/31 , C07C255/30 , C07D295/104 , C07D295/145 , G03C7/392 , G03C7/407 , G03C7/42 , G03C11/00
CPC分类号： C07D295/104 , C07C225/12 , C07C225/14 , C07C225/20 , C07C229/12 , C07C229/30 , C07C229/34 , C07C233/31 , C07C255/30 , C07D295/145 , G03C7/39208 , G03C7/407 , C07C2101/14 , C07C2101/16
摘要： The storage stability of photographic color images obtained by chromogenic development may be improved by compounds of the formula I, which are capable of reacting with primary amines, in particular color developer compounds (reagent for primary amines). The compounds of the formula may be added to the color photographic recording material or to a treatment bath downstream from color development. Compounds of the formula I are moreover suitable as an additive to a spent photographic processing bath or its overflow in order to reduce therein the content of color developer compounds before the processing bath or the overflow is disposed of or regenerated for further use. ##STR1## In formula I: A means --OR.sup.2, --SR.sup.2 or --NR.sup.2 R.sup.3 ; R.sup.1 means H, alkyl, aryl, acyl, sulphonyl or a residue as in A or a residue which, together with A or together with Z.sup.1, completes a ring;R.sup.2 means H, alkyl, aryl, acyl, sulphonyl; R.sup.3 means a residue as in R.sup.2 or optionally a residue which, together with R.sup.2 and the N atom, forms a heterocyclic ring, Z.sup.1 and Z.sup.2 mutually independently mean: H, halogen, cyano, alkyl, aryl, acyl, a heterocyclic group, alkoxycarbonyl, aroxycarbonyl, sulphonyl, imino, imido, sulphamoyl, carbonamido or sulphonamido; wherein Z.sup.1 and Z.sup.2, together with the C atom to which they are attached, may form a carbocyclic or heterocyclic ring system.
摘要翻译：通过显影发展获得的照相彩色图像的储存稳定性可以通过能够与伯胺反应的式I化合物，特别是彩色显影剂化合物（伯胺试剂）来改善。可以将该配方化合物加入到彩色照相记录材料中，或加入到显影下游的处理浴中。此外，式I化合物适合作为用过的照相处理槽或其溢流剂的添加剂，以便在处理槽或溢出处理或再生以供进一步使用之前将其中的显色剂化合物的含量减少。（I）式Ⅰ中，A表示-OR2，-SR2或-NR2R3; R1表示H中的H，烷基，芳基，酰基，磺酰基或残基，或与A或与Z1一起形成环的残基; R2表示H，烷基，芳基，酰基，磺酰基; R3表示残基，如R2或任选残基，其与R2和N原子一起形成杂环，Z1和Z2相互独立地表示：H，卤素，氰基，烷基，芳基，酰基，杂环基，烷氧基羰基，芳氧基羰基，磺酰基，亚氨基，亚氨基，氨磺酰基，碳酰氨基或磺酰氨基; 其中Z1和Z2与它们所连接的C原子一起可以形成碳环或杂环系。

49. 发明授权

US5510538A Process for the oxidation of primary and secondary alcohols to aldehydes and ketones and for the oxidation of 1,2-diols to .alpha.-ketols and .alpha.-diketones 失效
标题翻译：将伯醇和仲醇氧化成醛和酮以及将1,2-二醇氧化成α-酮和α-二酮的方法
公开(公告)号：US5510538A
公开(公告)日：1996-04-23
申请号：US356971
申请日：1994-12-16
申请人： Marco Frigerio , Simona Sputore , Marco Santagostino
发明人： Marco Frigerio , Simona Sputore , Marco Santagostino
IPC分类号： C07D339/06 , C07B41/06 , C07C45/29 , C07C45/30 , C07C47/115 , C07C47/228 , C07C47/42 , C07C47/54 , C07C49/12 , C07C49/403 , C07C49/433 , C07C49/437 , C07C49/513 , C07C51/373 , C07C62/38 , C07C63/04 , C07C63/70 , C07C221/00 , C07C225/12 , C07C225/16 , C07C319/20 , C07C323/22 , C07D209/12 , C07D213/48 , C07D307/46 , C07D307/48 , C07D471/14 , C07D501/26 , C07J1/00 , C07J9/00
CPC分类号： C07B41/06 , C07C45/30 , C07D213/48 , C07D307/48 , C07J1/0011 , C07J9/00
摘要： A process for the selective oxidation of a primary or secondary alcohol to an aldehyde or ketone and for the oxidation of a 1,2-diol to an .alpha.-ketol or .alpha.-diketone, which comprises contacting the alcohol or 1,2-diol with o-iodoxybenzoic acid. This process is suited for selective oxidation of alcohols containing easily oxidizable groups, such as amino or thioether groups and easily oxidizable heterocycles.
摘要翻译：将伯醇或仲醇选择性氧化成醛或酮并将1,2-二醇氧化成α-酮醇或α-二酮的方法，该方法包括使醇或1,2-二醇与邻碘苯甲酸。该方法适合于选择性氧化含有易氧化基团的醇，例如氨基或硫醚基团和易于氧化的杂环。

50. 发明申请

WO2004020391A1 VERFAHREN ZUR HERSTELLUNG VON MONOALKYLAMINOKETONEN 审中-公开
标题翻译：用于生产MONOALKYLAMINOKETONEN
公开(公告)号：WO2004020391A1
公开(公告)日：2004-03-11
申请号：PCT/EP2003/008514
申请日：2003-08-01
申请人： MERCK PATENT GMBH , FABIAN, Kai , NIESERT, Claus-Peter , KRALIK, Joachim , GLÜSENKAMP, Karl-Heinz
发明人： FABIAN, Kai , NIESERT, Claus-Peter , KRALIK, Joachim , GLÜSENKAMP, Karl-Heinz
IPC分类号： C07C225/12
CPC分类号： C07D333/22 , C07C225/16
摘要： Die Erfindung betrifft Monoalkylaminoketone der Formel (I), worin R 1 und R 2 die angegebenen Bedeutungen aufweisen.
摘要翻译：本发明涉及式（I）的Monoalkylaminoketone其中R <1>和R <2>的含义给出。

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