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11. 发明授权

US4874420A Herbicidal substituted triazines 失效
标题翻译：除草剂取代三嗪
公开(公告)号：US4874420A
公开(公告)日：1989-10-17
申请号：US220036
申请日：1988-07-15
申请人： Heinz-Jurgen Wroblowsky , Joachim Kluth , Klaus-Gunther Tietjen , Hans-Joachim Santel , Robert R. Schmidt , Harry Strang
发明人： Heinz-Jurgen Wroblowsky , Joachim Kluth , Klaus-Gunther Tietjen , Hans-Joachim Santel , Robert R. Schmidt , Harry Strang
IPC分类号： A01N43/68 , A01N43/70 , C07D251/16 , C07D251/18 , C07D251/42 , C07D251/44 , C07D251/50 , C07D251/52 , C07D251/54 , C07D251/70 , C07D401/06 , C07D401/12 , C07D405/06 , C07D405/12
CPC分类号： C07D401/12 , A01N43/68 , A01N43/70 , C07D251/50 , C07D251/52 , C07D251/54 , C07D405/12
摘要： Herbicidal substituted triazines of the formula ##STR1## in which A.sup.1 represents optionally branched and optionally aryl-substituted alkanediyl,A.sup.2 represents optionally branched alkanediyl,Q represents oxygen, sulphur, NH or N-alkyl,R.sup.1 represents hydrogen, hydroxyl, nitro, cyano, cyanoamino, azido, halogen, alkoxy, alkylthio (which is optionally substituted by halogen or cyano), alkyl, alkoxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, amino, alkylamino or dialkylamino,R.sup.2 represents hydrogen, alkyl, alkenyl or alkinyl,R.sup.3 represents optionally substituted aryl or heteroaryl,R.sup.4 represents hydrogen, alkyl, alkenyl or alkinyl andR.sup.5 represents hydrogen or alkyl.
摘要翻译：其中A 1表示任选支链和任选芳基取代的烷二基的除草取代三嗪，A 2表示任选支链烷二基，Q表示氧，硫，NH或N-烷基，R 1表示氢，羟基，硝基，氰基，氰基氨基，叠氮基，卤素，烷氧基，烷硫基（其任选被卤素或氰基取代），烷基，烷氧基羰基，氨基羰基，烷基氨基羰基，二烷基氨基羰基，氨基，烷基氨基或二烷基氨基，R 2表示氢，烷基，烯基或炔基，芳基或杂芳基，R 4表示氢，烷基，链烯基或炔基，R 5表示氢或烷基。

12. 发明授权

US4636245A Herbicidal tetrahydrothiopyran-2,4-dione derivatives, compositions, and method of use therefor 失效
标题翻译：除草四氢噻喃-2,4-二酮衍生物，组合物及其使用方法
公开(公告)号：US4636245A
公开(公告)日：1987-01-13
申请号：US737292
申请日：1985-05-23
申请人： Heinz-Jurgen Wroblowsky , Jorg Stetter , Ludwig Eue , Robert R. Schmidt , Hans-Joachim Santel
发明人： Heinz-Jurgen Wroblowsky , Jorg Stetter , Ludwig Eue , Robert R. Schmidt , Hans-Joachim Santel
IPC分类号： A01N43/14 , A01N43/18 , A01N43/80 , C07D335/02 , C07D409/12 , C07D413/12 , C07D417/12 , C07D521/00
CPC分类号： C07D409/12 , A01N43/18 , C07D335/02 , C07D413/12 , C07D417/12
摘要： Novel substituted tetrahydrothiopyran-2,4-dione herbicides of the formula ##STR1## in which R.sup.1 is hydrogen, alkyl, alkenyl, alkinyl, alkoxyalkyl, alkylthioalkyl, halogenoalkyl, cycloalkyl or optionally substituted aryl,R.sup.2 is alkyl, alkenyl, alkinyl, alkoxyalkyl, alkylthioalkyl, halogenoalkyl, halogenoalkenyl, alkoxycarbonylalkyl, alkoximinoalkyl, optionally substituted aralkyl or optionally substituted heterocyclylalkyl, andR.sup.3 and R.sup.4 each independently is hydrogen, alkyl, alkoxyalkyl, alkylthioalkyl, cycloalkyl, optionally substituted aryl, optionally substituted aryloxyalkyl or optionally substituted aralkyl,or metal salts thereof.
摘要翻译：式中：R 1为氢，烷基，烯基，炔基，烷氧基烷基，烷基硫代烷基，卤代烷基，环烷基或任选取代的芳基的新型取代的四氢噻喃-2,4-二酮除草剂，R2为烷基，烯基，炔基，烷氧基烷基，烷硫基烷基，卤代烷基，卤代烯基，烷氧基羰基烷基，肟基烷基，任选取代的芳烷基或任选取代的杂环基烷基，R 3和R 4各自独立地为氢，烷基，烷氧基烷基，烷硫基烷基，环烷基，任选取代的芳基，任选取代的芳氧基烷基或任选取代的芳烷基，其中。

13. 发明授权

US4614533A Herbicidal 5-amino-1-phenylpyrazoles 失效
标题翻译：除草剂5-氨基-1-苯基吡唑
公开(公告)号：US4614533A
公开(公告)日：1986-09-30
申请号：US690347
申请日：1985-01-10
申请人： Otto Schallner , Reinhold Gehring , Erich Klauke , Jorg Stetter , Heinz-Jurgen Wroblowsky , Robert R. Schmidt , Hans-Joachim Santel
发明人： Otto Schallner , Reinhold Gehring , Erich Klauke , Jorg Stetter , Heinz-Jurgen Wroblowsky , Robert R. Schmidt , Hans-Joachim Santel
IPC分类号： A01N43/56 , A01N47/02 , A01N47/18 , A01N47/22 , A01N47/36 , A01N53/00 , A01N57/22 , A01N57/24 , C07C67/00 , C07C253/00 , C07C255/66 , C07C317/32 , C07C317/48 , C07C323/48 , C07D231/38 , C07D231/40 , C07F9/40 , C07F9/6509 , A01N57/16
CPC分类号： C07D231/38 , A01N43/56 , A01N47/02 , A01N47/18 , A01N47/22 , A01N47/36 , A01N53/00 , A01N57/22 , C07D231/40 , C07F9/4015 , C07F9/650935
摘要： Herbicidally active 5-amino-1-phenyl-pyrazoles, most of which are new, of the formula ##STR1##
摘要翻译：抗除草活性的5-氨基-1-苯基 - 吡唑，其中大部分是新的，具有式（IMAGE）

14. 发明申请

US20050079979A1 Substituted benzoylisoxazoles and the use thereof as herbicides 审中-公开
标题翻译：取代的苯甲酰基异恶唑及其作为除草剂的用途
公开(公告)号：US20050079979A1
公开(公告)日：2005-04-14
申请号：US10954396
申请日：2004-09-30
申请人： Klaus-Helmut Muller , Stefan Lehr , Otto Schallner , Hans-Georg Schwarz , Heinz-Jurgen Wroblowsky , Mark Drewes , Dieter Feucht , Rolf Pontzen , Ingo Wetcholowsky
发明人： Klaus-Helmut Muller , Stefan Lehr , Otto Schallner , Hans-Georg Schwarz , Heinz-Jurgen Wroblowsky , Mark Drewes , Dieter Feucht , Rolf Pontzen , Ingo Wetcholowsky
IPC分类号： A01N43/80 , A01N43/824 , A01N43/90 , A01P13/00 , C07D209/48 , C07D231/12 , C07D233/32 , C07D239/10 , C07D249/12 , C07D253/08 , C07D261/08 , C07D275/06 , C07D413/10 , C07D487/04 , A01N43/84
CPC分类号： C07D413/10 , A01N43/80 , A01N43/90 , C07D249/12 , C07D261/08
摘要： The invention relates to novel substituted benzoylisoxazoles of the general formula (I), in which n, A, R1, R2, R3, R4, and Z are defined herein, and to processes for their preparation and to their use as herbicides.
摘要翻译：本发明涉及通式（I）的新型取代的苯甲酰基异恶唑，其中n，A，R 1，R 2，R 3，R 4和Z如本文所定义，用于制备和用作除草剂。

15. 发明授权

US5977401A Process and novel intermediates for preparing triazolinones 失效
标题翻译：制备三唑啉酮的方法和新型中间体
公开(公告)号：US5977401A
公开(公告)日：1999-11-02
申请号：US291318
申请日：1999-04-14
申请人： Heinz-Jurgen Wroblowsky
发明人： Heinz-Jurgen Wroblowsky
IPC分类号： C07C281/02 , C07C281/04 , C07D249/12 , C07C229/24 , C07C241/02 , C07C243/14 , C07C243/24
CPC分类号： C07C281/02 , C07C281/04 , C07D249/12
摘要： The present invention relates to a novel intermediate compound for preparing optionally substituted 1,2,4-triazolinones and a process for preparing that intermediate compound.
摘要翻译：本发明涉及用于制备任选取代的1,2,4-三唑啉酮的新型中间体化合物及其制备方法。

16. 发明授权

US5710303A Process for the preparation of alkoxytriazolinones 失效
标题翻译：制备烷氧基三唑啉酮的方法
公开(公告)号：US5710303A
公开(公告)日：1998-01-20
申请号：US723706
申请日：1996-09-30
申请人： Heinz-Jurgen Wroblowsky , Klaus Konig
发明人： Heinz-Jurgen Wroblowsky , Klaus Konig
IPC分类号： C07C281/04 , C07C281/16 , C07D249/12 , C07C275/70
CPC分类号： C07D249/12 , C07C281/04
摘要： Alkoxytriazolinones of the formula (I), ##STR1## are obtained in good yields and in high purity by reacting iminocarbonic diesters (II) with carbazinic esters (III) ##STR2## at -20.degree. C. to +120.degree. C. (1st step) and subjecting the semicarbazide derivatives (IV) formed in this process with elimination of R.sup.2 --OH ##STR3## to a cyclizing condensation reaction in the presence of a base at 20.degree. C. to 150.degree. C. with elimination of R.sup.3 --OH, if appropriate (2nd step) and, finally, by reacting the resulting 5-alkoxytriazolinones of the formula (V) �=formula (I) where R.sup.1 =H! with an alkylating agent of the formula R.sup.1 --X (VI) at 0.degree. C. to 150.degree. C., if appropriate in the presence of a base.
摘要翻译：通过使亚氨基碳酸二酯（II）与咔嗪酸酯（III）在-20℃至+ 120℃下反应，以良好的产率和高纯度获得式（I），（IMAGE）（I）的烷氧基三唑啉酮（第1步），在20℃〜150℃下，在碱的存在下，将在该工序中形成的氨基脲衍生物（Ⅳ）与R2-OH的反应进行环化缩合反应，（Ⅴ）[=式（I）其中R1 = H）与式R1-X（Ⅵ）的烷基化剂反应得到的5-烷氧基三唑啉酮）在0℃至150℃，如果合适，在碱的存在下。

17. 发明授权

US5594147A Process for the preparation of alkoxytriazolinones 失效
标题翻译：制备烷氧基三唑啉酮的方法
公开(公告)号：US5594147A
公开(公告)日：1997-01-14
申请号：US528584
申请日：1995-09-15
申请人： Heinz-Jurgen Wroblowsky , Klaus Konig
发明人： Heinz-Jurgen Wroblowsky , Klaus Konig
IPC分类号： C07C281/06 , C07D249/12
CPC分类号： C07D249/12 , C07C281/06
摘要： Alkoxytriazolinones of the general formula (I), ##STR1## in which R.sup.1 represents hydrogen, or represents in each case optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkylalkyl, aryl or arylalkyl, andR.sup.2 represents in each case optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkylalkyl, aryl or arylalkyl,(which can be used as intermediates for the preparation of herbicidal active compounds) are obtained in very good yields and in high purity by reacting imino(thio)carbonic esters (II) with alkoxyethyl carbazinates (III) ##STR2## in which Q represents O or S, R.sup.3 represents (for example) alkyl, aryl or aralkyl and R.sup.4 represents (for example) alkyl,at -20.degree. C. to +150.degree. C. (1st step) and subjecting the new semicarbazide derivatives (IV) ##STR3## which are formed with elimination of R.sup.3 --QH, if appropriate after intermediate isolation, to a cyclizing condensation reaction at 0.degree. C. to 200.degree. C., without the addition of a base, advantageously under reduced pressure, with the elimination of alkoxyethanols (2nd step).
摘要翻译：通式（I）的烷氧基三唑啉酮，其中R 1表示氢，或在每种情况下表示任选取代的烷基，烯基，炔基，环烷基，环烷基烷基，芳基或芳基烷基，和R 2表示在各种情况下任选取代的烷基，烯基，炔基，环烷基，环烷基烷基，芳基或芳基烷基（可用作制备除草活性化合物的中间体）以非常好的产率和高纯度通过使亚氨基（硫代）碳酸酯（II）其中Q代表O或S，R3代表（例如）烷基，芳基或芳烷基，R4代表（例如）烷基，在-20℃至+ 150℃（第1步），在0℃〜200℃进行环化缩合反应，在中间分离后，如果合适，将R3-QH所形成的新的氨基脲衍生物（IV）没有添加基础，优势我们在减压下，消除烷氧基乙醇（第二步）。

18. 发明授权

US5174808A Herbicidal pyrazolin-5-one derivatives, compositions and use 失效
标题翻译：除草剂吡唑啉-5-酮衍生物，组合物和用途
公开(公告)号：US5174808A
公开(公告)日：1992-12-29
申请号：US610597
申请日：1990-11-08
申请人： Heinz-Jurgen Wroblowsky , Peter Babczinski , Klaus Lurssen , Hans-Joachim Santel , Robert R. Schmidt
发明人： Heinz-Jurgen Wroblowsky , Peter Babczinski , Klaus Lurssen , Hans-Joachim Santel , Robert R. Schmidt
IPC分类号： A01N43/56 , C07D231/22 , C07D401/04 , C07D405/04 , C07D405/06 , C07D409/04 , C07D409/06
CPC分类号： C07D401/04 , C07D231/22 , C07D405/04 , C07D409/04 , C07D409/06
摘要： Herbicidal pyrazolin-5-one derivatives of the formula ##STR1## in which R.sup.1 represents alkyl, cycloalkyl, halogenoalkyl, alkenyl, alkynyl, alkenyl or alkynyl substituted by optionally substituted phenyl, halogenoalkenyl, alkoxy, alkoxyalkyl, alkylthioalkyl, alkylsulphonylalkyl, alkylsulphinylalkyl, alkoxycarbonylalkyl, in each case optionally substituted aryl, aralkyl, aryloxyalkyl or arylthioalkyl, an optionally substituted heterocycle, heterocyclylalkyl or the --NH--CO--R.sup.3 or --CO--O--R.sup.4 groups, in which R.sup.3 and R.sup.4 in each case independently of one another represent alkyl or aryl,R.sup.2 represents hydrogen, alkyl, cycloalkyl, halogenoalkyl, alkenyl, alkinyl, halogenoalkenyl, alkoxyalkyl, alkylthioalkyl, alkylsulphonylalkyl, alkylsuslphinylalkyl or alkoxycarbonylalkyl andAr represents optionally substituted aryl or a heterocycle which is optionally substituted and optionally fused,excluding the compounds 1-(3-chlorophenyl)-3-methylthiomethyl-4-(N-hydroxyaminomethylidene)-pyrazoline-5-one, 1-(4-chlorophenyl)-3-methylthiomethyl-4-(N-hydroxyaminomethylidene)-pyrazolin-5-one, 1-(4-trifluoronethylphenyl-3-methylthiomethyl-4-(N-hydroxyaminomethylidene))-pyrazolin-5-one and 1-(4-n-nitrophenyl)-3-methylthiomethyl-4-(N-hydroxyaminomethylidene)-pyrazolin-5-one.
摘要翻译：式（Ⅰ）的除草吡唑啉-5-酮衍生物，其中R 1表示被任选取代的苯基，卤代烯基，烷氧基，烷氧基烷基，烷基硫代烷基，烷基磺酰基烷基，烷基亚磺酰基烷基，烷基磺酰基烷基，烷氧基羰基烷基，在各种情况下均为任选取代的芳基，芳烷基，芳氧基烷基或芳硫基烷基，任选取代的杂环，杂环基烷基或-NH-CO-R 3或-CO-O-R 4基团，其中R 3和R 4各自独立地为另一个代表烷基或芳基，R 2表示氢，烷基，环烷基，卤代烷基，烯基，炔基，卤代烯基，烷氧基烷基，烷基硫代烷基，烷基磺酰基烷基，烷基磺酰基烷基或烷氧基羰基烷基，Ar表示任选取代的芳基或任选被取代和任选稠合的杂环，化合物1-（3-氯苯基）-3-甲硫基甲基-4-（N-羟基氨基亚甲基） - 吡唑并-5-酮， 1-（4-氯苯基）-3-甲基硫代甲基-4-（N-羟基氨基亚甲基） - 吡唑啉-5-酮，1-（4-三氟甲基苯基-3-甲硫基甲基-4-（N-羟基氨基甲基二烯） 5-（1-硝基苯基）-3-甲基硫代甲基-4-（N-羟基氨基亚甲基） - 对]吡唑-5-酮。

19. 发明授权

US6028200A Process for preparing 2-chloro-benzimidazole derivatives 失效
标题翻译： 2-氯 - 苯并咪唑衍生物的制备方法
公开(公告)号：US6028200A
公开(公告)日：2000-02-22
申请号：US307591
申请日：1999-05-07
申请人： Michael Conrad , Lutz Assmann , Heinz-Jurgen Wroblowsky , Carl Casser , Dietmar Bielefeldt
发明人： Michael Conrad , Lutz Assmann , Heinz-Jurgen Wroblowsky , Carl Casser , Dietmar Bielefeldt
IPC分类号： B01J27/06 , B01J27/14 , C07B61/00 , C07D491/04 , C07D491/056 , C07D235/02
CPC分类号： C07D491/04
摘要： A novel process for the preparation of 2-chloro-benzimidazole derivatives of the formula in whichA represents optionally halogenated alkylene having 1 or 2 carbon atoms,which process comprises reacting 1,3-dihydro-benzimidazol(ethi)ones of the formula ##STR1## in which X represents oxygen or sulphur,with phosphorus oxychloride.Novel 1,3-dihydro-benzimidazol(ethi)ones of the formula (II) and processes for their preparation.
摘要翻译：一种用于制备下式的2-氯 - 苯并咪唑衍生物的新方法，其中A表示任选地具有1或2个碳原子的卤代亚烷基，该方法包括使下式的1,3-二氢 - 苯并咪唑（ethi） X表示氧或硫，与磷酰氯反应。新的式（II）的1,3-二氢 - 苯并咪唑（ethi）及其制备方法。

20. 发明授权

US5965768A Process and novel intermediates for preparing triazolinones 失效
标题翻译：制备三唑啉酮的方法和新型中间体
公开(公告)号：US5965768A
公开(公告)日：1999-10-12
申请号：US114681
申请日：1998-07-13
申请人： Heinz-Jurgen Wroblowsky
发明人： Heinz-Jurgen Wroblowsky
IPC分类号： C07C281/02 , C07C281/04 , C07D249/12 , C07C229/30 , C07C243/16 , C07C243/24
CPC分类号： C07C281/02 , C07C281/04 , C07D249/12
摘要： The present invention relates to a novel process for preparing a hydrazinecarboxylic ester of the formula (III) ##STR1## wherein R represents C.sub.1-4 -alkyl, which is optionally substituted by halogen or C.sub.1-4 -alkoxy, or represents phenyl, which is optionally substituted by halogen or C.sub.1-4 -alkyl, andR.sup.1 represents halogenoalkyl which is useful as an intermediate for preparing triazolinones.
摘要翻译：本发明涉及一种制备式（III）的肼羧酸酯的新方法，其中R表示任选被卤素或C 1-4 - 烷氧基取代的C 1-4 - 烷基，或代表苯基，其任选被卤素或C 1-4 - 烷基，R 1表示可用作制备三唑啉酮的中间体的卤代烷基。

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