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81. 发明申请

US20070265267A1 FUNGICIDAL COMPOSITIONS 有权
标题翻译：杀真菌剂
公开(公告)号：US20070265267A1
公开(公告)日：2007-11-15
申请号：US11696908
申请日：2007-04-05
申请人： Harald WALTER , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hans Tobler
发明人： Harald WALTER , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hans Tobler
IPC分类号： A01N43/56 , A01N43/40 , A01N43/52 , A01N43/78 , A01N43/84 , A01N43/653 , A01N43/54
CPC分类号： A01N43/56 , A01N45/02 , A01N37/34 , A01N37/38 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/653 , A01N43/84 , A01N43/90 , A01N47/24 , A01N61/00 , A01N2300/00
摘要： A method of controlling phytopathogenic diseases on useful plants or on propagation material thereof, which comprises applying to the useful plants, the locus thereof or propagation material thereof a combination of components A) and B) in a synergistically effective amount, wherein component A) is a compound of formula I wherein R1 is difluoromethyl or trifluoromethyl; Y is —CHR2— or and R2 is hydrogen or C1-C6alkyl; or a tautomer of such a compound; and component B) is a compound selected from compounds known for their fungicidal and/or insecticidal activity, is particularly effective in controlling or preventing fungal diseases of useful plants.
摘要翻译：一种在有用植物或繁殖材料上控制植物病原性疾病的方法，其包括以协同有效量施用于有用植物，其基因座或繁殖材料的组合物A）和B）的组合，其中组分A）为式I的化合物，其中R 1是二氟甲基或三氟甲基; Y是-CHR 2 - 或 - 或R 2是氢或C 1 -C 6烷基; 或这种化合物的互变异构体; 和组分B）是选自其杀真菌和/或杀虫活性已知的化合物的化合物，在控制或预防有用植物的真菌疾病方面特别有效。

82. 发明申请

US20060287328A1 Silicon compounds with microbiocidal activity 失效
公开(公告)号：US20060287328A1
公开(公告)日：2006-12-21
申请号：US10569343
申请日：2004-09-08
申请人： Josef Ehrenfreund , Clemens Lamberth , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Clemens Lamberth , Hans Tobler , Harald Walter
IPC分类号： C07D417/02 , C07D413/02 , C07D409/02 , C07D403/02 , A01N43/54 , A01N43/80 , A01N43/76 , A01N43/64
CPC分类号： C07F7/0812 , A01N55/00
摘要： Fungicidal compounds of formula (1): where X is O or S; RING is phenyl or thienyl; Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by one to four groups R4; R1 is hydrogen, optionally substituted (C1-4)alkyl, formyl, optionally substituted (C1-4)alkylC(═O), optionally substituted (C1-4)alkylC(═O)O, optionally substituted (C1-4)alkoxy(C1-4)alkyl, optionally substituted allyl, optionally substituted propargyl or optionally substituted allenyl; each R2 is, independently, halogen, optionally substituted (C1-4)alkyl, optionally substituted (C1-4)alkoxy or optionally substituted (C1-4)alkoxy(C1-4)alkyl; R3 is (CRaRb)m-Cy-(CRcRd)n—Y; each R4 is, independently, selected from halogen, C1-3 alkyl, C1-3 haloalkyl, C1-3alkoxy(C1-3)alkyl and cyano; Ra, Rb, Rc and Rd are each, independently, hydrogen or optionally substituted (C1-4)alkyl; Cy is an optionally substituted carbocyclic or heterocyclic 3-7 membered ring which may be saturated, unsaturated or aromatic and which optionally contains a silicon atom as a ring member; (CRaRb)m and (CRcRd), may be bound either to the same carbon or silicon atom of Cy or to different atoms separated by 1, 2 or 3 ring members; Y is Si(OpZ1)(OqZ2)(O5Z) and provided that Cy contains a silicon atom as a ring member then Y may also be hydrogen; Z is C1-4 alkyl or C2-4 alkenyl (each of which is optionally interrupted by one heteroatom selected from O, S and N and is optionally substituted by one to three independently selected halogen atoms); Z1 and Z2 are, independently, methyl or ethyl; in and n are each, independently, 0, 1, 2 or 3; p, q and s are each, independently, 0 or 1; and r is 0, 1 or 2; or an N-oxide thereof; novel intermediates used in the preparation of these compounds, agrochemical compositions which comprise at least one of the novel compounds as active ingredient and the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.

83. 发明申请

US20060030567A1 Cyclopropyl-thienyl-carboxamide as fungicides 失效
公开(公告)号：US20060030567A1
公开(公告)日：2006-02-09
申请号：US10532847
申请日：2003-10-24
申请人： Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： C07D409/02 , A01N43/64 , A01N43/54
CPC分类号： C07D409/12 , C07D333/36 , C07D411/12 , C07D417/12
摘要： A fungicidally active compound of formula (I): where X is (X1), (X2) or (X3); Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, provided that the ring is not 1,2,3-triazole, the ring being substituted by groups R4, R5 and R6; R1 and R2 are each, independently, hydrogen, halo or methyl; R3 is optionally substituted C2-12 alkyl, optionally substituted C2-12 alkenyl, optionally substituted C2-12 alkynyl, optionally substituted C3−12 cycloalkyl, optionally substituted phenyl or optionally substituted heterocyclyl; R4, R5 and R6 are each, independently, selected from hydrogen, halo, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkylene and C1-4 haloalkoxy(C1-4)alkylene, provided that at least one of R4, R5 and R6 is not hydrogen; and R7 and R8 are each, independently, hydrogen, halogen, C1-4 alkyl or Clue haloalkyl; the invention also relates to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to the preparation of intermediates, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.

84. 发明申请

US20050182107A1 Siliconated phenyl amides derivatives useful as microbiocide 失效
公开(公告)号：US20050182107A1
公开(公告)日：2005-08-18
申请号：US10509607
申请日：2003-03-21
申请人： Josef Ehrenfreund , Pierre Joseph Jung , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Pierre Joseph Jung , Hans Tobler , Harald Walter
IPC分类号： A01N55/00 , A01N55/10 , C07F7/08 , C07F7/10 , C07D213/46 , A01N43/36 , A01N43/40
CPC分类号： C07F7/0812 , A01N55/00
摘要： A fungicidal compound of formula (1): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by groups R7, R8 and R9; R1 is hydrogen, optionally substituted (C1-4)alkylC(═O), optionally substituted (C1-4)alkylC(═O)O, optionally substituted (C1-4)alkoxy(C1-4)alkyl, optionally substituted allyl, optionally substituted propargyl or optionally substituted allenyl; R2, R3, R4 and R5 are each, independently, hydrogen, halogen, optionally substituted (C1-4)alkoxy(C1-4)alkoxy or optionally substituted (C1-4)alkoxy(C1)alkyl; R6 is an organic group containing three to thirteen carbon atoms and at least one silicon atom and, optionally, one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, and is optionally substituted by one to four independently selected halogen atoms; R7, R8 and R9 are each, independently, hydrogen, halogen, C1-3alkyl, C1-3haloalkyl, C1-3alkoxy(C1-3)alkyl or cyano, where at least one of R7, R8 and R9 is not hydrogen; and X is O or S; or an N-oxide thereof; and when present, each optional substituent on alkyl moieties, allyl, propargyl and allenyl is, independently, selected from halogen, hydroxy, cyano, methoxycarbonyl, ethoxycarbonyl, methoxy, ethoxy, methylsulfonyl, ethylsulfonyl, diflouromethoxy, trifluoromethoxy and trifluorothiomethoxy.

85. 发明授权

US4908383A N-phenyl-N-carboxythioureas and their use in the control of pests 失效
标题翻译： N-苯基-N-羧基硫脲及其在防治害虫中的应用
公开(公告)号：US4908383A
公开(公告)日：1990-03-13
申请号：US356665
申请日：1989-05-23
申请人： Jozef Drabek , Josef Ehrenfreund
发明人： Jozef Drabek , Josef Ehrenfreund
IPC分类号： A01N47/34 , C07C335/28 , C07C335/38
CPC分类号： A01N47/34 , C07C335/28 , C07C335/38 , C07C2101/08 , C07C2101/10
摘要： Novel N-phenyl-N-carboxythioureas of the formula I ##STR1## in which R.sub.1 and R.sub.2 each represents C.sub.1 -C.sub.10 alkyl, C.sub.3 -C.sub.7 cycloalkyl or C.sub.5 -C.sub.6 cycloalkenyl,R.sub.3 represents hydrogen, halogen, C.sub.1 -C.sub.10 alkyl, C.sub.1 -C.sub.10 alkoxy or C.sub.1 -C.sub.10 alkylthio,R.sub.4 represents C.sub.1 -C.sub.10 alkyl, C.sub.2 -C.sub.10 alkenyl, C.sub.2 -C.sub.10 alkynyl or phenyl-C.sub.1 -C.sub.7 alkyl; C.sub.1 -C.sub.10 alkyl, C.sub.2 -C.sub.10 alkenyl, C.sub.2 -C.sub.10 alkynyl or phenyl-C.sub.1 -C.sub.7 alkyl each mono- or poly-substituted by halogen or interrupted one or several times by oxygen and/or sulphur; C.sub.3 -C.sub.8 cycloalkyl; or C.sub.3 -C.sub.8 cycloalkyl mono- or poly-substituted by halogen or by C.sub.1 -C.sub.5 alkyl, andR.sub.5 represents C.sub.1 -C.sub.10 alkyl; phenyl-C.sub.1 -C.sub.7 alkyl; C.sub.1 -C.sub.10 alkyl or phenyl-C.sub.1 -C.sub.7 alkyl each mono- or poly-substituted by halogen or interrupted one or several times by oxygen and/or sulphur; C.sub.3 -C.sub.8 cycloalkyl; or C.sub.3 -C.sub.8 cycloalkyl mono- or poly-substituted by halogen or by C.sub.1 -C.sub.5 alkyl, processes and salts of corresponding isothioureas as intermediates for their preparation, their use in pest control, and pesticidal compositions that contain at least one compound of the formula I or an active intermediate, are disclosed. The preferred field of application is the control of pests on animals and plants.
摘要翻译：新的式I的N-苯基-N-羧基硫脲，其中R 1和R 2各自表示C 1 -C 10烷基，C 3 -C 7环烷基或C 5 -C 6环烯基，R 3表示氢，卤素，C 1 -C 10烷基，C 1 -C 10烷氧基或C 1 -C 10烷硫基，R 4表示C 1 -C 10烷基，C 2 -C 10烯基，C 2 -C 10炔基或苯基-C 1 -C 7烷基; C 1 -C 10烷基，C 2 -C 10烯基，C 2 -C 10炔基或苯基-C 1 -C 7烷基，其各自被卤素单取代或多取代，或被氧和/或硫中断一次或数次; C 3 -C 8环烷基; 或被卤素或C 1 -C 5烷基单取代或多取代的C 3 -C 8环烷基，R 5表示C 1 -C 10烷基; 苯基-C 1 -C 7烷基; 每个被卤素单取代或多取代的C 1 -C 10烷基或苯基-C 1 -C 7烷基，或被氧和/或硫中断一个或几个; C 3 -C 8环烷基; 或被卤素或C 1 -C 5烷基单取代或多取代的C 3 -C 8环烷基，相应的异硫脲的方法和盐作为其制备的中间体，其在病虫害防治中的用途，以及含有至少一种式I化合物或公开了一种活性中间体。优选的应用领域是控制动物和植物上的害虫。

86. 发明授权

US4870184A 1.4-bis-pyridyl-2,3-diazabutadienes 失效
标题翻译： 1,4-双 - 吡啶-2,3-二氮杂双环
公开(公告)号：US4870184A
公开(公告)日：1989-09-26
申请号：US288756
申请日：1988-12-22
申请人： Saleem Farooq , Josef Ehrenfreund , Hans-Rudolf Waespe
发明人： Saleem Farooq , Josef Ehrenfreund , Hans-Rudolf Waespe
IPC分类号： A01N43/82 , A01N43/824 , C07D213/76 , C07D417/04 , C07D417/14
CPC分类号： C07D417/04 , A01N43/82 , C07D417/14
摘要： The invention relates to novel 2-pyridyl-4,5-dihydro-1,3,4-thiadiazoles of formula ##STR1## wherein A is the 2-, 3- or 4-pyridyl radical,B is hydrogen, C.sub.1 -C.sub.4 alkyl or the 2, 3- or 4-pyridyl radical,R is hydrogen, C.sub.1 -C.sub.4 alkyl, benzyl, aryl or aryl which is substituted by halogen, nitro, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy-C.sub.1 -C.sub.4 alkyl or halo-C.sub.1 -C.sub.4 alkyl.The invention further relates to the preparation of these novel compounds and to the use thereof in pest control.
摘要翻译：本发明涉及式（I）的新的2-吡啶基-4,5-二氢-1,3,4-噻二唑，其中A是2-，3-或4-吡啶基，B是氢，C1 C 1-4烷基或2,3-或4-吡啶基，R是氢，被卤素，硝基，C 1 -C 4烷基，C 1 -C 4烷氧基-C 1 -C 4烷基或卤代-C 1烷基取代的C 1 -C 4烷基，苄基，芳基或芳基 -C 1-4烷基。本发明还涉及这些新化合物的制备及其在病虫害防治中的应用。

87. 发明授权

US4725302A Substituted phenylhydrazines and phenyloxadiazolinones and pesticidal usage thereof 失效
标题翻译：取代苯肼和苯基恶二唑啉酮及其农药使用
公开(公告)号：US4725302A
公开(公告)日：1988-02-16
申请号：US800179
申请日：1985-11-20
申请人： Josef Ehrenfreund
发明人： Josef Ehrenfreund
IPC分类号： A01N43/82 , A01N43/824 , A01N47/24 , C07D271/06 , C07D271/07 , C07D307/12 , C07D307/20 , C07D309/12 , C07D413/12 , A61K31/42 , C07D271/10 , C07D307/04 , C07D309/04
CPC分类号： C07D271/07 , A01N43/82 , A01N47/24 , C07D307/12 , C07D307/20 , C07D309/12 , C07D413/12
摘要： Phenylhydrazines of the formula I ##STR1## wherein R.sub.1 is --A--R--Z,A is oxygen, sulfur, ##STR2## R is C.sub.1 -C.sub.6 -alkylene, C.sub.1 -C.sub.6 -haloalkyl-C.sub.1 -C.sub.6 -alkylene, C.sub.1 -C.sub.6 -alkoxy-C.sub.1 -C.sub.6 -alkylene or C.sub.1 -C.sub.6 -alkylthio-C.sub.1 -C.sub.6 -alkylene,Z is halogen, C.sub.1 -C.sub.6 -haloalkyl, C.sub.1 -C.sub.6 -alkoxy, C.sub.1 -C.sub.6 -alkylthio, C.sub.1 -C.sub.6 -alkylsulfinyl or C.sub.1 -C.sub.6 -alkylsulfonyl, orR and Z together are ##STR3## R.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -alkoxy, C.sub.1 -C.sub.6 -alkylthio or (C.sub.1 -C.sub.6 -alkyl).sub.2 amino,n is a number from 1-4, and R.sub.2 can be different when n is one of the numbers 2-4,R.sub.3 is halogen,R.sub.4 is hydrogen,R.sub.5 is --COOR.sub.6, orR.sub.3, R.sub.4 and R.sub.5 together form a bridge member of the formula ##STR4## and R.sub.6 is C.sub.1 -C.sub.6 -alkyl, C.sub.2 -C.sub.6 -alkenyl or C.sub.2 -C.sub.6 -alkynyl.A process for producing these phenylhydrazines and their use for controlling pests are described.
摘要翻译：式I的苯肼（I）其中R 1是-ARZ，A是氧，硫，R 2是C 1 -C 6亚烷基，C 1 -C 6卤代烷基-C 1 -C 6亚烷基，C 1 -C 6 - 烷氧基-C 1 -C 6亚烷基或C 1 -C 6烷硫基-C 1 -C 6亚烷基，Z为卤素，C 1 -C 6卤代烷基，C 1 -C 6烷氧基，C 1 -C 6烷硫基，C 1 -C 6烷基亚磺酰基或C 1 -C 6 - C6-烷基磺酰基或R和Z一起是R 2是氢，卤素，C 1 -C 6烷基，C 1 -C 6 - 烷氧基，C 1 -C 6 - 烷硫基或（C 1 -C 6烷基）2氨基，n为1-4的数，当n为2-4时，R2为可以不同，R3为卤素，R4为氢，R5为-COOR6或R3，R4和R5一起形成桥构件式为“IMAGE”，R6为C1-C6-烷基，C2-C6-烯基或C2-C6-炔基。描述了制备这些苯肼的方法及其用于防治害虫的用途。

88. 发明授权

US4675046A Fused N-phenylsulfonyl-N'-pyrimidinylureas 失效
标题翻译：熔融的N-苯基磺酰基-N'-嘧啶基脲
公开(公告)号：US4675046A
公开(公告)日：1987-06-23
申请号：US825283
申请日：1986-02-03
申请人： Josef Ehrenfreund , Werner Fory
发明人： Josef Ehrenfreund , Werner Fory
IPC分类号： A01N47/36 , C07D217/24 , C07D279/02 , C07D311/18 , C07D311/76 , C07D327/06 , C07D335/06 , C07D339/08 , C07D401/12 , C07D411/12 , C07D521/00 , C07D239/69 , A01N43/54
CPC分类号： C07D521/00 , A01N47/36 , C07D217/24 , C07D327/06
摘要： N-phenylsulfonyl-N'-pyrimidinylureas of the formula ##STR1## wherein Z is oxygen or sulfur,R.sup.1 is hydrogen, halogen, nitro, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, cyano, or a --X--R.sup.5, --CO--X--R.sup.6, --CO--NR.sup.7 R.sup.8, --SO--R.sup.9 or --SO.sub.2 --R.sup.10 group,R.sup.2 is hydrogen, C.sub.1 -C.sub.4 alkyl or C.sub.1 -C.sub.4 alkoxy,R.sup.3 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy or C.sub.3 -C.sub.6 cycloalkyl,R.sup.4 is hydrogen, halogen, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.2 -C.sub.4 alkoxyalkoxy, C.sub.3 -C.sub.6 cycloalkyl or --NR.sup.11 R.sup.12,R.sup.5 is C.sub.3 -C.sub.5 alkynyl or C.sub.1 -C.sub.4 alkyl which is unsubstituted or substituted by halogen or C.sub.1 -C.sub.4 -alkoxy, or is C.sub.3 -C.sub.5 alkenyl, which is unsubstituted or is substituted by halogen or C.sub.1 -C.sub.4 -alkoxy,R.sup.6 and R.sup.9 are each independently C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkoxyalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl, phenyl or benzyl,R.sup.7 and R.sup.8 are each independently hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkoxyalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl, phenyl or benzyl,R.sup.10 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy or --NR.sup.13 R.sup.14,R.sup.11 and R.sup.12 are each independently hydrogen or C.sub.1 -C.sub.4 alkyl,R.sup.13 and R.sup.14 are each independently hydrogen C.sub.1 -C.sub.4 alkyl C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkoxyalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl, phenyl or benzyl, andX is oxygen or sulfur,or a salt thereof have good pre and post-emergence selective herbicidal and growth regulating properties.
摘要翻译： N-苯基磺酰基-N'-嘧啶基脲，其中Z是氧或硫，R 1是氢，卤素，硝基，C 1 -C 4烷基，C 1 -C 4卤代烷基，氰基或-X-R 5，-CO-X -R6，-CO-NR7R8，-SO-R9或-SO2-R10基团，R2是氢，C1-C4烷基或C1-C4烷氧基，R3是C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或C3 -C 6环烷基，R 4是氢，卤素，C 1 -C 4卤代烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷氧基，C 2 -C 4烷氧基烷氧基，C 3 -C 6环烷基或-NR 11 R 12，R 5是未被取代或被卤素或C1取代的C 3 -C 5炔基或C 1 -C 4烷基 C 4 - 烷氧基，或者是未被取代或被卤素或C 1 -C 4烷氧基取代的C 3 -C 5烯基，R 6和R 9各自独立地为C 1 -C 4烷基，C 1 -C 4卤代烷基，C 2 -C 4烷氧基烷基，C 3 -C 5烯基， C 3 -C 5炔基，苯基或苄基，R 7和R 8各自独立地为氢，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 2 -C 4烷氧基烷基，C 3 -C 5烯基，C 3 -C 5炔基，苯基或苄基，R 10为C 1 -C 4烷基，C 1 -C 4烷氧基， C1-C4卤代烷氧基或-NR13R14，R11和R12各自独立地表示 R 13和R 14各自独立地为C 1 -C 4烷基C 1 -C 4卤代烷基，C 2 -C 4烷氧基烷基，C 3 -C 5烯基，C 3 -C 5炔基，苯基或苄基，X为氧或硫或其盐具有良好的前期和后期选择性除草和生长调节性质。

89. 发明授权

US4589911A Fused N-phenylsulfonyl-N-triazinylureas 失效
标题翻译：熔融的N-苯基磺酰基-N-三嗪基脲
公开(公告)号：US4589911A
公开(公告)日：1986-05-20
申请号：US606076
申请日：1984-05-01
申请人： Josef Ehrenfreund , Werner Fory
发明人： Josef Ehrenfreund , Werner Fory
IPC分类号： A01N47/36 , C07D217/24 , C07D279/02 , C07D311/18 , C07D311/76 , C07D327/06 , C07D335/06 , C07D339/08 , C07D401/12 , C07D411/12 , C07D521/00 , A01N43/68 , A01N43/70
CPC分类号： C07D521/00 , A01N47/36 , C07D217/24 , C07D327/06
摘要： Fused N-phenylsulfonyl-N'-triazinylurea of formula I ##STR1## wherein Z is oxygen or sulfur,R.sup.1 is hydrogen, halogen, nitro, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, cyano, or a --X--R.sup.5, --CO--X--R.sup.6, --CO--NR.sup.7 R.sup.8, --SO--R.sup.9 or --SO.sub.2 --R.sup.10 group,R.sup.2 is hydrogen, C.sub.1 -C.sub.4 alkyl or C.sub.1 -C.sub.4 alkoxy,R.sup.3 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy or C.sub.3 -C.sub.6 cycloalkyl,R.sup.4 is hydrogen, halogen, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.2 -C.sub.4 alkoxyalkoxy, C.sub.3 -C.sub.6 cycloalkyl or --NR.sup.11 R.sup.12,R.sup.5 is C.sub.3 -C.sub.5 alkynyl or C.sub.1 -C.sub.4 alkyl which is unsubstituted or substituted by halogen or C.sub.1 -C.sub.4 -alkoxy, or is C.sub.3 -C.sub.5 alkenyl, which is unsubstituted or is substituted by halogen or C.sub.1 -C.sub.4 -alkoxy,R.sup.6 and R.sup.9 are each independently C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkoxyalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl, phenyl or benzyl,R.sup.7 and R.sup.8 are each independently hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkoxyalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl, phenyl or benzyl,R.sup.10 is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy or --NR.sup.13 R.sup.14,R.sup.11 and R.sup.12 are each independently hydrogen or C.sub.1 -C.sub.4 alkyl,R.sup.13 and R.sup.14 are each independently hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.2 -C.sub.4 alkoxyalkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl, phenyl or benzyl, andX is oxygen or sulfur,or a salt thereof have good pre and post-emergence selective herbicidal and growth regulating properties.
摘要翻译：熔融的式I的N-苯基磺酰基-N'-三嗪基脲其中Z是氧或硫，R 1是氢，卤素，硝基，C 1 -C 4烷基，C 1 -C 4卤代烷基，氰基或-X-R 5， -CO-X-R6，-CO-NR7R8，-SO-R9或-SO2-R10基，R2是氢，C1-C4烷基或C1-C4烷氧基，R3是C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1 C 4卤代烷氧基或C 3 -C 6环烷基，R 4是氢，卤素，C 1 -C 4卤代烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷氧基，C 2 -C 4烷氧基烷氧基，C 3 -C 6环烷基或-NR 11 R 12，R 5是未被取代或取代的C 3 -C 5炔基或C 1 -C 4烷基或未被取代或被卤素或C 1 -C 4 - 烷氧基取代的C 3 -C 5烯基，R 6和R 9各自独立地为C 1 -C 4烷基，C 1 -C 4卤代烷基，C 2 -C 4烷氧基烷基，C 3 -C 4烷氧基， C5链烯基，C3-C5炔基，苯基或苄基，R7和R8各自独立地为氢，C1-C4烷基，C1-C4卤代烷基，C2-C4烷氧基烷基，C3-C5烯基，C3-C5炔基，苯基或苄基，R10为C1-C4烷基，C1- C4烷氧基，C1-C4卤代烷氧基或-NR13R14，R11和R12各自为吲哚基 R 1和R 4各自独立地为氢，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 2 -C 4烷氧基烷基，C 3 -C 5烯基，C 3 -C 5炔基，苯基或苄基，X为氧或硫或其盐具有良好的芽前和出苗后选择性除草和生长调节性质。

90. 发明授权

US4348412A Insecticidal phenylureas and methods of use thereof 失效
标题翻译：杀虫苯脲及其使用方法
公开(公告)号：US4348412A
公开(公告)日：1982-09-07
申请号：US166634
申请日：1980-07-07
申请人： Josef Ehrenfreund
发明人： Josef Ehrenfreund
IPC分类号： A01N47/34 , C07C275/54 , A01N47/28 , C07C127/22
CPC分类号： C07C275/54 , A01N47/34
摘要： Novel halogen-substituted N-(3-trifluoromethyl-4-halogenoalkoxyphenyl)-N'-benzoylureas of the formula ##STR1## wherein R.sub.1 is a C.sub.1 -C.sub.4 -alkyl group which is substituted at least twice by fluorine, chlorine or bromine, R.sub.2 is fluorine or chlorine, and R.sub.3 is hydrogen, fluorine or chlorine; processes for producing these compounds, as well as compositions containing them, for use in combating pests, particularly for combating insects which infest plants and animals. The novel compounds are especially effective against larval stages of insects which damage plants by eating.
摘要翻译：式（I）的新型卤素取代的N-（3-三氟甲基-4-卤代烷氧基苯基）-N'-苯甲酰脲其中R1是被氟，氯或氯原子取代至少两次的C 1 -C 4烷基溴，R2是氟或氯，R3是氢，氟或氯; 用于生产这些化合物的方法，以及含有它们的组合物，用于防治害虫，特别是用于防治侵染植物和动物的昆虫。这些新颖的化合物对于通过进食损害植物的昆虫的幼虫阶段是特别有效的。

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