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1. 发明申请

WO9309099A3 SULFONAMIDE HERBICIDES 审中-公开
标题翻译：磺胺类除草剂
公开(公告)号：WO9309099A3
公开(公告)日：1993-06-10
申请号：PCT/EP9202558
申请日：1992-11-02
申请人： SCHERING AGROCHEMICALS LTD
发明人： GATES PETER STUART , JONES GRAHAM PETER , SAUNDERS DAVID EDWARD
IPC分类号： A01N43/54 , A01N43/56 , A01N43/66 , C07D239/26 , C07D239/34 , C07D239/38 , C07D239/42 , C07D239/52 , C07D251/20 , C07D251/60 , C07D401/06 , C07D401/12 , C07D403/06 , C07D403/12 , C07D409/12 , C07D417/06 , C07D239/60
CPC分类号： C07D401/06 , A01N43/54 , A01N43/56 , A01N43/66 , C07D239/52 , C07D251/20 , C07D251/60 , C07D403/06 , C07D403/12 , C07D409/12
摘要： Herbicidal sulfonamides of formula (I) and salts thereof, where A represents a substituted or unsubstituted benzene ring, or a 5- or 6-membered substituted or unsubstituted heteroaromatic ring; Q is -O-, -S- or a group -CXX'-; X and X', which may be the same or different, are each hydrogen, halogen, cyano, an optionally-substituted alkyl group, or a group -ORa, -SRa, or -CORb; or one of X and X' represents hydroxy and the other is as defined above; or X and X' together represent =O or =S; Ra is an optionally-substituted alkyl, aryl or acyl group; Rb is an optionally-substituted alkyl or aryl group, or a group -OR?c or -NRcRd; Rc and Rd¿, which may be the same or different, are each hydrogen, or an optionally-substituted alkyl or aryl group; Y is nitrogen or a group CR9; R1 is an optionally-substituted alkyl, alkenyl, alkynyl, cycloalkyl, aryl, heterocyclyl, benzoheterocyclyl or amino group; R2 is hydrogen, an optionally-substituted alkyl or carboxylic acyl group, or a group -SO¿2?R?1; R3 and R4¿, which may be the same or different, are each hydrogen, halo, an optionally substituted alkyl, alkoxy, cycloalkyl or amino group, or an optionally-substituted heterocyclyl group; and R9 represents hydrogen or an optionally-substituted alkyl group.

2. 发明申请

WO2023286725A1 紫外線吸収剤及びその製造方法、組成物、成形体、塗膜审中-公开
公开(公告)号：WO2023286725A1
公开(公告)日：2023-01-19
申请号：PCT/JP2022/027201
申请日：2022-07-11
申请人：東洋インキＳＣホールディングス株式会社 , トーヨーカラー株式会社
发明人：千葉　優美香 , 辰巳　僚一 , 槇　大輔
IPC分类号： C09K3/00 , C07D251/20 , C08K5/3492 , C08L101/00
摘要：下記一般式（１）～（３）で示す化合物からなる群から選ばれる１種以上の紫外線吸収色素、ならびにＮａ、Ｍｇ、Ａｌ、Ｋ、Ｃａ、およびＦｅからなる群から選ばれる１種以上の金属原子を含む金属成分を含む紫外線吸収剤であって、前記金属成分の含有量が前記紫外線吸収剤に対して０．１～５００００ｐｐｍである、紫外線吸収剤。

3. 发明申请

WO2012084857A3 METHOD FOR PRODUCING 2-(TRIAZINYLCARBONYL) SULFONANILIDES 审中-公开
标题翻译： 2-（三苄基羰基）磺酰苯胺的制备方法
公开(公告)号：WO2012084857A3
公开(公告)日：2012-08-16
申请号：PCT/EP2011073287
申请日：2011-12-19
申请人： BAYER CROPSCIENCE AG , KARIG GUNTER , FORD MARK JAMES , SIEGEL KONRAD
发明人： KARIG GUNTER , FORD MARK JAMES , SIEGEL KONRAD
IPC分类号： C07D403/04 , A01N43/66 , C07D251/20
CPC分类号： C07D251/20 , A01N43/66 , C07D403/04
摘要： The invention relates to a method, which is based on the oxidative ring opening of a compound with an oxindole structure, for producing substituted 2-(triazinylcarbonyl) sulfonanilides of formula (1-1) proceeding from an N-sulfonyl-substituted 3-triazinyl oxindole of formula (2-1), to the thus produced 2-(triazinylcarbonyl) sulfonanilides of formula (1-1), and to the use thereof as intermediate products for the synthesis of fine chemicals and active substances in the agricultural field. Furthermore, the invention relates to a multistage method for producing N-alkyl-N-[2-(1,3,5-triazin-2-ylcarbonyl)phenyl]alkansulfonamides of formula (4-1) proceeding from a 3-(alkylsulfanyl)-1,3-dihydro-2H-indol-2-on of formula (7-1), wherein the multistage method also has said oxidative opening as a sub-step, and to the 2-(triazinylcarbonyl) sulfonanilides of formula (1-1), said sulfonanilides being obtained by means of the oxidative ring opening and used as intermediates in the multistage method.
摘要翻译：本申请涉及一种方法，该方法是基于具有Oxindolstruktur的化合物的氧化开环，制备式（1-1）的取代的2-（Triazinylcarbonyl）sulfonaniliden的制备从N-3-sulfonylsubstituierten Triazinyloxindol启动式（2-1）和如此制备的式（1-1）的2-（三嗪基 - 羰基）磺酰苯胺及其作为用于合成农业中的精细化学品和活性成分的中间体的用途。此外，本发明涉及一种多级方法用于制备N-烷基-N- [2-（1,3,5-三嗪-2-基羰基）苯基]从3-（烷基硫基）启动式（4-1）的alkanesulfonamides -1,3-二氢-2H-吲哚-2-酮的式（7-1），其中，所述多阶段工艺包括如步骤的一部分的，所述式氧化开环和通过氧化开环得到的2-（Triazinylcarbonyl）磺酰苯胺（1-1），它们在多阶段过程中用作中间体。

4. 发明申请

WO9608949A3 NOVEL MONOMERIC AND POLYMERIC CYCLIC AMINE AND N-HALAMINE COMPOUNDS 审中-公开
标题翻译：新型单体和聚合物循环胺和N-哈马林化合物
公开(公告)号：WO9608949A3
公开(公告)日：1996-10-03
申请号：PCT/IB9500885
申请日：1995-09-22
申请人： UNIV AUBURN
发明人： WORLEY SHELLEY D , SUN GANG , SUN WANYING , CHEN TAY-YUAN
IPC分类号： A01N59/00 , C07D233/74 , C07D251/10 , C07D251/20 , C07D263/22 , C08F8/30 , C08F8/48 , C08F12/26
CPC分类号： C07D233/74 , A01N59/00 , C07D251/20 , C08F8/30 , C08F8/48 , C08F12/26 , Y02W10/37
摘要： Cyclic amine monomers and polymers and N-halamine biocidal polymer compounds are provided. Methods of making and using the same wherein the functional groups unhalogenated or halogenated hydantoins, triazine diones, imidazolidinones, and pyrimidinones are substituted onto inexpensive polymer units such as polystyrene, polyethylene, and modified polymethacrylamide are provided. The cyclic amine monomers and polymers can be utilized to form a biocidal N-halamine polymers. These N-halamine polymers are stable, insoluble biocides which release only small amounts of free halogen and other impurities. They can be useful as disinfectants for potable water, swimming pools, hot tubs, industrial water systems, cooling towers, air-conditioning systems, gas streams, paints, oils, ointments, fabrics, rubber materials, sterile bandages, coatings, hard surfaces, liners of containers, and the like.

5. 发明申请

WO2020000832A1 一种奧替拉西钾的合成方法审中-公开
公开(公告)号：WO2020000832A1
公开(公告)日：2020-01-02
申请号：PCT/CN2018/113332
申请日：2018-11-01
申请人：山东新时代药业有限公司
发明人：张贵民 , 朱安国 , 刘东
IPC分类号： C07D251/20
摘要：本发明提供了一种奧替拉西钾的合成方法。所述方法包括步骤：室温下，将2-氨甲酰胺基-2-氧乙酸，尿素，催化剂加入溶剂中，升温环化反应，检测至反应结束，降温，调节反应液的pH值并成钾盐，搅拌养晶，后抽滤，滤饼依次用纯化水，冷无水醇类洗涤，真空干燥后即得奥替拉西钾。与现有技术相比，整个工艺过程原料简单易得、操作简便、反应条件温和、质量稳定、收率较高、对环境也不会造成污染，适合工业化生产。

6. 发明申请

WO0246172A3 SUBSTITUTED 1, 3, 5-TRIAZINES AND PYRIMIDINES AS ABCA-1 ELEVATING COMPOUNDS AGAINST CORONARY ARTERY DISEASE OR ATHEROSCLEROSIS 审中-公开
标题翻译：作为ABCA-1替代化合物，针对冠状动脉疾病或甲状腺功能亢进的化合物替代1,3,5-二噻吩和嘧啶
公开(公告)号：WO0246172A3
公开(公告)日：2003-02-06
申请号：PCT/US0146387
申请日：2001-12-03
申请人： CV THERAPEUTICS INC
发明人： CAMPBELL MICHAEL , ZABLOCKI JEFF A , IBRAHIM PRABHA N
IPC分类号： A61K45/00 , A61K31/085 , A61K31/136 , A61K31/16 , A61K31/165 , A61K31/167 , A61K31/17 , A61K31/18 , A61K31/357 , A61K31/435 , A61K31/47 , A61K31/472 , A61K31/495 , A61K31/505 , A61K31/506 , A61K31/53 , A61K45/06 , A61P3/06 , A61P9/00 , A61P9/10 , A61P43/00 , C07C237/04 , C07C237/06 , C07C237/22 , C07C237/40 , C07C275/26 , C07C311/20 , C07C323/36 , C07C323/40 , C07C323/60 , C07C327/42 , C07C327/44 , C07C327/48 , C07C335/16 , C07D215/38 , C07D217/24 , C07D239/48 , C07D251/16 , C07D251/22 , C07D251/52 , C07D319/08 , C07D319/18 , C07D401/12 , C07D405/12 , C07D409/12 , C07D409/14 , C07D413/12 , C07D413/14 , C07D251/20 , C07D251/46 , C07D403/12
CPC分类号： C07D319/08 , A61K31/53 , A61K45/06 , C07C237/06 , C07C237/22 , C07C237/40 , C07C275/26 , C07C311/20 , C07C323/36 , C07C323/40 , C07C323/60 , C07C327/42 , C07C327/48 , C07C2601/08 , C07C2601/14 , C07C2602/10 , C07C2602/40 , C07C2602/42 , C07C2603/74 , C07D251/16 , C07D251/52 , C07D409/12 , A61K2300/00
摘要： The present invention provides compounds that elevate cellular expression of the ABCA-1 gene, promoting cholesterol efflux from cells and increasing HDL levels in the plasma of a mammal, in particular humans. The compounds are useful for treating coronary artery disease.
摘要翻译：本发明提供了提高ABCA-1基因的细胞表达，促进来自细胞的胆固醇流出并增加哺乳动物，特别是人的血浆中的HDL水平的化合物。该化合物可用于治疗冠状动脉疾病。

7. 发明申请

WO99067225A1 BENZOCYCLE-SUBSTITUTED TRIAZINE AND PYRIMIDINE ULTRAVIOLET LIGHT ABSORBERS 审中-公开
标题翻译：苯并噻唑啉和紫杉醇紫外线吸收剂
公开(公告)号：WO99067225A1
公开(公告)日：1999-12-29
申请号：PCT/US1999/013708
申请日：1999-06-17
IPC分类号： A61K8/49 , A61Q17/04 , C07D239/26 , C07D239/32 , C07D251/20 , C07D251/22 , C07D251/24 , C08K5/3492 , A61K7/42
CPC分类号： A61K8/4966 , A61Q17/04 , C07D239/26 , C07D251/20 , C07D251/22 , C07D251/24 , C08K5/3492
摘要： This invention relates generally to benzocycle-substituted pyrimidines and triazines and the use thereof to protect against degradation by environmental forces, inclusive of ultraviolet light, actinic radiation, oxidation, moisture, atmospheric pollutants and combinations thereof. The new class of benzocycle-substituted pyrimidines and triazines comprises a benzocycle attached to the triazine or pyrimidine ring, and preferably an additional aryl ring containing a hydroxyl group, either free or blocked to form a latent stabilizer, ortho- to the point of attachment to the triazine or pyrimidine ring. These materials may, under the appropriate circumstances, be bonded to formulations comprising coatings, polymers, resins, organic compounds and the like via reaction of the bondable functionality with the materials of the formulation. A method for stabilizing a material by incorporating such benzocycle-substituted pyrimidines and triazines is also disclosed.
摘要翻译：本发明一般涉及苯并环取代的嘧啶和三嗪及其用于防止包括紫外光，光化辐射，氧化，水分，大气污染物及其组合在内的环境力降解的用途。新类型的苯并环取代的嘧啶和三嗪包括与三嗪或嘧啶环连接的苯并环，并且优选含有游离或封闭以形成潜稳定剂的羟基的另外的芳环，三嗪或嘧啶环。这些材料可以在适当的情况下通过可结合的官能团与制剂的材料的反应与包含涂料，聚合物，树脂，有机化合物等的制剂结合。还公开了通过掺入这种苯并环取代的嘧啶和三嗪来稳定材料的方法。

8. 发明申请

WO1996008949A2 NOVEL MONOMERIC AND POLYMERIC CYCLIC AMINE AND N-HALAMINE COMPOUNDS 审中-公开
标题翻译：新型单体和聚合物循环胺和N-哈马林化合物
公开(公告)号：WO1996008949A2
公开(公告)日：1996-03-28
申请号：PCT/IB1995000885
申请日：1995-09-22
申请人： AUBURN UNIVERSITY
发明人： AUBURN UNIVERSITY , WORLEY, Shelley, D. , SUN, Gang , SUN, Wanying , CHEN, Tay-Yuan
IPC分类号： A01N59/00 , C07D233/74 , C07D251/10 , C07D251/20 , C07D263/22 , C08F8/30 , C08F8/48 , C08F12/26
CPC分类号： C07D233/74 , A01N59/00 , C07D251/20 , C08F8/30 , C08F8/48 , C08F12/26 , Y02W10/37
摘要： Cyclic amine monomers and polymers and N-halamine biocidal polymer compounds are provided. Methods of making and using the same wherein the functional groups unhalogenated or halogenated hydantoins, triazine diones, imidazolidinones, and pyrimidinones are substituted onto inexpensive polymer units such as polystyrene, polyethylene, and modified polymethacrylamide are provided. The cyclic amine monomers and polymers can be utilized to form a biocidal N-halamine polymers. These N-halamine polymers are stable, insoluble biocides which release only small amounts of free halogen and other impurities. They can be useful as disinfectants for potable water, swimming pools, hot tubs, industrial water systems, cooling towers, air-conditioning systems, gas streams, paints, oils, ointments, fabrics, rubber materials, sterile bandages, coatings, hard surfaces, liners of containers, and the like.
摘要翻译：提供了环胺单体和聚合物以及N-卤胺杀生物聚合物化合物。提供了制备和使用其的方法，其中将官能团的未卤化或卤代乙内酰脲，三嗪二酮，咪唑烷酮和嘧啶酮取代到廉价的聚合物单元如聚苯乙烯，聚乙烯和改性的聚甲基丙烯酰胺上。环胺单体和聚合物可用于形成杀生物N-卤代胺聚合物。这些N-卤代胺聚合物是仅释放少量游离卤素和其它杂质的稳定的不溶性杀生物剂。它们可用作饮用水，游泳池，热水浴缸，工业水系统，冷却塔，空调系统，气体流，油漆，油，软膏，织物，橡胶材料，无菌绷带，涂层，硬表面的消毒剂，容器内衬等。

9. 发明申请

WO2017076264A1 一类对GPR84具有激动作用的化合物及其制备方法和用途审中-公开
公开(公告)号：WO2017076264A1
公开(公告)日：2017-05-11
申请号：PCT/CN2016/104165
申请日：2016-11-01
申请人：中国科学院上海药物研究所
发明人：南发俊 , 谢欣 , 刘阳 , 张庆 , 陈林海 , 杨慧
IPC分类号： C07D239/60 , C07D239/54 , C07D309/38 , C07D213/69 , C07C49/825 , C07C39/08 , C07D239/56 , C07D239/48 , C07D251/20 , C07D239/545 , A61K31/505
CPC分类号： A61K31/505 , C07C39/08 , C07C49/825 , C07D213/69 , C07D239/48 , C07D239/54 , C07D239/545 , C07D239/56 , C07D239/60 , C07D251/20 , C07D309/38
摘要：本发明涉及一类通式Ⅰ所示的化合物或其药学上可接受的盐、其制备方法，以及其作为GPR84激动剂工具小分子中的应用，和其在制备治疗败血症的药物中的应用。

10. 发明申请

WO2013084013A1 CYCLOALKANE CARBOXYLIC ACID DERIVATIVES AS CXCR3 RECEPTOR ANTAGONISTS 审中-公开
标题翻译：作为CXCR3受体拮抗剂的环己烷羧酸衍生物
公开(公告)号：WO2013084013A1
公开(公告)日：2013-06-13
申请号：PCT/HU2012/000128
申请日：2012-12-03
申请人： SANOFI
发明人： BATA, Imre , BUDZER-LANTOS, Péter , VASAS, Attila , BARTÁNÉ BODOR, Veronika , FERENCZY, György , TÖMÖSKÖZI, Zsuzsanna , SZELECZKY, Gábor , BÁTORI, Sándor , SMRCINA, Martin , PATEK, Marcel , WEICHSEL, Aleksandra , S.THORPE, David
IPC分类号： A61K31/4025 , C07D207/40 , C07D209/48 , C07D209/94 , C07D221/20 , C07D233/74 , C07D239/54 , C07D251/20 , C07D263/44 , C07D277/34 , C07D405/12 , C07D413/12 , C07D417/12 , A61P37/08
CPC分类号： C07D207/408 , A61K31/4015 , A61K31/403 , A61K31/4035 , A61K31/4166 , A61K31/421 , A61K31/426 , A61K31/427 , A61K31/438 , A61K31/45 , A61K31/506 , A61K31/513 , A61K31/53 , C07D207/40 , C07D209/48 , C07D209/52 , C07D209/94 , C07D211/88 , C07D221/20 , C07D233/74 , C07D239/54 , C07D251/20 , C07D263/44 , C07D277/34 , C07D405/12 , C07D413/12 , C07D417/12
摘要： The present invention relates to compounds of formula 1 that are useful as an active ingredient of a medicament for preventive and/or therapeutic treatment of diseases caused by abnormal activation of CXCR3 chemokines. The invention relates furthermore to a process for the preparation of said compounds, to pharmaceutical compositions containing said compounds and to the novel intermediates used in the preparation of said compounds.
摘要翻译：本发明涉及可用作用于预防和/或治疗由CXCR3趋化因子的异常活化引起的疾病的药物的活性成分的式1化合物。本发明还涉及制备所述化合物的方法，含有所述化合物的药物组合物和用于制备所述化合物的新型中间体。

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