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11. 发明授权

US06255311B1 Fungicidal fused bicyclic pyrimidinones 有权
标题翻译：杀真菌融合双环嘧啶酮
公开(公告)号：US06255311B1
公开(公告)日：2001-07-03
申请号：US09260339
申请日：1999-03-02
申请人： James Francis Bereznak , Zen-Yu Chang , Thomas Paul Selby , Charlene Gross Sternberg
发明人： James Francis Bereznak , Zen-Yu Chang , Thomas Paul Selby , Charlene Gross Sternberg
IPC分类号： A01N4354
CPC分类号： C07D239/95 , A01N43/54 , A01N43/84
摘要： A method for controlling wheat powdery mildew is provided which encompasses applying to the plant, seed, seedling or portion of the plant to be protected, or, to its growing media, an effective amount of a compound of Formula II where Q is O, n is 0, R3 is halogen, R4 is halogen or hydrogen, R5 is an alkyl group having from three to five carbon atoms and R6 is an alkyl group having from three to eight carbon atoms. Also provided are certain compositions for controlling wheat powdery mildew which contain a compound of Formula II together with a surfactant, an organic solvent and/or a solid or liquid diluent. Also provided are certain fungicidal compounds within Formula II for controlling wheat powdery mildew.
摘要翻译：提供了一种控制小麦白粉病的方法，其包括向植物，种子，幼苗或待保护植物的一部分施用，或向其生长培养基施用有效量的其中Q为O的式II化合物，n为 0，R3为卤素，R4为卤素或氢，R5为碳原子数为3〜5的烷基，R6为碳原子数为3〜8的烷基。还提供了用于控制小麦白粉病的某些组合物，其含有式II化合物与表面活性剂，有机溶剂和/或固体或液体稀释剂。还提供了用于控制小麦白粉病的式II中的某些杀真菌化合物。

12. 发明授权

US06239074B1 Substituted 3-phenyluracils 失效
标题翻译：取代的3-苯基尿嘧啶
公开(公告)号：US06239074B1
公开(公告)日：2001-05-29
申请号：US08774722
申请日：1997-01-03
申请人： Ralf Klintz , Peter Schaefer , Gerhard Hamprecht , Elisabeth Heistracher , Hans-Josef Wolf , Karl-Otto Westphalen , Matthias Gerber , Uwe Kardorff , Helmut Walter , Klaus Grossmann
发明人： Ralf Klintz , Peter Schaefer , Gerhard Hamprecht , Elisabeth Heistracher , Hans-Josef Wolf , Karl-Otto Westphalen , Matthias Gerber , Uwe Kardorff , Helmut Walter , Klaus Grossmann
IPC分类号： A01N4354
CPC分类号： C07D239/54 , A01N43/54 , C07C265/12 , C07C271/04 , C07C271/22 , C07C275/32 , C07C275/38 , C07C275/40 , C07C275/42 , C07D317/28 , C07D405/04
摘要： A substituted 3-phenyluracil of the formula I where X1 and X2 are each oxygen; W is —C(R8)=X5, where X5 is oxygen, sulfur, or a radical —NR14; R14 is hydroxyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, cycloalkenyloxy, haloalkoxy, haloalkenyloxy, hydroxyalkoxy, cyanoalkoxy, cycloalkylalkoxy, alkoxyalkoxy, alkoxyalkenyloxy, alkylcarbonyloxy, haloalkylcarbonyloxy, alkylcarbamoyloxy, haloalkylcarbamoyloxy, alkoxycarbonylalkoxy, alkylthioalkoxy, dialkylaminoalkoxy, R8 is hydrogen, cyano or alkyl; R1 is halogen or cyano; R2 is hydrogen or halogen; R3 is hydrogen or alkyl; R4 is cyano, alkyl or haloalkyl; R5 is hydrogen, halogen or alkyl; or a salt or enol ether of a compound I wherein R3 is hydrogen, or its tautomeric forms, for the desiccation and defoliation of plants or as an insecticide or herbicide.
摘要翻译：式I其中X 1和X 2的取代的3-苯基尿嘧啶各自为氧; W为-C（R8）= X5，其中X5为氧，硫或-NR4; R14为羟基，烷氧基，烯氧基，炔氧基，环烷氧基，环烯氧基卤代烷氧基，卤代烷氧基，羟基烷氧基，氰基烷氧基，烷基羰基氧基，卤代烷基羰氧基，烷基氨基甲酰氧基，卤代烷基氨基甲酰氧基，烷氧基羰基烷氧基，烷基硫代烷氧基，二烷基氨基烷氧基，R8是氢，氰基或烷基; R1是卤素或氰基; R2是氢或卤素; R3 R4是氰基，烷基或卤代烷基; R5是氢，卤素或烷基;或其中R3是氢的化合物I或其互变异构形式的盐或烯醇醚，用于植物的干燥和脱叶或作为杀虫剂或除草剂。

13. 发明授权

US06228808B1 Carbamoylphenylsulfonylureas, processes for their preparation and their use as herbicides and plant growth regulators 失效
标题翻译：氨基甲酰基苯基磺酰脲，其制备方法及其作为除草剂和植物生长调节剂的用途
公开(公告)号：US06228808B1
公开(公告)日：2001-05-08
申请号：US09182763
申请日：1998-10-30
申请人： Heinz Kehne , Lothar Willms , Christian Waldraff , Hansjörg Dietrich , Hermann Bieringer , Christopher Rosinger , Thomas Auler
发明人： Heinz Kehne , Lothar Willms , Christian Waldraff , Hansjörg Dietrich , Hermann Bieringer , Christopher Rosinger , Thomas Auler
IPC分类号： A01N4354
CPC分类号： C07D275/06 , C07C311/16 , C07D521/00
摘要： Compounds of the formula (I) or salts thereof in which R1, R3=H, (subst.) hydrocarbon radical (HC) or (subst.) heterocyclyl which, including substituents, have 1-30 carbon atoms, R2=R0—Q0—, in which R0=H, (subst.) HC or (subst.) heterocyclyl radical, in each case having 1-30 carbon atoms including substituents, and Q0=a direct bond or —O—, —SO2-, —NH—, —N[(C1-C6)alkyl]-, —CO—, —CO—NH— or —O—CO—NH—; R4=H, halogen, NO2, CN, (C1-C4)alkyl, (C1-C4)alkoxy, [(C1-C4)alkyl]carbonyl or [(C1-C4)alkoxy]carbonyl, where each of the last four radicals may be halogenated; R5=H or (C1-C4)alkyl; Q=O or NR*; R*=H. (C1-C4)alkyl, (C3-C4)alkenyl or (C3-C4)alkynyl, where each of the last three radicals may be substituted by halogen, (C1-C4)alkoxy and/or (C1-C4)alkylthio, W=O or S; X,Y=H, halogen, (C1-C4)alkyl, (C1-C4)alkoxy, (C1-C4)alkylthio, where each of the last three radicals may be substituted by halogen, (C1-C4)alkoxy and/or (C1-C4)alkylthio, or mono- or di[(C1-C4)alkyl]amino, (C3-C4)cycloalkyl, (C2-C5)alkenyl, (C2-C5)alkynyl, (C2-C5)alkenyloxy or (C2-C5)alkynyloxy, Z=CH or N, are suitable as herbicides or plant growth regulators, for example for controlling harmful plants in crop plants, including transgenic crop plants. They can be prepared by processes according to claim 6, via intermediates, some of which are novel.
摘要翻译：式（I）化合物或其盐，其中R 1，R 3 = H，（取代）烃基（HC）或（取代）杂环基，其包括取代基，具有1-30个碳原子，R 2 = R 0 -Q 0-，其中R 0 = H，（低级）HC或（取代）杂环基，在每种情况下具有包含取代基的1-30个碳原子，Q 0 =直接键或-O-，-SO 2 - ， - NH-， -N [（C 1 -C 6）烷基] - ， - CO - ， - CO-NH-或-O-CO-NH-; R4 = H，卤素，NO2，CN，（C1-C4）烷基，（C1-C4）烷氧基，[（C1-C4）烷基]羰基或[（C1-C4）烷氧基]羰基，自由基可以被卤化; R5 = H或（C1-C4）烷基; Q = O或NR *; R * = H。（C 1 -C 4）烷基，（C 3 -C 4）烯基或（C 3 -C 4）炔基，其中最后三个基团中的每一个可以被卤素，（C 1 -C 4）烷氧基和/或（C 1 -C 4）烷硫基取代， W = O或S; X，Y = H，卤素，（C1-C4）烷基，（C1-C4）烷氧基，（C1-C4）烷硫基，其中最后三个基团中的每一个可以被卤素，（C 1 -C 4）烷氧基和/ 或（C 1 -C 4）烷硫基或单或二[（C 1 -C 4）烷基]氨基，（C 3 -C 4）环烷基，（C 2 -C 5）烯基，（C 2 -C 5）炔基，（C 2 -C 5）或（C 2 -C 5）炔氧基Z = CH或N适合作为除草剂或植物生长调节剂，例如用于控制作物植物（包括转基因作物植物）中的有害植物。它们可以通过根据权利要求6的方法通过中间体制备，其中一些是新颖的。

14. 发明授权

US06211189B1 Amino-spiro-quinazoline compounds 失效
标题翻译：氨基螺 - 喹唑啉化合物
公开(公告)号：US06211189B1
公开(公告)日：2001-04-03
申请号：US09583775
申请日：2000-05-31
申请人： Peter Hamley , Austen Pimm , Alan Tinker
发明人： Peter Hamley , Austen Pimm , Alan Tinker
IPC分类号： A01N4354
CPC分类号： C07D471/20 , C07D471/22 , C07D495/22
摘要： There are provided novel compounds of formula (I) wherein A represents an aromatic carbocyclic ring or a 5- or 6-membered heterocyclic aromatic ring containing 1 to 3 heteroatoms which may be the same or different and are selected from O, N and S; X represents —(CH2)n— wherein n represents zero or 1; and R1, R2 and R3 are as defined in the specification, and pharmaceutically acceptable salts thereof, and enantiomers and tautomers thereof; together with processes for their preparation, compositions containing them and their use in therapy. The compounds are inhibitors of nitric oxide synthase and are thereby particularly useful in the treatment or prophylaxis of inflammatory disease and pain.
摘要翻译：提供新的式（I）化合物，其中A表示芳族碳环或含有1至3个可相同或不同并且选自O，N和S的杂原子的5-或6-元杂环芳环; X表示 - （CH 2）n - ，其中n表示0或1; 并且R1，R2和R3如说明书中所定义，及其药学上可接受的盐，及其对映异构体和互变异构体; 以及其制备方法，含有它们的组合物及其在治疗中的用途。这些化合物是一氧化氮合酶的抑制剂，因此特别可用于治疗或预防炎性疾病和疼痛。

15. 发明授权

US06187779B1 Method for inhibiting neoplastic cells and related conditions by exposure to 2,8-disubstituted quinazoline derivatives 失效
标题翻译：通过暴露于2,8-二取代喹唑啉衍生物抑制肿瘤细胞和相关病症的方法
公开(公告)号：US06187779B1
公开(公告)日：2001-02-13
申请号：US09197311
申请日：1998-11-20
申请人： Rifat Pamukcu , Gary A. Piazza
发明人： Rifat Pamukcu , Gary A. Piazza
IPC分类号： A01N4354
CPC分类号： A61K31/505
摘要： A method for inhibiting neoplastic cells and related conditions by exposing them to 2,8 disubstituted quinazolinone compounds.
摘要翻译：一种通过将其暴露于2,8二取代喹唑啉酮化合物来抑制肿瘤细胞和相关病症的方法。

16. 发明授权

US06780821B1 Substituted phenyl uracils 失效
标题翻译：取代苯基尿嘧啶
公开(公告)号：US06780821B1
公开(公告)日：2004-08-24
申请号：US09720892
申请日：2002-06-20
申请人： Roland Andree , Mark Wilhelm Drewes , Dieter Feucht , Rolf Pontzen , Ingo Wetcholowsky , Hans-Georg Schwarz
发明人： Roland Andree , Mark Wilhelm Drewes , Dieter Feucht , Rolf Pontzen , Ingo Wetcholowsky , Hans-Georg Schwarz
IPC分类号： A01N4354
CPC分类号： C07D239/54 , A01N43/54 , C07C217/90 , C07C255/59 , C07C265/12 , C07C271/28 , C07C327/48 , C07D239/553 , C07D239/557
摘要： The invention relates to new substituted phenyluracils of the general formula (I) in which n, Q, R1, R2, R3, R4, R5 and X have the meanings given in the description, to process and new intermediates for their preparation, and to their use as herbicides.
摘要翻译：本发明涉及通式（I）的新的取代的苯基尿嘧啶，其中n，Q，R 1，R 2，R 3，R 4，R 5和X具有描述，处理和新的中间体的制备，以及它们作为除草剂的用途。

17. 发明授权

US06683027B2 Herbicidal mixtures 失效
标题翻译：除草混合物
公开(公告)号：US06683027B2
公开(公告)日：2004-01-27
申请号：US09938370
申请日：2001-08-24
申请人： Helmut Siegfried Baltruschat , Astrid Brandt
发明人： Helmut Siegfried Baltruschat , Astrid Brandt
IPC分类号： A01N4354
CPC分类号： A01N43/54 , A01N47/36 , A01N47/30 , A01N43/90 , A01N43/82 , A01N43/76 , A01N43/653 , A01N43/56 , A01N43/40 , A01N39/04 , A01N37/46 , A01N37/34 , A01N33/18 , A01N25/32 , A01N2300/00
摘要： The invention relates to a herbicidal composition comprising a herbicidally acceptable carrier and/or surface active agent and, as active ingredient, a synergistically effective amount of (1) at least one compound of formula I: in which R1, R2, A, m and n are as defined in claim 1; and (2) at least one additional herbicidal compound, which is active against broad-leaved weeds and/or annual grasses; and/or (3) at least one additional safening compound; which provides a synergistic effect against a broad spectrum of weed species, e.g., in cereal crops and/or reduces crop injuries. The invention also provides a respective method for controlling weeds and/or reducing crop injuries.
摘要翻译：本发明涉及除草组合物，其包含除草剂可接受的载体和/或表面活性剂，并且作为活性成分，协同有效量的（1）至少一种式I化合物：其中R 1，R 2 >，A，m和n如权利要求1所定义; 和（2）至少一种另外的除草化合物，其对阔叶杂草和/或一年生草有活性; 和/或（3）至少一种另外的安全化合物;其对广泛的杂草种类提供协同效应，例如在谷物作物中和/或减少作物损伤。本发明还提供了控制杂草和/ 或减少作物受伤。

18. 发明授权

US06680325B2 Agents for combating plant pests 有权
标题翻译：防治植物害虫的代理人
公开(公告)号：US06680325B2
公开(公告)日：2004-01-20
申请号：US10173062
申请日：2002-06-17
申请人： Christoph Erdelen , Wolfram Andersch , Klaus Stenzel , Astrid Mauler-Machnik , Wolfgang Krämer
发明人： Christoph Erdelen , Wolfram Andersch , Klaus Stenzel , Astrid Mauler-Machnik , Wolfgang Krämer
IPC分类号： A01N4354
CPC分类号： C07D277/32 , A01N51/00 , A01N37/46 , A01N37/50 , A01N43/36 , A01N43/54 , A01N43/653 , A01N43/707 , A01N43/80 , A01N43/82 , A01N47/26 , A01N2300/00
摘要： The present invention provides compositions for controlling plant pests, which contain the compound of the formula (I) in a mixture with fungicidally active compounds, except for cyclopropylcarboxamide derivatives and azolylmethylcycloalkanes.
摘要翻译：本发明提供用于控制植物害虫的组合物，除了环丙基甲酰胺衍生物和唑基甲基环烷烃之外，其含有与杀真菌活性化合物的混合物中的式（I）化合物。

19. 发明授权

US06664214B1 Uracil compounds and use thereof 失效
标题翻译：尿嘧啶化合物及其用途
公开(公告)号：US06664214B1
公开(公告)日：2003-12-16
申请号：US10019950
申请日：2002-01-07
申请人： Akira Shuto
发明人： Akira Shuto
IPC分类号： A01N4354
CPC分类号： C07D239/54 , A01N43/54
摘要： The invention provides an uracil compound represented by the general formula: wherein W represents oxygen or sulfur; R1 represents C1- to C3-alkyl or C1- to C3-haloalkyl; R2 represents C1- to C3-alkyl or C1- to C3-haloalkyl; R3 represents hydrogen, C1- to C3-alkyl, phenyl, C1- to C3-haloalkyl or cyano; R4 represents hydrogen or C1- to C3-alkyl; R5 represents C1- to C6-alkyl, C1- to C6-haloalkyl, C3- to C6-alkenyl, C3- to C6-haloalkenyl, C3- to C6-alkynyl or C3- to C6-haloalkynyl; X1 represents halogen; X2 represents hydrogen or halogen; X3 and X4 are independent with each other and each represents hydrogen, halogen, C1- to C6-alkyl, C1- to C6-haloalkyl, C2- to C6-alkenyl, C2- to C6-haloalkenyl, C3- to C6-alkynyl, C3- to C6-haloalkynyl, C1- to C6-alkoxy-C1- to C6-alkyl, C1- to C6-alkoxy, C1- to C6-haloalkoxy or cyano; and n represents an integer of 1 to 4. The uracil compound has an excellent herbicidal effect against various weeds and therefore it is useful as an active ingredient for a herbicide.
摘要翻译：本发明提供一种由通式表示的尿嘧啶化合物：其中W表示氧或硫; R 1表示C 1至C 3 - 烷基或C 1 -C 3 - 卤代烷基; R 2表示C 1至C 3 - 烷基或C 1 -C 3 - 卤代烷基; R 3表示氢，C 1至C 3 - 烷基，苯基，C 1至C 3 - 卤代烷基或氰基; R 4表示氢或C 1至C 3 - 烷基; R 5表示C 1〜C 6烷基，C 1〜C 6卤代烷基，C 3〜C 6链烯基，C 3〜C 6卤代链烯基，C 3〜C 6炔基或C 3〜C 6卤代炔基。 X 1表示卤素; X 2表示氢或卤素; X 3和X 4彼此独立，各自表示氢，卤素，C 1至C 6 - 烷基，C 1至C 6 - 卤代烷基，C 2至C 6 - 烯基，C 2至C 6 - 卤代烯基，C 3 至C 6 - 炔基，C 3 -C 6 - 卤代炔基，C 1至C 6 - 烷氧基-C 1至C 6 - 烷基，C 1至C 6 - 烷氧基，C 1至C 6 - 卤代烷氧基或氰基; 并且n表示1〜4的整数。尿嘧啶化合物对各种杂草具有优异的除草效果，因此可用作除草剂的活性成分。

20. 发明授权

US06645969B1 Aryl and heteroaryl quinazoline compounds which inhibit CSF-1R receptor tyrosine kinase 失效
标题翻译：抑制CSF-1R受体酪氨酸激酶的芳基和杂芳基喹唑啉化合物
公开(公告)号：US06645969B1
公开(公告)日：2003-11-11
申请号：US08521852
申请日：1995-05-18
申请人： Michael R. Myers , Alfred P. Spada , Martin P. Maguire , Paul E. Persons , Asher Zilberstein , Chin-Yi Jenny Hsu , Susan E. Johnson
发明人： Michael R. Myers , Alfred P. Spada , Martin P. Maguire , Paul E. Persons , Asher Zilberstein , Chin-Yi Jenny Hsu , Susan E. Johnson
IPC分类号： A01N4354
CPC分类号： C07D213/30 , A61K31/517 , A61K31/5377 , C07C43/2055 , C07C43/225 , C07C43/23 , C07D213/64 , C07D215/14 , C07D215/18 , C07D215/20 , C07D215/233 , C07D215/50 , C07D239/74 , C07D239/88 , C07D239/91 , C07D239/93 , C07D239/94 , C07D241/42 , C07D241/52 , C07D265/22 , C07D277/64 , C07D401/04 , C07D403/04 , C07D403/12 , C07D405/04 , C07D405/12 , C07D409/04 , C07D471/04
摘要： This invention relates to the modulation and/or inhibition of cell signaling, cell proliferation, cell inflammatory response, the control of abnormal cell growth and cell reproduction. More specifically, this invention relates to the use of mono- and/or bicyclic aryl or heteroaryl quinazoline compounds in inhibiting cell proliferation, including compounds which are useful protein tyrosine kinase (PTK) inhibitors. The method of treating cell proliferation and/or differentiation or mediator release using said quinazoline compounds and their use in pharmaceutical compositions is described.
摘要翻译：本发明涉及细胞信号调节和/或抑制，细胞增殖，细胞炎症反应，异常细胞生长和细胞繁殖的控制。更具体地，本发明涉及单和/或双环芳基或杂芳基喹唑啉化合物在抑制细胞增殖中的用途，包括有用的蛋白酪氨酸激酶（PTK）抑制剂的化合物。描述了使用所述喹唑啉化合物治疗细胞增殖和/或分化或介体释放的方法及其在药物组合物中的用途。

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