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21. 发明授权

US07678924B2 Process for the preparation of pyrazoles 有权
标题翻译：制备吡唑的方法
公开(公告)号：US07678924B2
公开(公告)日：2010-03-16
申请号：US11577511
申请日：2005-10-19
申请人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hans Tobler
发明人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hans Tobler
IPC分类号： C07D231/10
CPC分类号： C07D231/14
摘要： The present invention relates to a process for the preparation of compounds of formula I wherein R1 is C1-C4haloalkyl; R2 is C1-C6alkyl and R3 is methyl or ethyl, by reaction of compounds of formula II wherein the substituents are as defined for formula I, with compounds of formula III wherein R3 is as defined for formula I and n is 0 or 1.
摘要翻译：本发明涉及制备式Ⅰ化合物的方法，其中R 1是C 1 -C 4卤代烷基; R 2是C 1 -C 6烷基，R 3是甲基或乙基，其中取代基如式I所定义的式II化合物与式III化合物反应，其中R 3如式I所定义，n是0或1。

22. 发明申请

US20090221856A1 PROCESS FOR THE PREPARATION OF AMINES 有权
标题翻译：制备氨基酸的方法
公开(公告)号：US20090221856A1
公开(公告)日：2009-09-03
申请号：US12096796
申请日：2006-12-11
申请人： Hans Tobler , Harald Walter , Camilla Corsi , Josef Ehrenfreund , Fanny Giordano , Martin Zeller
发明人： Hans Tobler , Harald Walter , Camilla Corsi , Josef Ehrenfreund , Fanny Giordano , Martin Zeller
IPC分类号： C07C211/31
CPC分类号： C07C209/62 , C07B2200/09 , C07C17/23 , C07C17/30 , C07C17/354 , C07C25/22 , C07C25/24 , C07C209/10 , C07C209/70 , C07C211/61 , C07C2603/66 , C07C23/10
摘要： The present invention relates to a novel a process for the preparation of the compound of the general formula (I), wherein R1 and R2 are independently H or C1-6 alkyl, which comprises treating with a reducing agent either a compound of the general formula (II), wherein R1 and R2 have the meanings given for the compound of the formula (I), R3 is H or C1-4alkyl and Ph is phenyl, or a compound of the general formula (III), wherein R1, R2, R3 and Ph have the meanings given for the compound of the formula (II), the reducing agent being effective to cleave the benzyl moiety Ph-CH(R3)— from the benzylamino moiety PhCH(R3)NH— in the compound of the formula (II) or in the compound of the formula (III) to leave an amino group and, in addition, in the case of the compound of the formula (III), to reduce both the 2,3-double bond and the double bond joining the R1R2C— moiety to the 9-position of the benzonorbornene ring to single bonds. It also relates to processes for the preparation of the compounds (II) and (III) and their precursors and to the compounds (II) and (III) themselves and certain of their precursors, which are novel compounds. The compounds (I) are useful for the preparation of various fungicidal heterocyclyl-carboxylic acid benzonorbornen-5-yl-amides.
摘要翻译：本发明涉及一种制备通式（I）化合物的方法，其中R 1和R 2独立地为H或C 1-6烷基，其包括用还原剂处理通式（II）化合物，其中R1和R2具有式（I）化合物所给出的含义，R 3是H或C 1-4烷基，Ph是苯基，或通式（III）的化合物，其中R1，R2， R3和Ph具有式（II）化合物所给出的含义，还原剂有效地从式（II）化合物中的苄基氨基部分PhCH（R3）NH-切割苄基部分Ph-CH（R3）（II）化合物或式（III）化合物中，以留下氨基，另外，在式（III）化合物的情况下，为了还原2,3-双键和双键将R1R2C-部分连接到苯并降冰片烯环的9位到单键。它还涉及制备化合物（II）和（III）及其前体以及化合物（II）和（III）本身及其某些新型化合物的前体的方法。化合物（I）可用于制备各种杀真菌性杂环基 - 羧酸苯并降冰片烯-5-基 - 酰胺。

23. 发明申请

US20090177011A1 PROCESS FOR THE PRODUCTION OF ANILINES 审中-公开
标题翻译：生产过程的过程
公开(公告)号：US20090177011A1
公开(公告)日：2009-07-09
申请号：US11720692
申请日：2005-12-08
申请人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hans Tobler
发明人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hans Tobler
IPC分类号： C07C209/06
CPC分类号： C07C209/10 , C07C2601/02 , C07C211/45
摘要： The present invention relates to a process for the preparation of compounds of formula (I) wherein R1, R2 and R3 are each independently of the others hydrogen or methyl, by reaction of compounds of formula (II) wherein R1, R2 and R3 are as defined for formula (I) and X is bromine or chlorine, with ammonia in the presence of a catalytic amount of at least one copper-containing compound.
摘要翻译：本发明涉及式（Ⅰ）化合物的制备方法，其中R 1，R 2和R 3各自独立地为氢或甲基，其中R 1，R 2和R 3为对于式（I）定义，X是溴或氯，与氨在催化量的至少一种含铜化合物的存在下反应。

24. 发明申请

US20090163569A1 PROCESS FOR THE PRODUCTION OF AMIDES 有权
标题翻译：生产助剂的方法
公开(公告)号：US20090163569A1
公开(公告)日：2009-06-25
申请号：US12066683
申请日：2006-09-14
申请人： Hans Tobler , Harald Walter , Josef Ehrenfreund , Camilla Corsi , Fanny Giordano , Martin Zeller , Gottfried Seifert , Shailesh Shah , Neil George , Ian Kevin Jones , Paul Edward Bonnett
发明人： Hans Tobler , Harald Walter , Josef Ehrenfreund , Camilla Corsi , Fanny Giordano , Martin Zeller , Gottfried Seifert , Shailesh Shah , Neil George , Ian Kevin Jones , Paul Edward Bonnett
IPC分类号： A01N43/56 , C07D231/14 , C07C211/45 , C07C205/11 , C07D403/12 , A01P7/00
CPC分类号： C07C211/61 , A01N43/56 , C07C205/06 , C07C209/325 , C07C209/70 , C07C2603/66 , C07D231/14
摘要： The present invention relates to a process for the preparation of compounds of formula (I) wherein R1 and R2 are each independently of the other hydrogen or C1-C5alkyl and R3 is CF3 or CF2H, by a) reaction of a compound of formula (II) wherein R1 and R2 are as defined for formula (I), with at least one reducing agent to form a compound of formula (III) wherein R1 and R2 are as defined for formula (I), and b) reaction of that compound with at least one reducing agent to form a compound of formula (IV) wherein R1 and R2 are as defined for formula (I), and (c) reaction of that compound with a compound of formula (V) wherein Q is chlorine, fluorine, bromine, iodine, hydroxy or C1-C6alkoxy and R3 is as defined for formula (I), to form the compound of formula (I); and to novel intermediates for use in that process.
摘要翻译：本发明涉及制备式（I）化合物的方法，其中R 1和R 2各自独立地为氢或C 1 -C 5烷基，R 3为CF 3或CF 2 H，通过a）式（Ⅱ）化合物）其中R1和R2如式（I）所定义，与至少一种还原剂形成式（III）化合物，其中R 1和R 2如式（I）所定义，和b）该化合物与至少一种还原剂形成式（Ⅳ）化合物，其中R1和R2如式（Ⅰ）所定义，和（c）该化合物与式（Ⅴ）化合物的反应其中Q是氯，氟，溴，碘，羟基或C 1 -C 6烷氧基，R 3如式（I）所定义，形成式（I）化合物; 以及用于该过程的新型中间体。

25. 发明申请

US20080132557A1 Heterocyclic Carboxamides with Microbiocidal Activity 失效
标题翻译：具有杀微生物活性的杂环羧酰胺
公开(公告)号：US20080132557A1
公开(公告)日：2008-06-05
申请号：US11570796
申请日：2005-06-21
申请人： Clemens Lamberth , Camilla Corsi , Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Clemens Lamberth , Camilla Corsi , Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： A61K31/4155 , C07D403/12
CPC分类号： C07D403/12 , C07D231/40 , C07D333/20 , C07D409/12
摘要： Compounds of the formula (I), in which the substituents are as defined in claim 1 are suitable for use as microbiocides.
摘要翻译：其中取代基如权利要求1中所定义的式（I）化合物适合用作杀微生物剂。

26. 发明授权

US07355065B2 Process for the preparation of 4,4-difluoro-3-oxobutanoic acid esters 有权
标题翻译：制备4,4-二氟-3-氧代丁酸酯的方法
公开(公告)号：US07355065B2
公开(公告)日：2008-04-08
申请号：US11572053
申请日：2005-07-13
申请人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hans Tobler
发明人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hans Tobler
IPC分类号： C07C69/72
CPC分类号： C07C67/343 , C07C69/716
摘要： The present invention relates to a process for the preparation of a compound of the formula (I), wherein R is C1−12 alkyl, by the contact of a compound of the general formula (II), wherein R1 and R2 are each, independently, C1−12 alkyl; or R1 and R2 join together with the nitrogen atom to which they are attached to form an alicyclic amine ring containing 4 to 7 carbon atoms or a morpholine ring, with an acetic acid ester of the general formula (III) CH3COOR, wherein R is as defined under formula (I), in the presence of a base.
摘要翻译：本发明涉及制备式（I）化合物的方法，其中R是C 1-12烷基，通过通式（II）的化合物与其中R 1和R 2各自独立地为C 1-12烷基; 或R 1和R 2 2与它们所连接的氮原子一起形成含有4至7个碳原子的脂环族胺环或吗啉环，其中（III）CH 3 COOR的乙酸酯，其中R如式（I）所定义，在碱的存在下。

27. 发明授权

US08198215B2 Methods for protecting seeds 有权
标题翻译：保护种子的方法
公开(公告)号：US08198215B2
公开(公告)日：2012-06-12
申请号：US11573411
申请日：2005-08-11
申请人： Harald Walter , Ronald Zeun , Josef Ehrenfreund , Hans Tobler , Camilla Corsi , Clemens Lamberth
发明人： Harald Walter , Ronald Zeun , Josef Ehrenfreund , Hans Tobler , Camilla Corsi , Clemens Lamberth
IPC分类号： A01N43/56 , A01P3/00
CPC分类号： A01N43/56
摘要： A method of controlling phytopathogenic diseases on useful plants or plant propagation material thereof, which comprises applying to said plant propagation material a fungicidally effective amount of a compound of formula (I) wherein R1 is trifluoromethyl or difluoromethyl and R2 is hydrogen or methyl, or a tautomer of such a compound, is particularly effective in controlling or preventing fungal diseases of crop plants.
摘要翻译：一种控制有用植物或其植物繁殖材料上的植物病原性疾病的方法，其包括向所述植物繁殖材料施用杀真菌有效量的式（I）化合物，其中R 1为三氟甲基或二氟甲基且R 2为氢或甲基，或这种化合物的互变异构体在控制或预防作物植物的真菌病害中特别有效。

28. 发明授权

US08124567B2 Fungicidal compositions 有权
标题翻译：杀真菌剂
公开(公告)号：US08124567B2
公开(公告)日：2012-02-28
申请号：US11696908
申请日：2007-04-05
申请人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hans Tobler
发明人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hans Tobler
IPC分类号： A01N43/64 , A01N43/00
CPC分类号： A01N43/56 , A01N45/02 , A01N37/34 , A01N37/38 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/653 , A01N43/84 , A01N43/90 , A01N47/24 , A01N61/00 , A01N2300/00
摘要： A method of controlling phytopathogenic diseases on useful plants or on propagation material thereof, which comprises applying to the useful plants, the locus thereof or propagation material thereof a combination of components A) and B) in a synergistically effective amount, whereincomponent A) is a compound of formula I wherein R1 is difluoromethyl or trifluoromethyl; Y is —CHR2— or and R2 is hydrogen or C1-C6alkyl; or a tautomer of such a compound; and component B) is a compound selected from compounds known for their fungicidal and/or insecticidal activity, is particularly effective in controlling or preventing fungal diseases of useful plants.
摘要翻译：一种在有用植物或繁殖材料上控制植物病原性疾病的方法，其包括以协同有效量施用于有用植物，其基因座或繁殖材料的组合物A）和B）的组合，其中组分A）为式Ⅰ化合物，其中R 1是二氟甲基或三氟甲基; Y是-CHR2-或R2是氢或C1-C6烷基; 或这种化合物的互变异构体; 和组分B）是选自其杀真菌和/或杀虫活性已知的化合物的化合物，在控制或预防有用植物的真菌疾病方面特别有效。

29. 发明授权

US08124566B2 Synergistic fungicidal compositions 有权
标题翻译：协同杀菌组合物
公开(公告)号：US08124566B2
公开(公告)日：2012-02-28
申请号：US11576719
申请日：2005-10-06
申请人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hans Tobler
发明人： Harald Walter , Camilla Corsi , Josef Ehrenfreund , Clemens Lamberth , Hans Tobler
IPC分类号： A01N43/64 , A01N43/00
CPC分类号： A01N43/56 , A01N45/02 , A01N37/34 , A01N37/38 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/653 , A01N43/84 , A01N43/90 , A01N47/24 , A01N61/00 , A01N2300/00
摘要： A method of controlling phytopathogenic diseases on useful plants or on propagation material thereof, which comprises applying to the useful plants, the locus thereof or propagation material thereof a combination of components A) and B) in a synergistically effective amount, wherein component A) is a compound of formula (I), wherein R1 is difluoromethyl or trifluoromethyl; Y is —CHR2— or formula (DD) and R2 is hydrogen or C1-C6alkyl; or a tautomer of such a compound; and component B) is a compound selected from compounds known for their fungicidal and/or insecticidal activity, is particularly effective in controlling or preventing fungal diseases of useful plants.
摘要翻译：一种在有用植物或繁殖材料上控制植物病原性疾病的方法，其包括以协同有效量施用于有用植物，其基因座或繁殖材料的组合物A）和B）的组合，其中组分A）为式（I）的化合物，其中R 1是二氟甲基或三氟甲基; Y是-CHR2-或式（DD），R 2是氢或C 1 -C 6烷基; 或这种化合物的互变异构体; 和组分B）是选自其杀真菌和/或杀虫活性已知的化合物的化合物，在控制或预防有用植物的真菌疾病方面特别有效。

30. 发明授权

US07553798B2 Heterocyclic carboxamides with microbiocidal activity 失效
标题翻译：具有杀菌活性的杂环羧酰胺
公开(公告)号：US07553798B2
公开(公告)日：2009-06-30
申请号：US11570796
申请日：2005-06-21
申请人： Clemens Lamberth , Camilla Corsi , Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Clemens Lamberth , Camilla Corsi , Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： A01N43/40 , A01N43/78 , A01N43/56 , A01N43/36 , C07D213/44 , C07D417/02 , C07D401/02 , C07D409/02 , C07D277/20 , C07D403/02 , C07D231/10
CPC分类号： C07D403/12 , C07D231/40 , C07D333/20 , C07D409/12
摘要： Compounds of the formula (I), in which the substituents are as defined in claim 1 are suitable for use as microbiocides.
摘要翻译：其中取代基如权利要求1中所定义的式（I）化合物适合用作杀微生物剂。

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