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41. 发明申请

WO1997047333A1 NOVEL DEVICES FOR TRANSDERMAL ADMINISTERING OF TRIMEGESTONE 审中-公开
标题翻译：用于TRIMEGESTONE的超导管理的新设备
公开(公告)号：WO1997047333A1
公开(公告)日：1997-12-18
申请号：PCT/FR1997001023
申请日：1997-06-10
申请人： ROUSSEL UCLAF , DUBOIS, Jean-Luc
发明人： ROUSSEL UCLAF
IPC分类号： A61L15/44
CPC分类号： A61K9/7061 , A61K9/7069 , A61K9/7092 , A61K31/575
摘要： The invention discloses devices for transdermal administering characterised in that they contain: a protective film (a), a unilayer, two-layered or three-layered matrix loaded with Trimegestone and optionally a matrix loaded with oestrogen, a peelable protective film (b), their method of preparation and their application as medicine.
摘要翻译：本发明公开了用于透皮给药的装置，其特征在于它们包含：保护膜（a），负载三美顿孕酮的单层，双层或三层基质和任选的载有雌激素的基质，可剥离保护膜（b），其制备方法及其作为药物的应用。

42. 发明申请

WO1997047305A1 TRANSDERMAL SYSTEMS CONTAINING TWO ACTIVE PRINCIPLES IN SEPARATE COMPARTMENTS, THEIR METHOD OF PREPARATION AND APPLICATION AS MEDICINE 审中-公开
标题翻译：包含两个活动原则的分离式系统，其制备和应用方法作为医学
公开(公告)号：WO1997047305A1
公开(公告)日：1997-12-18
申请号：PCT/FR1997001024
申请日：1997-06-10
申请人： ROUSSEL UCLAF , DUBOIS, Jean-Luc
发明人： ROUSSEL UCLAF
IPC分类号： A61K31/575
CPC分类号： A61K9/7061 , A61K9/7069 , A61K9/7092 , A61K31/575
摘要： The invention discloses a device for transdermal administering of two active principles (I) and (II) constituted in two compartments (A) and (B), compartment (A) containing a matrix loaded with (I), and compartment (B) containing a matrix loaded with (II), each of these matrices being respectively coated with a protective film, identical in nature or not, (a) and (a'), characterised in that (A) is separated from (B) by an empty space of 1 to 10 mm and characterised in that (A) and (B) are supported by the same seelable protective film (b). Their method of preparation and their application as medicine are also disclosed.
摘要翻译：本发明公开了一种用于经皮施用两个隔室（A）和（B）中构成的两种活性成分（I）和（II）的装置，含有载有（I）的基质的隔室（A）和含有加载有（II）的基质，这些基体中的每一个分别涂覆有保护膜，其性质或不相同（a）和（a'），其特征在于（A）通过空白空间为1〜10mm，其特征在于，（A）和（B）由相同的可剥离保护膜（b）支撑。他们的制备方法及其作为药物的应用也被公开。

43. 发明申请

WO1997028116A1 BIPHENYL COMPOUNDS AND USE THEREOF AS OESTROGENIC AGENTS 审中-公开
标题翻译：联苯化合物及其作为致癌剂的用途
公开(公告)号：WO1997028116A1
公开(公告)日：1997-08-07
申请号：PCT/FR1997000184
申请日：1997-01-30
申请人： ROUSSEL UCLAF , LESUISSE, Dominique
发明人： ROUSSEL UCLAF
IPC分类号： C07C217/20
CPC分类号： C07C39/38 , C07C39/15 , C07C217/20
摘要： Compounds of formula (I), wherein [X] represents aromatic carbocyclic rings (A) and (B), where R1, R2, R3, R4, R5, R6 and R7 are as defined in the description, salts thereof, a method and intermediates for preparing same, the use thereof as drugs, and pharmaceutical compositions containing same, are disclosed.
摘要翻译：式（I）化合物，其中[X]表示芳族碳环（A）和（B），其中R1，R2，R3，R4，R5，R6和R7如说明书中所定义，其盐，公开了制备它们的中间体，其作为药物的用途以及含有它们的药物组合物。

44. 发明申请

WO1997023464A1 PHENYLIMIDAZOLIDINES AND USE THEREOF AS AN ANTIANDROGENIC AGENT 审中-公开
标题翻译：苯并咪唑并作为抗原剂使用
公开(公告)号：WO1997023464A1
公开(公告)日：1997-07-03
申请号：PCT/FR1996002029
申请日：1996-12-19
申请人： ROUSSEL UCLAF , CLAUSSNER, André , GOUBET, François , TEUTSCH, Jean-Georges
发明人： ROUSSEL UCLAF
IPC分类号： C07D233/72
CPC分类号： C07D233/78
摘要： Products of formula (I), wherein R1 and R2 are particularly cyano and trifluoromethyl, R3 is particularly alkyl, alkenyl or alkynyl optionally substituted by nitrooxy or carbonyloxy, R4 and R5 are particularly methyl optionally substituted by fluorine, and X and Y are particularly oxygen, as well as salts and isomers thereof, are disclosed.
摘要翻译：式（I）的产物，其中R 1和R 2特别是氰基和三氟甲基，R 3特别是任选被硝基氧基或羰氧基取代的烷基，烯基或炔基，R 4和R 5特别是任选被氟取代的甲基，X和Y特别是氧，以及其盐和异构体。

45. 发明申请

WO1996012706A1 NOVEL ACID PYRAZOLE AND PYRAZOLONE DERIVATIVES FOR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS 审中-公开
标题翻译：用作内皮素受体拮抗剂的新型吡咯和吡唑啉酮衍生物
公开(公告)号：WO1996012706A1
公开(公告)日：1996-05-02
申请号：PCT/FR1995001386
申请日：1995-10-20
申请人： ROUSSEL UCLAF , FORTIN, Michel , ZHANG, Jidong
发明人： ROUSSEL UCLAF
IPC分类号： C07D231/20
CPC分类号： C07D405/06 , C07D231/22
摘要： Products of formula (I) wherein R1 and R2 are hydrogen or optionally substituted alkyl, aryl, arylalkyl or alkylaryl, R3, R4 and R5 are keto, -(CH2)n-R6, -CH=CH-(CH2)n-R6 or -C &cir& C-(CH2)n-R6, where n is 0-4 and R6 is hydroxyl, a lkoxy and aryloxy, alkylthio, arylthio, carboxy, cyano, alkyl, aryl, amino, mono- or dialkylamino, acylamino, and (a), -(NH)m-SO2-W, where m is 0 or 1, W is -NH-R7, (b), (c), (d) or -R7, R7 is hydrogen, alkyl or aryl and R8 is R7 except for hydrogen, or one of R3, R4 and R5 is hydrogen, and all the possible isomeric forms of the products of formula (I), are disclosed.
摘要翻译：式（I）的产物，其中R 1和R 2是氢或任选取代的烷基，芳基，芳基烷基或烷基芳基，R 3，R 4和R 5是酮， - （CH 2）n -R 6，-CH = CH-（CH 2）n -R 6 或-C（C 1 -C 6 - ） - （CH 2）n -R 6，其中n为0-4且R 6为羟基，烷氧基和芳氧基，烷硫基，芳硫基，羧基，氰基，烷基，芳基，氨基，单或二烷基氨基，酰氨基，和（a）， - （NH）m -SO 2 -W，其中m为0或1，W为-NH-R7，（b），（c），（d）或-R7，R7为氢，烷基或芳基和R 8为R 7，除了氢，或者R 3，R 4和R 5中的一个为氢，并且公开了式（I）的产物的所有可能的异构形式。

46. 发明申请

WO1995029929A1 NOVEL ERYTHROMYCIN DERIVATIVES, METHOD FOR THEIR PREPARATION AND THEIR USE AS DRUGS 审中-公开
标题翻译：新型红霉素衍生物，其制备方法及其作为药物使用
公开(公告)号：WO1995029929A1
公开(公告)日：1995-11-09
申请号：PCT/FR1995000565
申请日：1995-05-02
申请人： ROUSSEL UCLAF , AGOURIDAS, Constantin , CHANTOT, Jean-François , DENIS, Alexis , GOUIN D'AMBRIERES, Solange , LE MARTRET, Odile
发明人： ROUSSEL UCLAF
IPC分类号： C07H17/08
CPC分类号： C07H17/08 , C07H17/00
摘要： Compounds of formula (I) in which R is a -(CH2)nAr radical, n is 3, 4 or 5, Ar is an optionally substituted heterocyclic radical and Z is a hydrogen atom or an acid residue. The compounds of formula (I) have useful antibiotic properties.
摘要翻译：其中R为 - （CH 2）n Ar基的式（I）化合物，n为3,4或5，Ar为任选取代的杂环基，Z为氢原子或酸残基。式（I）化合物具有有用的抗生素性质。

47. 发明申请

WO1995027720A1 NOVEL ERYTHROMYCIN DERIVATIVES, METHOD FOR PREPARING SAME AND USE THEREOF AS DRUGS 审中-公开
标题翻译：新型红霉素衍生物，其制备方法和作为药物使用的方法
公开(公告)号：WO1995027720A1
公开(公告)日：1995-10-19
申请号：PCT/FR1995000441
申请日：1995-04-06
申请人： ROUSSEL UCLAF , AGOURIDAS, Constantin , BENEDETTI, Yannick , CHANTOT, Jean-François , DENIS, Alexis , LE MARTRET, Odile
发明人： ROUSSEL UCLAF
IPC分类号： C07H17/08
CPC分类号： C07H17/08 , C07H17/00
摘要： Compounds of general formula (I), wherein R1 and R2, which are the same or different, are a hydrogen atom or a saturated or unsaturated hydrocarbon radical having up to 24 carbon atoms and being optionally interrupted by one or more heteroatoms and provided with one or more functional groupings; or R1 and R2, taken together with the nitrogen atom to which they are attached, form a heterocyclic ring optionally containing one or more heteroatoms selected from nitrogen, oxygen and sulphur; or R1 and R2, taken together, form a radical (a), wherein R'1 and R'2, which are the same or different, are a hydrogen atom or a saturated or unsaturated hydrocarbon radical having up to 23 carbon atoms and being optionally interrupted by one or more heteroatoms and provided with one or more functional groupings, and Z is a hydrogen atom or a carboxylic acid residue having up to 18 carbon atoms; as well as acid addition salts thereof. The compounds of formula (I) have valuable antibiotic properties.
摘要翻译：通式（I）的化合物，其中相同或不同的R 1和R 2是氢原子或具有至多24个碳原子的饱和或不饱和烃基，并且任选地被一个或多个杂原子中断并且具有一个或更多功能组; 或R 1和R 2与它们所连接的氮原子一起形成任选地含有一个或多个选自氮，氧和硫的杂原子的杂环; 或R 1和R 2一起形成基团（a），其中R 1和R 2相同或不同，为氢原子或具有至多23个碳原子的饱和或不饱和烃基，并且为任选被一个或多个杂原子中断并提供一个或多个官能团，Z是氢原子或具有至多18个碳原子的羧酸残基; 以及其酸加成盐。式（I）化合物具有有价值的抗生素特性。

48. 发明申请

WO1994016969A1 MULTIPLE PACKAGE FOR THE SIMULTANEOUS ADMINISTRATION OF TWO OR MORE LIQUIDS IN A PREPARATION 审中-公开
标题翻译：在制备中同时管理两种或多种液体的多个包装
公开(公告)号：WO1994016969A1
公开(公告)日：1994-08-04
申请号：PCT/FR1994000100
申请日：1994-01-27
申请人： ROUSSEL UCLAF , WOLFF, Jan
发明人： ROUSSEL UCLAF
IPC分类号： B65D81/32
CPC分类号： B65D81/3283 , G01F11/286
摘要： Unit consisting, according to one embodiment of the invention, of two non-rigid bottles (A, B) which, uncovered, are intended for different liquids. By applying manual pressure (P) on the non-rigid bottles (A, B), the liquids are transferred with the aid of linking tubes (T) to a dosing/dispensing container (C) shared by both bottles. Marks (M) are included on the walls of said container, indicating the volume, so that the final liquid, dosed and mixed in the doser/dispenser is dispensed, using a suitable application system, especially the pour-on system. Optionally, the unit can also consist of a package of two or more bottles having a similar liquid transfer and dosing/dispersing system.
摘要翻译：根据本发明的一个实施方案，由两个非刚性瓶（A，B）组成的单元，其未被覆盖，用于不同的液体。通过在非刚性瓶（A，B）上施加手动压力（P），借助于连接管（T）将液体转移到由两个瓶共享的计量/分配容器（C）。标记（M）被包括在所述容器的壁上，指示体积，使得使用合适的应用系统，特别是倾倒系统来分配在给料器/分配器中给药和混合的最终液体。任选地，该单元还可以由具有类似液体转移和剂量/分散系统的两个或更多个瓶子的包装组成。

49. 发明申请

WO1993013123A1 NOVEL 19-NOR STEROIDS HAVING A THIOCARBON-CONTAINING CHAIN IN THE 11BETA POSITION, A METHOD FOR PREPARING SAME AND INTERMEDIATES THEREFOR, MEDICINAL USES THEREOF AND COMPOSITIONS CONTAINING SAID STEROIDS 审中-公开
标题翻译：具有11BETA位置中的含硫链的新型19-非甾体类抗生素，其制备方法及其中间体，其药物用途及含有STEROIDS的组合物
公开(公告)号：WO1993013123A1
公开(公告)日：1993-07-08
申请号：PCT/FR1992001193
申请日：1992-12-17
申请人： ROUSSEL-UCLAF , CLAUSSNER, André , NIQUE, François , TEUTSCH, Jean-Georges , VAN DE VELDE, Patrick
发明人： ROUSSEL-UCLAF
IPC分类号： C07J43/00
CPC分类号： C07J31/006 , C07J41/0005 , C07J41/0016 , C07J41/0083 , C07J43/003
摘要： Compounds of formula (I), wherein R17 and R'17 are such that: either R17 and R'17 together form ketone, hydrazono, oxime or methylene, or R17 is hydroxyl, hydroxymethyl or acyloxy and R'17 is hydrogen, alkyl or optionally substitued alkenyl or alkynyl; R3 is hydrogen or alkyl; R16 is hydrogen, halogen or alkyl; m is 0, 1 or 2; X, Y and Z are such that: X is methylene, arylene or arylenoxy bonded to the steroid by a carbon atom; Y is a saturated or unsaturated straight or branched aliphatic chain which is optionally interrupted by oxygen; and Z is aryl, arylalkyl or straight or branched alkyl; addition salts thereof, a preparation method therefor, medicinal uses thereof, compositions containing said compounds, and resulting novel intermediates.

50. 发明申请

WO1993007750A1 CONTROL OF INSECTS 审中-公开
标题翻译：管理控制
公开(公告)号：WO1993007750A1
公开(公告)日：1993-04-29
申请号：PCT/EP1992002345
申请日：1992-10-12
申请人： ROUSSEL-UCLAF , MARTIN, Robert , CAYLEY, George, R. , THACKER, J., Richard, M. , HALL, Franklin, R.
发明人： ROUSSEL-UCLAF
IPC分类号： A01N53/00
CPC分类号： A01N53/00 , A01N25/04 , A01N2300/00
摘要： A method of controlling insects on plants which comprises the application to the plant of an effective amount of an aqueous formulation that contains a pyrethroid insecticide as active ingredient, an evaporation retardant and an emulsifier, optionally together with a carrier or solvent for the active ingredient, which the formulation satisfies the formula: mass of oil phase/mass of retardant )]]/C] where L is less than or equal to 15, A = 700376, B = -1.51, C = 0.8472, Moil is the weighted average relative molar mass of the oil phase, Mretardant is the average molar mass of the retardant, and X = Moil / Y where Y is the molar solubility ratio of the formulation, defined as the minimum number of moles of oil phase which will dissolve the retardant, divided by the number of moles of retardant, provided that, in the formula above, any solvent which has no liquid phase at 27 DEG C at atmospheric pressure is excluded.
摘要翻译：一种控制植物昆虫的方法，其包括向植物施用有效量的含有拟除虫菊酯杀虫剂作为活性成分的水性制剂，蒸发阻燃剂和乳化剂，任选地与活性成分的载体或溶剂一起使用，该配方满足以下公式：油相质量/阻燃剂质量/摩尔/摩擦剂。 X Exp [[ln（L / 4）+ [C x ln（AX B）]] / C]其中L小于或等于15，A = 700376，B = -1.51，C = 0.8472，是油相的加权平均相对摩尔质量，Mretardant是阻燃剂的平均摩尔质量，X = Moil <1.8> / Y，其中Y是制剂的摩尔溶解度比，定义为最小摩尔数将阻燃剂溶解的油相除以阻燃剂的摩尔数，条件是在上式中，排除了在27℃下在大气压下没有液相的任何溶剂。

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