发明公开
EP2035424A1 AMINO-IMIDAZOLONES AND THEIR USE AS A MEDICAMENT FOR TREATING COGNITIVE IMPAIRMENT, ALZHEIMER DISEASE, NEURODEGENERATION AND DEMENTIA.
审中-公开
![AMINO-IMIDAZOLONES AND THEIR USE AS A MEDICAMENT FOR TREATING COGNITIVE IMPAIRMENT, ALZHEIMER DISEASE, NEURODEGENERATION AND DEMENTIA.](/ep/2009/03/18/EP2035424A1/abs.jpg.150x150.jpg)
基本信息:
- 专利标题: AMINO-IMIDAZOLONES AND THEIR USE AS A MEDICAMENT FOR TREATING COGNITIVE IMPAIRMENT, ALZHEIMER DISEASE, NEURODEGENERATION AND DEMENTIA.
- 专利标题(中):AMINOIMIDAZOLONE和它们作为治疗认知障碍阿尔茨海默氏症,老年痴呆症和神经变性治疗
- 申请号:EP07748235.4 申请日:2007-06-12
- 公开(公告)号:EP2035424A1 公开(公告)日:2009-03-18
- 发明人: BERG, Stefan , HOLENZ, Jörg , HÖGDIN, Katharina , KIHLSTRÖM, Jacob , KOLMODIN, Karin , LINDSTRÖM, Johan , PLOBECK, Niklas , ROTTICCI, Didier , SEHGELMEBLE, Fernando , EK, Maria
- 申请人: AstraZeneca AB , Astex Therapeutics Limited
- 申请人地址: 151 85 Södertälje SE
- 专利权人: AstraZeneca AB,Astex Therapeutics Limited
- 当前专利权人: AstraZeneca AB,Astex Therapeutics Limited
- 当前专利权人地址: 151 85 Södertälje SE
- 优先权: US813767P 20060614; US896992P 20070326
- 国际公布: WO2007145569 20071221
- 主分类号: C07D487/04
- IPC分类号: C07D487/04 ; A61K31/519 ; A61P25/28
摘要:
This invention relates to novel compounds having the structural formula (I) and to their pharmaceutically acceptable salt, compositions and methods of use. These novel compounds provide a treatment or prophylaxis of cognitive impairment, Alzheimer Disease, neurodegeneration and dementia.
IPC结构图谱:
C | 化学;冶金 |
--C07 | 有机化学 |
----C07D | 杂环化合物 |
------C07D487/00 | 在稠环系中含有氮原子作为仅有的杂环原子的杂环化合物,不包含在C07D451/00至C07D477/00组中 |
--------C07D487/02 | .在稠合系中含有两个杂环 |
----------C07D487/04 | ..邻位稠合系 |