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    • 3. 发明申请
    • COMPOSITIONS FOR PROVIDING HEPATOPROTECTIVE EFFECT
    • 用于提供肝脏保护作用的组合物
    • WO2008049265A1
    • 2008-05-02
    • PCT/CN2006/002828
    • 2006-10-23
    • SIMPSON BIOTECH CO., LTD.MASAO, HattoriSHEU, Chia,Chin
    • MASAO, HattoriSHEU, Chia,Chin
    • A61K31/715A61K36/06A61P1/16
    • A61K31/715A61K36/07
    • This invention relates to a composition for injection comprising a neutral polysaccharide of Antrodia camphorata having characteristics as follows: (a) appearance: colorless and shapeless powder, (b) pH: neutral, (c) molecular weight: 899.5~1670.5 kDa determined by HPLC as shown in (4), (d) rotatory power: (α) D +115.0 º (c = 0.4433, H 2 O), (e) intrinsic viscosity: (ŋ) = 0.03971~0.06255 dl ·g -1 , (f) specific heat Cp: 0.2536~0.3995 Cal/g · ºC, (g) IR spectrum: as shown in (5), (h) 1 H-NMR spectrum: as shown in (6), (i) 13 C-NMR spectrum: as shown in (7), and (j) GC-MS analysis: as shown in (8). This invention also relates to a composition for oral administering comprising a neutral polysaccharide of Antrodia camphorata having characteristics (a)-(j) as above.
    • 本发明涉及一种注射用组合物,其特征在于:(a)外观:无色无定形粉末,(b)pH:中性,(c)通过HPLC测定的分子量:899.5〜1670.5kDa 如(4)所示,(d)旋转动力:(a)D + 1151°(c = 0.4433,H 2 O),(e)特性粘度: (ν)= 0.03971〜0.06255 dl·g -1,(f)比热Cp:0.2536〜0.3995 Cal / g·ºC,(g)IR光谱:如(5),( h)1 H-NMR光谱如(6)所示,(i)13 C-NMR光谱:如(7)所示,和(j)GC -MS分析:如(8)所示。 本发明还涉及用于口服给药的组合物,其包含具有上述特征(a) - (j)的樟脑的中性多糖。