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21. 发明授权

US6051709A Process for the diastereoselective synthesis of nucleoside analogues 失效
标题翻译：非对映选择性合成核苷类似物的方法
公开(公告)号：US6051709A
公开(公告)日：2000-04-18
申请号：US722224
申请日：1996-12-24
申请人： Michael David Goodyear , P. Owen Dwyer , Malcolm Leithead Hill , Andrew Jonathan Whitehead , Roy Hornby , Peter Hallett
发明人： Michael David Goodyear , P. Owen Dwyer , Malcolm Leithead Hill , Andrew Jonathan Whitehead , Roy Hornby , Peter Hallett
IPC分类号： C07D20060101 , C07D327/04 , C07D339/06 , C07D411/04 , C07D473/00 , C07D473/18 , C07D473/34 , C07D407/04 , C07D409/04
CPC分类号： C07D473/00 , C07D327/04 , C07D411/04
摘要： The invention relates to a diastereoselective process for the preparation of compounds of formula (I), wherein W is S, S.dbd.O, SO.sub.2 or O; X is S, S.dbd.O, SO.sub.2 or O; R.sub.1 is hydrogen or acyl, and R.sub.2 is a purine or pyrimidine base or an analogue or derivative thereof. ##STR1##
摘要翻译： PCT No.PCT / EP95 / 01503 Sec。 371日期：1996年12月24日 102（e）日期1996年12月24日PCT提交1995年4月21日PCT公布。公开号WO95 / 29174 日期：1月2日，1 9日本发明涉及制备式（I）化合物的非对映选择性方法，其中W为S，S = O，SO 2或O; X是S，S = O，SO 2或O; R1是氢或酰基，R2是嘌呤或嘧啶碱基或其类似物或衍生物。

22. 发明授权

US5817603A Substituted cyclohexene-1,2-dicarboxylic acid derivatives and intermediates for their preparation 失效
标题翻译：取代的环己烯-1,2-二羧酸衍生物及其制备中间体
公开(公告)号：US5817603A
公开(公告)日：1998-10-06
申请号：US798539
申请日：1997-02-11
申请人： Ralf Klintz , Elisabeth Heistracher , Peter Schaefer , Gerhard Hamprecht , Peter Plath , Uwe Kardorff , Matthias Gerber , Karl-Otto Westphalen , Helmut Walter
发明人： Ralf Klintz , Elisabeth Heistracher , Peter Schaefer , Gerhard Hamprecht , Peter Plath , Uwe Kardorff , Matthias Gerber , Karl-Otto Westphalen , Helmut Walter
IPC分类号： C07D317/30 , A01N37/30 , A01N37/32 , A01N37/34 , A01N37/46 , A01N43/12 , A01N43/16 , A01N43/18 , A01N43/28 , A01N43/32 , A01N43/38 , A01N43/40 , A01N43/74 , A01N43/78 , C07C233/57 , C07C233/60 , C07C233/61 , C07C233/62 , C07C233/63 , C07C237/42 , C07C251/48 , C07C251/60 , C07C255/13 , C07C255/24 , C07C255/42 , C07C255/46 , C07C255/58 , C07C271/62 , C07D209/48 , C07D295/185 , C07D307/12 , C07D307/90 , C07D309/06 , C07D335/02 , C07D339/06 , C07D339/08 , C07D401/10 , C07D413/06 , C07D413/10 , C07D417/06 , C07D417/10
CPC分类号： C07D209/48 , A01N37/30 , A01N37/32 , A01N37/34 , A01N37/46 , A01N43/12 , A01N43/16 , A01N43/40 , A01N43/74 , C07C233/61 , C07C233/63 , C07C255/13 , C07C255/46 , C07D295/185 , C07D307/12 , C07D307/90 , C07D309/06 , C07D339/08 , C07D401/10 , C07D413/10 , C07D417/10
摘要： Substituted cyclohexene-1,2-dicarboxylic acid derivatives I ##STR1## where R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5 and R.sup.6 are herein defined, or the agriculturally useful salts of Ia and Ib and intermediates for their preparation, which compounds are useful as herbicides and for the desiccation/defoliation of plants.
摘要翻译：本文定义R1，R2，R3，R4，R5和R6的取代的环己烯-1,2-二羧酸衍生物，或其农业上可用的Ia和Ib盐及其制备中间体，哪些化合物可用作除草剂和用于植物的干燥/脱叶。

23. 发明授权

US5693787A Intermediates in the synthesis of 1,3-oxathiolanyl cytosine nucleoside analogues 失效
标题翻译：中间体合成1,3-氧硫杂环戊烷胞嘧啶核苷类似物
公开(公告)号：US5693787A
公开(公告)日：1997-12-02
申请号：US464317
申请日：1995-06-05
申请人： Tarek Mansour , Haolun Jin , Allan H. L. Tse , M. Arshad Siddiqui
发明人： Tarek Mansour , Haolun Jin , Allan H. L. Tse , M. Arshad Siddiqui
IPC分类号： C07H19/00 , A61K31/513 , A61P31/12 , B01J31/02 , C07B53/00 , C07B61/00 , C07C13/10 , C07D20060101 , C07D207/00 , C07D231/04 , C07D233/02 , C07D261/02 , C07D263/04 , C07D275/02 , C07D277/04 , C07D285/04 , C07D291/04 , C07D307/04 , C07D307/16 , C07D307/18 , C07D307/24 , C07D317/08 , C07D317/24 , C07D317/32 , C07D317/34 , C07D323/02 , C07D327/04 , C07D333/48 , C07D339/02 , C07D339/06 , C07D341/00 , C07D403/04 , C07D405/04 , C07D407/04 , C07D409/04 , C07D411/04 , C07D411/12 , C07D411/14 , C07D413/04 , C07D419/04 , C07D471/00 , C07D473/00 , C07D473/06 , C07D473/30 , C07D473/34 , C07H19/04 , C07H19/06 , C07H19/16 , C07D333/36 , C07D333/42
CPC分类号： C07D405/04 , C07D307/24 , C07D317/32 , C07D317/34 , C07D327/04 , C07D339/06 , C07D409/04 , C07D411/04 , C07H19/04 , C07H19/06 , C07H19/16
摘要： The present invention relates to highly diastereoselective processes for production of cis-nucleosides and nucleoside analogues and derivatives in high optical purity and intermediates useful in those processes.
摘要翻译：本发明涉及用于生产高光学纯度的顺式核苷和核苷类似物和衍生物的高度非对映选择性方法以及在这些方法中有用的中间体。

24. 发明授权

US5631277A (2-one (or thione)-1,3-dithiole 4,5-diyl) bis(thiocyanate) compounds, compositions containing the compounds and their use as an antimicrobial and marine antifouling agents 失效
标题翻译：（2-酮（或硫酮）-1,3-二硫杂-4,5-二基）双（硫氰酸酯）化合物，含有这些化合物的组合物及其作为抗微生物剂和海洋防污剂的用途
公开(公告)号：US5631277A
公开(公告)日：1997-05-20
申请号：US676621
申请日：1996-07-10
申请人： Duane R. Romer , Weishi W. Wu , Ravi B. Shankar , R. Garth Pews
发明人： Duane R. Romer , Weishi W. Wu , Ravi B. Shankar , R. Garth Pews
IPC分类号： A01N43/28 , C07D339/06 , C09D5/14 , C09D5/16
CPC分类号： C09D5/1625 , A01N43/28 , C07D339/06 , C09D5/14
摘要： Disclosed is (2-thione-1,3-dithiole 4,5-diyl) bis(thiocyanate), its preparation and its use as an antimicrobial and marine antifouling agent.
摘要翻译：公开了（2-硫酮-1,3-二硫杂环戊烷4,5-二基）双（硫氰酸酯），其制备及其作为抗微生物剂和海洋防污剂的用途。

25. 发明授权

US5530141A 2,4-diaryl-1,3-dithiolanes; 2,4-diaryl-1,3-dioxolanes; 2,4-diaryl-1,3-oxathiolanes; and 2,5-diaryl-1,3-oxathiolanes for the treatment of disorders mediated by platelet activating factor or products of 5-lipoxygenase 失效
标题翻译： 2,4-二芳基-1,3-二硫戊环; 2,4-二芳基-1,3-二氧戊环; 2,4-二芳基-1,3-氧硫杂环戊烷; 和2,5-二芳基-1,3-氧硫杂环戊烷，用于治疗血小板活化因子或5-脂氧合酶产物介导的病症
公开(公告)号：US5530141A
公开(公告)日：1996-06-25
申请号：US944845
申请日：1992-09-14
申请人： T. Y. Shen , David M. Goldstein
发明人： T. Y. Shen , David M. Goldstein
IPC分类号： C07D317/28 , C07D327/04 , C07D339/06 , C07D409/12 , C07D339/02
CPC分类号： C07D409/12 , C07D317/28 , C07D327/04 , C07D339/06
摘要： 2,4-Diaryl-1,3-dithiolanes; 2,4-diaryl-1,3-dioxolanes; 2,4-diaryl-1,3-oxathiolanes; and 2,5-diaryl-1,3-oxathiolanes are disclosed that reduce the chemotaxis and respiratory burst leading to the formation of damaging oxygen radicals of polymorphonuclear leukocytes during an inflammatory or immune response. The compounds exhibit this biological activity by acting as PAF receptor antagonists, by inhibiting the enzyme 5-lipoxygenase, or by exhibiting dual activity, i.e., by acting as both a PAF receptor antagonist and inhibitor of 5-lipoxygenase.A method to treat disorders mediated by PAF or leukotrienes is also disclosed, that includes administering an effective amount of one or more of the above-identified compounds or a pharmaceutically acceptable salt thereof, optionally in a pharmaceutically acceptable carrier.
摘要翻译： 2,4-二芳基-1,3-二硫戊环; 2,4-二芳基-1,3-二氧戊环; 2,4-二芳基-1,3-氧硫杂环戊烷; 并且公开了2,5-二芳基-1,3-氧硫杂环戊烷，其减少趋化性和呼吸道爆发，导致在炎性或免疫反应期间形成多形核白细胞的有害氧自由基。该化合物通过作为PAF受体拮抗剂，通过抑制酶5-脂氧合酶，或通过显示双重活性，即作为PAF受体拮抗剂和5-脂肪氧合酶抑制剂两者而表现出该生物学活性。还公开了治疗由PAF或白细胞三烯介导的病症的方法，其包括任选地在药学上可接受的载体中施用有效量的一种或多种上述化合物或其药学上可接受的盐。

26. 发明授权

US5508412A Phthalimides useful as intermediate compounds 失效
标题翻译：邻苯二甲酰亚胺可用作中间体化合物
公开(公告)号：US5508412A
公开(公告)日：1996-04-16
申请号：US508044
申请日：1995-07-27
申请人： Juergen Kast , Norbert Meyer , Ulf Misslitz , Albrecht Harreus , Harald Rang , Matthias Gerber , Helmut Walter , Karl-Otto Westphalen
发明人： Juergen Kast , Norbert Meyer , Ulf Misslitz , Albrecht Harreus , Harald Rang , Matthias Gerber , Helmut Walter , Karl-Otto Westphalen
IPC分类号： A01N35/10 , A01N43/14 , A01N49/00 , C07C239/20 , C07C251/42 , C07C251/52 , C07C251/54 , C07C251/58 , C07C255/64 , C07C317/28 , C07C323/47 , C07D213/30 , C07D261/08 , C07D275/02 , C07D307/12 , C07D307/52 , C07D309/06 , C07D309/22 , C07D309/28 , C07D317/26 , C07D317/28 , C07D333/20 , C07D333/22 , C07D339/06 , C07D405/12 , C07D409/12 , C07D413/12 , C07D209/48
CPC分类号： C07D213/30 , A01N35/10 , A01N43/14 , A01N49/00 , C07C239/20 , C07C251/42 , C07C251/52 , C07C317/28 , C07C323/47 , C07D261/08 , C07D307/12 , C07D309/06 , C07D309/22 , C07D309/28 , C07D317/26 , C07D333/22 , C07D339/06 , C07D405/12 , C07D409/12 , C07D413/10 , C07D413/12 , C07C2101/02 , C07C2101/08 , C07C2101/14 , C07C2101/16
摘要： Unsaturated cyclohexenone oxime ethers I ##STR1## (Q.dbd.H, alkylcarbonyl, benzoyl, alkali metal or alkaline earth metal ion, substituted or unsubstituted ammonium ion, phosphonium ion, sulfonium ion, sulfoxonium ion, an equivalent of a transition metal cation;W=--C.tbd.C-- or --CH.dbd.CH--;R.sup.1 =substituted or unsubstituted cycloalkyl, cycloalkenyl or 6-membered heterocyclic group which has 1-2 oxygen and/or sulfur atoms and can be saturated or partially unsaturated; substituted or unsubstituted 5-membered saturated heterocycle with 1-2 oxygen and/or sulfur atoms; substituted or unsubstituted 5-membered heteroaromatic group with 1-2 nitrogen atoms and/or 1 oxygen or sulfur atom; substituted or unsubstituted phenyl, pyridyl or R.sup.9 -X-substituted alkyl with X=O, S, --SO--, --SO.sub.2 -- and R.sup.9 =alkyl, phenyl, 5/6-membered hetaryl with 1-3 hetero atoms;R.sup.2 =alkyl;R.sup.3 =H, alkyl;R.sup.4 =H, halogen, alkyl;R.sup.5 =H, alkyl;or R.sup.3 +R.sup.4, R.sup.3 +R.sup.5 or R.sup.4 +R.sup.5 together form C.sub.2 -C.sub.4 -alkylene or C.sub.2 -C.sub.4 -alkenylene;R.sup.6 =H, alkyl, unsubstituted or phenyl-substituted haloalkyl, alkenyl, alkoxyalkyl, alkylthioalkyl, substituted or unsubstituted cycloalkyl or cycloalkenyl; substituted or unsubstituted phenyl or pyridyl) are suitable as herbicides.
摘要翻译：不饱和环己烯酮肟醚I（Q = H，烷基羰基，苯甲酰基，碱金属或碱土金属离子，取代或未取代的铵离子，鏻离子，锍离子，氧锍离子，当量的过渡金属阳离子; W = -C 3BOND C-或-CH = CH-; R 1 =具有1-2个氧和/或硫原子并且可以是饱和或部分不饱和的取代或未取代的环烷基，环烯基或6元杂环基;取代或未取代的5 具有1-2个氧和/或硫原子的饱和杂环;具有1-2个氮原子和/或1个氧或硫原子的取代或未取代的5元杂芳基;取代或未取代的苯基，吡啶基或R9-X取代的具有X = O，S，-SO - ， - SO 2 - 和R 9 =烷基的苯基，具有1-3个杂原子的5-6元杂芳基; R 2 =烷基; R 3 = H，烷基; R 4 = H，卤素，烷基; R 5 = H，烷基或R 3 + R 4，R 3 + R 5或R 4 + R 5一起形成C 2 -C 4亚烷基或C 2 -C 4亚烯基; R 6 = H，或苯基取代的卤代烷基，烯基，烷氧基烷基，烷硫基烷基，取代或未取代的环烷基或环烯基; 取代或未取代的苯基或吡啶基）适合作为除草剂。

27. 发明授权

US5407896A Unsaturated cyclohexenone oxime ethers and herbicidal compositions thereof 失效
标题翻译：不饱和环己烯酮肟醚及其除草组合物
公开(公告)号：US5407896A
公开(公告)日：1995-04-18
申请号：US10318
申请日：1993-01-28
申请人： Juergen Kast , Norbert Meyer , Ulf Misslitz , Albrecht Harreus , Harald Rang , Matthias Gerber , Helmut Walter , Karl-Otto Westphalen
发明人： Juergen Kast , Norbert Meyer , Ulf Misslitz , Albrecht Harreus , Harald Rang , Matthias Gerber , Helmut Walter , Karl-Otto Westphalen
IPC分类号： A01N35/10 , A01N43/14 , A01N49/00 , C07C239/20 , C07C251/42 , C07C251/52 , C07C251/54 , C07C251/58 , C07C255/64 , C07C317/28 , C07C323/47 , C07D213/30 , C07D261/08 , C07D275/02 , C07D307/12 , C07D307/52 , C07D309/06 , C07D309/22 , C07D309/28 , C07D317/26 , C07D317/28 , C07D333/20 , C07D333/22 , C07D339/06 , C07D405/12 , C07D409/12 , C07D413/12 , A01N43/16 , C07D309/34
CPC分类号： C07D213/30 , A01N35/10 , A01N43/14 , A01N49/00 , C07C239/20 , C07C251/42 , C07C251/52 , C07C317/28 , C07C323/47 , C07D261/08 , C07D307/12 , C07D309/06 , C07D309/22 , C07D309/28 , C07D317/26 , C07D333/22 , C07D339/06 , C07D405/12 , C07D409/12 , C07D413/10 , C07D413/12 , C07C2101/02 , C07C2101/08 , C07C2101/14 , C07C2101/16
摘要： Unsaturated cyclohexenone oxime ethers I ##STR1## (Q=H, alkylcarbonyl, benzoyl, alkali metal or alkaline earth metal ion, substituted or unsubstituted ammonium ion, phosphonium ion, sulfonium ion, sulfoxonium ion, an equivalent of a transition metal cation;W=--C.tbd.C-- or --CH.dbd.CH--;R.sup.1 =substituted or unsubstituted cycloalkyl, cycloalkenyl or 6-membered heterocyclic group which has 1-2 oxygen and/or sulfur atoms and can be saturated or partially unsaturated; substituted or unsubstituted 5-membered saturated heterocycle with 1-2 oxygen and/or sulfur atoms; substituted or unsubstituted 5-membered heteroaromatic group with 1-2 nitrogen atoms and/or 1 oxygen or sulfur atom; substituted or unsubstituted phenyl, pyridyl or R.sup.9 --X-substituted alkyl with X=O, S, --SO--, --SO.sub.2 -- andR.sup.9 =alkyl, phenyl, 5/6-membered hetaryl with 1-3 hetero atoms;R.sup.2 =alkyl;R.sup.3 =H, alkyl;R.sup.4 =H, halogen, alkyl;R.sup.5 =H, alkyl;or R.sup.3 +R.sup.4, R.sup.3 +R.sup.5 or R.sup.4 +R.sup.5 together form C.sub.2 -C.sub.4 -alkylene or C.sub.2 -C.sub.4 -alkenylene;R.sup.6 =H, alkyl, unsubstituted or phenyl-substituted haloalkyl, alkenyl, alkoxyalkyl, alkylthioalkyl, substituted or unsubstituted cycloalkyl or cycloalkenyl; substituted or unsubstituted phenyl or pyridyl) are suitable as herbicides.
摘要翻译：不饱和环己烯酮肟醚I（Q = H，烷基羰基，苯甲酰基，碱金属或碱土金属离子，取代或未取代的铵离子，鏻离子，锍离子，氧锍离子，当量的过渡金属阳离子; W = -C 3BOND C-或-CH = CH-; R 1 =具有1-2个氧和/或硫原子并且可以是饱和或部分不饱和的取代或未取代的环烷基，环烯基或6元杂环基;取代或未取代的5 具有1-2个氧和/或硫原子的饱和杂环;具有1-2个氮原子和/或1个氧或硫原子的取代或未取代的5元杂芳基;取代或未取代的苯基，吡啶基或R9-X取代的具有X = O，S，-SO - ， - SO 2 - 和R 9 =烷基的苯基，具有1-3个杂原子的5-6元杂芳基; R 2 =烷基; R 3 = H，烷基; R 4 = H，卤素，烷基; R 5 = H，烷基或R 3 + R 4，R 3 + R 5或R 4 + R 5一起形成C 2 -C 4亚烷基或C 2 -C 4亚烯基; R 6 = H，或苯基取代的卤代烷基，烯基，烷氧基烷基，烷硫基烷基，取代或未取代的环烷基或环烯基; 取代或未取代的苯基或吡啶基）适合作为除草剂。

28. 发明授权

US5399710A Protein labeling reagents 失效
公开(公告)号：US5399710A
公开(公告)日：1995-03-21
申请号：US994939
申请日：1992-12-22
申请人： Sudhakar Kasina , Ananthachari Srinivasan , James Sanderson , Alan R. Fritzberg
发明人： Sudhakar Kasina , Ananthachari Srinivasan , James Sanderson , Alan R. Fritzberg
IPC分类号： A61K51/10 , C07C319/18 , C07C323/52 , C07D307/60 , C07D339/06 , C07D495/04 , C07D487/04 , C07D207/38 , C07C101/04
CPC分类号： C07D495/04 , A61K51/1093 , C07C319/18 , C07D307/60 , C07D339/06 , A61K2123/00 , Y02P20/55
摘要： Novel labeling reagents are useful for radiolabeling proteins such as antibodies with radionuclide metals such as .sup.99m Tc, .sup.186 Re, and .sup.188 Re. The reagents are of the following formula: ##STR1## wherein: each X is independently chosen from O, S, NH, or NR.sub.2, wherein R.sub.2 is a protecting group or an electron withdrawing group;R.sub.1 represents a protecting group, wherein each R.sub.1 is a separate protecting group or the two R.sub.1 symbols are taken together to represent a single protecting group; andeach T is independently chosen from hydrogen, lower alkyl groups of from 1 to about 6 carbon atoms, electron withdrawing groups, and lower alkyl groups of from 1 to about 6 carbon atoms substituted with electron withdrawing group(s).

29. 发明授权

US5378744A Synthetic polymer compositions containing charge transfer complexes, their preparation and the use thereof 失效
标题翻译：含有电荷转移络合物的合成聚合物组合物及其制备及其应用
公开(公告)号：US5378744A
公开(公告)日：1995-01-03
申请号：US7426
申请日：1993-01-22
申请人： Peter Chetcuti
发明人： Peter Chetcuti
IPC分类号： C08K5/00 , C07D339/06 , C07D345/00 , C08K5/45 , C08K5/48 , C08L101/00 , H01B1/00 , H01B1/12 , H01B1/20 , C08K5/3415 , C08K5/3417
CPC分类号： H01B1/121 , C07D339/06 , C07D345/00 , C08K5/45 , C08K5/48
摘要： A composition comprising a) a thermosetting, thermoplastic or structurally crosslinked polymer and b) a charge transfer complex of formula I in the form of a network of crystal needles in the polymer matrix[A].sup..crclbar. B.sup..sym. (I),wherein A is a compound of formula II or a mixture of compounds of formula II ##STR1## wherein the R substituents are identical and are H or C.sub.1 -C.sub.4 alkyl, or the adjacent R substituents, taken together, are --(CH.sub.2).sub.3 --or --(CH.sub.2).sub.4 --; R.sub.1 or C.sub.1 -C.sub.4 alkyl; and H.sub.1 is .dbd.N--CN, and X.sub.2, X.sub.3 and X.sub.4 are each independently of one another .dbd.O or .dbd.N--CN, and B is a compound of formula III or IIIa ##STR2## wherein R.sub.2, R.sub.3, R.sub.4 and R.sub.5 are each independently of one another H, linear or branched C.sub.1 -C.sub.18 -alkyl-(Z.sub.1).sub.n --, phenyl-(Z.sub.1).sub.n - or benzyl-(Z.sub.1).sub.n --which are unsubstituted or substituted by C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy or C.sub.1 -C.sub.4 alkylthio, or R.sub.2 and R.sub.3 as well as R.sub.4 and R.sub.5 are together, each independently of the other, trimethylene, tetramethylene, --Z.sub.2 --(CH.sub.2)--Z.sub.2 --, --Z.sub.2 --(CH.sub.2).sub.2 --Z.sub.2 --, --Z.sub.1 --CH.dbd.CH--Z.sub.1 --or --CH.dbd.CH--CH.dbd.CH--, each unsubstituted or substituted by C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy or C.sub.1 -C.sub.4 alkylthio, n is 0 or 1 steht, Y.sub.1 and Y.sub.2 are each independently of the other --S--or --Se--, Z.sub.1 is --S-- or --Se--, Z.sub.2 is --O--, --S--or --Se--, Z is --S--, --Se--or NR.sub.7, and R.sub.7 is H, C.sub.1 -C.sub.6 alkyl, phenyl or benzyl, and R.sub.6 is H, C.sub.1 -C.sub.4 alkyl, phenyl or benzyl. The composition is an electric conductor.
摘要翻译：一种组合物，其包含a）热固性，热塑性或结构交联的聚合物和b）聚合物基质[A]（ - ）B（+）（I）中的结晶针网络形式的式I的电荷转移络合物，其中A是式II化合物或式II化合物齿状且为H或C 1 -C 4烷基或相邻R取代基的化合物一起为 - （CH 2）3 - 或 - （CH 2）4 - ; R1或C1-C4烷基; 并且H 1是= N-CN，且X 2，X 3和X 4各自独立地为= O或= N-CN，B为式III或IIIa的化合物。（III）（IIIa）其中R 2，R 3，R 4和R 5彼此独立地为H，直链或支链C 1 -C 18烷基 - （Z 1）n - ，苯基 - （Z 1）n或苄基 - （Z 1）n - 是未取代的或被C 1 -C 4烷基，C 1 -C 4烷基，C 1 -C 4烷氧基或C 1 -C 4烷硫基取代，或者R 2和R 3以及R 4和R 5各自独立地为三亚甲基，四亚甲基，-Z 2 - （CH 2），-Z2-（CH2）2-Z2-，-Z1-CH = CH-Z1-或-CH = CH-CH = CH-，各自未被取代或被C1-C4烷基，C1-C4烷氧基或C1-C4烷硫基取代，n 为0或1个，Y1和Y2各自独立地为-S-或-Se-，Z1为-S-或-Se-，Z2为-O - ， - S-或-Se-，Z为 - S-，-Se-或NR7，R7是H，C1-C6烷基，苯基或苄基，R6是H，C1-C4烷基，苯基或苄基。组合物是电导体。

30. 发明授权

US5374609A Cyclohexenone oxime ethers and their use as herbicides 失效
标题翻译：环己烯酮肟醚及其作为除草剂的用途
公开(公告)号：US5374609A
公开(公告)日：1994-12-20
申请号：US65912
申请日：1993-05-25
申请人： Juergen Kast , Norbert Meyer , Ulf Misslitz , Albrecht Harreus , Thomas Kuekenhoehner , Harald Rang , Matthias Gerber , Karl-Otto Westphalen , Helmut Walter
发明人： Juergen Kast , Norbert Meyer , Ulf Misslitz , Albrecht Harreus , Thomas Kuekenhoehner , Harald Rang , Matthias Gerber , Karl-Otto Westphalen , Helmut Walter
IPC分类号： A01N35/10 , A01N37/22 , A01N37/34 , A01N43/08 , A01N43/10 , A01N43/14 , A01N43/16 , A01N43/28 , A01N43/80 , A01P13/00 , C07C239/20 , C07C249/08 , C07C251/42 , C07C251/52 , C07C251/54 , C07C251/58 , C07C251/60 , C07C255/62 , C07C323/47 , C07D213/30 , C07D261/08 , C07D275/02 , C07D307/10 , C07D309/06 , C07D309/08 , C07D309/20 , C07D317/14 , C07D333/06 , C07D335/02 , C07D339/06 , A01N33/24 , C07C251/50
CPC分类号： C07D213/30 , A01N35/10 , A01N43/14 , C07C239/20 , C07C251/42 , C07C251/52 , C07D261/08 , C07D309/06 , C07D309/08 , C07D335/02 , C07C2101/12 , C07C2101/14
摘要： Cyclohexenone oxime ethers I ##STR1## where R.sup.1 is C.sub.1 -C.sub.6 -alkyl, A is unsubstituted or substituted C.sub.3 -C.sub.6 -alkynylene, Z is unsubstituted or substituted phenyl or a 5-membered or 6-membered heteroaromatic and R.sup.2 is C.sub.1 -C.sub.4 -alkoxy-C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.4 -alkylthio-C.sub.1 -C.sub.6 -alkyl, unsubstituted or substituted C.sub.3 -C.sub.7 -cycloalkyl or C.sub.5 -C.sub.7 -cycloalkenyl, an unsubstituted or substituted 5-membered saturated heterocyclic structure having one or two hetero atoms, an unsubstituted or substituted 6-membered or 7-membered saturated or monounsaturated or diunsaturated heterocyclic structure having one or two hetero atoms, an unsubstituted or substituted 5-membered heteroaromatic having one to three hetero atoms or unsubstituted or substituted phenyl or pyridyl, and their agriculturally useful salts and esters of C.sub.1 -C.sub.10 -carboxylic acids and inorganic acids, are suitable as herbicides.
摘要翻译：环己烯酮肟醚I（I）其中R1是C1-C6-烷基，A是未取代或取代的C3-C6-亚炔基，Z是未取代或取代的苯基或5元或6元杂芳族，R2是C1 C 1 -C 4 - 烷氧基-C 1 -C 6 - 烷基，C 1 -C 4 - 烷硫基-C 1 -C 6 - 烷基，未取代或取代的C 3 -C 7 - 环烷基或C 5 -C 7 - 环烯基，未取代或取代的5元饱和杂环结构，或两个杂原子，具有一个或两个杂原子的未取代或取代的6元或7元饱和或单不饱和或不饱和杂环结构，未取代或取代的具有1至3个杂原子的5元杂芳基或未取代或取代的苯基或吡啶基及其农业上有用的C1-C10-羧酸和无机酸的盐和酯类，适用作除草剂。

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