发明申请
WO2004113294A1 PROCESS AND INTERMEDIATES FOR THE PREPARATION OF (1R, 2S, 5S)-3-AZABICYCLO[3, 1, 0]HEXANE-2-CARBOXAMIDE, N-[3-AMINO-1-(CYCLOBUTYLMETHYL)-2, 3-DIOXOPROPYL] ]-3-[(2S)-2-[[[1, 1-DIMETHYLETHYL]AMINO]CARBONYLAMINO]-3, 3-DIMETHYL-1-OXOBUTYL]-6, 6-DIMETHYL
审中-公开
基本信息:
- 专利标题： PROCESS AND INTERMEDIATES FOR THE PREPARATION OF (1R, 2S, 5S)-3-AZABICYCLO[3, 1, 0]HEXANE-2-CARBOXAMIDE, N-[3-AMINO-1-(CYCLOBUTYLMETHYL)-2, 3-DIOXOPROPYL] ]-3-[(2S)-2-[[[1, 1-DIMETHYLETHYL]AMINO]CARBONYLAMINO]-3, 3-DIMETHYL-1-OXOBUTYL]-6, 6-DIMETHYL
- 专利标题（中）：（1R，2S，5S）-3-亚氨基] [3,1,0]庚烷-2-羧酰胺，N- [3-氨基-1-（环己基甲基）-2,3-二氧杂环戊烯]的制备方法和中间体 ] -3 - [（2S）-2 - [[[1,1-二甲基氨基]氨基]羰基氨基] -3,3-二甲基-1-氧代丁基] -6,6-二甲基
- 申请号：PCT/US2004/018914 申请日：2004-06-15
- 公开(公告)号：WO2004113294A1 公开(公告)日：2004-12-29
- 发明人： SUDHAKAR, Anantha , DAHANUKAR, Vilas , ZAVIALOV, Ilia, A. , ORR, Cecilia , NGUYEN, Hoa, N. , WEBER, Juergen , JEON, Ingyu , CHEN, Minzhang , GREEN, Michael, D. , WONG, George, S. , PARK, Jeonghan , IWAMA, Tetsuo
- 申请人： SCHERING CORPORATION , SUDHAKAR, Anantha , DAHANUKAR, Vilas , ZAVIALOV, Ilia, A. , ORR, Cecilia , NGUYEN, Hoa, N. , WEBER, Juergen , JEON, Ingyu , CHEN, Minzhang , GREEN, Michael, D. , WONG, George, S. , PARK, Jeonghan , IWAMA, Tetsuo
- 申请人地址： 2000 Galloping Hill Road, Kenilworth, NJ 07033-0530 US
- 专利权人： SCHERING CORPORATION,SUDHAKAR, Anantha,DAHANUKAR, Vilas,ZAVIALOV, Ilia, A.,ORR, Cecilia,NGUYEN, Hoa, N.,WEBER, Juergen,JEON, Ingyu,CHEN, Minzhang,GREEN, Michael, D.,WONG, George, S.,PARK, Jeonghan,IWAMA, Tetsuo
- 当前专利权人： SCHERING CORPORATION,SUDHAKAR, Anantha,DAHANUKAR, Vilas,ZAVIALOV, Ilia, A.,ORR, Cecilia,NGUYEN, Hoa, N.,WEBER, Juergen,JEON, Ingyu,CHEN, Minzhang,GREEN, Michael, D.,WONG, George, S.,PARK, Jeonghan,IWAMA, Tetsuo
- 当前专利权人地址： 2000 Galloping Hill Road, Kenilworth, NJ 07033-0530 US
- 代理机构： KALYANARAMAN, Palaiyur, S.
- 优先权： US60/479,517 20030617
- 主分类号： C07D209/52
- IPC分类号： C07D209/52
摘要：
In one embodiment, the present application relates to a process of making a compound of formula (I): and to certain intermediate compounds that are made within the process of making the compound of formula (I).
摘要（中）：
在一个实施方案中，本申请涉及制备式（I）化合物的方法：和在制备式（I）化合物的过程中制备的某些中间体化合物。
IPC结构图谱:
| C | 化学；冶金 |
| --C07 | 有机化学 |
| ----C07D | 杂环化合物 |
| ------C07D209/00 | 杂环化合物，含五元环、与其他环稠合、带1个氮原子作为惟一的杂环原子 |
| --------C07D209/02 | .与一个碳环稠合 |
| ----------C07D209/52 | ..与一非六元环稠合 |