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1. 发明申请

US20150183785A1 ANTIPARISITIC DIHYDROAZOLE COMPOUNDS AND COMPOSITIONS COMPRISING SAME 有权
标题翻译：抗生素二氢化合物及其组合物
公开(公告)号：US20150183785A1
公开(公告)日：2015-07-02
申请号：US14658668
申请日：2015-03-16
申请人： MERIAL, INC.
发明人： Loic Patrick Le Hir de Fallois , Hyoung Ik Lee , Douglas Edward Wilkinson , Brent Christopher Beck
IPC分类号： C07D471/04 , A01N43/90
CPC分类号： C07D471/04 , A01N43/80 , A01N43/90 , A61K31/365 , A61K31/437 , A61K31/495 , A61K38/05 , A61K45/06 , C07K5/06 , A61K2300/00
摘要： The present invention relates to novel dihydroazole of formula (I) and salts thereof: Wherein R1, A1, A2, G, X and Y are as defined in the description, compositions thereof, processes for their preparation and their uses to prevent or treat parasitic infections or infestations in animals and as pesticides.
摘要翻译：本发明涉及式（I）的新型二氢唑及其盐：其中R1，A1，A2，G，X和Y如说明书中所定义，其组成，其制备方法及其用于预防或治疗寄生虫感染或感染动物和农药。

2. 发明申请

US20180362589A1 ANTHELMINTIC DEPSIPEPTIDE COMPOUNDS 审中-公开
公开(公告)号：US20180362589A1
公开(公告)日：2018-12-20
申请号：US16111027
申请日：2018-08-23
申请人： MERIAL INC.
发明人： Loic Le Hir de Fallois , Greg Pacofsky , Alan Long , Charles Meng , Hyoung Ik Lee , Cyprian O. Ogbu
IPC分类号： C07K11/02 , C07D273/00
摘要： The present invention provides cyclic depsipeptide compounds of formula (I) and compositions comprising the compounds that are effective against parasites that harm animals. The compounds and compositions may be used for combating parasites in or on mammals and birds. The invention also provides for an improved method for eradicating, controlling and preventing parasite infestation in birds and mammals.

3. 发明授权

US10081656B2 Anthelmintic depsipeptide compounds 有权
公开(公告)号：US10081656B2
公开(公告)日：2018-09-25
申请号：US15160577
申请日：2016-05-20
申请人： MERIAL INC.
发明人： Loic Le Hir de Fallois , Greg Pacofsky , Alan Long , Charles Meng , Hyoung Ik Lee , Cyprian O. Ogbu
IPC分类号： A61P33/00 , C07K11/02 , A01N43/72 , C07D273/00 , A61K38/00
CPC分类号： C07K11/02 , A01N43/72 , A61K38/00 , C07D273/00 , A01N37/46 , A01N43/90
摘要： The present invention provides cyclic depsipeptide compounds of formula (I) and compositions comprising the compounds that are effective against parasites that harm animals. The compounds and compositions may be used for combating parasites in or on mammals and birds. The invention also provides for an improved method for eradicating, controlling and preventing parasite infestation in birds and mammals.

4. 发明申请

US20170022197A1 ANTIPARISITIC DIHYDROAZOLE COMPOUNDS AND COMPOSITIONS COMPRISING SAME 有权
标题翻译：抗生素二氢化合物及其组合物
公开(公告)号：US20170022197A1
公开(公告)日：2017-01-26
申请号：US15191163
申请日：2016-06-23
申请人： MERIAL, INC.
发明人： Loic Patrick Le Hir de Fallois , Hyoung Ik Lee , Douglas Edward Wilkinson , Brent Christopher Beck
IPC分类号： C07D471/04 , A61K31/437 , A61K38/05 , C07K5/06 , A01N43/90
CPC分类号： C07D471/04 , A01N43/80 , A01N43/90 , A61K31/365 , A61K31/437 , A61K31/495 , A61K38/05 , A61K45/06 , C07K5/06 , A61K2300/00
摘要： The present invention relates to novel dihydroazole of formula (I) and salts thereof: Wherein R1, A1, A2, G, X and Y are as defined in the description, compositions thereof, processes for their preparation and their uses to prevent or treat parasitic infections or infestations in animals and as pesticides.
摘要翻译：其中R1，A1，A2，G，X和Y如说明书中所定义，其组合物，其制备方法及其用于预防或治疗动物和农药中的寄生虫感染或侵染的用途。

5. 发明申请

US20170233438A1 ANTHELMINTIC DEPSIPEPTIDE COMPOUNDS 审中-公开
公开(公告)号：US20170233438A1
公开(公告)日：2017-08-17
申请号：US15378219
申请日：2016-12-14
申请人： MERIAL INC.
发明人： Loic Le Hir de Fallois , Greg Pacofsky , Alan Long , Charles Q. Meng , Hyoung Ik Lee
IPC分类号： C07K11/02 , A61K45/06 , A61K38/15
CPC分类号： C07K11/02 , A01N43/72 , A61K38/15 , A61K45/06 , C07D273/00 , C07D413/14
摘要： The present invention provides cyclic depsipeptide compounds of formula (I) and compositions comprising the compounds that are effective against parasites that harm animals, including humans. The compounds and compositions may be used for combating parasites in or on animals including mammals and birds. The invention also provides for an improved method for eradicating, controlling and preventing parasite infestation in animals, including birds and mammals.

6. 发明申请

US20170022253A1 ANTHELMINTIC DEPSIPEPTIDE COMPOUNDS 审中-公开
标题翻译：安全性杀虫剂化合物
公开(公告)号：US20170022253A1
公开(公告)日：2017-01-26
申请号：US15160577
申请日：2016-05-20
申请人： MERIAL INC.
发明人： Loic Le Hir de Fallois , Greg Pacofsky , Alan Long , Charles Meng , Hyoung Ik Lee , Cyprian O. Ogbu
IPC分类号： C07K11/02
CPC分类号： C07K11/02 , A01N43/72 , A61K38/00 , C07D273/00 , A01N37/46 , A01N43/90
摘要： The present invention provides cyclic depsipeptide compounds of formula (I) and compositions comprising the compounds that are effective against parasites that harm animals. The compounds and compositions may be used for combating parasites in or on mammals and birds. The invention also provides for an improved method for eradicating, controlling and preventing parasite infestation in birds and mammals.
摘要翻译：本发明提供式（I）的环状缩肽化合物和包含有效对抗伤害动物的寄生虫的化合物的组合物。化合物和组合物可用于对抗哺乳动物和鸟类中或哺乳动物上的寄生虫。本发明还提供了用于消除，控制和预防鸟类和哺乳动物中的寄生虫感染的改进方法。

7. 发明授权

US09376434B2 Antiparisitic dihydroazole compounds and compositions comprising same 有权
公开(公告)号：US09376434B2
公开(公告)日：2016-06-28
申请号：US14658668
申请日：2015-03-16
申请人： MERIAL, INC.
发明人： Loic Patrick Le Hir de Fallois , Hyoung Ik Lee , Douglas Edward Wilkinson , Brent Christopher Beck
IPC分类号： A61K31/495 , A61K31/365 , C07D471/04 , A01N43/90 , A01N43/80 , A61K31/437 , A61K38/05 , A61K45/06 , C07K5/06
CPC分类号： C07D471/04 , A01N43/80 , A01N43/90 , A61K31/365 , A61K31/437 , A61K31/495 , A61K38/05 , A61K45/06 , C07K5/06 , A61K2300/00
摘要： The present invention relates to novel dihydroazole of formula (I) and salts thereof: Wherein R1, A1, A2, G, X and Y are as defined in the description, compositions thereof, processes for their preparation and their uses to prevent or treat parasitic infections or infestations in animals and as pesticides.

8. 发明授权

US09776999B2 Antiparisitic dihydroazole compounds and compositions comprising same 有权
公开(公告)号：US09776999B2
公开(公告)日：2017-10-03
申请号：US15191163
申请日：2016-06-23
申请人： MERIAL, INC.
发明人： Loic Patrick Le Hir de Fallois , Hyoung Ik Lee , Douglas Edward Wilkinson , Brent Christopher Beck
IPC分类号： A61K31/495 , A61K31/365 , C07D471/04 , A01N43/90 , A01N43/80 , A61K31/437 , A61K38/05 , A61K45/06 , C07K5/06
CPC分类号： C07D471/04 , A01N43/80 , A01N43/90 , A61K31/365 , A61K31/437 , A61K31/495 , A61K38/05 , A61K45/06 , C07K5/06 , A61K2300/00
摘要： The present invention relates to novel dihydroazole of formula (I) and salts thereof: Wherein R1, A1, A2, G, X and Y are as defined in the description, compositions thereof, processes for their preparation and their uses to prevent or treat parasitic infections or infestations in animals and as pesticides.

9. 发明授权

US09339033B2 1-aryl-5-alkyl pyrazole derivative compounds, processes of making and methods of using thereof 有权
标题翻译： 1-芳基-5-烷基吡唑衍生物化合物，其制备方法及其使用方法
公开(公告)号：US09339033B2
公开(公告)日：2016-05-17
申请号：US14325761
申请日：2014-07-08
申请人： MERIAL, INC.
发明人： Loic Patrick Le Hir de Fallois , Hyoung Ik Lee , Philip Reid Timmons , William Glenn Cawthorne, Jr. , Adalberto Perez de Leon
IPC分类号： A01N43/56 , C07D401/04 , C07D231/18 , A01N47/02 , A61K31/415 , A61K31/4439 , A61K45/06 , A01N25/02
CPC分类号： A01N43/56 , A01N25/02 , A01N47/02 , A61K31/415 , A61K31/4439 , A61K45/06 , C07D231/18 , C07D401/04
摘要： Provided are 1-aryl-5-alkyl pyrazole compounds, of formula (I): wherein: R1 is hydrogen, cyano, halogen, R8, formyl, —C(O)R8, —C(O)OR8, —C(O)NR9R10, or —C(S)NH2; R2 is R8 or —S(O)mR11; R3 is methyl, ethyl or C1-C4 haloalkyl; R4, R5 and R7 are independently hydrogen, halogen, alkyl, haloalkyl, cyano or nitro; R6 is halogen, alkyl, haloalkyl, alkoxy, haloalkyloxy, cyano, nitro, —C(O)R12, —S(O)nR12 or SF5; Z is a nitrogen atom or C—R13; R8 is alkyl, haloalkyl, cycloalkyl or halocycloalkyl; R9 is hydrogen, alkyl, haloalkyl or alkoxy; R10 is hydrogen, alkyl, haloalkyl or alkoxy; R11 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl or cycloalkyl; R12 is alkyl or haloalkyl; R13 is hydrogen, halogen, cyano, nitro, alkyl, haloalkyl, alkoxy or haloalkoxy; m is 0, 1 or 2; and n is 0, 1 or 2; or a salt thereof, the method of making compounds of formula (I) and the use of these compounds against ectoparasites, endoparasites and pests.
摘要翻译：提供式（I）的1-芳基-5-烷基吡唑化合物：其中：R 1是氢，氰基，卤素，R 8，甲酰基，-C（O）R 8，-C（O）OR 8，-C ）NR 9 R 10或-C（S）NH 2; R2是R8或-S（O）mR11; R3是甲基，乙基或C1-C4卤代烷基; R4，R5和R7独立地是氢，卤素，烷基，卤代烷基，氰基或硝基; R 6是卤素，烷基，卤代烷基，烷氧基，卤代烷氧基，氰基，硝基，-C（O）R 12，-S（O）n R 12或SF 5; Z是氮原子或C-R13; R8是烷基，卤代烷基，环烷基或卤代环烷基; R9是氢，烷基，卤代烷基或烷氧基; R 10是氢，烷基，卤代烷基或烷氧基; R11是烷基，卤代烷基，烯基，卤代烯基，炔基，卤代炔基或环烷基; R12是烷基或卤代烷基; R 13是氢，卤素，氰基，硝基，烷基，卤代烷基，烷氧基或卤代烷氧基; m为0,1或2; 且n为0,1或2; 或其盐，制备式（I）化合物的方法以及这些化合物对外寄生虫，内寄生虫和害虫的用途。

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