专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

2. 发明申请

US20060229206A1 Acylated thiosemicarbazides as herbicides 失效
标题翻译：酰化硫代氨基脲作为除草剂
公开(公告)号：US20060229206A1
公开(公告)日：2006-10-12
申请号：US11386499
申请日：2006-03-22
申请人： Shy-Fuh Lee , Vivian Du , Richard Anderson
发明人： Shy-Fuh Lee , Vivian Du , Richard Anderson
IPC分类号： A01N43/40 , A01N47/34 , A01N43/02 , C07D213/46 , C07C335/20
CPC分类号： A01N47/34 , C07C337/06 , C07D213/56
摘要： The present invention provides compounds of Formula I: wherein Ar1 is aryl or heteroaryl, Ar2 is aryl or heteroaryl, and R is a suitable organic group. Herbicidal composition comprising such active compounds, and methods for controlling undesirable plants by applying such compounds, are also described.
摘要翻译：本发明提供式I化合物：其中Ar 1为芳基或杂芳基，Ar 2为芳基或杂芳基，R为合适的有机基团。还描述了包含这种活性化合物的除草组合物，以及通过应用这些化合物来控制不期望的植物的方法。

3. 发明申请

US20030199579A1 Ectoparasitic insect pest controllers for animals and their usage 有权
标题翻译：用于动物的寄生虫害虫控制器及其用途
公开(公告)号：US20030199579A1
公开(公告)日：2003-10-23
申请号：US10399327
申请日：2003-05-21
发明人： Rikio Yamaguchi , Tetsuyoshi Nishimatsu , Kazuhiro Takagi
IPC分类号： A01N037/12 , A01N047/34 , A01N037/44 , A01N037/34
CPC分类号： A01N37/18 , A01N37/24 , A01N37/34 , A01N37/44 , A01N47/34 , A01N47/40 , C07C243/22 , C07C251/44 , C07C251/86 , C07C255/66 , C07C281/06 , C07C281/14 , C07C317/42 , C07C323/44 , C07C337/06 , C07C337/08
摘要： 1 Ectoparasitic insect pest controllers for animals, containing hydrazine derivatives of the general formula (I) as the active ingredient, and methods for application of the same: (I) nullwherein A is (II), (III), (IV), (V) (wherein R4 and R5 are each H, C1-6alkyl, or the like; and X is H, or one to five substituents selected from among halogeno and optionally halogenated C1-6alkyl groups); R1 is H or C1-6alkyl; R2 and R3 are each H, OH, C1-6alkyl, phenylcarbonyl, or the like; Y is H, or one to five substituents selected from among halogeno, nitro, and cyano; Z is halogeno, cyano, C1-6alkyl, or the like; and W is O or Snull. The insect pest controllers exert remarkable controlling effects on parasitic insect pests harmful to domestic or pet animals, e.g. fleas, lice, ticks.
摘要翻译：含有通式（I）的肼衍生物作为活性成分的动物的寄生虫害虫控制剂及其应用方法：（I）[其中A是（II），（III），（IV）， V）（其中R 4和R 5各自为H，C 1-6烷基等; X为H，或1至5个选自卤代和任意卤代的C 1-6烷基的取代基）; R 1是H或C 1-6烷基; R 2和R 3各自为H，OH，C 1-6烷基，苯基羰基等; Y是H或选自卤代，硝基和氰基的一至五个取代基; Z是卤代，氰基，C 1-6烷基等; W为O或S]。昆虫害虫控制剂对对家畜或宠物有害的寄生昆虫害虫具有显着的防治作用，跳蚤，虱子，蜱虫。

4. 发明申请

US20030194371A1 (Ethylene)-(propylene) - triaminepentaacetic acid derivatives, process for their production, and their use for the production of pharmaceutical agents 审中-公开
标题翻译：（乙烯） - （丙烯） - 三氨基五乙酸衍生物，其生产方法及其用于生产药剂
公开(公告)号：US20030194371A1
公开(公告)日：2003-10-16
申请号：US10191987
申请日：2002-07-10
申请人： Schering AG
发明人： Lutz Lehmann , Matthias Friebe , Christoph-Stephan Hilger , Ulrich Niedballa , Johannes Platzek , Bernd Raduchel
IPC分类号： A61K051/00 , A61K049/00 , C07F005/00 , C07H021/04
CPC分类号： C07D207/452 , C07C229/16 , C07C229/76 , C07C233/43 , C07C331/28 , C07C337/06 , C07C2601/08 , C07C2601/14
摘要： The invention relates to (ethylene)-(propylene)-triaminepentaacetic acid derivatives that are substituted on both the ethylene bridge and the propylene bridge, as well as conjugates of these compounds with biomolecules. The compounds and conjugates are suitable as agents for NMR diagnosis and radiodiagnosis as well as for radiotherapy.
摘要翻译：本发明涉及在乙烯桥和丙烯桥上取代的（乙烯） - （丙烯） - 三氨基五乙酸衍生物，以及这些化合物与生物分子的缀合物。化合物和缀合物适合作为核磁共振诊断和放射诊断以及放射治疗的试剂。

5. 发明申请

US20020026058A1 Method for producing triazolinthion derivatives 有权
标题翻译：三唑衍生物的制备方法
公开(公告)号：US20020026058A1
公开(公告)日：2002-02-28
申请号：US09795062
申请日：2001-02-26
发明人： Manfred Jautelat , Achim Hupperts , Reinhard Lantzsch
IPC分类号： C07D249/08
CPC分类号： C07D249/12 , C07C337/06
摘要： According to a novel process, it is possible to prepare triazolinethione derivatives of the formula 1 in which R1 and R2 are each as defined in the description by a) reacting hydrazine derivatives of the formula 2 nullor their acid addition salts with an inorganic or organic acid with thiocyanate of the formula 3 nullin which Y represents sodium, potassium or ammonium nullin the presence of a diluent and, if appropriate, in the presence of a catalyst and b) reacting the resulting thiosemicarbazide derivatives of the formula 4 nullwith formic acid, if appropriate in the presence of a catalyst and if appropriate in the presence of a diluent. The thiosemicarbazide derivatives of the formula (IV) are novel.
摘要翻译：根据新的方法，可以制备下式的三唑啉硫酮衍生物，其中R1和R2各自如说明书中所定义：a）使下式的肼衍生物或其酸加成盐与无机或有机酸与硫氰酸酯反应其中Y表示钠，钾或铵，在稀释剂存在下，如果合适的话，在催化剂存在下，和b）使所得到的硫代氨基脲衍生物与甲酸反应，如果合适的话，在催化剂和如果合适的话，在稀释剂存在下。式（IV）的硫代氨基脲衍生物是新颖的。

6. 发明授权

US5585468A Substituted thioureas as bifunctional chelators 失效
标题翻译：取代硫脲作为双功能螯合剂
公开(公告)号：US5585468A
公开(公告)日：1996-12-17
申请号：US204197
申请日：1994-06-27
申请人： Daniel J. Coughlin , Benjamin A. Belinka, Jr.
发明人： Daniel J. Coughlin , Benjamin A. Belinka, Jr.
IPC分类号： G01N33/58 , A61K39/44 , A61K47/48 , A61K51/00 , A61K51/08 , A61K51/10 , C07C335/06 , C07C335/14 , C07C335/16 , C07C335/22 , C07C337/06 , C07D207/44 , C07D207/452 , C07D213/34 , C07D213/71 , C09K3/00
CPC分类号： C07D207/452 , A61K47/48 , A61K51/082 , A61K51/088 , A61K51/1093 , C07C335/22 , C07C337/06 , C07D213/71 , A61K2121/00 , A61K2123/00
摘要： This invention relates to chelating agents useful for coupling metal ions to biologically active molecules. In particular, substantial thioureas for chelating metals such as technetium are provided that can be conjugated to a targeting molecule such as an antibody, a peptide or a protein.
摘要翻译： PCT No.PCT / US93 / 03208 Sec。 371日期1994年6月27日第 102（e）日期1994年6月27日PCT提交1993年4月8日PCT公布。出版物WO93 / 21151 日期：1993年10月28日本发明涉及用于将金属离子与生物活性分子偶联的螯合剂。特别地，提供了用于螯合金属例如锝的大量硫脲，其可以与靶向分子例如抗体，肽或蛋白质缀合。

7. 发明授权

US5527885A Bifunctional isothiocyanate derived thiocarbonyls as ligands for metal binding 失效
标题翻译：双官能异硫氰酸酯衍生的硫代羰基作为金属结合的配体
公开(公告)号：US5527885A
公开(公告)日：1996-06-18
申请号：US268445
申请日：1994-06-30
申请人： Daniel J. Coughlin , Benjamin A. Belinka, Jr.
发明人： Daniel J. Coughlin , Benjamin A. Belinka, Jr.
IPC分类号： G01N33/58 , A61K39/44 , A61K47/48 , A61K51/00 , A61K51/08 , A61K51/10 , C07C335/06 , C07C335/14 , C07C335/16 , C07C335/22 , C07C337/06 , C07D207/44 , C07D207/452 , C07D213/34 , C07D213/71 , C09K3/00 , A61K35/14
CPC分类号： C07D207/452 , A61K47/48 , A61K51/082 , A61K51/088 , A61K51/1093 , C07C335/22 , C07C337/06 , C07D213/71 , A61K2121/00 , A61K2123/00
摘要： This invention relates to chelating agents useful for coupling metal ions to biologically active molecules. In particular, isothiocyanate derived thiocarbonyls for chelating metals such as technetium are provided that can be conjugated to a targeting molecule such as an antibody, a peptide or a protein.
摘要翻译：本发明涉及用于将金属离子与生物活性分子偶联的螯合剂。特别地，提供了用于螯合金属例如锝的异硫氰酸酯衍生的硫代羰基，其可以与靶向分子例如抗体，肽或蛋白质缀合。

8. 发明授权

US4294985A Production of thiocarbohydrazide on a commercial scale 失效
标题翻译：以商业规模生产硫代碳酰肼
公开(公告)号：US4294985A
公开(公告)日：1981-10-13
申请号：US48856
申请日：1979-06-15
申请人： Gunther Cramm , Karl H. Blocher
发明人： Gunther Cramm , Karl H. Blocher
IPC分类号： C07C327/56 , C01B20060101 , C07C20060101 , C07C67/00 , C07C325/00 , C07C335/40 , C07C337/06 , C07C159/00
CPC分类号： C07C337/06
摘要： In the production of thiocarbohydrazide by reacting hydrazine hydrate with carbon disulphide in the presence of water to form in a first stage hydrazinium dithiocarbazinate, subsequently thermally decomposing the hydrazinium dithiocarbazinate in a second stage to form thiocarbohydrazide, and recovering the thiocarbohydrazide from the reaction medium, the improvement which comprises effecting the entire reaction in the mother liquor of a preceding batch, carrying out the first reaction stage at a temperature between about 25.degree. C. and 45.degree. C., with injection of carbon disulphide below the surface of the reaction mixture; carrying out the second stage at about 62.degree. to 65.degree. C. without prior isolation of the intermediate product; filtering off the thiocarbohydrazide formed after cooling, separating the amount of mother liquor in excess of that required for the next batch, and feeding the balance of the mother liquor to the next batch. The excess mother liquor not required for the next batch is heated to about 70.degree. to 75.degree. C., and after separating off the thiocarbohydrazide, the remaining mother liquor is subjected to combustion.
摘要翻译：在硫代碳酰肼的制备中，通过在水存在下使水合肼与二硫化碳反应，在第一阶段中形成二硫代肼基肼，然后在第二阶段热分解二硫代肼基肼，形成硫代碳酰肼，并从反应介质中回收硫代碳酰肼，其包括进行前一批次的母液中的整个反应，在约25℃至45℃的温度下进行第一反应阶段，在反应混合物的表面下注入二硫化碳; 在大约62°至65℃进行第二阶段，而不预先分离中间产物; 过滤冷却后形成的硫代碳酰肼，将母液的量分离超过下一批所需的母液量，并将母液的余量送入下一批。将下一批不需要的过量母液加热至约70℃至75℃，分离硫代碳酰肼后，将剩余的母液进行燃烧。

9. 发明授权

US3929877A Process for the production of thiocarbohydrazide 失效
标题翻译：硫代碳酰肼的生产工艺
公开(公告)号：US3929877A
公开(公告)日：1975-12-30
申请号：US52493174
申请日：1974-11-18
申请人： AKZO N V OF ARNHEM HOLLAND
发明人： TOTH ANTON , RUPP HANS-DIETER , MEYER GERHARD
IPC分类号： C07C337/06 , C07C67/00 , C07C325/00 , C07C157/02
CPC分类号： C07C337/06
摘要： Process for producing thiocarbohydrazide in high yields above 75%, especially above 90%, by heating hydrazine-dithiocarbazinate at about 20*-85*C. in an aqueous or a water-free hydrazine hydrate containing hydrogen sulfide, for example in an amount of at least about 1% and preferably about 2 to 36% by weight H2S. The heating or thermal treatment is carried out at about 20*C. to 85*C., preferably 50*-80*C. and especially 72*-78*C. Almost quantitative yields can be achieved in producing the thiocarbohydrazide which is of known utility, especially in producing biocides for the agricultural industry.
摘要翻译：通过在含有硫化氢的含水或无水肼水合物中，在约20-85℃加热肼二硫代肼基甲酸酯，生产硫代碳酰肼的高产率高于75％，特别是高于90％的方法，至少约1％，优选约2至36％H 2 S。加热或热处理在约20℃至85℃，优选50-80℃，特别是72℃-78℃下进行。在制备硫代碳酰肼中可以实现几乎定量的产率特别是生产农业生物杀虫剂。

10. 发明授权

US2731496A Method of making thiosemicarbazide 失效
标题翻译：制备硫代氨基脲的方法
公开(公告)号：US2731496A
公开(公告)日：1956-01-17
申请号：US33384053
申请日：1953-01-28
申请人： MONSANTO CHEMICALS
发明人： TAYLOR GEORGE E
CPC分类号： C07C337/06

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式