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    • 27. 发明申请
    • NOVEL IMIDAZOLE DERIVATIVES HAVING MICROBIOCIDAL ACTIVITY
    • 具有微生物活性的新咪唑烷衍生物
    • WO2009127615A1
    • 2009-10-22
    • PCT/EP2009/054389
    • 2009-04-14
    • SYNGENTA PARTICIPATIONS AGDUMEUNIER, RaphaelLAMBERTH, ClemensTRAH, Stephan
    • DUMEUNIER, RaphaelLAMBERTH, ClemensTRAH, Stephan
    • C07D233/60C07D233/68C07D403/12A01N43/50A61K31/4489A61P35/00
    • C07D233/68C07D233/60C07D403/12
    • The present invention relates to novel imidazole derivatives of formula I as active ingredients which have microbiocidal activity, in particular fungicidal activity wherein (I) wherein R 1 is halogen, C 1 -C 4 alkyl or C 1 -C 4 haloalkyl, R 2 is an optionally substituted aryl, R 3 is halogen or OR 7 , R 4 and R 5 are, independently of each other, hydrogen, halogen or OR 7 , R 6 is halogen or C 1 -C 4 alkyl, and R 7 is hydrogen, C 1 -C 6 alkyl, C 3 -C 7 cycloalkyl, C 3 -C 10 cycloalkylalkyl, C 1 -C 6 haloalkyl, C 2 -C 6 alkenyl, C 2 -C 6 haloalkenyl, C3-C7 cycloalkenyl, C 2 -C 6 alkynyl, C 2 -C 6 haloalkynyl, C 2 -C 6 alkyloxyalkyl, C 3 -C 8 dialkylaminoalkyl, C 4 -C 10 cycloalkylaminoalkyl or C4-C10 heterocyclylalkyl, or an agrochemically usable salt form thereof, provided that when R 3 is halogen, at least one of R 4 or R 5 is OR 7 , or when R 3 is OR7, at least one of R 4 or R 5 is OR 7 or halogen
    • 本发明涉及式I的新型咪唑衍生物,其具有杀微生物活性,特别是杀真菌活性的活性成分,其中(I)其中R1是卤素,C1-C4烷基或C1-C4卤代烷基,R2是任选取代的芳基,R3是卤素 或OR7,R4和R5彼此独立地为氢,卤素或OR7,R6为卤素或C1-C4烷基,R7为氢,C1-C6烷基,C3-C7环烷基,C3-C10环烷基烷基,C1- C 6卤代烷基,C 2 -C 6烯基,C 2 -C 6卤代烯基,C 3 -C 7环烯基,C 2 -C 6炔基,C 2 -C 6卤代炔基,C 2 -C 6烷氧基烷基,C 3 -C 8二烷基氨基烷基,C 4 -C 10环烷基氨基烷基或C 4 -C 10杂环基烷基, 条件是当R 3为卤素时,R 4或R 5中的至少一个为OR 7,或者当R 3为OR 7时,R 4或R 5中的至少一个为OR 7或卤素
    • 29. 发明申请
    • NOVEL PYRIDOPYRAZINE DERIVATIVES
    • 新型吡咯烷酮衍生物
    • WO2008031566A2
    • 2008-03-20
    • PCT/EP2007/007912
    • 2007-09-11
    • SYNGENTA PARTICIPATIONS AGSYNGENTA LIMITEDCROWLEY, Patrick, JelfLAMBERTH, ClemensWENDEBORN, Sebastian, VolkerTRAH, Stephan
    • CROWLEY, Patrick, JelfLAMBERTH, ClemensWENDEBORN, Sebastian, VolkerTRAH, Stephan
    • C07D471/04A01N43/90
    • The present invention relates to novel N -oxide derivatives of pyridopyrazines of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity :wherein X is N + -O" and Y is N; or X is N and Y is N + -O"; or X and Y are both N + -O"; R is for example H, halo, cyano, C 1-6 alkyl or C 1-6 alkoxy; R 1 is optionally substituted aryl or heteroaryl; R 2 is for example halo, C 1-8 alkyl, C 3-8 CycloaIkyI, aryl, or heteroaryl; R 3 and R 4 independently of each other are for example H, C 1-8 alkyl, halo(d-8)alkyl, C 2-8 alkenyl, C 2-8 alkynyl or aryl; or R 3 and R 4 together with the nitrogen atom to which they are attached form a C 3-10 alkylene chain or C 3-7 alkenylene chain optionally substituted with halo, C 1-4 alkyl, C 1-4 haloalkyl, C1-4 alkoxy; or R 3 and R 4 together with the nitrogen atom to which they are attached form for example a morpholine, thiomorpholine or thiomorpholine S-oxide ring; or R 3 and R 4 together with the nitrogen atom to which they are attached form a bicyclic annelated or fused ring; and R 7 and R 8 independently of each other are for example H, halo, cyano, C 1-4 alkyl, C 1-4 aIkoxy or halo(C 1-4 )alkyl.
    • 本发明涉及式(I)吡啶并吡嗪的新型N-氧化物衍生物作为具有杀微生物活性,特别是杀真菌活性的活性成分:其中X为N + -O,Y为N; 或X为N且Y为N + O“; 或X和Y均为N + O-O“; R为例如H,卤素,氰基,C 1-6烷基或C 1-6烷基, R 1是任选取代的芳基或杂芳基; R 2是例如卤素,C 1-8烷基,C 1-4烷基, 环烷基,芳基或杂芳基; R 3和R 4彼此独立地是例如H,C 1〜 烷基,卤代(C 1-8)烷基,C 2-8链烯基,C 2-8炔基或芳基;或R 3, R 4和R 4与它们所连接的氮原子一起形成C 3-10亚烷基链或C 3-7亚烷基, 任选被卤素取代的亚烯基链,C 1-4烷基,C 1-4卤代烷基,C 1-4烷氧基或R 3和R 3 与它们所连接的氮原子一起形成例如吗啉,硫代吗啉或硫代吗啉S-氧化物环;或R 3和R 4, SUP与它们所连接的氮原子一起形成a 双环环或稠环; R 7和R 8彼此独立地是例如H,卤素,氰基,C 1-4烷基,C 1 -C 4烷基, 1-4烷氧基或卤代(C 1-4烷基)烷基。