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21. 发明授权

US4581453A Guanidinothiazole derivatives containing alkylene bridges, and their use for influencing lipid metabolism 失效
标题翻译：含有亚烷基桥的胍基噻唑衍生物及其用于影响脂质代谢的用途
公开(公告)号：US4581453A
公开(公告)日：1986-04-08
申请号：US492776
申请日：1983-05-09
申请人： Joachim Ippen , Elisabeth Perzborn , Walter Puls , Klaus Schaller , Friedel Seuter
发明人： Joachim Ippen , Elisabeth Perzborn , Walter Puls , Klaus Schaller , Friedel Seuter
IPC分类号： A61K31/425 , A61K31/505 , A61P3/00 , A61P3/06 , A61P7/02 , A61P9/10 , A61P31/04 , A61P31/10 , C07D239/16 , C07D249/08 , C07D277/22 , C07D277/32 , C07D277/34 , C07D277/48 , C07D417/12 , C07D417/14 , C07D239/02 , A61K31/495
CPC分类号： C07D417/12 , C07D239/16 , C07D277/48 , C07D417/14
摘要： The invention relates to guanidinothiazol derivatives of Formula (I) as defined herein, said compounds being useful for influencing lipid metabolism, as antithombotic agents and as antimycotic agents. Also included in the invention are compositions containing said guanidinothiazol derivatives of Formula (I) and the use of said compounds and compositions for treatment of the above-mentioned conditions. In addition, the invention includes methods for the manufacture of the guanidinothiazole derivatives of Formula (I).
摘要翻译：本发明涉及如本文所定义的式（I）的胍基噻唑衍生物，所述化合物可用于影响脂质代谢，作为抗栓剂和抗真菌剂。本发明还包括含有式（I）的胍基噻唑衍生物的组合物以及所述化合物和组合物用于治疗上述病症的用途。此外，本发明包括制备式（I）的胍基噻唑衍生物的方法。

22. 发明授权

US4558139A Bafilomycin pesticides 失效
标题翻译：巴法洛霉素农药
公开(公告)号：US4558139A
公开(公告)日：1985-12-10
申请号：US589380
申请日：1984-03-14
申请人： Hans-Paul Hagenmaier , Gerhard Werner , Hannelore Drautz , Hartwig Holst , Hans Zahner , Wilhelm Brandes , Paul Reinecke , Gerhard Zoebelein , Wilhelm Stendel , Peter Andrews , Klaus Schaller
发明人： Hans-Paul Hagenmaier , Gerhard Werner , Hannelore Drautz , Hartwig Holst , Hans Zahner , Wilhelm Brandes , Paul Reinecke , Gerhard Zoebelein , Wilhelm Stendel , Peter Andrews , Klaus Schaller
IPC分类号： C12P17/16 , A01N43/22 , A01N63/02 , A61K31/365 , A61P33/10 , C07D407/06 , C07H7/06 , C12P19/02 , C12P19/44
CPC分类号： C12R1/465 , C07H7/06 , C12P19/02 , C12P19/44
摘要： Bafilomycins of the formula ##STR1## in which R.sup.1 is hydrogen or CH.sub.3, andR.sup.2 is hydrogen, or the group ##STR2## are produced by culturing certain streptomyces, e.g. Tu 1922, Tu 2437 and Tu 2599. Those wherein at least one of the OH groups is acylated are new. The compounds are pesticidally active.
摘要翻译： R1为氢或CH3，R2为氢的式（Ⅰ）的Bafilomycins或通过培养某些链霉菌如 Tü1922，Tü2437和Tü2599.其中至少一个OH基团被酰化的那些是新的。该化合物具有杀虫活性。

23. 发明申请

US20060028718A1 Illuminating device and optical object-analyzing device 有权
标题翻译：照明装置和光学物体分析装置
公开(公告)号：US20060028718A1
公开(公告)日：2006-02-09
申请号：US10520954
申请日：2003-07-10
申请人： Matthias Seel , Klaus Schaller , Ines Schaller
发明人： Matthias Seel , Klaus Schaller , Ines Schaller
IPC分类号： G02B21/06
CPC分类号： G01N21/6458
摘要： Disclosed is an illuminating device (10) comprising a light source (12), optical components (16, 18, 20) that define a plurality of light paths (14) originating from the light source, a light-conditioning array (22) on at least one of said light paths, a least one light output (34) to which an associated device that is to be supplied with light or conditioned light is or can be connected, at least one light path-selecting unit (24) which is provided with several input light path sections associated with another light path and at least one output light path section leading to said light output or another associated light output. Each light path can optionally be connected to the light output via the output light path section or to a predefined or selected light output via a predefined or selected output light path section as the selected light path in a corresponding selection mode of the light path-selecting unit by means of the light path-selecting unit that can be switched between several selection modes.
摘要翻译：公开了一种照明装置（10），包括光源（12），光学部件（16,18,20），其限定源自光源的多个光路（14），光调节阵列（22），至少一个所述光路，至少一个光输出（34），待供应光或调节光的相关联装置可连接至该光输出（34），至少一个光路选择单元（24）设置有与另一光路相关联的多个输入光路部分以及导致所述光输出或另一相关光输出的至少一个输出光路部分。每个光路可以可选地经由输出光路部分连接到光输出，或者通过预定义或选择的输出光路部分连接到预定义或选择的光输出，作为在光路选择的相应选择模式中的所选光路通过可以在几种选择模式之间切换的光路选择单元来实现。

24. 发明授权

US06204272B1 Use of aminothiazoles for treating wounds and skin 失效
标题翻译：使用氨基噻唑治疗伤口和皮肤
公开(公告)号：US06204272B1
公开(公告)日：2001-03-20
申请号：US09319974
申请日：1999-08-10
申请人： Klaus Schaller , Bernd Baasner , Magdalena Liszkay , Hans-Otto Werling , Ehrhardt Proksch
发明人： Klaus Schaller , Bernd Baasner , Magdalena Liszkay , Hans-Otto Werling , Ehrhardt Proksch
IPC分类号： A61K31505
CPC分类号： A61K31/506
摘要： The invention relates to the use of substituted 2-aminothiazoles for promoting wound healing.
摘要翻译：本发明涉及取代的2-氨基噻唑用于促进伤口愈合的用途

25. 发明授权

US5104879A Antimycotically active substituted 2-aminothiazoles 失效
标题翻译：抗微生物活性取代的2-氨基丁酸
公开(公告)号：US5104879A
公开(公告)日：1992-04-14
申请号：US596626
申请日：1990-10-11
申请人： Joachim Ippen , Bernd Baasner , Klaus Schaller , Miklos von Bittera
发明人： Joachim Ippen , Bernd Baasner , Klaus Schaller , Miklos von Bittera
IPC分类号： A61K31/505 , A61P31/04 , C07C45/00 , C07C45/63 , C07C49/80 , C07C49/84 , C07D417/12 , C07D417/14
CPC分类号： C07D417/12 , C07C45/004 , C07C45/63 , C07C49/80 , C07C49/84 , C07D417/14
摘要： Antimicotically active 2-aminothiazoles have been found having the formula ##STR1## in which R.sup.1 represents hydrogen or alkyl andR.sup.2 represents optionally substituted cyclohexyl or phenyl which is substituted by halogen, alkyl, halogenoalkyl, halogenoalkoxy, dioxyhalogenoalkyl or halogenoalkylthio,and their physiologically tolerable acid addition salts,with the exception of the compounds 4-(4-chlorophenyl)-2-[2-(1,4,5,6-tetrahydropyrimidinyl)-amino]thiazole and 4-(2,4-dichlorophenyl)-2-[2-(1,4,5,6-tetrahydropyrimidinyl)-amino]-thiazole and 4-(4-chloro-2-methylphenyl)-2-[2-(1,4,5,6-tetrahydropyrimidinyl)-amino]-thiazole and with the exception of the physiologically tolerable acid addition salts of these compoundshave been found.
摘要翻译：已经发现具有式“IMAGE”的反活性2-氨基噻唑，其中R1代表氢或烷基，R2代表任选取代的环己基或被卤素，烷基，卤代烷基，卤代烷氧基，二卤基烷基或卤代烷硫基取代的苯基，以及它们的生理可耐受酸加成盐，除4-（4-氯苯基）-2- [2-（1,4,5,6-四氢嘧啶基） - 氨基]噻唑和4-（2,4-二氯苯基）-2- [2-（1,4,5,6-四氢嘧啶基） - 氨基] - 噻唑和4-（4-氯-2-甲基苯基）-2- [2-（1,4,5,6-四氢嘧啶基） - 氨基] - 噻唑，除了这些化合物的生理可耐受酸加成盐之外。

26. 发明授权

US5096889A Antimycotic compositions of nikkomycin compounds and azole antimycotics 失效
标题翻译：尼科霉素化合物和唑类抗霉素的抗真菌组合物
公开(公告)号：US5096889A
公开(公告)日：1992-03-17
申请号：US640769
申请日：1991-01-14
申请人： Richard F. Hector , Klaus Schaller , Heinrich F. Moeschler , Manfred Plempel
发明人： Richard F. Hector , Klaus Schaller , Heinrich F. Moeschler , Manfred Plempel
IPC分类号： A61K31/415 , A61K31/70
CPC分类号： A61K31/70
摘要： Nikkomycin compounds have been found to be orally or parenterally effective as anti-fungals in animals. They may be used alone or, preferably, in combination with azole antimycotics for a synergistic anti-fungal effect.
摘要翻译：已经发现尼古霉素化合物在动物中作为抗真菌剂是口服或肠胃外有效的。它们可以单独使用或优选与唑类抗霉素组合使用，用于协同的抗真菌作用。

27. 发明授权

US5091375A Nikkomycin derivatives 失效
标题翻译：尼古霉素衍生物
公开(公告)号：US5091375A
公开(公告)日：1992-02-25
申请号：US464087
申请日：1990-01-12
申请人： Richard F. Hector , Klaus Schaller , Heinrich F. Moeschler , Manfred Blempel
发明人： Richard F. Hector , Klaus Schaller , Heinrich F. Moeschler , Manfred Blempel
IPC分类号： A61K38/00 , C07H19/06 , C07K5/06 , C07K5/065 , C07K5/078 , C07K5/083 , C07K5/087 , C07K5/09 , C07K5/093 , C07K9/00
CPC分类号： C07H19/06 , C07K5/06034 , C07K5/0606 , C07K5/06078 , C07K5/06139 , C07K5/06156 , C07K5/06191 , C07K5/0806 , C07K5/0808 , C07K5/0812 , C07K5/0815 , C07K5/0819 , C07K9/003 , C07K9/008 , A61K38/00
摘要： Nikkomycin derivatives have been found to be orally or parenterally effective as anti-fungals in animals. They may be used alone or, preferably, in combination with azole antimycotics for a synergistic anti-fungal effect.
摘要翻译：已经发现尼古霉素衍生物在动物中作为抗真菌剂是口服或非肠道有效的。它们可以单独使用或优选与唑类抗霉素组合使用，用于协同的抗真菌作用。

28. 发明授权

US5019560A Method for treating fungal infections with nikkomycin derivatives 失效
标题翻译：用尼科霉素衍生物治疗真菌感染的方法
公开(公告)号：US5019560A
公开(公告)日：1991-05-28
申请号：US252613
申请日：1988-10-03
申请人： Richard F. Hector , Klaus Schaller , Heinrich F. Moeschler , Manfred Plempel
发明人： Richard F. Hector , Klaus Schaller , Heinrich F. Moeschler , Manfred Plempel
IPC分类号： A61K31/70 , A61K31/7042 , A61K31/7052 , A61K31/7056 , A61K31/7064 , A61K31/7072 , A61P31/04 , A61P31/10 , C07H19/052 , C07H19/06
CPC分类号： C07H19/06 , C07H19/052
摘要： A method of treating a mammal infected with a dimorphic, highly chitinous fungi, the method comprising administering to the mammal therapeutically effective amounts of a nikkomycin derivative having the following structure: ##STR1##

29. 发明授权

US5011850A Substituted diazolylalkyl-carbinols, a process for their preparation and their use as antimycotic agents 失效
标题翻译：取代的二唑基烷基 - 甲醇，其制备方法及其作为抗真菌剂的用途
公开(公告)号：US5011850A
公开(公告)日：1991-04-30
申请号：US915435
申请日：1986-10-06
申请人： Hans-Ludwig Elbe , Erik Regel , Karl H. Buchel , Klaus Schaller , Manfred Plempel
发明人： Hans-Ludwig Elbe , Erik Regel , Karl H. Buchel , Klaus Schaller , Manfred Plempel
IPC分类号： A61K31/41 , A61K31/415 , A61P31/04 , C07C45/63 , C07C49/00 , C07D20060101 , C07D233/60 , C07D249/08 , C07D403/06 , C07D405/06 , C07D521/00
CPC分类号： C07D231/12 , C07C45/63 , C07D233/56 , C07D249/08
摘要： The invention relates to compounds and their derivatives, said compounds being described herein as those of Formula (I). The compounds and compositions containing them are effective antimycotic agents and the invention includes methods for the use of said compounds and compositions.
摘要翻译：本发明涉及化合物及其衍生物，所述化合物在本文中被描述为式（I）的化合物。含有它们的化合物和组合物是有效的抗真菌剂，本发明包括使用所述化合物和组合物的方法。

30. 发明授权

US4914087A Nikkomycin derivatives, antimycotic compositions of nikkomycin derivatives and azole antimycotics 失效
标题翻译：尼古霉素衍生物，尼科霉素衍生物的抗真菌组合物和唑类抗霉素
公开(公告)号：US4914087A
公开(公告)日：1990-04-03
申请号：US161645
申请日：1988-02-29
申请人： Richard F. Hector , Klaus Schaller , Heinrich F. Moeschler , Manfred Plempel
发明人： Richard F. Hector , Klaus Schaller , Heinrich F. Moeschler , Manfred Plempel
IPC分类号： A61K31/41 , A61K31/70 , A61K31/7042 , A61K31/7052 , A61K31/7064 , A61K31/7072 , A61K38/00 , A61P31/00 , A61P31/04 , A61P31/10 , C07D249/08 , C07H19/06 , C07K5/06 , C07K5/065 , C07K5/078 , C07K5/083 , C07K5/087 , C07K5/09 , C07K5/093 , C07K9/00
CPC分类号： C07H19/06 , C07K5/06078 , C07K5/06139 , C07K5/06191 , C07K5/0806 , C07K5/0808 , C07K5/0812 , C07K5/0815 , C07K5/0819 , C07K9/003 , C07K9/008 , A61K38/00
摘要： Nikkomycin derivatives have been found to be orally or parenterally effective as anti-fungals in animals. They may be used alone or, preferably, in combination with azole antimycotics for a synergistic anti-fungal effect.

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