基本信息:
- 专利标题： 아실옥시알킬 카르바메이트 프로드러그, 합성 및 사용 방법
- 专利标题（英）：Acyloxyalkyl carbamate prodrugs, methods of synthesis and use
- 专利标题（中）：丙烯酰基碳酸酯产品，合成和使用方法
- 申请号：KR1020067003464 申请日：2004-08-20
- 公开(公告)号：KR101140559B1 公开(公告)日：2012-07-05
- 发明人： 갤럽마크에이 , 야오펀메이 , 루드비코우마리아제이 , 판투 , 펑거
- 申请人： 제노포트 인코포레이티드
- 申请人地址： **** CENTRAL EXPRESSWAY, SANTA CLARA, CA *****, U.S.A.
- 专利权人： 제노포트 인코포레이티드
- 当前专利权人： 제노포트 인코포레이티드
- 当前专利权人地址： **** CENTRAL EXPRESSWAY, SANTA CLARA, CA *****, U.S.A.
- 代理人： 특허법인코리아나
- 优先权： US10/932,374 2004-08-13; US60/496,938 2003-08-20
- 国际申请： PCT/US2004/027330 2004-08-20
- 国际公布： WO2005019163 2005-03-03
- 主分类号： C07C271/22
- IPC分类号： C07C271/22 ; C07D207/416 ; C07D333/38 ; C07D401/04
The present specification are generally (±) -4- amino-3- (4-chlorophenyl) portion acyloxyalkyl carbamate prodrugs, thereof the pharmaceutical composition of the acid and analogs thereof, (±) -4- amino-3 (4-chlorophenyl) butanoic acid and analogs thereof of the method of producing a prodrug, and for example, seizures, and / or typical disease and / or for treating or preventing a disorder (±) -4, such as acid reflux disease -amino-3 relates to a use of (4-chlorophenyl) portion and a prodrug thereof the pharmaceutical composition of the acid and its analogs. The present specification is also directed to the appropriate (±) -4- amino-3- (4-chlorophenyl) butanoic acid and its acyloxyalkyl carbamate prodrugs thereof, and the sustained release oral dosage forms of the analogs of water for oral administration.
公开/授权文献:
- KR1020060126899A 아실옥시알킬 카르바메이트 프로드러그, 합성 및 사용 방법 公开/授权日：2006-12-11
信息查询:
EspacenetIPC结构图谱:
| C | 化学；冶金 |
| --C07 | 有机化学 |
| ----C07C | 无环或碳环化合物 |
| ------C07C271/00 | 氨基甲酸衍生物，即含有如下任何基团的化合物NCOO，NCOHal，NCOO，NCOHal或NCHalHal或氮原子不属于硝基或亚硝基 |
| --------C07C271/06 | .氨基甲酸酯 |
| ----------C07C271/08 | ..氨基甲酸酯基的氧原子连接非环碳原子 |
| ------------C07C271/10 | ...氨基甲酸酯基的氮原子连接氢原子或非环碳原子 |
| --------------C07C271/22 | ....连接由羧基取代的烃基的碳原子 |