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1. 发明申请

WO2008007930A9 MELANOCORTIN RECEPTOR AGONISTS 审中-公开
公开(公告)号：WO2008007930A9
公开(公告)日：2008-01-17
申请号：PCT/KR2007/003429
申请日：2007-07-13
申请人： LG LIFE SCIENCES LTD. , CHOI, Sung Pil , AHN, In Ae , LEE, Sang Hyup , LEE, Sang Dae , SHIN, Mi Sook , LEE, Koo , CHOI, Deog Young , SHIM, Dong Sup , YIM, Hyeon Joo , YOON, Min Kyung , CHUNG, Soo Yong , LEE, Jung Ae , HA, Yong Hwa , KIM, Young Kwan , PARK, Oeuk , LEE, Hyun Min , KIM, Youn Hoa
发明人： CHOI, Sung Pil , AHN, In Ae , LEE, Sang Hyup , LEE, Sang Dae , SHIN, Mi Sook , LEE, Koo , CHOI, Deog Young , SHIM, Dong Sup , YIM, Hyeon Joo , YOON, Min Kyung , CHUNG, Soo Yong , LEE, Jung Ae , HA, Yong Hwa , KIM, Young Kwan , PARK, Oeuk , LEE, Hyun Min , KIM, Youn Hoa
IPC分类号： C07D403/06
摘要： The present invention relates to a compound of the following formula 1, pharmaceutically acceptable salt and isomer thereof effective as agonist of melanocortin receptor, and an agonistic composition of melanocortin receptor comprising the same as active ingredient.

2. 发明申请

WO2008007930A1 MELANOCORTIN RECEPTOR AGONISTS 审中-公开
标题翻译：梅兰康汀受体激动剂
公开(公告)号：WO2008007930A1
公开(公告)日：2008-01-17
申请号：PCT/KR2007003429
申请日：2007-07-13
申请人： LG LIFE SCIENCES LTD , CHOI SUNG PIL , AHN IN AE , LEE SANG HYUP , LEE SANG DAE , SHIN MI SOOK , LEE KOO , CHOI DEOG YOUNG , SHIM DONG SUP , YIM HYEON JOO , YOON MIN KYUNG , CHUNG SOO YONG , LEE JUNG AE , HA YONG HWA , KIM YOUNG KWAN , PARK OEUK , LEE HYUN MIN , KIM YOUN HOA
发明人： CHOI SUNG PIL , AHN IN AE , LEE SANG HYUP , LEE SANG DAE , SHIN MI SOOK , LEE KOO , CHOI DEOG YOUNG , SHIM DONG SUP , YIM HYEON JOO , YOON MIN KYUNG , CHUNG SOO YONG , LEE JUNG AE , HA YONG HWA , KIM YOUNG KWAN , PARK OEUK , LEE HYUN MIN , KIM YOUN HOA
IPC分类号： C07D403/06
CPC分类号： C07D207/16 , C07D207/48 , C07D401/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14
摘要： The present invention relates to a compound of the following formula 1, pharmaceutically acceptable salt and isomer thereof effective as agonist of melanocortin receptor, and an agonistic composition of melanocortin receptor comprising the same as active ingredient.
摘要翻译：本发明涉及有效作为黑皮质素受体激动剂的下式1化合物，其药学上可接受的盐和异构体，以及包含与活性成分相同的黑皮质素受体激动剂组合物。

3. 发明申请

WO2006057505A1 NOVEL COMPOUNDS AS AGONIST FOR PPARγ AND PPARα, METHOD FOR PREPARATION OF THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME 审中-公开
标题翻译：新的化合物作为PPAR的助剂？和PPARα，其制备方法和含有其的药物组合物
公开(公告)号：WO2006057505A1
公开(公告)日：2006-06-01
申请号：PCT/KR2005/003943
申请日：2005-11-22
申请人： LG Life Sciences, Ltd. , KIM, Geun Tae , KOH, Jong Sung , HAN, Hee Oon , KIM, Seung Hae , KIM, Kyoung-Hee , CHUNG, Hee-Kyung , HONG, Sung Woon , LEE, Chang-Seok , KOO, Ki Dong , YIM, Hyeon Joo , HUR, Gwong-Cheung , KIM, Hye Jin , PARK, Ok Ku , LEE, Hyun Mi , WOO, Sung Ho
发明人： KIM, Geun Tae , KOH, Jong Sung , HAN, Hee Oon , KIM, Seung Hae , KIM, Kyoung-Hee , CHUNG, Hee-Kyung , HONG, Sung Woon , LEE, Chang-Seok , KOO, Ki Dong , YIM, Hyeon Joo , HUR, Gwong-Cheung , KIM, Hye Jin , PARK, Ok Ku , LEE, Hyun Mi , WOO, Sung Ho
IPC分类号： C07C251/34
CPC分类号： C07C309/66 , C07D263/32 , C07D265/22 , C07D271/06 , C07D277/24
摘要： The present invention relates to novel compounds accelerating the activity of Peroxisome proliferator-activated receptor gamma (PPARγ) and alpha (PPARα), processes of preparing the same, and pharmaceutical compositions containing the same as an active agent.
摘要翻译：本发明涉及促进过氧化物酶体增殖物激活受体γ（PPARγ）和α（PPARα）的活性的新化合物，其制备方法以及含有它们作为活性剂的药物组合物。

4. 发明申请

WO2005047253A1 MELANOCORTIN RECEPTOR AGONISTS 审中-公开
标题翻译：梅兰康汀受体激动剂
公开(公告)号：WO2005047253A1
公开(公告)日：2005-05-26
申请号：PCT/KR2004/002930
申请日：2004-11-12
申请人： LG LIFE SCIENCES LTD. , YAMANOUCHI PHARMACEUTICAL CO., LTD. , LEE, Koo , PARK, Heui-Sul , AHN, In-Ae , YOO, Hyun-Ju , CHOI, Sung-Pil , CHOI, Deog-Young , YIM, Hyeon-Joo , KWON, O-Hwan , KONDOH, Yutaka
发明人： LEE, Koo , PARK, Heui-Sul , AHN, In-Ae , YOO, Hyun-Ju , CHOI, Sung-Pil , CHOI, Deog-Young , YIM, Hyeon-Joo , KWON, O-Hwan , KONDOH, Yutaka
IPC分类号： C07D211/34
CPC分类号： C07D401/04 , C07D211/22 , C07D211/26 , C07D211/32 , C07D211/34 , C07D211/58 , C07D401/14
摘要： The present invention relates a compound of formula 1, and pharmaceutically acceptable salt, hydrate, solvate, or isomer thereof effective as agonist of melanocortin receptor, and an agonistic composition of melanocortin receptor comprising the same as active ingredient.
摘要翻译：本发明涉及有效作为黑皮质素受体激动剂的式1化合物及其药学上可接受的盐，水合物，溶剂化物或异构体，以及包含与活性成分相同的黑皮质素受体激动剂组合物。

5. 发明申请

WO2005047251A1 MELANOCORTIN RECEPTOR AGONISTS 审中-公开
标题翻译：黑色素受体激动剂
公开(公告)号：WO2005047251A1
公开(公告)日：2005-05-26
申请号：PCT/KR2004/002929
申请日：2004-11-12
申请人： LG LIFE SCIENCES LTD. , YAMANOUCHI PHARMACEUTICAL CO., LTD. , LEE, Koo , PARK, Heui-Sul , AHN, In-Ae , YOO, Hyun-Ju , KIM, Jong-Yup , CHOI, Deog-Young , YIM, Hyeon-Joo , CHUNG, Kyung-Ha , SHIM, Dong-Sup , LEE, Sang-Kyun , KONDOH, Yutaka , HIRABAYASHI, Ryoji , HONDA, Shugo , KAKU, Hidetaka , SHISHIKURA, Jun-Ichi , ITO, Hiroyuki , KURAMA, Takeshi
发明人： LEE, Koo , PARK, Heui-Sul , AHN, In-Ae , YOO, Hyun-Ju , KIM, Jong-Yup , CHOI, Deog-Young , YIM, Hyeon-Joo , CHUNG, Kyung-Ha , SHIM, Dong-Sup , LEE, Sang-Kyun , KONDOH, Yutaka , HIRABAYASHI, Ryoji , HONDA, Shugo , KAKU, Hidetaka , SHISHIKURA, Jun-Ichi , ITO, Hiroyuki , KURAMA, Takeshi
IPC分类号： C07D207/16
CPC分类号： C04B35/632 , C07D205/04 , C07D207/14 , C07D211/58 , C07D401/12 , C07D403/12 , C07D405/12
摘要： The present invention relates a compound of formula 1, and pharmaceutically acceptable salt, hydrate, solvate, or isomer thereof effective as agonist of melanocortin receptor, and an agonistic composition of melanocortin receptor comprising the same as active ingredient.
摘要翻译：本发明涉及作为黑皮质素受体激动剂有效的式1化合物及其药学上可接受的盐，水合物，溶剂化物或异构体，以及包含其作为活性成分的黑皮质素受体激动剂组合物

6. 发明申请

WO1992003445A1 NOVEL CEPHALOSPORIN COMPOUNDS AND PROCESSES FOR PREPARATION THEREOF 审中-公开
标题翻译：新型CEPHOROSPORIN化合物及其制备方法
公开(公告)号：WO1992003445A1
公开(公告)日：1992-03-05
申请号：PCT/KR1991000013
申请日：1991-05-01
申请人： LUCKY LTD. , KIM, Yong, Zu , OH, Hung, Seung , YEO, Jae, Hong , LIM, Jong, Chan , BANG, Chan, Sik , KIM, Won, Sup , YIM, Hyeon, Joo
发明人： LUCKY LTD.
IPC分类号： C07D501/36
CPC分类号： C07D501/00
摘要： The present invention provides a cephalosporin compound represented by formulas (I-S) and (I-R), wherein R is a C1-4 alkyl, C3-4 alkenyl, C3-4 cycloalkyl, amino optionally substituted with a C1-4 alkyl radical, phenyl, or 2-, 4- or 6- substituted phenyl group with two or fewer substituents chosen from C1-4 alkyl, C1-3 alkoxy, halogen and hydroxy radicals; R is hydrogen or a C1-4 alkyl group; R and R , which should be different from each other, are hydrogen or a C1-4 alkyl group; and Q is N or CH, and the pharmaceutically acceptable non-toxic salts, physiologically hydrolyzable esters, hydrates and solvates thereof, which possess potent and broad antibacterial activities. The invention also provides processes for preparing these compounds and to pharmaceutical compositions containing them as active ingredients.
摘要翻译：本发明提供由式（IS）和（IR）表示的头孢菌素化合物，其中R 1为C 1-4烷基，C 3-4烯基，C 3-4环烷基，任选被C 1-4烷基取代的氨基苯基或2-，4-或6-取代的苯基，其具有两个或更少个选自C 1-4烷基，C 1-3烷氧基，卤素和羟基的取代基; R 2是氢或C 1-4烷基; R a和R b彼此不同的是氢或C 1-4烷基; 和Q是N或CH，以及其药学上可接受的无毒盐，生理上可水解的酯，水合物和溶剂合物，其具有有效和广泛的抗菌活性。本发明还提供了制备这些化合物的方法和含有它们作为活性成分的药物组合物。

7. 发明申请

WO2009082134A3 DIPEPTIDYL PEPTIDASE-IV INHIBITING COMPOUNDS, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS ACTIVE AGENT 审中-公开
标题翻译：二肽基肽酶-IV抑制化合物，其制备方法以及含有该化合物作为活性剂的药物组合物
公开(公告)号：WO2009082134A3
公开(公告)日：2009-09-24
申请号：PCT/KR2008007543
申请日：2008-12-19
申请人： LG LIFE SCIENCES LTD , LEE CHANG-SEOK , YIM HYEON JOO , KIM KYOUNG-HEE , LEE JAEICK , LEE SUNG-HACK , LEE KYU WOONG , LEE HEE BONG , PARK WAN SU , MIN CHANGHEE
发明人： LEE CHANG-SEOK , YIM HYEON JOO , KIM KYOUNG-HEE , LEE JAEICK , LEE SUNG-HACK , LEE KYU WOONG , LEE HEE BONG , PARK WAN SU , MIN CHANGHEE
IPC分类号： C07D471/04
CPC分类号： C07D471/04
摘要： Disclosed herein are novel compounds of Formula (1) as defined in the specification having excellent inhibitory activity against dipeptidyl peptidase-IV (DPP-IV), methods of preparing the same and pharmaceutical compositions comprising the same as an active agent.
摘要翻译：本文公开了如本说明书中所定义的具有优异的抗二肽基肽酶-IV（DPP-IV）抑制活性的式（1）化合物，其制备方法和包含其作为活性剂的药物组合物。

8. 发明申请

WO2009082134A2 DIPEPTIDYL PEPTIDASE-IV INHIBITING COMPOUNDS, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS ACTIVE AGENT 审中-公开
标题翻译： DIPEPTIDYL PEPTIDASE-IV抑制化合物，其制备方法和含有它们作为活性代谢物的药物组合物
公开(公告)号：WO2009082134A2
公开(公告)日：2009-07-02
申请号：PCT/KR2008/007543
申请日：2008-12-19
申请人： LG LIFE SCIENCES, LTD. , LEE, Chang-Seok , YIM, Hyeon Joo , KIM, Kyoung-Hee , LEE, Jaeick , LEE, Sung-Hack , LEE, Kyu Woong , LEE, Hee Bong , PARK, Wan Su , MIN, Changhee
发明人： LEE, Chang-Seok , YIM, Hyeon Joo , KIM, Kyoung-Hee , LEE, Jaeick , LEE, Sung-Hack , LEE, Kyu Woong , LEE, Hee Bong , PARK, Wan Su , MIN, Changhee
IPC分类号： C07D471/04
CPC分类号： C07D471/04
摘要： Disclosed herein are novel compounds of Formula (1) as defined in the specification having excellent inhibitory activity against dipeptidyl peptidase-IV (DPP-IV), methods of preparing the same and pharmaceutical compositions comprising the same as an active agent.
摘要翻译：本文公开的是具有对二肽基肽酶-IV（DPP-IV）具有优异抑制活性的本说明书中定义的新颖的式（1）化合物，其制备方法和包含其作为活性剂的药物组合物。

9. 发明申请

WO2007058504A1 NOVEL COMPOUNDS AS AGONIST FOR PPAR GAMMA AND PPAR ALPHA, METHOD FOR PREPARATION OF THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME 审中-公开
标题翻译：作为PPAR GAMMA和PPAR ALPHA的激动剂的新型化合物，其制备方法和含有它们的药物组合物
公开(公告)号：WO2007058504A1
公开(公告)日：2007-05-24
申请号：PCT/KR2006/004867
申请日：2006-11-18
申请人： LG LIFE SCIENCES, LTD. , KIM, Geun Tae , HAN, Hee Oon , KOH, Jong Sung , KIM, Seung Hae , KIM, Kyoung-Hee , CHUNG, Hee-kyung , PARK, Ok Ku , JEON, Sang Kweon , WOO, Sung Ho , YIM, Hyeon Joo , HUR, Gwong-Cheung , HONG, Sung Woon , KOO, Ki Dong , LEE, Chang-Seok , CHANG, Min Sun , KOO, Sun-Young , JOO, Hyun Woo , SONG, Jeong Uk , MOON, Sang Pil , SONG-Mi-a
发明人： KIM, Geun Tae , HAN, Hee Oon , KOH, Jong Sung , KIM, Seung Hae , KIM, Kyoung-Hee , CHUNG, Hee-kyung , PARK, Ok Ku , JEON, Sang Kweon , WOO, Sung Ho , YIM, Hyeon Joo , HUR, Gwong-Cheung , HONG, Sung Woon , KOO, Ki Dong , LEE, Chang-Seok , CHANG, Min Sun , KOO, Sun-Young , JOO, Hyun Woo , SONG, Jeong Uk , MOON, Sang Pil , SONG-Mi-a
IPC分类号： C07C251/34 , A61K45/00 , A61K31/192
CPC分类号： A61K31/192 , C07C251/48 , C07C309/65 , C07C2601/08 , C07D209/22 , C07D209/42 , C07D213/643 , C07D239/34 , C07D261/08 , C07D263/20 , C07D265/36 , C07D271/10 , C07D277/28 , C07D401/12 , C07D413/06 , C07D413/12
摘要： The present invention relates to novel compounds accelerating the activity of Peroxisome proliferator-activated receptor gamma (PPARγ) and alpha (PPARα), processes of preparing the same, and pharmaceutical compositions containing the same as an active agent.
摘要翻译：本发明涉及促进过氧化物酶体增殖物激活受体γ（PPARγ）和α（PPARα）的活性的新化合物，其制备方法以及含有它们作为活性剂的药物组合物。

10. 发明申请

WO2006104356A1 DIPEPTIDYL PEPTIDASE-IV INHIBITING COMPOUNDS, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT 审中-公开
标题翻译： DIPEPTIDYL PEPTIDASE-IV抑制化合物，其制备方法和含有它们的药物组合物作为活性剂
公开(公告)号：WO2006104356A1
公开(公告)日：2006-10-05
申请号：PCT/KR2006/001169
申请日：2006-03-30
申请人： LG LIFE SCIENCES, LTD. , LEE, Chang-Seok , KOH, Jong Sung , KOO, Ki Dong , KIM, Geun Tae , KIM, Kyoung-Hee , HONG, Sang Yong , KIM, Sungsub , KIM, Min-Jung , YIM, Hyeon Joo , LIM, Dongchul , KIM, Hye Jin , HAN, Hee Oon , BU, Seong Cheol , KWON, Oh Hwan , KIM, Sung Ho , HUR, Gwong-Cheung , KIM, Ji Young , YEOM, Zi-Ho , YEO, Dong-Jun
发明人： LEE, Chang-Seok , KOH, Jong Sung , KOO, Ki Dong , KIM, Geun Tae , KIM, Kyoung-Hee , HONG, Sang Yong , KIM, Sungsub , KIM, Min-Jung , YIM, Hyeon Joo , LIM, Dongchul , KIM, Hye Jin , HAN, Hee Oon , BU, Seong Cheol , KWON, Oh Hwan , KIM, Sung Ho , HUR, Gwong-Cheung , KIM, Ji Young , YEOM, Zi-Ho , YEO, Dong-Jun
IPC分类号： C07D471/04
CPC分类号： C07D487/04 , C07D401/06 , C07D413/06 , C07D471/04 , C07D498/04 , C07D513/04
摘要： The present invention relates to novel compounds exhibiting good inhibitory activity versus Dipeptidyl Peptidase-IV(DPP-IV), methods of preparing the same and pharmaceutical compositions containing the same as an active agent.
摘要翻译：本发明涉及相对于二肽基肽酶-IV（DPP-IV）显示出良好抑制活性的新化合物，其制备方法和含有该活性剂的药物组合物。

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