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11. 发明授权

US5468775A Enaminone esters 失效
标题翻译：烯胺酯
公开(公告)号：US5468775A
公开(公告)日：1995-11-21
申请号：US024970
申请日：1993-03-02
申请人： Kenneth R. Scott , Jesse M. Nicholson , Ivan O. Edafiogho
发明人： Kenneth R. Scott , Jesse M. Nicholson , Ivan O. Edafiogho
IPC分类号： C07C45/51 , C07C225/20 , C07C229/48 , C07C237/24 , C07C243/22 , C07D295/30 , A61K31/24
CPC分类号： C07D295/30 , C07C225/20 , C07C229/48 , C07C237/24 , C07C243/22 , C07C45/512 , C07C2101/16
摘要： The present invention concerns enaminones having the formula: ##STR1## wherein R is from the group consisting of COOCH.sub.3 and COOC.sub.2 H.sub.5 ; R.sup.1 is from the group consisting of H and CH.sub.3 ; R.sup.2 is from the group consisting of H when R.sup.1 is CH.sub.3 and CH.sub.3 when R.sup.1 is H; and R.sup.3 is from the group of first radicals consisting of benzyl, phenethyl, disubstituted phenyl and trisubstituted phenyl. The substituted species are second radicals having positive lipophilicity selected from the group consisting of F, Cl, Br, and I.
摘要翻译：本发明涉及具有下式的烯胺基酮：其中R为COOCH 3和COOC 2 H 5; R1来自H和CH3组成的组; 当R1为CH3时，R2为H，当R1为H时为CH3; 并且R 3是由苄基，苯乙基，二取代的苯基和三取代的苯基组成的一组基团。取代的物质是具有选自F，Cl，Br和I的正亲油性的第二基团。

12. 发明授权

US5466684A 7-(substituted)-9-[(substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines 失效
标题翻译： 7-（取代的）-9 - [（取代的甘氨酰基）酰胺基] -6-脱甲基-6-脱氧四环素
公开(公告)号：US5466684A
公开(公告)日：1995-11-14
申请号：US304731
申请日：1994-09-12
申请人： Phaik-Eng Sum , Ving J. Lee , Raymond T. Testa
发明人： Phaik-Eng Sum , Ving J. Lee , Raymond T. Testa
IPC分类号： A61K31/16 , A61K31/40 , A61K31/403 , A61K31/425 , A61K31/428 , A61K31/65 , A61P31/04 , C07C20060101 , C07C231/12 , C07C237/26 , C07C255/50 , C07C255/52 , C07C317/28 , C07D207/16 , C07D209/02 , C07D211/14 , C07D211/22 , C07D211/26 , C07D213/36 , C07D213/38 , C07D233/56 , C07D233/64 , C07D237/26 , C07D249/04 , C07D249/08 , C07D261/08 , C07D265/30 , C07D277/64 , C07D293/00 , C07D295/12 , C07D295/13 , C07D295/14 , C07D295/15 , C07D295/22 , C07D295/30 , C07D307/32
CPC分类号： C07D295/30 , C07C237/26 , C07D207/16 , C07D213/38 , C07D295/13 , C07D295/15 , C07C2101/02 , C07C2103/46
摘要： The invention provides compounds of the formula: ##STR1## wherein R, R.sup.3, R.sup.4 and W are defined in the specification. These compounds are useful as antibiotic agents.
摘要翻译：本发明提供下式的化合物：其中R，R 3，R 4和W在说明书中定义。这些化合物可用作抗生素。

13. 发明授权

US5214152A Halogen substituted 5-thiazole methane amine compounds 失效
标题翻译：卤素取代的5-噻唑甲胺化合物
公开(公告)号：US5214152A
公开(公告)日：1993-05-25
申请号：US655072
申请日：1991-02-14
申请人： Isao Minamida , Koichi Iwanaga , Tetsuo Okauchi
发明人： Isao Minamida , Koichi Iwanaga , Tetsuo Okauchi
IPC分类号： C07D213/61 , A01N33/18 , A01N35/08 , A01N43/40 , A01N43/42 , A01N43/60 , A01N43/78 , A01N47/24 , A01N55/00 , C07C211/22 , C07C211/29 , C07C229/34 , C07C243/10 , C07C311/50 , C07D20060101 , C07D213/24 , C07D213/38 , C07D213/40 , C07D213/42 , C07D213/64 , C07D213/70 , C07D213/74 , C07D213/77 , C07D215/12 , C07D215/38 , C07D239/26 , C07D241/12 , C07D277/20 , C07D277/22 , C07D277/28 , C07D277/32 , C07D277/38 , C07D277/42 , C07D295/13 , C07D295/30 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14 , C07D413/12 , C07D413/14 , C07D417/12 , C07D417/14 , C07F7/08
CPC分类号： C07D213/40 , A01N35/08 , A01N43/40 , A01N43/42 , A01N43/60 , A01N43/78 , A01N47/24 , A01N55/00 , C07C211/29 , C07D213/38 , C07D213/42 , C07D213/61 , C07D213/64 , C07D213/70 , C07D213/74 , C07D215/12 , C07D239/26 , C07D241/12 , C07D277/28 , C07D277/32 , C07D277/42 , C07D401/06 , C07F7/0812
摘要： .alpha.-Unsaturated amines of the formula: ##STR1## wherein X.sup.1 and X.sup.2 are such that one is an electron-attracting group with the other being a hydrogen atom or an electron-attracting group; R.sup.1 is a group attached through a nitrogen atom; R.sup.2 is a hydrogen atom or a group attached through a carbon, nitrogen or oxygen atom; n is an integer equal to 0, 1 or 2; A is a heterocyclic group or a cyclic hydrocarbon group, and salts thereof and their agrochemical use as insecticidal and/or miticidal agents are described.
摘要翻译： α-不饱和胺，其具有下式：其中X1和X2使得一个是吸电子基团，另一个是吸电子基团或吸电子基团; R1是通过氮原子连接的基团; R2是氢原子或通过碳，氮或氧原子连接的基团; n是等于0,1或2的整数; A是杂环基或环状烃基，其盐及其作为杀虫剂和/或杀螨剂的农药用途被描述。

14. 发明授权

US4665174A Production of cyclopentenone derivatives 失效
标题翻译：环戊烯酮衍生物的生产
公开(公告)号：US4665174A
公开(公告)日：1987-05-12
申请号：US377050
申请日：1982-05-11
申请人： Masayoshi Minai , Tadashi Katsura
发明人： Masayoshi Minai , Tadashi Katsura
IPC分类号： C07C45/71 , C07C49/753 , C07C69/708 , C07C225/00 , C07C225/20 , C07C327/22 , C07D213/36 , C07D213/38 , C07D295/116 , C07D295/30 , C07D307/00 , C07D307/32 , C07D307/33 , C07D307/42 , C07D317/64 , C07D333/14 , C07D333/20 , C07D333/34 , C07D493/04 , C07D493/06 , C07H15/203 , C07D279/10 , C07C85/02 , C07C87/50 , C07D265/30
CPC分类号： C07D295/30 , C07C321/00 , C07C323/00 , C07C327/00 , C07C45/71 , C07D213/38 , C07D295/116 , C07D307/33 , C07D307/42 , C07D317/64 , C07D333/20 , C07D333/34 , C07H15/203
摘要： A process for preparing cyclopentenone derivatives of the formula: ##STR1## wherein R.sup.1 is hydrogen, lower alkyl or lower alkenyl, R.sup.2 is hydrogen, lower alkyl, lower alkenyl, lower alkynyl, cycloalkyl, substituted or unsubstituted aryl or substituted or unsubstituted ar(lower)alkyl and A is the residue of a nucleophilic agent from which a hydrogen atom is excluded, which comprises reacting a 3-hydroxy-4-cyclopentenone compound of the formula: ##STR2## wherein R.sup.1 and R.sup.2 are each as defined above with a nucleophilic agent of the formulaA--H (III)wherein A is as defined above.The cyclopentenone derivatives of the formula (I) are useful as pharmaceuticals, agricultural chemicals, perfumes and as intermediates for the preparation of agricultural chemicals, pharmaceuticals and perfumes.
摘要翻译：制备下式的环戊烯酮衍生物的方法：其中R 1是氢，低级烷基或低级链烯基，R 2是氢，低级烷基，低级烯基，低级炔基，环烷基，取代或未取代的芳基或取代或未取代的芳基 Ar（低级）烷基，A是除去氢原子的亲核剂的残基，其包括使下式的3-羟基-4-环戊烯酮化合物：其中R 1和R 2各自为如上定义的具有式AH（III）的亲核剂，其中A如上所定义。式（I）的环戊烯酮衍生物可用作药物，农药，香料以及用于制备农药，药物和香料的中间体。

15. 发明授权

US4564677A Preparation of N-amino compounds 失效
标题翻译： N-氨基化合物的制备
公开(公告)号：US4564677A
公开(公告)日：1986-01-14
申请号：US571977
申请日：1984-01-19
申请人： Martin L. Kantor
发明人： Martin L. Kantor
IPC分类号： C07D209/08 , C07D295/30 , C07B31/00 , C07B43/02
CPC分类号： C07D295/30 , C07D209/08
摘要： Disclosed is a method of preparing N-amino compounds from corresponding secondary amines by reacting a secondary amine with nitrous acid and zinc in a neutral pH reaction media to form the corresponding N-amine.
摘要翻译：公开了通过在中性pH反应介质中使仲胺与亚硝酸和锌反应形成相应的N-胺，从相应的仲胺制备N-氨基化合物的方法。

16. 发明授权

US4180568A Control of phytopathogens with certain 2,6-dinitroanilines 失效
标题翻译：用某些2,6-二硝基苯胺控制植物病原体
公开(公告)号：US4180568A
公开(公告)日：1979-12-25
申请号：US878370
申请日：1978-02-16
申请人： James R. Beck , Joseph A. Yahner
发明人： James R. Beck , Joseph A. Yahner
IPC分类号： C07D207/50 , C07D295/30 , A01N9/20
CPC分类号： C07D295/30 , C07D207/50
摘要： It has been discovered that fungal foliar phytopathogens may be controlled by the use of a broad class of 2,6-dinitroanilines. The fungicidally-effective compounds may bear a broad range of substituent groups on the anilino nitrogen and in the 3- and 4-positions of the benzene ring.
摘要翻译：已经发现真菌叶片植物病原体可以通过使用广泛的2,6-二硝基苯胺来控制。杀真菌有效的化合物可以在苯胺基氮和苯环的3-和4-位上具有宽范围的取代基。

17. 发明授权

US4138244A Nitrophenylhydrazine compounds 失效
标题翻译：硝基苯肼化合物
公开(公告)号：US4138244A
公开(公告)日：1979-02-06
申请号：US713463
申请日：1976-08-11
申请人： Don L. Hunter , William G. Woods , James D. Stone , Cecil W. LeFevre
发明人： Don L. Hunter , William G. Woods , James D. Stone , Cecil W. LeFevre
IPC分类号： A01N33/26 , C07D295/22 , C07D295/30 , A01N9/20 , A01N9/22 , A01N9/28
CPC分类号： C07D295/30 , A01N33/26 , C07C243/00
摘要： N-Amino substituted aniline and 1,3-phenylenediamine compounds having 1 or 2 nitro groups on the aromatic ring. The compounds are useful as herbicides and as intermediates for peparing herbicides.
摘要翻译：在芳环上具有1或2个硝基的N-氨基取代苯胺和1,3-苯二胺化合物。该化合物可用作除草剂和作为除草剂的中间体。

18. 发明授权

US3928593A Antiviral compositions containing piperazine derivatives and method of use 失效
标题翻译：含有哌嗪衍生物的抗病毒组合物及其使用方法
公开(公告)号：US3928593A
公开(公告)日：1975-12-23
申请号：US13655871
申请日：1971-04-22
申请人： LEPETIT SPA
发明人： LANCINI GIANCARLO , THIRY LISE
IPC分类号： C07D295/30 , C07D487/08 , A61K31/495
CPC分类号： C07D295/30 , C07D487/08
摘要： Compositions and methods for controlling viral infections comprising a piperazine compound corresponding to the formula

WHEREIN R represents hydrogen, lower alkyl, lower acyl or phenyl-lower-alkyl; R1, R2, R3 and R4 each represents hydrogen or lower alkyl; each of the pairs R1 and R2 or R3 and R4 may also represent a lower alkylene group bridging the piperazine ring; X is selected from H2, benzylidene and (H, lower acyl); and pharmaceutically acceptable acid addition salts of such compounds.
摘要翻译：用于控制病毒感染的组合物和方法，包括对应于式WHEREIN R的哌嗪化合物代表氢，低级烷基，低级酰基或苯基 - 低级 - 烷基; R1，R2，R3和R4各自表示氢或低级烷基; 对R1和R2或R3和R4中的每一个也可以代表桥接哌嗪环的低级亚烷基; X选自H 2，亚苄基和（H，低级酰基）; 和这些化合物的药学上可接受的酸加成盐。

19. 发明授权

US3891706A 2-Amino-2,6-dinitrophenylhydrazines 失效
标题翻译： 2-氨基-2,6-二硝基苯肼
公开(公告)号：US3891706A
公开(公告)日：1975-06-24
申请号：US29414772
申请日：1972-10-02
申请人： WILCOX MERRILL
发明人： WILCOX MERRILL
IPC分类号： A01N33/18 , A01N33/26 , A01N37/34 , A01N37/44 , A01N37/48 , A01N51/00 , C07C243/38 , C07D295/06 , C07D295/22 , C07D295/30 , C07C109/04
CPC分类号： C07D295/30 , C07C243/00 , C07C243/38
摘要： 3-amino-2,6-dinitrophenylhydrazines of the formula

WHEREIN Y is halogen, haloalkyl carbamyl, lower alkyl substituted carbamyl, carboxyl, lower alkoxy carbonyl, trifluoromethyl, nitro or cyano; Z is amino which is optionally substituted with lower alkyl, lower alkoxy, substituted lower alkyl, substituted lower alkoxy or mono or di-lower alkylamino, with the proviso that not more than one of the substituents is alkoxy, substituted alkoxy or mono or di-lower alkylamino; R1 is H, lower alkyl or lower alkenyl, said alkyl and alkenyl groups are optionally substituted with halogen, lower alkoxy, phenyl or cycloalkyl; R2 and R3 are independently H, C1-C5 alkyl, C2-C5 alkenyl, said alkyl and alkenyl groups are optionally substituted with cycloalkyl groups; R2 and R3 can also be taken together with the nitrogen atom to which they are linked forming the ring structures piperidino, hexamethylenimino, morpholino, or 4methylpiperazino. These compounds are very active plant growth regulators and are particularly useful as herbicides and in tobacco sucker control.
摘要翻译： 3-氨基-2,6-二硝基苯肼，其结构式为：Y是卤素，卤代烷基氨基甲酰基，低级烷基取代的氨基甲酰基，羧基，低级烷氧基羰基，三氟甲基，硝基或氰基; Z是任选被低级烷基，低级烷氧基，取代的低级烷基，取代的低级烷氧基或单或二低级烷基氨基取代的氨基，条件是不超过一个取代基是烷氧基，取代的烷氧基或单或二 - 低级烷基氨基; R 1是H，低级烷基或低级烯基，所述烷基和烯基任选被卤素，低级烷氧基，苯基或环烷基取代; R2和R3独立地为H，C1-C5烷基，C2-C5烯基，所述烷基和烯基任选被环烷基取代; R2和R3也可以与它们所连接的氮原子一起形成环结构哌啶子基，六亚甲基亚氨基，吗啉代或4-甲基哌嗪基。

20. 发明授权

US3297689A 1-arylidenemaino-4-(4-benzhydryl-1-piperazinylcarbonyl) piperazines and intermediate herefor 失效
标题翻译： 1-亚芳基新亚胺-4-（4-二苯甲基-1-哌嗪基羰基）哌嗪及其中间体
公开(公告)号：US3297689A
公开(公告)日：1967-01-10
申请号：US42358265
申请日：1965-01-05
申请人： SEARLE & CO
发明人： CUSIC JOHN W , PETER YONAN
IPC分类号： C07D295/205 , C07D295/28 , C07D295/30 , C07D317/58
CPC分类号： C07D295/205 , C07D295/30 , C07D317/58

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