基本信息:
- 专利标题: P38 INHIBITORS AND METHODS OF USE THEREOF
- 专利标题(中):P38抑制剂及其使用方法
- 申请号:PCT/US2004005693 申请日:2004-02-25
- 公开(公告)号:WO2004078116A2 公开(公告)日:2004-09-16
- 发明人: MUNSON MARK , MARESKA DAVID A , KIM YOUNGBOO , GRONEBERG ROBERT , RIZZI JAMES , RODRIGUEZ MARTHA , KIM GANGHYEOK , VIGERS GUY , RAO CHANG , BALACHARI DEVAN , HARVEY DARREN
- 申请人: ARRAY BIOPHARMA INC , MUNSON MARK , MARESKA DAVID A , KIM YOUNGBOO , GRONEBERG ROBERT , RIZZI JAMES , RODRIGUEZ MARTHA , KIM GANGHYEOK , VIGERS GUY , RAO CHANG , BALACHARI DEVAN , HARVEY DARREN
- 专利权人: ARRAY BIOPHARMA INC,MUNSON MARK,MARESKA DAVID A,KIM YOUNGBOO,GRONEBERG ROBERT,RIZZI JAMES,RODRIGUEZ MARTHA,KIM GANGHYEOK,VIGERS GUY,RAO CHANG,BALACHARI DEVAN,HARVEY DARREN
- 当前专利权人: ARRAY BIOPHARMA INC,MUNSON MARK,MARESKA DAVID A,KIM YOUNGBOO,GRONEBERG ROBERT,RIZZI JAMES,RODRIGUEZ MARTHA,KIM GANGHYEOK,VIGERS GUY,RAO CHANG,BALACHARI DEVAN,HARVEY DARREN
- 优先权: US37816403 2003-03-03; US68884903 2003-10-15
- 主分类号: A61K
- IPC分类号: A61K20060101 ; A61K31/4745 ; A61K31/503 ; A61K31/675 ; C07D20060101 ; C07D231/56 ; C07D261/20 ; C07D401/14 ; C07D403/04 ; C07D413/12 ; C07D471/02 ; C07D471/04 ; C07D487/02 ; C07D491/02 ; A61K
摘要:
This invention relates to inhibitors of p38, and methods for producing these inhibitors. The invention also provides pharmaceutical compositions comprising the inhibitors of the invention and methods of utilizing the inhibitors and pharmaceutical compositions in the treatment and prevention of various disorders mediated by p38.
摘要(中):
本发明涉及p38的抑制剂及其制备方法。 本发明还提供包含本发明抑制剂的药物组合物和利用抑制剂和药物组合物治疗和预防由p38介导的各种疾病的方法。
公开/授权文献:
- WO2004078116A9 P38 INHIBITORS AND METHODS OF USE THEREOF 公开/授权日:2008-09-12
IPC结构图谱:
A | 人类生活必需 |
--A61 | 医学或兽医学;卫生学 |
----A61K | 医用、牙科用或梳妆用的配制品 |