基本信息:
- 专利标题: TREATMENT OF BREAST CANCER BRAIN METASTASES
- 专利标题(中):治疗乳腺癌脑转移瘤
- 申请号:PCT/IB2015/059525 申请日:2015-12-10
- 公开(公告)号:WO2016092508A1 公开(公告)日:2016-06-16
- 发明人: SHENG, Qing , JAIN, Rakesh K. , ASKOXYLAKIS, Vasileios , FERRARO, Gino B. , FUKUMURA, Dai , KODACK, David P.
- 申请人: MASSACHUSETTS GENERAL HOSPITAL , NOVARTIS AG , SHENG, Qing , JAIN, Rakesh K. , ASKOXYLAKIS, Vasileios , FERRARO, Gino B. , FUKUMURA, Dai , KODACK, David P.
- 申请人地址: 55 Fruit Street Boston, Massachusetts 02114 US
- 专利权人: MASSACHUSETTS GENERAL HOSPITAL,NOVARTIS AG,SHENG, Qing,JAIN, Rakesh K.,ASKOXYLAKIS, Vasileios,FERRARO, Gino B.,FUKUMURA, Dai,KODACK, David P.
- 当前专利权人: MASSACHUSETTS GENERAL HOSPITAL,NOVARTIS AG,SHENG, Qing,JAIN, Rakesh K.,ASKOXYLAKIS, Vasileios,FERRARO, Gino B.,FUKUMURA, Dai,KODACK, David P.
- 当前专利权人地址: 55 Fruit Street Boston, Massachusetts 02114 US
- 代理机构: RUECK, Sandra
- 优先权: US62/091,200 20141212
- 主分类号: A61K31/4741
- IPC分类号: A61K31/4741 ; A61K38/17 ; A61K45/00 ; A61K39/395
摘要:
The present invention relates to a pharmaceutical combination which comprises (a) a phosphatidylinositol 3-kinase inhibitor or pharmaceutically acceptable salt thereof, and (b) a Her3 antagonist, for simultaneous, separate or sequential administration for the treatment of breast cancer brain metastases; a method of treating a subject having a breast cancer brain metastases comprising administration of said combination to a subject in need thereof; use of such combination for the treatment of breast cancer brain metastases; and a commercial package comprising such combination.
摘要(中):
本发明涉及一种药物组合,其包含(a)磷脂酰肌醇3-激酶抑制剂或其药学上可接受的盐,和(b)Her3拮抗剂,用于同时,分别或连续施用以治疗乳腺癌脑转移瘤; 一种治疗患有乳腺癌脑转移的受试者的方法,包括向有需要的受试者施用所述组合; 使用这种组合治疗乳腺癌脑转移瘤; 以及包括这种组合的商业包装。
公开/授权文献:
- WO2016092508A9 TREATMENT OF BREAST CANCER BRAIN METASTASES 公开/授权日:2016-06-16
IPC结构图谱:
A | 人类生活必需 |
--A61 | 医学或兽医学;卫生学 |
----A61K | 医用、牙科用或梳妆用的配制品 |
------A61K31/00 | 含有机有效成分的医药配制品 |
--------A61K31/33 | .杂环化合物 |
----------A61K31/335 | ..仅有氧作为环杂原子的,例如制霉色基素 |
------------A61K31/40 | ...有仅以1个氮作为环杂原子的五元环的,例如舒必利、琥珀酰亚胺、托尔米丁、甲氧吡丁苯 |
--------------A61K31/47 | ....喹啉;异喹啉 |
----------------A61K31/4738 | .....与杂环邻位或迫位稠合的 |
------------------A61K31/4741 | ......与有氧作为环杂原子的环稠合的,例如筒箭毒碱衍生物、诺司卡品、荷包牡丹碱 |