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41. 发明授权

US5430158A Pyrazole derivatives 失效
标题翻译：吡唑衍生物
公开(公告)号：US5430158A
公开(公告)日：1995-07-04
申请号：US313975
申请日：1994-09-28
申请人： Ki J. Hwang , Kyung H. Park
发明人： Ki J. Hwang , Kyung H. Park
IPC分类号： C07D231/20 , A01N47/34 , C07D231/22
CPC分类号： A01N47/34 , C07D231/22
摘要： An anilin derivative which corresponds to the following formula: ##STR1## wherein, R.sub.2 is hydrogen, lower alkoxy group, a nitro group, or one or more halogen atoms selected from fluorine, chlorine and bromine; and X is a lower alkyl group or a phenyl substituent. The compounds are intermediates for insecticides.
摘要翻译：对应于下式的苯胺衍生物：其中，R 2为氢，低级烷氧基，硝基或选自氟，氯和溴的一个或多个卤素原子; X为低级烷基或苯基取代基。这些化合物是杀虫剂的中间体。

42. 发明授权

US5283341A N-alkylation of heterocyclic, aromatic amines 失效
标题翻译：杂环芳族胺的N-烷基化
公开(公告)号：US5283341A
公开(公告)日：1994-02-01
申请号：US880587
申请日：1992-05-08
申请人： Norio Tanaka , Masataka Hatanaka , Yoshihisa Watanabe
发明人： Norio Tanaka , Masataka Hatanaka , Yoshihisa Watanabe
IPC分类号： B01J27/13 , B01J31/24 , C07B61/00 , C07D231/12 , C07D231/20 , C07D231/22 , C07D231/38 , C07D233/54 , C07D233/58 , C07D249/04 , C07D249/06 , C07D249/08 , C07D249/18 , C07D249/20 , B01J23/46 , C07D249/22 , C07D403/02
CPC分类号： C07D231/12
摘要： A process for producing a heterocyclic tertiary amine of the formula (III): ##STR1## wherein A is a nitrogen atom or C-R.sup.5, B is a nitrogen atom or C-R.sup.6, is a single bond or a double bond, and each of R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5 and R.sup.6 which may be the same or different, is a hydrogen atom, an acyl group, a halogen atom, a cyano group, etc., provided that two of R.sup.1, R.sup.2, R.sup.3 and R.sup.4 may together form a 3-membered, 4-membered, 5-membered or 6-membered aliphatic ring, a heterocyclic rig or aromatic ring, and R.sup.7 is a C.sub.1-6 alkyl group which may be substituted, etc., which process comprises reacting a heterocyclic secondary amine of the formula (I): ##STR2## wherein A, B, , R.sup.1, R.sup.2, R.sup.3 and R.sup.4 are as defined above, with an alkylating agent of the formula (II):R.sup.7 --X (II)wherein R.sup.7 is as defined above, and X is a hydroxyl group, a halogen atom, a OSO.sub.3 R.sup.7 group, a OSO.sub.2 R.sup.7 group, a OCO.sub.2 R.sup.7 group, a OCOR.sup.7 group, a OP(O)(OR.sup.7) group, a OP(O)O(R.sup.7).sub.2 group or an amino group, in the presence of a catalyst of Group VIII of the Periodic Table.
摘要翻译：制备式（III）的杂环叔胺的方法：（*化学结构*）（III）其中A为氮原子或C-R5，B为氮原子或C-R6，为单键或双键，R 1，R 2，R 3，R 4，R 5和R 6可以相同或不同，为氢原子，酰基，卤素原子，氰基等，条件是两个 R 1，R 2，R 3和R 4可以一起形成3元，4元，5元或6元脂族环，杂环基或芳环，并且R 7为可被取代的C 1-6烷基，等等，该方法包括使式（I）的杂环仲胺：其中A，B，，R 1，R 2，R 3和R 4如上所定义的式（I）化合物与式（II）：其中R7如上定义的R7-X（II），X是羟基，卤素原子，OSO3R7基，OSO2R7基，OCO2R7基，OCOR7基，OP（O ）（OR 7）基，OP（O）O（R 7）2基或氨基， n元素周期表第VIII族催化剂的存在。

43. 发明授权

US5206256A Naphthalene derivatives 失效
标题翻译：萘衍生物
公开(公告)号：US5206256A
公开(公告)日：1993-04-27
申请号：US687802
申请日：1991-04-19
申请人： Marc Lang
发明人： Marc Lang
IPC分类号： A61K31/40 , A61K31/41 , A61K31/415 , A61K31/4184 , A61P35/00 , C07D207/32 , C07D231/12 , C07D231/22 , C07D233/56 , C07D233/64 , C07D235/06 , C07D249/04 , C07D249/06 , C07D249/08 , C07D249/10 , C07D249/12 , C07D249/18 , C07D249/20 , C07D257/04 , C07D521/00 , C12N9/99
CPC分类号： C07D231/12 , C07D233/56 , C07D249/04 , C07D249/06 , C07D249/08
摘要： Compounds of formula I ##STR1## wherein the dotted line, Az, Z, R.sub.1 and R.sub.2 are as defined in the description, have valuable pharmaceutical properties and are effective especially against tumors. They are prepared in a manner known per se.
摘要翻译：式I的化合物（I）其中虚线，Az，Z，R 1和R 2如说明书中所定义，具有有价值的药物性质，尤其对肿瘤有效。它们是以本身已知的方式准备的。

44. 发明授权

US5196532A Diaryl-substituted heterocyclic compounds, their preparation and drugs and cosmetics obtained therefrom 失效
公开(公告)号：US5196532A
公开(公告)日：1993-03-23
申请号：US717264
申请日：1991-06-18
申请人： Hans-Heiner Wuest , Bernd Janssen , William V. Murray , Michael P. Wachter , Stanley Bell
发明人： Hans-Heiner Wuest , Bernd Janssen , William V. Murray , Michael P. Wachter , Stanley Bell
IPC分类号： C07D207/32 , C07D207/323 , C07D207/325 , C07D207/337 , C07D231/06 , C07D231/12 , C07D231/22 , C07D231/24 , C07D233/54 , C07D233/84 , C07D237/08 , C07D239/36 , C07D261/08 , C07D263/04 , C07D263/10 , C07D263/32 , C07D271/06 , C07D271/10 , C07D271/107 , C07D277/30 , C07D307/36 , C07D307/38 , C07D307/40 , C07D307/54 , C07D333/08 , C07D333/18 , C07D333/24
CPC分类号： C07D207/323 , C07D207/325 , C07D207/337 , C07D231/06 , C07D231/12 , C07D231/22 , C07D231/24 , C07D233/64 , C07D233/84 , C07D237/08 , C07D239/36 , C07D261/08 , C07D263/04 , C07D263/10 , C07D263/32 , C07D271/06 , C07D271/107 , C07D277/30 , C07D307/36 , C07D307/38 , C07D307/40 , C07D307/54 , C07D333/08 , C07D333/18 , C07D333/24
摘要： Compounds of formula I ##STR1## where R.sup.1 and R.sup.2 are each hydrogen or methyl, A is an ethylene or methylene radical which is unsubstituted or substituted by methyl, hydroxyl or oxo,L is a saturated or unsaturated five-membered or six-membered heterocyclic structure which is unsubstituted or substituted by hydroxyl, mercapto, C.sub.1 -C.sub.6 -alkyl, or C.sub.1 -C.sub.4 -alkanoyl and has from 1 to 3 heteroatoms from the group consisting of N, O and S, the second and third heteroatoms being a nitrogen atom,R.sup.3 is hydrogen, a hydroxy or C.sub.1 -C.sub.6 -alkoxy group,R.sup.4 is hydrogen, C.sub.1 -C.sub.4 -alkyl, halogen or methoxy,R.sup.5 is hydrogen or methoxy or tert-butyl,R.sup.6 is hydrogen methyl, nitrile or a C.sub.2 -C.sub.10 -ketal group or the radical --CHR.sup.7 OR.sup.8 --CHR.sup.7 --NR.sup.9 R.sup.10, --COR.sup.11, --SR.sup.12, ##STR2## in which R.sup.7 is hydrogen or C.sub.1 -C.sub.4 -alkyl,R.sup.8 is hydrogen, C.sub.1 -C.sub.4 -alkyl or C.sub.1 -C.sub.20 -alkanoyl or is benzoyl which is unsubstituted or substituted by methoxy, nitro, methyl or chlorine,R.sup.9 and R.sup.10 are each hydrogen, C.sub.1 -C.sub.4 -alkyl or C.sub.1 -C.sub.6 -alkanoyl or are each benzoyl which is unsubstituted or substituted as for R.sup.8, or R.sup.9 and R.sup.10, together with the nitrogen atom to which they are bonded, form a saturated, 5-membered or 6-membered heterocyclic radical which may contain oxygen as the second heteroatom,R.sup.11 is hydrogen, C.sub.1 -C.sub.4 -alkyl, --OR.sup.13 or --NR.sup.14 R.sup.15, where R.sup.13 is hydrogen, unsubstituted or hydroxyl-substituted C.sub.1 -C.sub.8 -alkyl, aryl or aralkyl which is unsubstituted or substituted by chlorine, bromine, methyl, methoxy or nitro, substitution in the case of the aralkyl group being in the aryl moiety, and where R.sup.14 and R.sup.15 are each hydrogen, unsubstituted or hydroxyl-substituted C.sub.1 -C.sub.6 -alkyl or an aralkyl or aryl group which is unsubstituted or substituted as for R.sup.13, or R.sup.14 and R.sup.15, together with the nitrogen atom to which they are bonded, form a heterocyclic radical as defined above for R.sup.9 and R.sup.10, andR.sup.12 is C.sub.1 14 C.sub.4 -alkyl,and compounds of formula Ia ##STR3## where R.sup.3, R.sup.4, R.sup.6 and L have the abovementined meanings and R.sup.17 is hydrogen or hydroxyl, and their physiologically tolerated salts, processes for their preparation and drugs and cosmetics prepared therefrom.

45. 发明授权

US5162528A Herbicidal and fungicidal agents based on substituted pyrazolin-5-one derivatives 失效
标题翻译：基于取代的吡唑啉-5-酮衍生物的除草剂和杀真菌剂
公开(公告)号：US5162528A
公开(公告)日：1992-11-10
申请号：US650354
申请日：1991-02-04
申请人： Reinhold Gehring , Markus Lindig , Heinz-Jurgen Wroblowsky , Hans-Joachim Santel , Robert R. Schmidt , Wilhelm Brandes , Robert H. Strang
发明人： Reinhold Gehring , Markus Lindig , Heinz-Jurgen Wroblowsky , Hans-Joachim Santel , Robert R. Schmidt , Wilhelm Brandes , Robert H. Strang
IPC分类号： A01N43/56 , A01N43/78 , A01N47/02 , C07D231/22 , C07D231/24 , C07D231/26 , C07D231/30 , C07D231/32 , C07D231/44 , C07D231/52 , C07D401/04 , C07D405/04 , C07D405/06 , C07D409/04 , C07D409/06 , C07D417/04
CPC分类号： C07D401/04 , A01N43/56 , A01N43/78 , A01N47/02 , C07D231/22 , C07D231/24 , C07D231/26 , C07D231/30 , C07D231/32 , C07D231/44 , C07D231/52 , C07D405/04 , C07D405/06 , C07D409/04 , C07D409/06 , C07D417/04
摘要： The invention relates to the use of partly known substituted pyrazolin-5-one derivatives of the formula (I) ##STR1## as herbicides and fungicides, new substituted pyrazolin-5-one derivatives and processes for their preparation.
摘要翻译：本发明涉及部分已知的式（I）的取代吡唑啉-5-酮衍生物作为除草剂和杀真菌剂，新的取代的吡唑啉-5-酮衍生物及其制备方法。

46. 发明授权

US5087724A Substituted benzenes useful as intermediates 失效
标题翻译：取代的苯可用作中间体
公开(公告)号：US5087724A
公开(公告)日：1992-02-11
申请号：US519727
申请日：1990-05-07
申请人： Norio Tanaka , Takuya Kakuta , Eiichi Oya , Masatoshi Baba
发明人： Norio Tanaka , Takuya Kakuta , Eiichi Oya , Masatoshi Baba
IPC分类号： C07D231/20 , A01N43/56 , B01J27/128 , B01J31/28 , C07B61/00 , C07C25/13 , C07C43/174 , C07C63/70 , C07C245/20 , C07C255/50 , C07C255/53 , C07C255/54 , C07C317/14 , C07C317/22 , C07C317/32 , C07C317/44 , C07C317/46 , C07C323/09 , C07C323/19 , C07C323/20 , C07C323/48 , C07C323/62 , C07D231/22
CPC分类号： C07C323/19 , C07C317/14 , C07C317/22 , C07C317/44 , C07C323/09 , C07C323/20 , C07C323/62 , C07D231/22
摘要： A process for producing a 4-benzoyl-5-hydroxylpyrazole of the formula III: ##STR1## which comprises reacting carbon monoxide and a 5-hydroxypyrazole of the formula II: ##STR2## with a substituted benzene of the formula I: ##STR3## in the presence of a base and a catalyst of Group VIII of the Periodic Table.
摘要翻译：制备式III的4-苯甲酰基-5-羟基吡唑的方法：（III），其包括使一氧化碳与式II的5-羟基吡唑：（II）与取代的苯的式I化合物（Ⅰ）在碱的存在下和元素周期表第VIII族的催化剂存在下进行。

47. 发明授权

US5028717A Herbicidal and fungicidal agents based on substituted pyrazolin-5-one derivatives 失效
标题翻译：基于取代的吡唑啉-5-酮衍生物的除草剂和杀真菌剂
公开(公告)号：US5028717A
公开(公告)日：1991-07-02
申请号：US433483
申请日：1989-11-08
申请人： Reinhold Gehring , Markus Lindig , Heinz-Jurgen Wroblowsky , Hans-Joachim Santel , Robert R. Schmidt , Wilhelm Brandes , Robert H. Strang
发明人： Reinhold Gehring , Markus Lindig , Heinz-Jurgen Wroblowsky , Hans-Joachim Santel , Robert R. Schmidt , Wilhelm Brandes , Robert H. Strang
IPC分类号： A01N43/56 , A01N43/78 , A01N47/02 , C07D231/22 , C07D231/24 , C07D231/26 , C07D231/30 , C07D231/32 , C07D231/44 , C07D231/52 , C07D401/04 , C07D405/04 , C07D405/06 , C07D409/04 , C07D409/06 , C07D417/04
CPC分类号： C07D401/04 , A01N43/56 , A01N43/78 , A01N47/02 , C07D231/22 , C07D231/24 , C07D231/26 , C07D231/30 , C07D231/32 , C07D231/44 , C07D231/52 , C07D405/04 , C07D405/06 , C07D409/04 , C07D409/06 , C07D417/04
摘要： The invention relates to the use of partly known substituted pyrazolin-5-one derivatives of the formula (I) ##STR1## as herbicides and fungicides, new substituted pyrazolin-5-one derivatives and processes for their preparation.

48. 发明授权

US5021446A Pyrazole compounds, insecticidal and acaricidal compositions and use 失效
标题翻译：吡唑化合物，杀虫剂和杀螨剂的组合物和用途
公开(公告)号：US5021446A
公开(公告)日：1991-06-04
申请号：US569223
申请日：1990-08-17
申请人： Naoto Meki , Kazue Nishida , Tomotoshi Imahase
发明人： Naoto Meki , Kazue Nishida , Tomotoshi Imahase
IPC分类号： A01N43/56 , A01N49/00 , C07D231/18 , C07D231/22 , C07D401/12
CPC分类号： C07D401/12 , A01N43/56 , A01N49/00 , C07D231/18 , C07D231/22
摘要： There are disclosed a pyrazole compound represented by the formula, ##STR1## wherein the substituents of R.sub.1 to R.sub.8 and the symbol Z have the specified meanings as described in the text, an insecticidal and acaricidal composition containing the same, use of said composition for control of insects and mites and a method of preparing said compound, and its intermediate.

49. 发明授权

US4977073A Silver halide light-sensitive color photographic material 失效
公开(公告)号：US4977073A
公开(公告)日：1990-12-11
申请号：US290176
申请日：1988-12-23
申请人： Osamu Ishige , Toyoaki Masukawa , Shuji Kida , Shigeto Hirabayashi
发明人： Osamu Ishige , Toyoaki Masukawa , Shuji Kida , Shigeto Hirabayashi
IPC分类号： C07C307/10 , C07C311/08 , C07C311/29 , C07C311/39 , C07D231/22 , C07D231/52 , C07D295/26 , C07D307/66 , C07D307/68 , C07D403/12 , C07D487/04 , G03C7/305
CPC分类号： C07D295/26 , C07C307/10 , C07C311/08 , C07C311/29 , C07C311/39 , C07D231/22 , C07D231/52 , C07D307/66 , C07D307/68 , C07D403/12 , C07D487/04 , G03C7/30541 , Y10S430/156 , Y10S430/16
摘要： A silver halide light-sensitive color photographic material which comprises a coupler represented by formula [I]; ##STR1## wherein A represents a coupler residue that is capable of releasing the remaining group of said coupler upon reaction with an oxidation product of a developing agent; L represents a timing group which is capable of releasing the rest of the group after said remaining group being released from A; n represents 0 or 1; X represents an oxygen or sulfur atom; Y represents a --NHSO.sub.2 R.sub.1 ' group, a ##STR2## group or a --NHCOR.sub.1 ' group, in which formulas R.sub.1 ' and R.sub.2 ' independently represent a hydrogen atom, an aliphatic group, an aromatic group or a heterocyclic group; R.sub.1 and R.sub.2 independently represent a hydrogen atom, an aliphatic group, an aromatic group or a heterocyclic group; R.sub.3 represents a substituent group; m represents 0, 1 or 2, provided that when m is 2, two R.sub.3 s may be different, and that two of R.sub.1, R.sub.2 and R.sub.3 or two of R.sub.1 ', R.sub.2 ' and R.sub.3 ' may be divalent groups to form a ring structure.

50. 发明授权

US4950678A Substituted N-(heterocyclic-substituted phenyl)-N'-benzylureas 失效
标题翻译：取代的N-（杂环取代的苯基）-N-苄基脲
公开(公告)号：US4950678A
公开(公告)日：1990-08-21
申请号：US386333
申请日：1989-07-27
申请人： Robert L. Carney , John M. Gruber , Alfred S. T. Lui
发明人： Robert L. Carney , John M. Gruber , Alfred S. T. Lui
IPC分类号： C07D207/34 , C07D209/44 , C07D231/12 , C07D231/14 , C07D231/16 , C07D231/22 , C07D231/56 , C07D235/06 , C07D235/10 , C07D249/18 , C07D409/04 , C07D521/00
CPC分类号： C07D249/08 , C07D207/34 , C07D209/44 , C07D231/12 , C07D231/14 , C07D231/16 , C07D231/22 , C07D231/56 , C07D233/56 , C07D235/06 , C07D235/10 , C07D249/18 , C07D409/04
摘要： Novel substituted N-(heterocyclic-substituted phenyl)-N'-benzoyl-ureas, processed for producing these compounds, intermediates therefor, compositions thereof and the use of the compounds for the control of pests.
摘要翻译：用于制备这些化合物的新型取代的N-（杂环取代的苯基）-n'-苯甲酰基 - 脲，其中间体，其组合物以及该化合物用于防治害虫的用途。

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