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1. 发明申请

US20110224241A1 ISOTHIAZOLE AND PYRAZOLE DERIVATIVES AS FUNGICIDES 失效
标题翻译：异噻唑和吡唑衍生物作为杀真菌剂
公开(公告)号：US20110224241A1
公开(公告)日：2011-09-15
申请号：US12668435
申请日：2008-07-09
申请人： Peter Ackermann , Carla Bobbio , Camilla Corsi , Josef Ehrenfreund , Ann Monica McGinley , Andreas Verras , Ruud Titulaer
发明人： Peter Ackermann , Carla Bobbio , Camilla Corsi , Josef Ehrenfreund , Ann Monica McGinley , Andreas Verras , Ruud Titulaer
IPC分类号： A61K31/506 , C07D417/06 , A61K31/4439 , A01N43/80 , A61P31/10 , A01P3/00 , C07D401/06 , A01N43/56
CPC分类号： C07D417/06 , A01N43/56 , A01N43/80 , C07D401/06 , C07D417/14
摘要： The present invention relates to compounds of Formula (I) wherein R1, R2, R3 or R4 are as defined in claim 1 or a salt or N-oxide thereof and their use in methods for the control and/or prevention of fungal infection, particularly in plants. The compounds claimed are isothiazole and pyrazole derivatives.
摘要翻译：本发明涉及其中R 1，R 2，R 3或R 4如权利要求1所定义的式（I）化合物或其盐或N-氧化物及其在控制和/或预防真菌感染的方法中的用途，特别是在植物中。所要求的化合物是异噻唑和吡唑衍生物。

2. 发明授权

US08377953B2 Isothiazole and pyrazole derivatives as fungicides 失效
标题翻译：异噻唑和吡唑衍生物作为杀真菌剂
公开(公告)号：US08377953B2
公开(公告)日：2013-02-19
申请号：US12668435
申请日：2008-07-09
申请人： Peter Ackermann , Carla Bobbio , Camilla Corsi , Ann Monica McGinley , Andreas Verras , Ruud Titulaeu , Josef Ehrenfreund
发明人： Peter Ackermann , Carla Bobbio , Camilla Corsi , Ann Monica McGinley , Andreas Verras , Ruud Titulaeu , Josef Ehrenfreund
IPC分类号： A61K31/506 , A61K31/4439 , A01N43/56 , A01N43/80 , A01P3/00 , A61P31/10 , C07D401/06 , C07D417/06
CPC分类号： C07D417/06 , A01N43/56 , A01N43/80 , C07D401/06 , C07D417/14
摘要： The present invention relates to compounds of Formula (I) wherein R1, R2, R3 or R4 are as defined in claim 1 or a salt or N-oxide thereof and their use in methods for the control and/or prevention of fungal infection, particularly in plants. The compounds claimed are isothiazole and pyrazole derivatives.
摘要翻译：本发明涉及其中R 1，R 2，R 3或R 4如权利要求1所定义的式（I）化合物或其盐或N-氧化物及其在控制和/或预防真菌感染的方法中的用途，特别是在植物中。所要求的化合物是异噻唑和吡唑衍生物。

3. 发明申请

US20100292258A1 SUBSTITUTED AROMATIC HETEROCYCLIC COMPOUNDS AS FUNGICIDES 审中-公开
标题翻译：取代的芳香杂环化合物作为防腐剂
公开(公告)号：US20100292258A1
公开(公告)日：2010-11-18
申请号：US12601317
申请日：2008-06-16
申请人： Peter Ackermann , Carla Bobbio , Camilla Corsi , Josef Ehrenfreund , Ann Monica McGinley
发明人： Peter Ackermann , Carla Bobbio , Camilla Corsi , Josef Ehrenfreund , Ann Monica McGinley
IPC分类号： A61K31/506 , C07D401/06 , C07D403/06 , A61K31/444 , A61K31/4439 , A01N43/54 , A01N43/40 , A01P3/00 , A61P31/10
CPC分类号： C07D401/06 , C07D403/06 , C07D405/14 , C07D409/14
摘要： The present invention relates to compounds of formula (I) wherein R1, R2, R3, R4, R5 and R6 are as defined in claim 1 or a salt or N-oxide thereof and their use in methods for the control and/or prevention of fungal infection, particularly in plants.
摘要翻译：本发明涉及其中R 1，R 2，R 3，R 4，R 5和R 6如权利要求1中所定义的式（I）化合物或其盐或N-氧化物及其在控制和/或预防真菌感染，特别是在植物中。

4. 发明授权

US08389442B2 N-phenyl-′(4-pyridyl)-azinyl!amine derivatives as plant protection agents 失效
标题翻译： N-苯基 - （4-吡啶基） - 嗪基胺衍生物作为植物保护剂
公开(公告)号：US08389442B2
公开(公告)日：2013-03-05
申请号：US10549486
申请日：2004-03-25
申请人： Peter Ackermann , Daniel Stierli , Martin Diggelmann , Fredrik Cederbaum , Jean Wenger , Ruud Titulaer
发明人： Peter Ackermann , Daniel Stierli , Martin Diggelmann , Fredrik Cederbaum , Jean Wenger , Ruud Titulaer
IPC分类号： A01N43/66 , A01N43/54 , A01N43/40 , C07D403/00 , C07D251/00 , C07D237/00 , C07D237/02 , C07D213/04
CPC分类号： C07D401/04 , A01N43/40 , A01N43/54 , A01N43/66 , C07D401/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14
摘要： The use of fungicidal compounds of formula Ij wherein A and A′ are both N or A and A′ are both CH or A is CH and A′ is N; j is 0 or 1 and the R groups are as defined in claim 1; their preparation and compositions 10 comprising the compounds.
摘要翻译：使用式Ij的杀真菌化合物，其中A和A'都是N或A，A'都是CH或A是CH，A'是N; j为0或1，R基团如权利要求1所定义; 它们的制备方法和包含该化合物的组合物10。

5. 发明申请

US20070032490A1 N-Phenyl-'(4-pyridyl)-azinyl!amine derivatives as plant protection agents 失效
标题翻译： N-苯基 - （4-吡啶基） - 嗪基胺衍生物作为植物保护剂
公开(公告)号：US20070032490A1
公开(公告)日：2007-02-08
申请号：US10549486
申请日：2004-03-25
申请人： Peter Ackermann , Daniel Stierli , Martin Diggelmann , Fredrik Cederbaum , Jean Wenger , Ruud Titulaer
发明人： Peter Ackermann , Daniel Stierli , Martin Diggelmann , Fredrik Cederbaum , Jean Wenger , Ruud Titulaer
IPC分类号： A01N43/54 , A01N43/40 , A01N43/66
CPC分类号： C07D401/04 , A01N43/40 , A01N43/54 , A01N43/66 , C07D401/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14
摘要： The use of fungicidal compounds of formula Ij wherein A and A′ are both N or A and A′ are both CH or A is CH and A′ is N; j is 0 or 1 and the R groups are as defined in claim 1; their preparation and compositions 10 comprising the compunds.
摘要翻译：使用式I的杀真菌化合物其中A和A'都是N或A，A'都是CH或A是CH，A'是N; j为0或1，R基团如权利要求1所定义; 它们的制备方法和组合物10包括该组合物。

6. 发明授权

US5420301A Process for the preparation of substituted difluorobenzo-1,3-dioxoles 失效
标题翻译：制备取代的二氟苯-1,3-二氧杂环戊烯的方法
公开(公告)号：US5420301A
公开(公告)日：1995-05-30
申请号：US147617
申请日：1993-11-05
申请人： Peter Ackermann , Hans-Ruedi Kanel , Bruno Schaub
发明人： Peter Ackermann , Hans-Ruedi Kanel , Bruno Schaub
IPC分类号： A61K31/33 , C07D317/06 , C07D317/46 , C07D405/04 , C07F1/00 , C07F1/02 , C07F3/00 , C07F5/02 , C07F7/08 , C07F7/10 , C07F19/00 , C07D317/50 , C07D317/52 , C07D317/54
CPC分类号： C07D405/04 , C07D317/46 , C07F1/00 , C07F1/02 , C07F19/00 , C07F3/00 , C07F5/025 , C07F7/0814 , C07F7/10 , Y02P20/55
摘要： The reaction of 2,2-difluorobenzo-1,3-dioxole with (a) an alkali metal or an alkali metal compound and then (b) a compound R.sup.1 -Z.sup.1 in which Z.sup.1 is a leaving group, or with an aldehyde produces compounds of formula I ##STR1## wherein R.sup.1 is --OH, --SH, --CHO, --CN, --COOH, --B(OH).sub.2, --COX, with X being Cl or Br, or is --COOR.sup.2, --SiR.sub.3.sup.2 or --B(OR.sup.2).sub.2, with R.sup.2 being a C.sub.1 -C.sub.12 alcohol moiety without the hydroxy group, wherein R.sup.1 is further --C.sub.n H.sub.2n COOR.sup.2, with n being an integer from 1 to 4, or linear or branched C.sub.1 -C.sub.12 hydroxyalkyl which is unsubstituted or is substituted by --F, --CN, C.sub.1 -C.sub.6 alkoxy, phenyl, fluorophenyl, C.sub.1 -C.sub.4 alkoxy-phenyl, C.sub.1 -C.sub.4 alkylthio-phenyl, C.sub.1 -C.sub.4 alkyl-phenyl, C.sub.1 -C.sub.4 fluoroalkyl-phenyl, nitrophenyl or by cyanophenyl, or wherein R.sup.1 is a benzyl alcohol which is unsubstituted or is substituted by F, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 alkylthio, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 fluoroalkyl, nitro or by cyano, or is C.sub.1 -C.sub.12 acyl, or wherein R.sup.1 is a radical of formula II ##STR2## wherein R.sup.5 is --CN, --CF.sub.3, --COOR.sup.2, --CONH.sup.2, --CO--NHR.sup.2 or --CONR.sub.2.sup.2, R.sup.3 and R.sup.4 are a direct bond or each is H, or R.sup.3 is H and R.sup.4 independently has the meanings of R.sup.5, or R.sup.3 and R.sup.4 together are --CH.sub.2 --NR.sup.6 --CH.sub.2 --, --CH.sub.2 --NR.sup.6 --CO-- or --CO--NR.sup.6 --CO-- wherein R.sup.6 is the radical of a removable protecting group, or wherein further R.sup.1 is a radical of formula III ##STR3## Insecticides or fungicides can be prepared from the compounds of formula I.3-(2,2-difluorobenzodioxol-4-yl)-4-cyanopyrrole can be prepared by reacting 4-metallo-2,2-difluorobenzodioxole (III) with an unsaturated nitrile and then with a sulfonylmethyl isocyanide in a one-pot process. The compounds III are novel intermediates.
摘要翻译： 2,2-二氟苯-1,3-二氧杂环戊烯与（a）碱金属或碱金属化合物反应，然后（b）其中Z 1为离去基团的化合物R1-Z1或与醛反应生成化合物其中R 1是-OH，-SH，-CHO，-CN，-COOH，-B（OH）2，-COX，X是Cl或Br，或者是-COOR 2， - SiR 32或-B（OR 2）2，其中R 2是没有羟基的C 1 -C 12醇部分，其中R 1还是-C n H 2n NOR 2，n是1至4的整数，或未被取代的直链或支链C 1 -C 12羟基烷基被-F，-CN，C 1 -C 6烷氧基，苯基，氟苯基，C 1 -C 4烷氧基 - 苯基，C 1 -C 4烷硫基 - 苯基，C 1 -C 4烷基 - 苯基，C 1 -C 4氟烷基 - 苯基，硝基苯基或氰基苯基取代，或其中R 1为苄基醇，其未被取代或被F，C 1 -C 4烷氧基，C 1 -C 4烷硫基，C 1 -C 4烷基，C 1 -C 4氟烷基，硝基或氰基取代，或者是C 1 -C 12酰基，或其中R 1是式II基团。（II）其中R5是-CN，-CF3，-COOR2，-CONH2，-CO-NHR 2或-CONR 22，R 3和R 4是直接键或各自为H或R 3为H且R 4独立地具有R 5的含义，或者R 3和R 4一起为-CH 2 -NR 6 -CH 2 - ， - CH 2 -NR 6 -CO - 或-CO-NR 6 -CO-，其中R 6是可除去的保护基的基团，或其中R 1是式III的基团由式I化合物制备。3-（2,2-二氟苯并二氧杂环戊烯-4-基） 4-氰基吡咯可以通过4-金属-2,2-二氟苯并二氧杂环戊烯（III）与不饱和腈然后与一种磺酰基甲基异氰化物反应来制备。化合物III是新的中间体。

7. 发明授权

US4822806A .alpha.-methyl-(6-phenoxy)-2-picolyl cyclopropanecaraboxylates having pesticidal activity 失效
标题翻译：具有杀虫活性的α-甲基 - （6-苯氧基）-2-甲基吡咯烷基环丙烷甲醛
公开(公告)号：US4822806A
公开(公告)日：1989-04-18
申请号：US2370
申请日：1987-01-12
申请人： Peter Ackermann
发明人： Peter Ackermann
IPC分类号： A01N53/00 , A01N53/08 , C07D213/64 , C07D213/647 , A01N43/40
CPC分类号： C07D213/647 , A01N53/00
摘要： The invention relates to .alpha.-methyl-(6-phenoxy)-2-picolyl cyclopropanecarboxylates of the formula ##STR1## wherein X.sub.1 is methyl or halogen,R.sub.1 is hydrogen or halogen, andR.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 alkylthio, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 haloalkoxy, C.sub.1 -C.sub.4 haloalkylthio, C.sub.2 -C.sub.4 alkenyl, C.sub.2 -C.sub.4 alkynyl, nitro or cyano.The invention also relates to the preparation of these esters and to the use thereof in pest control.
摘要翻译：本发明涉及式（I）的α-甲基 - （6-苯氧基）-2-甲基吡咯烷基环丙烷羧酸酯，其中X 1是甲基或卤素，R 1是氢或卤素，R 2是氢，卤素，C 1 -C 4烷基 C1-C4烷氧基，C1-C4烷硫基，C1-C4卤代烷基，C1-C4卤代烷氧基，C1-C4卤代烷硫基，C2-C4链烯基，C2-C4炔基，硝基或氰基。本发明还涉及这些酯的制备及其在害虫防治中的应用。

8. 发明授权

US4786654A Substituted benzylcyclopropylmethyl ethers 失效
标题翻译：取代的苄基环丙基甲基醚
公开(公告)号：US4786654A
公开(公告)日：1988-11-22
申请号：US53911
申请日：1987-05-26
申请人： Laurenz Gsell , Peter Ackermann
发明人： Laurenz Gsell , Peter Ackermann
IPC分类号： C07C41/01 , A01N31/14 , A01N31/16 , C07C41/00 , C07C43/29 , C07C67/00 , C07C313/00 , C07C323/20 , C07C147/06 , C07C149/34
CPC分类号： C07C43/29 , A01N31/14 , A01N31/16
摘要： There are disclosed novel unsubstituted or substituted phenoxyfluorobenzyltetramethylcyclopropylmethyl ethers of formula ##STR1## wherein Y is hydrogen, halogen, C.sub.1 -C.sub.4 alkyl or C.sub.1 -C.sub.4 alkyl which is substituted by 1 to 9 halogen atoms, C.sub.1 -C.sub.4 alkoxy or C.sub.1 -C.sub.4 alkoxy which is substituted by 1 to 9 halogen atoms, C.sub.1 -C.sub.4 alkylthio or C.sub.1 -C.sub.4 alkylthio which is substituted by 1 to 9 halogen atoms, or is C.sub.2 -C.sub.4 alkenyl or C.sub.2 -C.sub.4 alkynyl and their benzyl ether intermediates of formula IV ##STR2## wherein X is halogen or p-tosyl. Also disclosed is a process for the preparation of these compounds and compositions containing them for use in pest control, especially for controlling insects that attack plants and animals, in particular their larval stages. The novel compounds are particularly effective against plant-destructive insects in rice crops.
摘要翻译：公开了式（I）的新的未取代或取代的苯氧基氟苄基四甲基环丙基甲基醚，其中Y是氢，卤素，C 1 -C 4烷基或被1至9个卤素原子取代的C 1 -C 4烷基，C 1 -C 4烷氧基或C 1 -C 4烷氧基，被1至9个卤素原子取代，被1至9个卤素原子取代的C 1 -C 4烷硫基或C 1 -C 4烷硫基，或者是C 2 -C 4烯基或C 2 -C 4炔基及其式IV的苄基醚中间体其中X 是卤素或对甲苯磺酰基。还公开了一种用于制备这些化合物和含有它们的组合物用于病虫害防治的方法，特别是用于防治攻击植物和动物，特别是其幼虫期的昆虫。新型化合物对水稻作物中的植物性破坏性昆虫特别有效。

9. 发明授权

US4782087A Insecticidal prop-1-ynyl-3-phenoxybenzyl-2,2-dimethyl-3-(2,2-dihalovinyl)-cyclopropan e-1-carboxylates 失效
标题翻译：杀虫剂丙-1-炔基-3-苯氧基苄基-2,2-二甲基-3-（2,2-二卤乙烯基） - 环丙烷-1-羧酸酯
公开(公告)号：US4782087A
公开(公告)日：1988-11-01
申请号：US501457
申请日：1983-06-06
申请人： Saleem Farooq , Peter Ackermann , Jozef Drabek , Laurenz Gsell , Odd Kristiansen , Rudolf Wehrli
发明人： Saleem Farooq , Peter Ackermann , Jozef Drabek , Laurenz Gsell , Odd Kristiansen , Rudolf Wehrli
IPC分类号： A01N53/00 , A01N53/08 , C07C41/30 , C07C43/295 , C07C69/743
CPC分类号： A01N53/00 , C07C41/30 , C07C69/743 , C07C2101/02
摘要： Prop-1-ynyl-3-phenoxybenzyl-2,2-dimethyl-3-(2',2'-dihalovinyl)-cyclopropane-1-carboxylates of the formula ##STR1## in which X.sub.1 if fluorine, chlorine or bromine, and their use in combating pests.
摘要翻译：具有式“IMAGE”的丙-1-炔基-3-苯氧基苄基-2,2-二甲基-3-（2'，2'-二卤乙烯基） - 环戊烷-1-羧酸酯，其中如果氟，氯或溴，及其在防治害虫方面的应用。

10. 发明授权

US4618615A Certain 6-phenoxy-2-pyridinyl-.alpha.-methyl-methylene esters of .alpha.-cyclopropyl-.alpha.-phenyl-acetic acid derivatives and their use for controlling pests 失效
标题翻译： α-环丙基-α-苯基 - 乙酸衍生物的某些6-苯氧基-2-吡啶基-α-甲基 - 亚甲基酯及其用于防治害虫
公开(公告)号：US4618615A
公开(公告)日：1986-10-21
申请号：US549149
申请日：1983-11-07
申请人： Peter Ackermann , Laurenz Gsell , Boris Kohler
发明人： Peter Ackermann , Laurenz Gsell , Boris Kohler
IPC分类号： A01N53/00 , C07D213/64 , C07D213/647 , C07D491/056 , A01N43/40
CPC分类号： C07D213/647 , A01N53/00
摘要： .alpha.-Cyclopropyl-.alpha.-phenylacetate and salts thereof, corresponding to the formula ##STR1## wherein R.sub.1 is hydrogen, methyl, cyano or ethinyl,X.sub.1 is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl, C.sub.1 -C.sub.5 -haloalkyl or C.sub.1 -C.sub.5 -alkoxy,X.sub.2 is hydrogen, halogen or C.sub.1 -C.sub.5 -alkyl, or together with X.sub.1 is methylenedioxy, andX.sub.3 and X.sub.4 are hydrogen or halogen.Processes for producing these .alpha.-cyclopropyl-.alpha.-phenylacetates and their use for controlling pests are described.
摘要翻译： α-环丙基-α-苯基乙酸酯及其盐，其对应于其中R 1是氢，甲基，氰基或乙炔基的式（I），X 1是氢，卤素，C 1 -C 5 - 烷基，C 1 -C 5 - 卤代烷基或 C 1 -C 5 - 烷氧基，X 2为氢，卤素或C 1 -C 5 - 烷基，或与X 1一起为亚甲二氧基，且X 3和X 4为氢或卤素。描述了制备这些α-环丙基-α-苯乙酸酯的方法及其用于防治害虫的用途。

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