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71. 发明授权

US5206242A Diaryl-substituted pyrazole compounds and drugs and cosmetics obtained therefrom 失效
公开(公告)号：US5206242A
公开(公告)日：1993-04-27
申请号：US753916
申请日：1991-09-03
申请人： Hans-Heiner Wuest , Bernd Janssen , William V. Murray , Michael P. Wachter , Stanley Bell
发明人： Hans-Heiner Wuest , Bernd Janssen , William V. Murray , Michael P. Wachter , Stanley Bell
IPC分类号： C07D207/32 , C07D207/323 , C07D207/325 , C07D207/337 , C07D231/06 , C07D231/12 , C07D231/22 , C07D231/24 , C07D233/54 , C07D233/84 , C07D237/08 , C07D239/36 , C07D261/08 , C07D263/04 , C07D263/10 , C07D263/32 , C07D271/06 , C07D271/10 , C07D271/107 , C07D277/30 , C07D307/36 , C07D307/38 , C07D307/40 , C07D307/54 , C07D333/08 , C07D333/18 , C07D333/24
CPC分类号： C07D207/323 , C07D207/325 , C07D207/337 , C07D231/06 , C07D231/12 , C07D231/22 , C07D231/24 , C07D233/64 , C07D233/84 , C07D237/08 , C07D239/36 , C07D261/08 , C07D263/04 , C07D263/10 , C07D263/32 , C07D271/06 , C07D271/107 , C07D277/30 , C07D307/36 , C07D307/38 , C07D307/40 , C07D307/54 , C07D333/08 , C07D333/18 , C07D333/24
摘要： Compounds of formula I ##STR1## where R.sup.1 and R.sup.2 are each hydrogen or methyl,A is en ethylene or methylene radical which is unsubstituted or substituted by methyl, hydroxyl or oxo,L is a saturated or unsaturated five-membered or six-membered heterocyclic structure which is unsubstituted or substituted by hydroxyl, mercapto, C.sub.1 -C.sub.6 -alkyl, or C.sub.1 -C.sub.4 -alkanoyl and has from 1 to 3 heteroatoms from the group consisting of N, O and S, the second and third heteroatoms being a nitrogen atom,R.sup.3 is hydrogen, a hydroxy or C.sub.1 -C.sub.6 -alkoxy group,R.sup.4 is hydrogen, C.sub.1 -C.sub.4 -alkyl, halogen or methoxy,R.sup.5 is hydrogen or methoxy or tert-butyl,R.sup.6 is hydrogen, methyl, nitrile or a C.sub.2 -C.sub.10 -ketal group or the radical --CHR.sup.7 OR.sup.8 --CHR.sup.7 --NR.sup.9 R.sup.10, --COR.sup.11, --SR.sup.12, ##STR2## in which R.sup.7 is hydrogen or C.sub.1 -C.sub.4 -alkyl,R.sup.8 is hydrogen, C.sub.1 -C.sub.4 -alkyl or C.sub.1 -C.sub.20 -alkanoyl or is benzoyl which is unsubstituted or substituted by methoxy, nitro, methyl or chlorine,R.sup.9 and R.sup.10 are each hydrogen, C.sub.1 -C.sub.4 -alkyl or C.sub.1 -C.sub.6 -alkanoyl or are each benzoyl which is unsubstituted or substituted as for R.sup.8, or R.sup.9 and R.sup.10, together with the nitrogen atom to which they are bonded, form a saturated, 5-membered or 6-membered heterocyclic radical which may contain oxygen as the second heteroatom,R.sup.11 is hydrogen, C.sub.1 -C.sub.4 -alkyl, --OR.sup.13 or --NR.sup.14 R.sup.15, where R.sup.13 is hydrogen, unsubstituted or hydroxyl-substituted C.sub.1 -C.sub.6 -alkyl, aryl or aralkyl which is unsubstituted or substituted by chlorine, bromine, methyl, methoxy or nitro, substitution in the case of the aralkyl group being in the aryl moiety, and where R.sup.14 and R.sup.15 are each hydrogen, unsubstituted or hydroxyl-substituted C.sub.1 -C.sub.6 -alkyl or an aralkyl or aryl group which is unsubstituted or substituted as for R.sup.13, or R.sup.14 and R.sup.15, together with the nitrogen atom to which they are bonded, form a heterocyclic radical as defined above for R.sup.9 and R.sup.10, andR.sup.12 is C.sub.1 -C.sub.4 -alkyl,and compounds of formula Ia ##STR3## where R.sup.3, R.sup.4, R.sup.6 and L have the abovementioned meanings and R.sup.17 is hydrogen or hydroxyl, and their physiologically tolerated salts, processes for their preparation and drugs and cosmetics prepared therefrom.

72. 发明授权

US5152824A Sulfamidosulfonamide derivatives and herbicides 失效
标题翻译：磺酰胺酰胺衍生物和除草剂
公开(公告)号：US5152824A
公开(公告)日：1992-10-06
申请号：US665557
申请日：1991-03-06
申请人： Kenzi Makino , Katsushi Morimoto , Shigeaki Akiyama , Hideaki Suzuki , Takeshi Nagaoka , Koichi Suzuki , Tsutomu Nawamaki , Shigeomi Watanabe
发明人： Kenzi Makino , Katsushi Morimoto , Shigeaki Akiyama , Hideaki Suzuki , Takeshi Nagaoka , Koichi Suzuki , Tsutomu Nawamaki , Shigeomi Watanabe
IPC分类号： A01N47/38 , A01N51/00 , C07D231/06 , C07D405/04 , C07D409/04 , C07D417/04 , C07D417/12 , C07D417/14 , C07D521/00
CPC分类号： C07D231/06 , A01N47/38 , A01N51/00 , C07D231/12 , C07D233/56 , C07D249/08 , C07D405/04 , C07D409/04 , C07D417/04 , C07D417/12 , C07D417/14
摘要： A sulfamidosulfonamide derivative of the formula (1) and an agriculturally suitable salt thereof: ##STR1## wherein Q is ##STR2## X is an oxygen atom or a sulfur atom; and G is ##STR3## which are useful as herbicide.
摘要翻译：式（1）的磺酰氨基磺酰胺衍生物及其农业上合适的盐：其中Q是氧原子或硫原子;其中Q是氧原子或硫原子; 而G是除去草剂之外的“IMAGE”。

73. 发明授权

US4992203A Non-linear optics 失效
标题翻译：非线性光学
公开(公告)号：US4992203A
公开(公告)日：1991-02-12
申请号：US420720
申请日：1989-10-13
申请人： Simon Allen , Paul F. Gordon , John O. Morley
发明人： Simon Allen , Paul F. Gordon , John O. Morley
IPC分类号： C07D231/06 , C09K19/52 , G02F1/065 , G02F1/35 , G02F1/355 , G02F1/361
CPC分类号： G02F1/3612 , C09K19/54 , C09K19/586 , G02F1/065
摘要： Optical elements having non-linear optical properties comprising a compound of the formula: ##STR1## wherein D is an electron donorA is an electron acceptor;and W, X, Y and Z are each independently H or any group capable of attachment to the pyrazolyl ring; in which the molecules of the compound are aligned so that the element has a net non-centrosymmetry, a method for their preparation, optical devices comprising such elements, and compounds of formula I.
摘要翻译：具有非线性光学性质的光学元件包括下式化合物：其中D是电子给体A是电子受体; 并且W，X，Y和Z各自独立地为H或能够连接至吡唑基环的任何基团; 其中化合物的分子对准，使得元件具有净非中心对称性，其制备方法，包含这些元件的光学器件和式I化合物。

74. 发明授权

US4924001A Process for preparing 5-cyano-4, 5-dihydro-3,4-dicarboxypyrazole derivatives 失效
标题翻译： 5-氰基-4,5-二氢-3,4-二羧基吡唑衍生物的制备方法
公开(公告)号：US4924001A
公开(公告)日：1990-05-08
申请号：US422922
申请日：1989-10-17
申请人： John R. Rizzo , Eddie V. P. Tao
发明人： John R. Rizzo , Eddie V. P. Tao
IPC分类号： C07D231/06
CPC分类号： C07D231/06
摘要： The present invention provides 5-cyano-4,5-dihydro-3,4-dicarboxypyrazoles and a process for preparing such compounds which comprises reacting a dialkyl fumarate with diazoacetonitrile.
摘要翻译：本发明提供5-氰基-4,5-二氢-3,4-二羧基吡唑及其制备方法，该方法包括使富马酸二烷基酯与重氮乙腈反应。

75. 发明授权

US4824960A Preparation of 1-aryl-5-amino-pyrazoles 失效
标题翻译： 1-芳基-5-氨基 - 吡唑的制备
公开(公告)号：US4824960A
公开(公告)日：1989-04-25
申请号：US34300
申请日：1987-04-03
申请人： Bernd Gallenkamp , Hermann Arold
发明人： Bernd Gallenkamp , Hermann Arold
IPC分类号： C07B61/00 , B01J31/00 , B01J31/02 , B01J31/04 , C07D231/06 , C07D231/38 , C07D401/04
CPC分类号： C07D231/38 , C07D401/04
摘要： A process for the preparation of a 1-aryl-5-amino-pyrazole of the formula ##STR1## in which Ar is in each case optionally substituted phenyl or pyridyl, comprising reacting an arylhydrazine of the formulaAr--NH--NH.sub.2with acrylonitrile of the formulaCH.sub.2 .dbd.CH--CNin a first stage in the presence of a diluent at a temperature between about 20.degree. C. and 100.degree. C. to form the arylhydrazine derivative of the formulaAr--NH--NH--CH.sub.2 --CH.sub.2 --CN, andin a second stage contacting such derivative with an oxidizing agent in the presence of a base at a temperature between about 0.degree. C. and 60.degree. C., thereby to effect oxidation and cyclization. The products are known intermediates for herbicides and insecticides.
摘要翻译：制备式“IMAGE”的1-芳基-5-氨基吡唑的方法，其中Ar各自为任选取代的苯基或吡啶基，包括使式Ar-NH-NH 2的芳基肼与在稀释剂存在下，在约20℃至100℃之间的第一阶段中，CH 2 = CH-CN的式CH = CN，形成式Ar-NH-NH-CH 2 -CH 2 CN的芳基肼衍生物，并且在第二阶段中，在约0℃至60℃的温度下，在碱的存在下，使这种衍生物与氧化剂接触，从而进行氧化和环化。该产品是除草剂和杀虫剂的已知中间体。

76. 发明授权

US4824859A Pyrazoline compounds compositions and use 失效
标题翻译：吡唑啉化合物组合物和用途
公开(公告)号：US4824859A
公开(公告)日：1989-04-25
申请号：US606867
申请日：1984-05-03
申请人： Sidney C. Burford , David N. Hardern
发明人： Sidney C. Burford , David N. Hardern
IPC分类号： C07D231/06 , C07D401/04 , C07D401/12 , A61K31/415
CPC分类号： C07D231/06 , C07D401/04 , C07D401/12
摘要： There are described compounds of formula I, ##STR1## in which Ar.sub.1 and Ar.sub.2, which may be the same or different, each independently represent phenyl or pyridinyl, the phenyl or the pyridinyl each optionally being substituted by one or more of halogen; hydroxy; --COOR.sub.12 ; trihalomethyl; alkoxy C1 to 6; alkyl C1 to 6; --NR.sub.1 R.sub.2 ; alkoxy C1 to 6 substituted by --NR.sub.1 R.sub.2 or by phenyl; or alkyl C1 to 6 substituted by --NR.sub.1 R.sub.2 or by --COOR.sub.12 ;R.sub.1 and R.sub.2, which may be the same or different, each independently represent hydrogen or alkyl C1 to 6,R.sub.3 represents hydrogen, alkyl C1 to 6, alkanoyl C1 to 6, benzoyl, --COOR.sub.8, or --CONHR.sub.11,R.sub.4, R.sub.5, R.sub.6 and R.sub.7, which may be the same or different each independently represent hydrogen, alkyl C1 to 6 or phenyl,R.sub.8 represents alkyl C1 to 6 or aryl,R.sub.11 represents alkyl C1 to 6 or aryl,R.sub.12 represents hydrogen or alkyl C1 to 6, and pharmaceutically acceptable derivatives thereof.There are also described compositions containing the compounds and methods for their preparation.The compounds are indicated for use as pharmaceutical, eg antiinflammatory agents.
摘要翻译：描述了式I的化合物，其中Ar 1和Ar 2可以相同或不同，各自独立地表示苯基或吡啶基，苯基或吡啶基各自任选被一个或多个卤素取代; 羟基; -COOR12; 三卤甲基烷氧基C1至6; 烷基C1至6; -NR1R2; 被-NR 1 R 2取代的C 1-6烷氧基或苯基取代; 或被-NR 1 R 2或-COOR 12取代的C 1-6的烷基; R1和R2可以相同或不同，各自独立地表示氢或C1至6的烷基，R3表示氢，C1至6的烷基，C1至6的烷酰基，苯甲酰基，-COOR8或-CONHR11，R4，R5，R6 和R 7可以相同或不同，各自独立地表示氢，烷基C1至6或苯基，R8表示烷基C1至6或芳基，R11表示烷基C1至6或芳基，R12表示氢或C1-6烷基，和药学上可接受的衍生物还描述了含有这些化合物的组合物及其制备方法。化合物被指示用作药物，例如抗炎剂。

77. 发明授权

US4816590A Pyrazoline compounds and method of whitening 失效
标题翻译：吡唑啉化合物和美白方法
公开(公告)号：US4816590A
公开(公告)日：1989-03-28
申请号：US935911
申请日：1986-11-28
申请人： Hans R. Meyer
发明人： Hans R. Meyer
IPC分类号： C07D231/06 , C09B67/22 , D06L3/12 , D06L3/06
CPC分类号： C07D231/06 , D06L3/1257
摘要： The invention relates to pyrazoline compounds of formula ##STR1## wherein R.sub.1 is hydrogen or methyl, R.sub.2 and R.sub.3 are each independently of the other methyl, ethyl or hydroxyethyl, R.sub.4 is hydrogen or chlorine, R.sub.5 and R.sub.6 are each independently of the other hydrogen or methyl, R.sub.7 is hydrogen, methyl or phenyl, n is 0 or 1, with the proviso that, if n is 0 and R.sub.4 to R.sub.7 are hydrogen, R.sub.2 is methyl and R.sub.3 is hydroxyethyl, and X.sup..crclbar. is a C.sub.1 -C.sub.3 alkanoate, C.sub.1 -C.sub.4 alkanephosphonate, C.sub.1 -C.sub.4 alkanesulfonate, phosphite, sulfamate or glycolate anion and, if R.sub.1 is methyl, X.sup..crclbar. is also a methosulfate, chloride or bromide ion, to the preparation of said compounds, to the use thereof as fluorescent whitening agents, and to novel hydrazine intermediates of formula ##STR2## wherein R.sub.2 and R.sub.3 are methyl, ethyl or hydroxyethyl, and the acetone hydrazones and salts thereof.
摘要翻译：本发明涉及式IMA的吡唑啉化合物，其中R 1是氢或甲基，R 2和R 3各自独立地是甲基，乙基或羟乙基，R 4是氢或氯，R 5和R 6各自独立地是氢或甲基，R 7为氢，甲基或苯基，n为0或1，前提条件是如果n为0，且R4至R7为氢，则R2为甲基，R3为羟乙基，X（ - ）为C1-C3烷酸酯 C1-C4烷基膦酸酯，C1-C4烷基磺酸盐，亚磷酸盐，氨基磺酸盐或乙醇酸盐阴离子，如果R1是甲基，X（ - ）也是一种硫酸盐，氯化物或溴离子，用于制备所述化合物，作为荧光增白剂试剂，以及式IMA图的新型肼中间体，其中R2和R3是甲基，乙基或羟乙基，以及丙酮腙及其盐。

78. 发明授权

US4780543A 1-phenyl-3-(2-nitroethenyl)pyrazoline and 1-phenyl-3-(2,2-dicyanoethenyl)pyrazoline 失效
标题翻译： 1-苯基-3-（2-硝基乙烯基）吡唑啉和1-苯基-3-（2,2-二氰基乙烯基）吡唑啉
公开(公告)号：US4780543A
公开(公告)日：1988-10-25
申请号：US98996
申请日：1987-09-21
申请人： Paul Gordon , Brian Bothwell
发明人： Paul Gordon , Brian Bothwell
IPC分类号： C07D231/06 , C09K19/34 , G02F1/361
CPC分类号： C07D231/06 , C09K19/3483 , G02F1/3612
摘要： A compound of the formula: ##STR1## wherein E is an ethenyl group of the formula: ##STR2## in which X is H when Y is NO.sub.2 ;Y is H when X is NO.sub.2 ; orX is CN when Y is CNwhich has the capacity to form a crystal in which the molecules are aligned substantially in the same manner giving it non-linear optical properties. The crystalline product is thus adapted for use in devices exhibiting non-linear optical effects.
摘要翻译：下式的化合物：其中E是下式的乙烯基：其中当Y是NO 2时X是H; 当X为NO2时，Y为H; 或者当Y是CN时，X是CN，其具有形成其中分子基本上以相同方式排列的晶体的能力，得到非线性光学性质。因此，结晶产品适用于显示非线性光学效应的装置。

79. 发明授权

US4767779A Pyrazoline-1-carboxamides, composition containing them, and insecticidal method of using them 失效
标题翻译：吡唑啉-1-甲酰胺，含有它们的组合物和使用它们的杀虫方法
公开(公告)号：US4767779A
公开(公告)日：1988-08-30
申请号：US849658
申请日：1986-04-09
申请人： Angelina J. Duggan
发明人： Angelina J. Duggan
IPC分类号： A01N47/38 , C07D231/06 , C07D405/04 , C07D405/12 , C07D405/14 , A01N43/56
CPC分类号： C07D231/06 , A01N47/38 , C07D405/04 , C07D405/12 , C07D405/14
摘要： Pyrazolines of the following formula are insecticides: ##STR1## wherein R.sub.A, R.sub.B and R.sub.C are aromatic groups; R.sub.N is hydrogen or lower alkyl; and W is oxygen or sulfur.
摘要翻译：下式的吡唑啉类是杀虫剂：其中RA，RB和RC是芳族基团; RN是氢或低级烷基; W是氧或硫。

80. 发明授权

US4724199A Silver halide photographic light sensitive materials 失效
标题翻译：卤化银照相感光材料
公开(公告)号：US4724199A
公开(公告)日：1988-02-09
申请号：US792187
申请日：1985-10-28
申请人： Hidetoshi Kobayashi , Masaharu Toriuchi , Isamu Itoh
发明人： Hidetoshi Kobayashi , Masaharu Toriuchi , Isamu Itoh
IPC分类号： C07D249/18 , C07D231/06 , C07D231/08 , C07D231/56 , C07D235/28 , C07D249/08 , C07D249/12 , C07D249/20 , C07D257/04 , C07D285/12 , C07D285/125 , C07D411/12 , G03C1/06 , G03C1/485 , G03C7/305 , G03C8/08 , G03C1/02 , G03C5/54 , G03C7/26
CPC分类号： C07D257/04 , C07D285/125 , G03C1/061 , G03C7/305 , G03C8/08 , Y10S430/156
摘要： A silver halide photographic light-sensitive material containing, in at least one layer thereof, a compound capable of releasing a fogging agent upon an oxidation-reduction reaction with an oxidation product of a developing agent under an alkaline condition. The material has an increased sensitivity, an increased contrast and an accelerated development rate.
摘要翻译：一种卤化银照相感光材料，其在至少一层中含有在碱性条件下与显影剂的氧化产物进行氧化还原反应时能够释放起雾剂的化合物。该材料具有增加的灵敏度，增加的对比度和加速的发展速度。

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