专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

11. 发明申请

WO1995004727A1 PROCESS FOR THE PREPARATION OF FLUOROATHENYLTHIO HETEROCYCLIC DERIVATIVES 审中-公开
标题翻译：制备氟尿嘧啶杂环衍生物的方法
公开(公告)号：WO1995004727A1
公开(公告)日：1995-02-16
申请号：PCT/GB1994001570
申请日：1994-07-20
申请人： ZENECA LIMITED , TURNBULL, Michael, Drysdale , WILLETTS, Nigel, James , FITZJOHN, Steven , KHOLIA, Prafula, Govind , SMITH, Alison, Mary , SALMON, Roger , BANSAL, Harjinder, Singh , WILLIAMS, Alfred, Glyn
发明人： ZENECA LIMITED
IPC分类号： C07D263/58
CPC分类号： C07D263/58 , C07C17/087 , C07C17/23 , C07C21/18 , C07C309/73 , C07D239/38 , C07D277/74
摘要： A process for the preparation of a compound of formula (I) : HetSCH2CH2CH=CF2 wherein Het is an optionally substituted 5- or 6-membered heterocyclic ring, which comprises reacting a compound of formula (II) : HetSH with a compound of formula (III) : CF2=CHCH2CH2L wherein L is chlorine or bromine or a group -OSO2R wherein R is a C1-4 alkyl group or a phenyl group optionally substituted by a C1-4 alkyl group.
摘要翻译：制备式（I）化合物的方法：HetSCH2CH2CH = CF2其中Het是任选取代的5或6元杂环，其包括使式（II）化合物：HetSH与式（I）化合物 III）：CF 2 = CHCH 2 CH 2 L其中L是氯或溴或基团-OSO 2 R a，其中R a是C 1-4烷基或任选被C 1-4烷基取代的苯基。

12. 发明申请

WO1994027951A1 PREPARATION OF CYCLOPROPANE ESTERS 审中-公开
标题翻译：环孢菌素的制备
公开(公告)号：WO1994027951A1
公开(公告)日：1994-12-08
申请号：PCT/GB1994001139
申请日：1994-05-25
申请人： ZENECA LIMITED , BOWDEN, Martin, Charles , TURNBULL, Michael, Drysdale
发明人： ZENECA LIMITED
IPC分类号： C07C69/743
CPC分类号： C07C43/32 , C07C69/65 , C07C69/743
摘要： There is disclosed a process for the preparation of a lower alkyl ester of 3-(2-chloro-3,3,3-trifluoroprop-1-en-1-yl)-2,2-dimethylcyclopropane carboxylic acid which comprises the steps of (a) reacting a compound of the formula (I): CF3-CXC1-CH(OH)-CH=C(CH3)2, wherein X is chloro or bromo, with a tri-lower-alkyl orthoacetate containing up to four carbon atoms in each alkyl group in the presence of at least a catalytic amount of an acid catalyst at an elevated temperature for a sufficient time to obtain a compound of the formula (III): CF3-CXC1-CH=CH-C(CH3)2-CH2CO2R, wherein R is an alkyl group containing up to four carbon atoms, and (b) treating said compound of formula (III) with at least one molar equivalent of a base to obtain said alkyl ester of 3-(2-chloro-3,3,3-trifluoroprop-1-en-1-yl)-2,2-dimethylcyclopropane carboxylic acid. The products are useful as intermediates for insecticides.
摘要翻译：公开了制备3-（2-氯-3,3,3-三氟丙-1-烯-1-基）-2,2-二甲基环丙烷羧酸的低级烷基酯的方法，该方法包括以下步骤：（a）使式（I）化合物：CF 3 -S CXCl-CH（OH）-CH = C（CH 3）2，其中X是氯或溴，与含有最多四个碳原子的三低级烷基原乙酸在至少催化量的酸催化剂存在下，在升高的温度下在足够的时间得到式（III）的化合物：CF 3 -CClCl-CH = CH-C（CH 3）2 -CH 2 CO 2 R，其中R是含有至多4个碳原子的烷基，和（b）用至少一摩尔当量碱处理式（III）化合物，得到所述3-（2-氯 - 3,3,3-三氟丙-1-烯-1-基）-2,2-二甲基环丙烷羧酸。该产品可用作杀虫剂的中间体。

13. 发明申请

WO1994006782A1 BENZOXAZOLE AND BEZOTHIAZOLE DERIVATIVES 审中-公开
标题翻译：苯并唑和异丁唑衍生物
公开(公告)号：WO1994006782A1
公开(公告)日：1994-03-31
申请号：PCT/GB1993001913
申请日：1993-09-10
申请人： ZENECA LIMITED , FITZJOHN, Steven , ROBINSON, Michael, Peter , TURNBULL, Michael, Drysdale , SMITH, Alison, Mary , SALMON, Roger , TAYLOR, Robin
发明人： ZENECA LIMITED
IPC分类号： C07D277/74
CPC分类号： C07D263/58 , A01N43/76 , A01N43/78 , A01N47/02 , C07C17/087 , C07C205/58 , C07C309/66 , C07C309/73 , C07D277/74 , C07D277/76 , C07C19/14
摘要： The invention provides novel compounds of formula (I) having nematicidal, insecticidal, acaricidal and fungicidal properties, compositions comprising them and processes and intermediates for their preparation, wherein X is oxygen or sulphur; n is 0, 1 or 2; R1, R2, R3, and R4 are independently selected from hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, alkylcycloalkyl, optionally substituted aryl, optionally substituted arylalkyl, optionally substituted aryloxy, optionally substituted arylalkoxy, alkoxy, alkenyloxy, alkynyloxy, hydroxyalkyl, alkoxyalkyl, alkylthio, alkenylthio, alkynylthio, haloalkyl, haloalkenyl, haloalkynyl, haloalkoxy, haloalkenyloxy, haloalkynyloxy, haloalkylthio, haloalkenylthio, haloalkynylthio, halogen, hydroxy, cyano, nitro, -NR5R6, -NR7COR8, -NR9SO2R10, -N(SO2-R11)(SO2-R12), -COR13, -CONR14R15, -COOR16, -OCOR17, -OSO2R18, -SO2NR19R20, -SO2R21, -SOR22, -CSNR23R24, -SiR25R26R27, -OCH2CO2R28, -OCH2CH2CO2R29, -CONR30SO2R31 and -SO2Z; or an adjacent pair of R1, R2, R3 and R4 when taken together form a fused 5- or 6-membered carbocyclic or heterocyclic ring; R5, R6, R7, R8, R9, R10, R11, R12, R13, R14, R15, R16, R17, R18, R19, R20, R21, R22, R23, R24, R25, R26, R27, R28, R29, R30 and R31 are independently selected from hydrogen, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, haloalkynyl, optionally substituted aryl and optionally substituted aryalkyl; and Z is halogen.
摘要翻译：本发明提供了具有杀线虫，杀虫，杀螨和杀真菌性质的新颖的式（I）化合物，包含它们的组合物及其制备方法和中间体，其中X是氧或硫; n为0,1或2; R 1，R 2，R 3和R 4独立地选自氢，烷基，烯基，炔基，环烷基，烷基环烷基，任选取代的芳基，任选取代的芳烷基，任选取代的芳氧基，任选取代的芳基烷氧基，烷氧基，烯氧基，炔氧基，羟烷基，烷氧基烷基，烷基硫代，链烯硫基，炔硫基，卤代烷基，卤代烯基，卤代炔基，卤代烷氧基，卤代烯基氧基，卤代炔基氧基，卤代烷硫基，卤代烯基硫基，卤代炔硫基，卤素，羟基，氰基，硝基，-NR5R6，-NR7COR8，-NR9SO2R10，-N（SO2-R11） -R12），-COR13，-CONR14R15，-COOR16，-OCOR17，-OSO2R18，-SO2NR19R20，-SO2R21，-SOR22，-CSNR23R24，-SiR25R26R27，-OCH2CO2R28，-OCH2CH2CO2R29，-CONR30SO2R31和-SO2Z; 或相邻的一对R 1，R 2，R 3和R 4一起形成稠合的5元或6元碳环或杂环; R5，R6，R7，R8，R9，R10，R11，R12，R13，R14，R15，R16，R17，R18，R19，R20，R21，R22，R23，R24，R25，R26，R27，R28， R30和R31独立地选自氢，烷基，烯基，炔基，卤代烷基，卤代烯基，卤代炔基，任选取代的芳基和任选取代的芳烷基; Z为卤素。

14. 发明申请

WO2009090402A3 HERBICIDAL COMPOUNDS 审中-公开
公开(公告)号：WO2009090402A3
公开(公告)日：2009-07-23
申请号：PCT/GB2009/000127
申请日：2009-01-16
申请人： SYNGENTA LIMITED , CORDINGLEY, Matthew, Robert , TURNBULL, Michael, Drysdale , CARTER, Neil, Brian , CROWLEY, Patrick, Jelf
发明人： CORDINGLEY, Matthew, Robert , TURNBULL, Michael, Drysdale , CARTER, Neil, Brian , CROWLEY, Patrick, Jelf
IPC分类号： A01N43/90 , A01P13/00
摘要： The present invention relates to a method of controlling plants or inhibiting plant growth which comprises applying to the plants or to the locus thereof a herbicidally effective amount of a compound of formula (I) wherein R 1 , R 2 , R 3 , R 4 and R 5 are as defined in claim 1; or a salt or TV-oxide thereof. Furthermore, the present invention relates to processes for preparing compounds of formula (I), to intermediates used in the preparation of compounds of formula (I), to herbicidal compositions comprising compounds of formula (I) and to certain novel pyridopyridines.

15. 发明申请

WO2008071918A1 PYRIDO-PYRAZINE DERIVATIVES USEFUL AS HERBICIDAL COMPOUNDS 审中-公开
标题翻译：吡咯并吡啶衍生物有效用作除草剂化合物
公开(公告)号：WO2008071918A1
公开(公告)日：2008-06-19
申请号：PCT/GB2007004662
申请日：2007-12-06
申请人： SYNGENTA LTD , CARTER NEIL BRIAN , CORDINGLEY MATTHEW ROBERT , CROWLEY PATRICK JEFF , TURNBULL MICHAEL DRYSDALE
发明人： CARTER NEIL BRIAN , CORDINGLEY MATTHEW ROBERT , CROWLEY PATRICK JEFF , TURNBULL MICHAEL DRYSDALE
IPC分类号： C07D471/04 , A01N43/90 , A01P13/00
CPC分类号： C07D471/04 , A01N43/90
摘要： The present invention relates to compounds of formula (I): wherein R 1 , R 2 , R 3 , R 4 and R 5 are as defined in claim 1; or a salt or N-oxide thereof. Furthermore, the present invention relates to processes for preparing compounds of formula (I), to methods of controlling plants and compositions comprising compounds of formula (I).
摘要翻译：本发明涉及式（I）的化合物：其中R 1，R 2，R 3，R 4， SUP＆gt;和R＆gt; 5如权利要求1中所定义; 或其盐或N-氧化物。此外，本发明涉及制备式（I）化合物的方法，涉及含有式（I）化合物的植物和组合物的控制方法。

16. 发明申请

WO2008009908A1 PYRIDO [2, 3-B] PYRAZINE DERIVATIVES USEFUL AS HERBICIDAL COMPOUNDS 审中-公开
标题翻译：吡咯并[2,3-B]吡嗪衍生物有效用作除草剂化合物
公开(公告)号：WO2008009908A1
公开(公告)日：2008-01-24
申请号：PCT/GB2007/002668
申请日：2007-07-16
申请人： SYNGENTA LIMITED , CARTER, Neil, Brian , CORDINGLEY, Matthew, Robert , CROWLEY, Patrick, Jeff , TURNBULL, Michael, Drysdale
发明人： CARTER, Neil, Brian , CORDINGLEY, Matthew, Robert , CROWLEY, Patrick, Jeff , TURNBULL, Michael, Drysdale
IPC分类号： C07D471/04 , A01N43/60
CPC分类号： C07D471/04 , A01N43/90
摘要： The present invention relates to a method of controlling plants or inhibiting plant growth which comprises applying to the plants or to the locus thereof a herbicidally effective amount of a compound of formula (I) wherein R 1 , R 2 , R 3 , R 4 and R 5 are as defined in claim 1; or salts or N-oxides thereof. Furthermore, the present invention relates to processes for preparing compounds of formula (I), to herbicidal compositions comprising compounds of formula (I) and to certain novel pyrido[2,3-b]pyrazines.
摘要翻译：本发明涉及一种控制植物或抑制植物生长的方法，包括向植物或其基因座施用除草有效量的式（I）化合物，其中R 1，R 2， R 2，R 3，R 4和R 5如权利要求1中所定义。或其盐或N-氧化物。此外，本发明涉及制备式（I）化合物的方法，其包含式（I）化合物和某些新的吡啶并[2,3-b]吡嗪的除草组合物。

17. 发明申请

WO1994027942A1 PREPARATION OF HALOGENATED ALCOHOLS 审中-公开
标题翻译：氢化酒精的制备
公开(公告)号：WO1994027942A1
公开(公告)日：1994-12-08
申请号：PCT/GB1994001140
申请日：1994-05-25
申请人： ZENECA LIMITED , BOWDEN, Martin, Charles , TURNBULL, Michael, Drysdale
发明人： ZENECA LIMITED
IPC分类号： C07C29/38
CPC分类号： C07C29/38 , C07C33/423
摘要： The invention discloses a process for the preparation of a halogenated alcohol of the formula (I): CF3-CXC1-CH(OH)-CH=C(CH3)2 wherein X is bromo or chloro which comprises reacting a compound of the formula (II): CF3CHXC1 with 3-methylbut-2-en-1-al in the presence of a strong base and an inert solvent. The products are useful intermediates for the manufacture of insecticides. 5-Bromo-5-chloro-4-hydroxy-2-methyl-6,6,6-trifluorohex-2-ene is new.
摘要翻译：本发明公开了制备式（I）的卤代醇的方法：CF 3 -S CXCl-CH（OH）-CH = C（CH 3）2，其中X是溴或氯，其包括使式 II）：具有3-甲基丁-2-烯-1-醇的CF 3 CHXCl在强碱和惰性溶剂的存在下反应。该产品是制造杀虫剂的有用中间体。 5-溴-5-氯-4-羟基-2-甲基-6,6,6-三氟己-2-烯是新的。

18. 发明申请

WO2008071918A8 PYRIDO-PYRAZINE DERIVATIVES USEFUL AS HERBICIDAL COMPOUNDS 审中-公开
公开(公告)号：WO2008071918A8
公开(公告)日：2008-06-19
申请号：PCT/GB2007/004662
申请日：2007-12-06
申请人： SYNGENTA LIMITED , CARTER, Neil, Brian , CORDINGLEY, Matthew, Robert , CROWLEY, Patrick, Jelf , TURNBULL, Michael, Drysdale
发明人： CARTER, Neil, Brian , CORDINGLEY, Matthew, Robert , CROWLEY, Patrick, Jelf , TURNBULL, Michael, Drysdale
IPC分类号： C07D471/04 , A01N43/90 , A01P13/00
摘要： The present invention relates to compounds of formula (I): wherein R 1 , R 2 , R 3 , R 4 and R 5 are as defined in claim 1; or a salt or N-oxide thereof. Furthermore, the present invention relates to processes for preparing compounds of formula (I), to methods of controlling plants and compositions comprising compounds of formula (I).

19. 发明申请

WO1996015672A1 FUNGICIDAL COMPOSITION 审中-公开
标题翻译：杀真菌剂
公开(公告)号：WO1996015672A1
公开(公告)日：1996-05-30
申请号：PCT/GB1995002576
申请日：1995-11-02
申请人： ZENECA LIMITED , TURNBULL, Michael, Drysdale , CROWLEY, Patrick, Jelf , CHRYSTAL, Ewan, James, Turner , CLOUGH, John, Martin , YOULE, David , BEAUTEMENT, Kevin , BARNETT, Susan, Patricia , PONSFORD, Roger, John , OUTRED, Dennis, James , MAMALIS, Patrick , HATTER, Glenn , SMITH, Peter, Duncan , BELLINI, Peter
发明人： ZENECA LIMITED
IPC分类号： A01N43/64
CPC分类号： C07D403/12 , A01N43/64 , C07D251/10 , C07D251/72 , C07F9/6521
摘要： A fungicidal composition comprising, as an active ingredient, a compound of formula (Ia) or (Ib) or a tautomer thereof, wherein R and R are, independently, hydrogen; C1-C6 alkyl, optionally substituted with OH or halo; C2-C6 alkenyl, optionally substituted with OH or halo; or R and R together form a 3 to 8 membered cycloalkyl or cycloalkenyl ring either of which is optionally substituted with C1-C6 alkyl, C2-C6 alkenyl, OH or halo; R is hydrogen, C1-C20 alkyl, C2-C20 alkenyl or C2-C20 alkynyl group, any of which is optionally substituted; R and R are, independently, hydrogen, CO2R , COR , CONR R , OCOR , CO2X, COX, SO2X or CONHX, wherein X is benzyl, phenyl, a 3 to 8 membered cycloalkyl, cycloalkenyl or saturated or unsaturated heterocyclic ring, or a fused ring system; R and R are, independently, hydrogen, C1-C8 alkyl, C2-C8 alkenyl, C1-C8 haloalkyl or C2-C8 haloalkenyl; or a salt or metal complex thereof; and a fungicidally acceptable carrier or diluent.
摘要翻译：一种杀真菌组合物，其包含作为活性成分的式（Ia）或（Ib）化合物或其互变异构体，其中R 1和R 2独立地是氢; 任选被OH或卤素取代的C 1 -C 6烷基; 任选被OH或卤素取代的C 2 -C 6烯基; 或R 1和R 2一起形成任选被C 1 -C 6烷基，C 2 -C 6烯基，OH或卤素取代的3至8元环烷基或环烯基环; R 3是氢，C 1 -C 20烷基，C 2 -C 20烯基或C 2 -C 20炔基，其中任何一个任选被取代; R 4和R 5独立地是氢，CO 2 R 9，COR 9，CONR 9 R 9，OCOR 9，CO 2 X，COX，SO 2 X或CONHX，其中X 是苄基，苯基，3至8元环烷基，环烯基或饱和或不饱和杂环，或稠环体系; R 9和R 9独立地是氢，C 1 -C 8烷基，C 2 -C 8烯基，C 1 -C 8卤代烷基或C 2 -C 8卤代烯基; 或其盐或金属络合物; 和杀真菌剂可接受的载体或稀释剂。

20. 发明申请

WO1996015671A1 HERBICIDES 审中-公开
标题翻译：除草剂
公开(公告)号：WO1996015671A1
公开(公告)日：1996-05-30
申请号：PCT/GB1995002575
申请日：1995-11-02
申请人： ZENECA LIMITED , TURNBULL, Michael, Drysdale , CROWLEY, Patrick, Jelf , CHRYSTAL, Ewan, James, Turner , CLOUGH, John, Martin , BRYAN, Ian, Bennett , BEAUTEMENT, Kevin , BARNETT, Susan, Patricia , PONSFORD, Roger, John , OUTRED, Dennis, James , MAMALIS, Patrick , HATTER, Glenn , SMITH, Peter, Duncan , BELLINI, Peter
发明人： ZENECA LIMITED
IPC分类号： A01N43/64
CPC分类号： C07D403/12 , A01N43/64 , C07D251/10 , C07D405/12 , C07F9/6521
摘要： Compositions containing 1,2-dihydro-1,3,5-triazines of general formulae (Ia) or (Ib), wherein R , R , R , R , R , R and R are various substituents, or their tautomers and salts and metal complexes thereof, have herbicidal activity and may be applied either pre- or post-emergence to control weeds. Some of the compounds of general formulae (Ia) and (Ib) are new.
摘要翻译：含有通式（Ia）或（Ib）的1,2-二氢-1,3,5-三嗪的组合物，其中R 1，R 2，R 3，R 4，R 4 R 5和R 5'是各种取代基，或它们的互变异构体及其盐和金属络合物，具有除草活性，并且可以在芽前或出苗后施用以控制杂草。一些通式（Ia）和（Ib）的化合物是新的。

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式