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141. 发明申请

US20080227796A1 7-Amino-6-Hetaryl-1,2,4-Triazolo[1,5-A]Pyrimidine Compounds and the Use Thereof for Controlling Pathogenic Fungi 审中-公开
公开(公告)号：US20080227796A1
公开(公告)日：2008-09-18
申请号：US11793286
申请日：2005-12-16
申请人： Oliver Wagner , Thomas Grote , Joachim Rheinheimer , Barbara Nave , Reinhard Stierl
发明人： Oliver Wagner , Thomas Grote , Joachim Rheinheimer , Barbara Nave , Reinhard Stierl
IPC分类号： A01N43/90 , C07D487/04 , A01P3/00
CPC分类号： A01N43/90 , C07D213/55 , C07D237/14 , C07D487/04
摘要： The present invention relates to novel 7-amino-6-hetaryl-1,2,4-triazolo[1,5-a]pyrimidine compounds and to their agriculturally acceptable salts, and also to their use for controlling harmful fungi, and also to crop protection compositions comprising at least one such compound as active component.The novel 7-amino-6-hetaryl-1,2,4-triazolo[1,5-a]pyrimidine compounds can be described by the formula I where the substituents R1, R2, Het, X and Y in formula I are as defined below: Het is a 6-membered heteroaromatic radical selected from the group consisting of pyridinyl, pyridazinyl, pyrazinyl, 1,2,4-triazinyl and 1,3,5-triazinyl, where the 6-membered heteroaromatic radical may have 1, 2 or 3 identical or different substituents L, R1, R2 independently of one another are hydrogen, C1-C8-alkyl, C1-C8-haloalkyl, C1-C8-alkoxy, C3-C8-cycloalkyl, C3-C8-cycloalkoxy, C5-C10-bicycloalkyl, C3-C8-halocycloalkyl, C2-C8-alkenyl, C2-C8-alkenyloxy, C4-C10-alkadienyl, C2-C8-haloalkenyl, C3-C8-cycloalkenyl, C3-C8-halocycloalkenyl, C2-C8-alkynyl, C2-C8-alkynyloxy, C2-C8-haloalkynyl, NH2, C1-C8-alkylamino, di-C1-C8-alkylamino, phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, X is hydrogen, halogen, OH, cyano, C1-C4-alkyl and the like, Y is hydrogen, halogen, cyano, C1-C4-alkyl and the like.

142. 发明授权

US06476061B1 Fungicides containing pyrrolidones as their active agents 失效
标题翻译：杀真菌剂含有吡咯烷酮作为其活性剂
公开(公告)号：US06476061B1
公开(公告)日：2002-11-05
申请号：US09831406
申请日：2001-05-09
申请人： Joachim Rheinheimer , Karl Eicken , Ingo Rose , Thomas Grote , Eberhard Ammermann , Gisela Lorenz , Siegfried Strathmann , Gerhard Hamprecht
发明人： Joachim Rheinheimer , Karl Eicken , Ingo Rose , Thomas Grote , Eberhard Ammermann , Gisela Lorenz , Siegfried Strathmann , Gerhard Hamprecht
IPC分类号： A61N4336
CPC分类号： C07D207/50 , A01N43/36
摘要： The invention relates to fungicides containing compounds of formula (I) as their active agents, the radicals in said formula (I) having the following meanings: R1 is hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-halogenalkylcarbonyl; R2 is hydrogen, C1-C6-alkyl or C1-C6-halogenalkyl; R3-R12 are hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, C1-C6-halogenalkyl, C1-C6-alkoxy, C1-C6-halogenalkoxy, C1-C6-alkylsulfonyl, C1-C6-halogenalkylsulfonyl, formyl, cyano, C1-C6-alkylthio or phenyl which can optionally be substituted by halogen atoms, C1-C6-alkyl or C1-C6-halogenalkyl groups, and to their agriculturally usable salts. The invention also relates to methods for combating fungi in plants using these fungicides.
摘要翻译：本发明涉及含有式（I）化合物作为其活性剂的杀真菌剂，所述式（I）中的基团具有以下含义：R 1是氢，C 1 -C 6 - 烷基，C 1 -C 6 - 烷基羰基，甲酰基或C 1 -C 6烷基， C6-卤代烷基羰基; R2是氢，C1-C6-烷基或C1-C6-卤代烷基; R3-R12是氢，卤素，C1-C8-环烷基，C1-C6-烷基，C1-C6-卤代烷基，C1-C6-烷氧基，C1-C6-卤代烷氧基，C1-C6-烷基磺酰基，C1-C6-卤代烷基磺酰基，甲酰基，氰基，C 1 -C 6 - 烷硫基或可以被卤素原子，C 1 -C 6烷基或C 1 -C 6 - 卤代烷基取代的苯基，以及它们的农业上可用的盐。本发明还涉及使用这些杀真菌剂防治植物中真菌的方法。

143. 发明授权

US06441044B1 Cycloalkyl carboxylic acid amides, their production and their use as fungicides in agriculture 失效
标题翻译：环烷基羧酸酰胺，它们的生产及其作为杀虫剂在农业中的应用
公开(公告)号：US06441044B1
公开(公告)日：2002-08-27
申请号：US09763685
申请日：2001-02-26
申请人： Ingo Rose , Frank Wetterich , Karl Eicken , Joachim Rheinheimer , Gisela Lorenz , Eberhard Ammermann , Thomas Grote , Siegfried Strathmann
发明人： Ingo Rose , Frank Wetterich , Karl Eicken , Joachim Rheinheimer , Gisela Lorenz , Eberhard Ammermann , Thomas Grote , Siegfried Strathmann
IPC分类号： A01N3718
CPC分类号： A01N53/00 , C07C233/58 , C07C255/48 , C07C271/24 , C07C2601/02
摘要： The present invention relates to cycloalkylcarboxamides of formula I where: A is optionally substituted C3-C6-cycloalkyl; Alk is straight-chain or branched C1-C6-alkylene; R1 is optionally substituted C1-C6-alkyl or C2-C6-alkenyl; R2, R3 is hydrogen, or is optionally halogenated C1-C6-alkyl or C2-C6-alkenyl; W is an optionally substituted fused bicyclic ring system having in each case six ring atoms, where one or two carbon ring atoms may be replaced by nitrogen atoms; and their agriculturally useful salts. Furthermore, the invention relates to fungicidal compositions comprising a compound of formula I as crop protection agent.
摘要翻译：本发明涉及式I的环烷基甲酰胺，其中：A为任选取代的C 3 -C 6 - 环烷基; Alk为直链或支链C 1 -C 6亚烷基; R 1为任选取代的C 1 -C 6 - 烷基或C 2 -C 6 - 烯基; R 2 ，R 3是氢，或任选被卤代的C 1 -C 6 - 烷基或C 2 -C 6 - 烯基; W是任选取代的稠合双环体系，其各自为六个环原子，其中一个或两个碳环原子可被氮取代原子及其农业上有用的盐。此外，本发明涉及杀真菌组合物，其包含式I化合物作为作物保护剂。

144. 发明授权

US07101900B2 Benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides 失效
标题翻译：苄基偕胺肟衍生物，中间产物及其生产和用作杀真菌剂的方法
公开(公告)号：US07101900B2
公开(公告)日：2006-09-05
申请号：US11061470
申请日：2005-02-22
申请人： Joachim Rheinheimer , Karl Eicken , Ingo Rose , Thomas Grote , Eberhard Ammermann , John-Bryan Speakman , Siegfried Strathmann , Gisela Lorenz
发明人： Joachim Rheinheimer , Karl Eicken , Ingo Rose , Thomas Grote , Eberhard Ammermann , John-Bryan Speakman , Siegfried Strathmann , Gisela Lorenz
IPC分类号： A61K31/15 , A61K31/381 , C07D213/44 , C07D333/20 , C07D251/158
CPC分类号： C07C259/14 , A01N37/52 , C07C2601/02
摘要： Novel benzamidoxime derivatives, processes and intermediates for their preparation and their use as fungicides are described.In the context of the present invention, benzamidoxime derivatives are compounds of the formula I where: A is an aryl or hetaryl radical; Y is a straight-chain or branched C1–C4-alkylene group, where one carbon can be replaced by oxygen, nitrogen or sulfur or by a cyclopropyl group; Rn1 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1–C6-alkyl, C1–C6-alkoxy, C1–C4-haloalkyl, C1–C4-haloalkoxy, C1–C4-alkylthio, C1–C4-alkoxyalkoxy; R2 is unsubstituted or substituted phenyl-C1–C6-alkyl, thienyl-C1–C4-alkyl, or pyrazolyl-C1–C4-alkyl, Rp3 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1–C6-alkyl, C1–C6-alkoxy, C1–C4-haloalkyl, C1–C4-haloalkoxy, C1–C4-alkylthio, C1–C4-alkoxyalkoxy, C1–C6-alkylcarbonyl; n is 0–5; p is, depending on the number of free valencies, 0–4.
摘要翻译：描述了新的苯甲酰胺肟衍生物，其制备方法和中间体及其作为杀真菌剂的用途。在本发明的上下文中，苯甲酰胺肟衍生物是式I的化合物，其中：A是芳基或杂芳基; Y是直链或支链C 1 -C 4 - 亚烷基，其中一个碳可被氧，氮或硫取代或被环丙基取代; R 1是与以下组成的组中的一至五个相同或不同的基团：氢，卤素，C 1 -C 6 C 1 -C 6烷基，C 1 -C 6 - 烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 卤代烷氧基，C 1 -C 4 - 烷硫基，C 1 -C 4 - 烷氧基烷氧基; R 2是未取代或取代的苯基-C 1 -C 6 - 烷基，噻吩基-C 1 -C 或 - 吡唑基-C 1 -C 4 - C 1-4 - 烷基，R 3 - （CH 3）3 - / SUP>是与由以下组成的组中的一至五个相同或不同的基团：氢，卤素，C 1 -C 6 - 烷基，C 1 - C 1 -C 6 - 烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 3 > 4个 - 卤代烷氧基，C 1 -C 4 - 烷硫基，C 1 -C 4 - - 烷氧基烷氧基，C 1 -C 6 - 烷基羰基; n为0-5; p取决于自由价格的数量，0-4。

145. 发明授权

US06881742B1 Benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides 失效
标题翻译：苄基偕胺肟衍生物，中间产物及其生产和用作杀真菌剂的方法
公开(公告)号：US06881742B1
公开(公告)日：2005-04-19
申请号：US10089148
申请日：2000-10-05
申请人： Joachim Rheinheimer , Karl Eicken , Ingo Rose , Thomas Grote , Eberhard Ammermann , John-Bryan Speakman , Siegfried Strathmann , Gisela Lorenz
发明人： Joachim Rheinheimer , Karl Eicken , Ingo Rose , Thomas Grote , Eberhard Ammermann , John-Bryan Speakman , Siegfried Strathmann , Gisela Lorenz
IPC分类号： A61P31/10 , A01N37/52 , A61K31/165 , C07C259/14 , A01N43/10 , A01N33/08 , A01N43/36 , A01N43/40 , A01N43/50 , C07D213/44 , C07D213/78 , C07D231/14 , C07D239/28 , C07D277/30
CPC分类号： C07C259/14 , A01N37/52 , C07C2601/02
摘要： Novel benzamidoxime derivatives, processes and intermediates for their preparation and their use as fungicides are described.In the context of the present invention, benzamidoxime derivatives are compounds of the formula I where: A is an aryl or hetaryl radical; Y is a straight-chain or branched C1-C4-alkylene group, where one carbon can be replaced by oxygen, nitrogen or sulfur or by a cyclopropyl group; Rn1 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkoxyalkoxy; R2 is unsubstituted or substituted phenyl-C1-C6-alkyl, thienyl-C1-C4-alkyl, or pyrazolyl-C1-C4-alkyl, Rp3 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkoxyalkoxy, C1-C6-alkylcarbonyl; n is 0-5; p is, depending on the number of free valencies, 0-4.
摘要翻译：描述了新的苯甲酰胺肟衍生物，其制备方法和中间体及其作为杀真菌剂的用途。在本发明的上下文中，苯甲酰胺肟衍生物是式I的化合物，其中：A是芳基或杂芳基; Y是直链或支链C 1 -C 4 - 亚烷基，其中一个碳可被氧，氮或硫取代或被环丙基取代; R 1是与以下组成的组中的一至五个相同或不同的基团：氢，卤素，C 1 -C 6 C 1 -C 6烷基，C 1 -C 6 - 烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 卤代烷氧基，C 1 -C 4 - 烷硫基，C 1 -C 4 - 烷氧基烷氧基; R 2是未取代或取代的苯基-C 1 -C 6 - 烷基，噻吩基-C 1 -C 或 - 吡唑基-C 1 -C 4 - C 1-4 - 烷基，R 3 - （CH 3）3 - / SUP>是与由以下组成的组中的一至五个相同或不同的基团：氢，卤素，C 1 -C 6 - 烷基，C 1 - C 1 -C 6 - 烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 3 > 4个 - 卤代烷氧基，C 1 -C 4 - 烷硫基，C 1 -C 4 - - 烷氧基烷氧基，C 1 -C 6 - 烷基羰基; n为0-5; p取决于自由价格的数量，0-4。

146. 发明授权

US06586369B1 Fungicidal agents containing pyrrolidones as their active agents and use thereof for treating plants 失效
标题翻译：含有吡咯烷酮作为其活性剂的杀真菌剂及其用于处理植物的用途
公开(公告)号：US06586369B1
公开(公告)日：2003-07-01
申请号：US10204349
申请日：2002-08-20
申请人： Joachim Rheinheimer , Karl Eicken , Ingo Rose , Thomas Grote , Eberhard Ammermann , John-Bryan Speakman , Siegfried Strathmann , Gisela Lorenz
发明人： Joachim Rheinheimer , Karl Eicken , Ingo Rose , Thomas Grote , Eberhard Ammermann , John-Bryan Speakman , Siegfried Strathmann , Gisela Lorenz
IPC分类号： C07D20718
CPC分类号： C07D207/50 , A01N37/32 , A01N37/36 , A01N37/38 , A01N41/02 , A01N41/10 , A01N43/36
摘要： Agrochemical compositions having fungicidal action and comprising as active compounds compounds of the formula I where R1 is hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-haloalkylcarbonyl; R2 is halogen, C1-C6-alkylthio, C1-C6-alkoxy, C3-C6-cycloalkyl-C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkyl, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, C1-C6-alkylsulfinyl, halo-C1-C6-alkylsulfonyl, cyano or a radical NR13R14; R3-R12 are hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, halo-C1-C6-alkyl, C1-C6-alkoxy, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, halo-C1-C6-alkylsulfonyl, formyl, C1-C6-alkylcarbonyl, cyano, C1-C6-alkylthio or phenyl, which may be unsubstituted or substituted by halogen, C1-C6-alkyl or halo-C1-C6-alkyl, R13 is hydrogen, C1-C6-alkyl, R14 is C1-C6-alkyl, C1-C8-cycloalkyl or, together with R13 and the nitrogen atom to which they are attached, a saturated or unsaturated heterocyclic five- or six-membered ring which contains one or two heteroatoms selected from the group consisting of nitrogen and oxygen, and their agriculturally useful salts are described.
摘要翻译：具有杀真菌作用的农药组合物，包含作为活性化合物的式I化合物，其中R 1是氢，C 1 -C 6烷基，C 1 -C 6烷基羰基，甲酰基或C 1 -C 6卤代烷基羰基; R 2是卤素，C 1 -C 6烷硫基， C 1 -C 6烷氧基，C 1 -C 6烷氧基，C 1 -C 6烷氧基，C 1 -C 6 - 烷基亚磺酰基， C 1 -C 6 - 烷基磺酰基，氰基或NR 13 R 14基; R 3 -R 12是氢，卤素，C 1 -C 8 - 环烷基，C 1 -C 6烷基，卤代-C 1 -C 6 - 烷基，C 1 -C 6 - 烷氧基， C 1 -C 6 - 烷基磺酰基，卤代-C 1 -C 6 - 烷基磺酰基，甲酰基，C 1 -C 6 - 烷基羰基，氰基，C 1 -C 6 - 烷硫基或苯基，其可以是未取代的或被卤素取代，或卤代-C 1 -C 6烷基，R 13是氢，C 1 -C 6烷基，R 14是C 1 -C 6 - 烷基，C 1 -C 8 - 环烷基，或者与R 13和它们所连接的氮原子一起是饱和或不饱和杂环五元或六元环，其含有一个或两个选自组的杂原子描述了氮和氧及其农业上有用的盐。

147. 发明授权

US06680283B1 Fungicidal compositions comprising as active compounds pyrrolidones, and their use in the treatment of plants 失效
标题翻译：包含作为活性化合物吡咯烷酮的杀真菌组合物及其在处理植物中的用途
公开(公告)号：US06680283B1
公开(公告)日：2004-01-20
申请号：US10410788
申请日：2003-04-11
申请人： Joachim Rheinheimer , Karl Eicken , Ingo Rose , Thomas Grote , Eberhard Ammermann , John-Bryan Speakman , Siegfried Strathmann , Gisela Lorenz
发明人： Joachim Rheinheimer , Karl Eicken , Ingo Rose , Thomas Grote , Eberhard Ammermann , John-Bryan Speakman , Siegfried Strathmann , Gisela Lorenz
IPC分类号： A01N4336
CPC分类号： A01N43/36 , A01N37/32 , A01N37/36 , A01N37/38 , A01N41/02 , A01N41/10 , C07D207/50
摘要： Agrochemical compositions having fungicidal action and comprising as active compounds compounds of the formula I where R1 is hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-haloalkylcarbonyl; R2 is halogen, C1-C6-alkylthio, C1-C6-alkoxy, C3-C6-cycloalkyl-C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkyl, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, C1-C6-alkylsulfinyl, halo-C1-C6-alkylsulfonyl, cyano or a radical NR13R14; R3-R12 are hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, halo-C1-C6-alkyl, C1-C6-alkoxy, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, halo-C1-C6-alkylsulfonyl, formyl, C1-C6-alkylcarbonyl, cyano, C1-C6-alkylthio or phenyl, which may be unsubstituted or substituted by halogen, C1-C6-alkyl or halo-C1-C6-alkyl, R13 is hydrogen, C1-C6-alkyl, R14 is C1-C6-alkyl, C1-C8-cycloalkyl or, together with R13 and the nitrogen atom to which they are attached, a saturated or unsaturated heterocyclic five- or six-membered ring which contains one or two heteroatoms selected from the group consisting of nitrogen and oxygen, and their agriculturally useful salts are described.
摘要翻译：具有杀真菌作用的农药组合物包含作为活性化合物的式I其中R 1为氢，C 1 -C 6烷基，C 1 -C 6烷基羰基，甲酰基或C 1 -C 6卤代烷基羰基; R 2为卤素， C 1 -C 6烷氧基，C 1 -C 6烷氧基，C 1 -C 6烷氧基，C 1 -C 6烷氧基，C 1 -C 6烷氧基， C 6 - 烷基亚磺酰基，卤代-C 1 -C 6 - 烷基磺酰基，氰基或基团NR 13 R 14; R 3 -R 12是氢，卤素，C 1 -C 8 - 环烷基，C 1 -C 6 - 烷基卤代-C 1 -C 6 - 烷基，C 1 -C 6 - 烷氧基，卤代-C 1 -C 6 - 烷氧基，C 1 -C 6烷基磺酰基，卤代-C 1 -C 6烷基磺酰基，甲酰基，C 1 -C 6烷基羰基，氰基，C 1 -C 6 - 烷硫基或苯基，其可以是未取代的或被卤素，C 1 -C 6 - 烷基或卤代-C 1 -C 6烷基取代，R 13是氢，C 1 -C 6烷基，R 14是C 1 -C 6 - 烷基，C 1 -C 8 - 环烷基或与R 13和它们所连接的氮原子一起是饱和或不饱和的杂环五元或六元环，其含有一个或两个选自以下的杂原子：描述了由氮和氧组成的组及其农业上有用的盐。

148. 发明申请

US20070197557A1 Fungicidal mixtures 审中-公开
标题翻译：杀菌混合物
公开(公告)号：US20070197557A1
公开(公告)日：2007-08-23
申请号：US11596468
申请日：2005-05-11
申请人： Jordi Tormo I Blasco , Thomas Grote , Maria Scherer , Reinhard Stierl , Siegfried Strathmann , Ulrich Schofl , Joachim Rheinheimer
发明人： Jordi Tormo I Blasco , Thomas Grote , Maria Scherer , Reinhard Stierl , Siegfried Strathmann , Ulrich Schofl , Joachim Rheinheimer
IPC分类号： A01N43/54 , A01N43/90
CPC分类号： A01N43/90 , A01N43/86 , A01N43/54 , A01N43/16 , A01N43/42 , A01N2300/00
摘要： Fungicidal mixtures comprising, as active components, 1) the triazolopyrimidine derivative of the formula I and 2) at least one compound of the formula II, in which the variables are as defined below: A is O or N; B is N or a direct bond; G is C or N; R1 alkyl; R2 alkoxy; and R3 is halogen; in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compound I with compounds II and the use of the compound I with compounds II for preparing such mixtures, and also compositions comprising these mixtures.
摘要翻译：作为活性组分的杀真菌混合物包括1）式I的三唑并嘧啶衍生物和2）至少一种式II化合物，其中变量如下所定义：A是O或N; B是N或直接键; G为C或N; R 1烷基; R 2烷氧基; R 3是卤素; 协同有效量的方法，使用化合物I与化合物II的混合物来控制有害真菌，以及化合物I与化合物II用于制备这种混合物的用途，以及包含这些混合物的组合物。

149. 发明申请

US20050187265A1 Novel benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides 失效
标题翻译：新型苄基偕胺肟衍生物，其生产和使用的中间产物和方法作为杀真菌剂
公开(公告)号：US20050187265A1
公开(公告)日：2005-08-25
申请号：US11061470
申请日：2005-02-22
申请人： Joachim Rheinheimer , Karl Eicken , Ingo Rose , Thomas Grote , Eberhard Ammermann , John-Bryan Speakman , Siegfried Strathmann , Gisela Lorenz
发明人： Joachim Rheinheimer , Karl Eicken , Ingo Rose , Thomas Grote , Eberhard Ammermann , John-Bryan Speakman , Siegfried Strathmann , Gisela Lorenz
IPC分类号： A61P31/10 , A01N37/52 , A61K31/165 , C07C259/14 , C07D333/22 , A61K31/381 , A61K31/415 , A61K31/44 , C07C259/10
CPC分类号： C07C259/14 , A01N37/52 , C07C2601/02
摘要： Novel benzamidoxime derivatives, processes and intermediates for their preparation and their use as fungicides are described. In the context of the present invention, benzamidoxime derivatives are compounds of the formula I where: A is an aryl or hetaryl radical; Y is a straight-chain or branched C1-C4-alkylene group, where one carbon can be replaced by oxygen, nitrogen or sulfur or by a cyclopropyl group; Rn1 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkoxyalkoxy; R2 is unsubstituted or substituted phenyl-C1-C6-alkyl, thienyl-C1-C4-alkyl, or pyrazolyl-C1-C4-alkyl, Rp3 are one to five identical or different radicals from the group consisting of: hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkoxyalkoxy, C1-C6-alkylcarbonyl; n is 0-5; p is, depending on the number of free valencies, 0-4.
摘要翻译：描述了新的苯甲酰胺肟衍生物，其制备方法和中间体及其作为杀真菌剂的用途。在本发明的上下文中，苯甲酰胺肟衍生物是式I的化合物，其中：A是芳基或杂芳基; Y是直链或支链C 1 -C 4 - 亚烷基，其中一个碳可被氧，氮或硫取代或被环丙基取代; R 1是与以下组成的组中的一至五个相同或不同的基团：氢，卤素，C 1 -C 6 C 1 -C 6烷基，C 1 -C 6 - 烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 卤代烷氧基，C 1 -C 4 - 烷硫基，C 1 -C 4 - 烷氧基烷氧基; R 2是未取代或取代的苯基-C 1 -C 6 - 烷基，噻吩基-C 1 -C 或 - 吡唑基-C 1 -C 4 - C 1-4 - 烷基，R 3 - （CH 3）3 - / SUP>是与由以下组成的组中的一至五个相同或不同的基团：氢，卤素，C 1 -C 6 - 烷基，C 1 - C 1 -C 6 - 烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 卤代烷氧基 C 1 -C 4 - 烷硫基，C 1 -C 4 - 烷氧基烷氧基，C 1 -C 4烷基硫基，C 1 -C 4 - -C 6 - 烷基羰基; n为0-5; p取决于自由价格的数量，0-4。

150. 发明授权

US08153820B2 Method for the production of N-substituted (3-dihalomethyl-1-methylpyrazol-4-yl) carboxamides 有权
标题翻译：制备N-取代的（3-二卤代甲基-1-甲基吡唑-4-基）甲酰胺的方法
公开(公告)号：US08153820B2
公开(公告)日：2012-04-10
申请号：US12601966
申请日：2008-05-30
申请人： Thomas Zierke , Joachim Rheinheimer , Michael Rack , Sebastian Peer Smidt , Ansgar Gereon Altenhoff , Joachim Schmidt-Leithoff , Nina Challand
发明人： Thomas Zierke , Joachim Rheinheimer , Michael Rack , Sebastian Peer Smidt , Ansgar Gereon Altenhoff , Joachim Schmidt-Leithoff , Nina Challand
IPC分类号： C07D231/10
CPC分类号： C07D231/14
摘要： The present invention relates to a process for preparing N-substituted (3-dihalomethylpyrazol-4-yl)carboxamides of the formula (I) in which R1 is optionally substituted phenyl or C3-C7-cycloalkyl, R1a is hydrogen or fluorine, or R1a together with R1 is optionally substituted C3-C5-alkanediyl or C5-C7-cycloalkanediyl, R2 is C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl or C1-C4-alkoxy-C1-C2-alkyl, X is F or Cl and n is 0, 1, 2 or 3; which comprises A) providing a compound of the formula (II) in which X is F or Cl, Y is Cl or Br and R2 has one of the meanings given above and B) reacting a compound of the formula (II) with carbon monoxide and a compound of the formula (III) in which R1, R1a and n have one of the meanings given above; in the presence of a palladium catalyst; to intermediates used for the preparation according to the process according to the invention, and also to processes for their preparation.
摘要翻译：本发明涉及式（I）的N-取代的（3-二卤代甲基吡唑-4-基）甲酰胺的制备方法，其中R 1为任选取代的苯基或C 3 -C 7 - 环烷基，R 1a为氢或氟，或R 1a R 1是C 1 -C 6 - 烷基，C 2 -C 6 - 烯基，C 2 -C 6炔基或C 1 -C 4 - 烷氧基-C 1 -C 2 - 烷基，其中R 1是任选取代的C 3 -C 5 - 烷二基或C 5 -C 7 - 环烷二基， X是F或Cl，n是0,1,2或3; 其包括A）提供其中X为F或Cl，Y为Cl或Br的式（II）化合物，R 2具有上述含义之一，B）使式（II）化合物与一氧化碳和其中R1，R1a和n具有上述含义之一的式（III）化合物; 在钯催化剂的存在下; 用于根据本发明的方法制备的中间体，以及其制备方法。

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