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41. 发明申请

US20080262242A1 Process For the Production of Carboxanilides 有权
标题翻译：碳酰苯胺生产工艺
公开(公告)号：US20080262242A1
公开(公告)日：2008-10-23
申请号：US12093619
申请日：2006-11-13
申请人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Hans Tobler
发明人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Hans Tobler
IPC分类号： C07D231/14
CPC分类号： C07D231/14
摘要： The present invention relates to a novel process for the preparation of a compound of general formula (I): wherein R1 is H or C1-4 alkyl and R2 is difluoromethyl or trifluoromethyl, which comprises reacting a compound of general formula (II): wherein R1 has the meaning given above and X is chloro or bromo, with a compound of general formula (III): wherein R2 has the meaning given above, in the presence of a base, a palladium catalyst and a ferrocenyl biphoshine ligand of the Josiphos type, the reaction being carried out in an ether solvent at a reflux temperature of at least 100° C.
摘要翻译：本发明涉及一种制备通式（I）化合物的新方法：其中R 1是H或C 1-4烷基，R SUP 其中R 2是二氟甲基或三氟甲基，其包括使通式（II）的化合物：其中R 1具有上面给出的含义和X是氯或溴的化合物与通式式（III）：其中R 2具有上面给出的含义，在Josiphos型的碱，钯催化剂和二茂铁基二膦配体的存在下，该反应在醚溶剂中进行在至少100℃的回流温度下

42. 发明授权

US07598395B2 Heterocyclocarboxamide derivatives 有权
标题翻译：杂环羧酰胺衍生物
公开(公告)号：US07598395B2
公开(公告)日：2009-10-06
申请号：US10530737
申请日：2003-10-14
申请人： Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： C07D231/00 , C07D207/00 , C07D295/00 , C09B5/00 , A01N47/36 , A01N43/58 , A01N43/647 , A01N43/36
CPC分类号： C07D213/82 , A01N43/32 , A01N43/36 , A01N43/40 , A01N43/56 , A01N43/76 , A01N43/78 , A01N43/90 , C07C211/61 , C07C2603/66 , C07D207/34 , C07D231/14 , C07D263/34 , C07D277/56 , C07D327/06 , C07D487/08 , C07D493/08 , C07D495/08
摘要： The invention relates to a fungicidally active compound of formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, provided that the ring is not 1,2,3-triazole, the ring being substituted by groups R8, R9 and R10; X is a single or double bond; Y is O, S, N(R11) or (CR12R13)(CR14R15)m(CR16R17)n; m is 0 or 1; n is 0 or 1; and R1 to R17 each, independently, have a range of values; to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.
摘要翻译：本发明涉及式（I）的杀真菌活性化合物：其中Het是含有一至三个杂原子的5-或6-元杂环，各自独立地选自氧，氮和硫，条件是环不为1，该环被R8，R9和R10基团取代; X是单键或双键; Y是O，S，N（R11）或（CR12R13）（CR14R15）m（CR16R17）n; m为0或1; n为0或1; 并且R 1至R 17各自独立地具有一定范围的值; 涉及这些化合物的制备，用于制备这些化合物的新型中间体，包括至少一种新化合物作为活性成分的农用化学组合物，所述组合物的制备以及使用活性成分或用于通过植物病原微生物，优选真菌控制或预防植物感染的农业或园艺成分。

43. 发明申请

US20090216027A1 MICROBIOCIDAL (E.G. FUNGICIDAL) 1,2,3-TRIAZOLE DERIVATIVES 有权
标题翻译： MICROBIOCIDAL（E.G. Fungicidal）1,2,3-三唑衍生物
公开(公告)号：US20090216027A1
公开(公告)日：2009-08-27
申请号：US12463449
申请日：2009-05-11
申请人： Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： C07D249/04 , C07D487/00
CPC分类号： C07D401/12 , A01N43/647 , A01N55/00 , C07D249/04 , C07D333/36 , C07D405/12 , C07D409/12 , C07D409/14 , C07D411/12 , C07D413/12 , C07D417/12 , C07D487/08 , C07D493/08 , C07D495/08
摘要： A compound of formula (I): where A is an ortho-substituted ring selected from a number of specified rings; R1 is halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 haloalkoxy or optionally substituted C2-4 alkenyl, optionally substituted C2-4 alkynyl or optionally substituted SO2(C1-4)alkyl (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R2 is C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkyl or C1-4 alkylthio(C1-4)alkyl or [optionally substituted aryl](C1-4)alkyl- or [optionally substituted aryl]oxy(C1-4)alkyl-(where the optionally substituted aryl moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R3 is hydrogen, CH2C≡CR4, CH2CR4═C(H)R4, CH═C═CH2 or COR5 or optionally substituted C1-4 alkyl, optionally substituted C1-4 alkoxy or optionally substituted (C1-4) alkylC(═O)O (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy, C1-4 alkyl, C1-2 haloalkoxy, hydroxy, cyano, carboxyl, methoxycarbonyl, ethoxycarbonyl, methylsulfonyl and ethylsulfonyl); each R4 is, independently, hydrogen, halogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 alkoxy(C1-4)alkyl; and R5 is hydrogen or optionally substituted C1-6 alkyl, optionally substituted C1-4 alkoxy, optionally substituted C1-4 alkoxy(C1-4)alkyl, optionally substituted C1-4 alkylthio(C1-4)alkyl or optionally substituted aryl (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen, C1-6 alkoxy, C1-6 haloalkoxy, cyano, hydroxy, methoxycarbonyl and ethoxycarbonyl).
摘要翻译：式（I）的化合物：其中A是选自多个指定环的邻位取代的环; R 1是卤素，氰基，硝基，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4卤代烷氧基或任选取代的C 2-4烯基，任选取代的C 2-4炔基或任选取代的SO 2（C 1-4）烷基（其中任选取代的部分可各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 2是C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4）烷基或C 1-4烷硫基（C 1-4）烷基或[任意取代的芳基]（C 1-4）烷基 - 或[ 芳基]氧基（C 1-4）烷基 - （其中任选取代的芳基部分可各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 3是氢，CH 2C≡CR4，CH 2 CR 4 -C（H）R 4，CH-C-CH 2或COR 5或任选取代的C 1-4烷基，任选取代的C 1-4烷氧基或任选取代的（C 1-4）烷基C（O） O（其中任选取代的部分可以各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基，C 1-4烷基，C 1-2卤代烷氧基，羟基，氰基，羧基，甲氧基羰基，乙氧基羰基，甲基磺酰基和乙基磺酰基） ; 每个R 4独立地是氢，卤素，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4烷氧基（C 1-4）烷基; 并且R 5为氢或任选取代的C 1-6烷基，任选取代的C 1-4烷氧基，任选取代的C 1-4烷氧基（C 1-4）烷基，任选取代的C 1-4烷硫基（C 1-4）烷基或任选取代的芳基（其中任选取代的部分各自可具有至多3个取代基，各自独立地选自卤素，C 1-6烷氧基，C 1-6卤代烷氧基，氰基，羟基，甲氧基羰基和乙氧基羰基）。

44. 发明授权

US07531559B2 Fungicidal 1,2,3 triazole derivatives 失效
标题翻译：杀真菌剂1,2,3三唑衍生物
公开(公告)号：US07531559B2
公开(公告)日：2009-05-12
申请号：US10524721
申请日：2003-08-18
申请人： Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： A61K31/41 , C07D249/00
CPC分类号： C07D401/12 , A01N43/647 , A01N55/00 , C07D249/04 , C07D333/36 , C07D405/12 , C07D409/12 , C07D409/14 , C07D411/12 , C07D413/12 , C07D417/12 , C07D487/08 , C07D493/08 , C07D495/08
摘要： A compound of formula (I):, where A is an ortho-substituted ring selected from a number of specified rings; R1 is halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 haloalkoxy or optionally substituted C2-4 alkenyl, optionally substituted C2-4 alkynyl or optionally substituted SO2(C1-4 alkyl) (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R2 is C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkyl or C1-4 alkylthio(C1-4)alkyl or [optionally substituted aryl](C1-4)alkyl- or [optionally substituted aryl]oxy(C1-4)alkyl (where the optionally substituted aryl moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R3 is hydrogen, CH2C≡CR4, CH2CR4═C(H)R4, CH═C═CH2 or COR5 or optionally substituted C1-4 alkyl, optionally substituted C1-4 alkoxy or optionally substituted (C1-4)alkylC(═O)O (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy, C1-4 alkyl, C1-2 haloalkoxy, hydroxy, cyano, carboxyl, methoxycarbonyl, ethoxycarbonyl, methylsulfonyl and ethylsulfonyl); each R4 is, independently, hydrogen, halogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 alkoxy(C1-4)alkyl; and R5 is hydrogen or optionally substituted C1-6 alkyl, optionally substituted C1-4 alkoxy, optionally substituted C1-4 alkoxy(C1-4)alkyl, optionally substituted C1-4 alkylthio(C1-4)alkyl or optionally substituted aryl (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen, C1-6 alkoxy, C1-6 haloalkoxy, cyano, hydroxy, methoxycarbonyl and ethoxycarbonyl).
摘要翻译：式（I）的化合物：其中A是选自若干指定环的邻位取代的环; R 1是卤素，氰基，硝基，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4卤代烷氧基或任选取代的C 2-4烯基，任选取代的C 2-4炔基或任选取代的SO 2（C 1-4烷基）（其中任选取代的部分可各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 2是C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4）烷基或C 1-4烷硫基（C 1-4）烷基或[任意取代的芳基]（C 1-4）烷基 - 或[ 芳基]氧基（C 1-4）烷基（其中任选取代的芳基部分可各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 3是氢，CH 2C≡CR4，CH 2 CR 4 -C（H）R 4，CH-C-CH 2或COR 5或任选取代的C 1-4烷基，任选取代的C 1-4烷氧基或任选取代的（C 1-4）烷基C（O） O（其中任选取代的部分可以各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基，C 1-4烷基，C 1-2卤代烷氧基，羟基，氰基，羧基，甲氧基羰基，乙氧基羰基，甲基磺酰基和乙基磺酰基） ; 每个R 4独立地是氢，卤素，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4烷氧基（C 1-4）烷基; 并且R 5为氢或任选取代的C 1-6烷基，任选取代的C 1-4烷氧基，任选取代的C 1-4烷氧基（C 1-4）烷基，任选取代的C 1-4烷硫基（C 1-4）烷基或任选取代的芳基（其中任选取代的部分各自可具有至多3个取代基，各自独立地选自卤素，C 1-6烷氧基，C 1-6卤代烷氧基，氰基，羟基，甲氧基羰基和乙氧基羰基）。

45. 发明授权

US07241721B2 Biphenyl derivatives and their use as fungicides 失效
公开(公告)号：US07241721B2
公开(公告)日：2007-07-10
申请号：US10540036
申请日：2003-12-15
申请人： Josef Ehrenfreund , Clemens Lamberth , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Clemens Lamberth , Hans Tobler , Harald Walter
IPC分类号： A01N43/56 , C07D231/18
CPC分类号： C07D213/82 , A01N43/06 , A01N43/14 , A01N43/32 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/74 , A01N43/80 , C07C25/24 , C07C211/45 , C07C211/52 , C07C217/76 , C07C219/32 , C07C233/03 , C07C2601/02 , C07C2601/08 , C07D207/34 , C07D231/14 , C07D231/16 , C07D237/24 , C07D239/28 , C07D239/30 , C07D263/34 , C07D277/56 , C07D307/68 , C07D309/28 , C07D327/06 , C07D333/38 , C07F7/0812
摘要： A fungicidally active compound of formula (I): where Het is a substituted 5- or 6-membered heterocyclic ring; R1 is hydrogen, formyl, CO—C1-4 alkyl, COO—C1-4 alkyl, C1-4 alkoxy(C1-4)alkylene, CO—C1-4 alkylenoxy(C1-4)alkyl, propargyl or allenyl; R2, R3, R4 and R5 are each, independently, hydrogen, halogen, methyl or CF3; each R6 is, independently, halogen, methyl or CF3; R7 is (Z)mC═C(Y1), (Z)mC(Y1)═C(Y2)(Y3) or tri(C1-4)alkylsilyl; X is O or S; Y1, Y2 and Y3 are each, independently, hydrogen, halogen, C1-6 alkyl [optionally substituted by one or more substituents each independently selected from halogen, hydroxy, C1-4 alkoxy, C1-4 haloalkoxy, C1-4 alkylthio, C1-4 haloalkylthio, C1-4 alkylamino, di(C1-4)alkylamino, C1-4 alkoxycarbonyl, C1-4 alkylcarbonyloxy and tri(C1-4)alkylsilyl], C2-4 alkenyl [optionally substituted by one or more substituents each independently selected from halogen], C2-4 alkynyl [optionally substituted by one or more substituents each independently selected from halogen], C3-7 cycloalkyl [optionally substituted by one or more substituents each independently selected from halogen, C1-4 alkyl and C1-4 haloalkyl] or tri(C1-4)alkylsilyl; Z is C1-4 alkylene [optionally substituted by one or more substituents each independently selected from hydroxy, cyano, C1-4 alkoxy, halogen, C1-4 haloalkyl, C1-4 haloalkoxy, C1-4 alkylthio, COOH and COO—C1-4 alkyl]; m is 0 or 1; and n is 0, 1 or 2; the invention also relates to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi

46. 发明申请

US20060154967A1 Chemical compounds 失效
公开(公告)号：US20060154967A1
公开(公告)日：2006-07-13
申请号：US10524721
申请日：2003-08-18
申请人： Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： A01N43/64 , A01N43/40 , C07D417/02 , C07D409/02 , C07D405/02 , C07D403/02
CPC分类号： C07D401/12 , A01N43/647 , A01N55/00 , C07D249/04 , C07D333/36 , C07D405/12 , C07D409/12 , C07D409/14 , C07D411/12 , C07D413/12 , C07D417/12 , C07D487/08 , C07D493/08 , C07D495/08
摘要： A compound of formula (I):, where A is an ortho-substituted ring selected from a number of specified rings; R1 is halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 haloalkoxy or optionally substituted C2-4 alkenyl, optionally substituted C2-4 alkynyl or optionally substituted SO2(C1-4 alkyl) (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R2 is C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkyl or C1-4 alkylthio(C1-4)alkyl or [optionally substituted aryl](C1-4)alkyl- or [optionally substituted aryl]oxy(C1-4)alkyl (where the optionally substituted aryl moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R3 is hydrogen, CH2C≡CR4, CH2CR4═C(H)R4, CH═C═CH2 or COR5 or optionally substituted C1-4 alkyl, optionally substituted C1-4 alkoxy or optionally substituted (C1-4)alkylC(═O)O (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy, C1-4 alkyl, C1-2 haloalkoxy, hydroxy, cyano, carboxyl, methoxycarbonyl, ethoxycarbonyl, methylsulfonyl and ethylsulfonyl); each R4 is, independently, hydrogen, halogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 alkoxy(C1-4)alkyl; and R5 is hydrogen or optionally substituted C1-6 alkyl, optionally substituted C1-4 alkoxy, optionally substituted C1-4 alkoxy(C1-4)alkyl, optionally substituted C1-4 alkylthio(C1-4)alkyl or optionally substituted aryl (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen, C1-6 alkoxy, C1-6 haloalkoxy, cyano, hydroxy, methoxycarbonyl and ethoxycarbonyl).

47. 发明申请

US20060100250A1 Biphenyl derivatives and their use as fungicides 失效
公开(公告)号：US20060100250A1
公开(公告)日：2006-05-11
申请号：US10540036
申请日：2003-12-15
申请人： Josef Ehrenfreund , Clemens Lamberth , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Clemens Lamberth , Hans Tobler , Harald Walter
IPC分类号： A01N43/36 , A01N43/40 , C07D213/46 , C07F7/02
CPC分类号： C07D213/82 , A01N43/06 , A01N43/14 , A01N43/32 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/74 , A01N43/80 , C07C25/24 , C07C211/45 , C07C211/52 , C07C217/76 , C07C219/32 , C07C233/03 , C07C2601/02 , C07C2601/08 , C07D207/34 , C07D231/14 , C07D231/16 , C07D237/24 , C07D239/28 , C07D239/30 , C07D263/34 , C07D277/56 , C07D307/68 , C07D309/28 , C07D327/06 , C07D333/38 , C07F7/0812
摘要： A fungicidally active compound of formula (1): where Het is a substituted 5- or 6-membered heterocyclic ring; R1 is hydrogen, formyl, CO-C1-4 alkyl, COO-C1-4 alkyl, C1-4 alkoxy(C1-4)alkylene, CO-C1-4 alkylenoxy(C1-4)alkyl, propargyl or allenyl; R2, R3, R4 and R5 are each, independently, hydrogen, halogen, methyl or CF3; each R6 is, independently, halogen, methyl or CF3; R7 is (Z)mC═C(Y1), (Z)mC(Y1)═C(Y2)(Y3) or tri(C1-4)alkylsilyl; X is O or S; Y1, Y2 and Y3 are each, independently, hydrogen, halogen, C1-6 alkyl [optionally substituted by one or more substituents each independently selected from halogen, hydroxy, C1-4 alkoxy, C1-4 haloalkoxy, C1-4 alkylthio, C1-4 haloalkylthio, C1-4 alkylamino, di(C1-4)alkylamino, C1-4 alkoxycarbonyl, C1-4 alkylcarbonyloxy and tri(C1-4)alkylsilyl], C2-4 alkenyl [optionally substituted by one or more substituents each independently selected from halogen], C2-4 alkynyl [optionally substituted by one or more substituents each independently selected from halogen], C3-7 cycloalkyl [optionally substituted by one or more substituents each independently selected from halogen, C1-4 alkyl and C1-4 haloalkyl] or tri(C1-4)alkylsilyl; Z is C1-4 alkylene [optionally substituted by one or more substituents each independently selected from hydroxy, cyano, C1-4 alkoxy, halogen, C1-4 haloalkyl, C1-4 haloalkoxy, C1-4 alkylthio, COOH and COO-C1-4 alkyl]; m is 0 or 1; and n is 0, 1 or 2; the invention also relates to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.

48. 发明申请

US20050221989A1 O-cyclopropyl-carboxanilides and their use as fungicides 有权
标题翻译： O-环丙基甲酰苯胺及其作为杀真菌剂的用途
公开(公告)号：US20050221989A1
公开(公告)日：2005-10-06
申请号：US10506918
申请日：2003-02-21
申请人： Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： A01N43/32 , A01N43/36 , A01N43/40 , A01N43/56 , A01N43/78 , A01N43/84 , C07B61/00 , C07C211/45 , C07C211/52 , C07C249/02 , C07C251/24 , C07D207/34 , C07D213/82 , C07D231/14 , C07D231/16 , C07D231/44 , C07D277/20 , C07D277/56 , C07D307/52 , C07D327/06 , C07D333/20 , C07D405/12 , C07D409/12 , C07D411/12 , C07D417/12 , A01N25/00 , A01N43/54 , A01N43/80 , A01N43/02 , A01N43/08
CPC分类号： C07D213/82 , A01N43/32 , A01N43/36 , A01N43/40 , A01N43/56 , A01N43/78 , A01N43/84 , C07D207/34 , C07D231/14 , C07D231/16 , C07D277/56 , C07D307/52 , C07D327/06 , C07D333/20 , C07D405/12 , C07D409/12 , C07D411/12 , C07D417/12
摘要： A compound of formula (1): F1 Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by groups R4, R5 and R6; R1 is hydrogen or halo; R2 is hydrogen or halo; R3 is optionally substituted C2-12 alkyl, optionally substituted C2-12 alkenyl, optionally substituted C2-12 alkynyl, optionally substituted C3-12 cycloalkyl, optionally substituted phenyl or optionally substituted heterocyclyl; and R4, R5 and R6 are, independently, selected from hydrogen, halo, cyano, nitro, C1-4 haloalkyl, C1-4 alkoxyl (C(1-4) alkoxyl (C1-4) alkyl and C1-4 haloalkoxy (C1-4) alkyl, provided that at least one of R4, R5 and R6 is not hydrogen. The compounds of formula (1) have plant-protective properties and are suitable for protecting plants against infestations by phytopathogenic microorganisms.
摘要翻译：式（1）的化合物：F1Het是含有一至三个杂原子的5-或6-元杂环，各自独立地选自氧，氮和硫，该环被基团R 4取代 >，R 5和R 6; R 1是氢或卤素; R 2是氢或卤素; R 3是任选取代的C 2-12烷基，任选取代的C 2-12链烯基，任选取代的C 2-12 - 任选取代的C 3-12环烷基，任选取代的苯基或任选取代的杂环基; R 4，R 5和R 6独立地选自氢，卤素，氰基，硝基，C 1〜 4个卤代烷基，C 1-4烷氧基（C 1-4（1-4））烷氧基（C 1-4 - ）烷基和C 1-4卤代烷氧基（C 1-4 - ）烷基，条件是R 4，R 5，O， >和R 6不是氢。式（1）化合物具有植物保护性质，并且适用于通过植物病原微生物保护植物免受侵袭。

49. 发明授权

US07956194B2 Microbiocidal (E.G. fungicidal) 1,2,3-triazole derivatives 有权
标题翻译：杀微生物剂（E.G.杀真菌剂）1,2,3-三唑衍生物
公开(公告)号：US07956194B2
公开(公告)日：2011-06-07
申请号：US12463449
申请日：2009-05-11
申请人： Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： C07D403/00 , C07C211/60
CPC分类号： C07D401/12 , A01N43/647 , A01N55/00 , C07D249/04 , C07D333/36 , C07D405/12 , C07D409/12 , C07D409/14 , C07D411/12 , C07D413/12 , C07D417/12 , C07D487/08 , C07D493/08 , C07D495/08
摘要： A compound of formula (I): where A is an ortho-substituted ring selected from a number of specified rings; R1 is halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 haloalkoxy or optionally substituted C2-4 alkenyl, optionally substituted C2-4 alkynyl or optionally substituted SO2(C1-4)alkyl (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R2 is C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkyl or C1-4 alkylthio(C1-4)alkyl or [optionally substituted aryl](C1-4)alkyl- or [optionally substituted aryl]oxy(C1-4)alkyl-(where the optionally substituted aryl moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R3 is hydrogen, CH2C≡CR4, CH2CR4═C(H)R4, CH═C═CH2 or COR5 or optionally substituted C1-4 alkyl, optionally substituted C1-4 alkoxy or optionally substituted (C1-4) alkylC(═O)O (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy, C1-4 alkyl, C1-2 haloalkoxy, hydroxy, cyano, carboxyl, methoxycarbonyl, ethoxycarbonyl, methylsulfonyl and ethylsulfonyl); each R4 is, independently, hydrogen, halogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 alkoxy(C1-4)alkyl; and R5 is hydrogen or optionally substituted C1-6 alkyl, optionally substituted C1-4 alkoxy, optionally substituted C1-4 alkoxy(C1-4)alkyl, optionally substituted C1-4 alkylthio(C1-4)alkyl or optionally substituted aryl (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen, C1-6 alkoxy, C1-6 haloalkoxy, cyano, hydroxy, methoxycarbonyl and ethoxycarbonyl).
摘要翻译：式（I）的化合物：其中A是选自多个指定环的邻位取代的环; R 1是卤素，氰基，硝基，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4卤代烷氧基或任选取代的C 2-4烯基，任选取代的C 2-4炔基或任选取代的SO 2（C 1-4）烷基（其中任选取代的部分可各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 2是C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4）烷基或C 1-4烷硫基（C 1-4）烷基或[任意取代的芳基]（C 1-4）烷基 - 或[ 芳基]氧基（C 1-4）烷基 - （其中任选取代的芳基部分可各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 3是氢，CH 2C≡CR4，CH 2 CR 4 = C（H）R 4，CH = C = CH 2或COR 5或任选取代的C 1-4烷基，任选取代的C 1-4烷氧基或任选取代的（C 1-4）烷基C（= O（其中任选取代的部分可以各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基，C 1-4烷基，C 1-2卤代烷氧基，羟基，氰基，羧基，甲氧基羰基，乙氧基羰基，甲基磺酰基和乙基磺酰基） ; 每个R 4独立地是氢，卤素，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4烷氧基（C 1-4）烷基; 并且R 5为氢或任选取代的C 1-6烷基，任选取代的C 1-4烷氧基，任选取代的C 1-4烷氧基（C 1-4）烷基，任选取代的C 1-4烷硫基（C 1-4）烷基或任选取代的芳基（其中任选取代的部分各自可具有至多3个取代基，各自独立地选自卤素，C 1-6烷氧基，C 1-6卤代烷氧基，氰基，羟基，甲氧基羰基和乙氧基羰基）。

50. 发明申请

US20100010063A1 HETEROCYCLOCARBOXAMIDE DERIVATIVES 有权
标题翻译：杂环碳酰胺衍生物
公开(公告)号：US20100010063A1
公开(公告)日：2010-01-14
申请号：US12549478
申请日：2009-08-28
申请人： Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： A01N43/38 , C07D209/58 , C07D307/87 , A01N43/08 , A01P1/00
CPC分类号： C07D213/82 , A01N43/32 , A01N43/36 , A01N43/40 , A01N43/56 , A01N43/76 , A01N43/78 , A01N43/90 , C07C211/61 , C07C2603/66 , C07D207/34 , C07D231/14 , C07D263/34 , C07D277/56 , C07D327/06 , C07D487/08 , C07D493/08 , C07D495/08
摘要： The invention relates to a fungicidally active compound of formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, provided that the ring is not 1,2,3-triazole, the ring being substituted by groups R8, R9 and R10; X is a single or double bond; Y is O, S, N(R11) or (CR12R13)(CR14R15)m(CR16R17)n; m is 0 or 1; n is 0 or 1; and R1 to R17 each, independently, have a range of values; to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.
摘要翻译：本发明涉及式（I）的杀真菌活性化合物：其中Het是含有一至三个杂原子的5-或6-元杂环，各自独立地选自氧，氮和硫，条件是环不为1，该环被R8，R9和R10基团取代; X是单键或双键; Y是O，S，N（R11）或（CR12R13）（CR14R15）m（CR16R17）n; m为0或1; n为0或1; 并且R 1至R 17各自独立地具有一定范围的值; 涉及这些化合物的制备，用于制备这些化合物的新型中间体，包括至少一种新化合物作为活性成分的农用化学组合物，所述组合物的制备以及使用活性成分或用于通过植物病原微生物，优选真菌控制或预防植物感染的农业或园艺成分。

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