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11. 发明授权

US08975252B2 Morpholine derivative 有权
标题翻译：吗啉衍生物
公开(公告)号：US08975252B2
公开(公告)日：2015-03-10
申请号：US12664637
申请日：2008-06-16
申请人： Hidenori Akatsuka , Hiroshi Sugama , Nobumasa Awai , Takayuki Kawaguchi , Yoichi Takahashi , Toru Iijima , Jingkang Shen , Guangxin Xia , Jianshu Xie
发明人： Hidenori Akatsuka , Hiroshi Sugama , Nobumasa Awai , Takayuki Kawaguchi , Yoichi Takahashi , Toru Iijima , Jingkang Shen , Guangxin Xia , Jianshu Xie
IPC分类号： A61K31/535 , C07D265/30 , C07D209/08 , C07D209/14 , C07D209/30 , C07D209/34 , C07D209/42 , C07D231/56 , C07D265/36 , C07D403/04 , C07D413/04 , C07D413/12 , C07D413/14 , C07D417/14 , C07D471/04
CPC分类号： C07D265/30 , C07D209/08 , C07D209/14 , C07D209/30 , C07D209/34 , C07D209/42 , C07D231/56 , C07D265/36 , C07D403/04 , C07D413/04 , C07D413/12 , C07D413/14 , C07D417/14 , C07D471/04
摘要： The present invention provides a morpholine derivative of the formula [I]; wherein R1 is a substituted alkyl group, an optionally substituted aryl group, an optionally substituted heterocyclo group, a cycloalkyl group or an alkyl group; R2 is a substituted alkyl group, an optionally substituted aryl group, an optionally substituted heterocyclo group, an optionally substituted alkylcarbonyl group, an optionally substituted arylcarbonyl group, an optionally substituted heterocyclo-substituted carbonyl group or a cycloalkylcarbonyl group; T is a methylene group or a carbonyl group; R3, R4, R5 and R6 are the same or different and a hydrogen atom, an optionally substituted carbamoyl group or an optionally substituted alkyl group; or pharmaceutically acceptable salts thereof. These compounds are useful as a renin inhibitor.
摘要翻译：本发明提供式[I]的吗啉衍生物。其中R1是取代的烷基，任选取代的芳基，任选取代的杂环基，环烷基或烷基; R 2是取代的烷基，任选取代的芳基，任选取代的杂环基，任选取代的烷基羰基，任选取代的芳基羰基，任选取代的杂环取代的羰基或环烷基羰基; T是亚甲基或羰基; R3，R4，R5和R6相同或不同，氢原子，任选取代的氨基甲酰基或任选取代的烷基; 或其药学上可接受的盐。这些化合物可用作肾素抑制剂。

12. 发明授权

US08410166B2 Fused bicyclic compound 有权
标题翻译：稠合双环化合物
公开(公告)号：US08410166B2
公开(公告)日：2013-04-02
申请号：US13561662
申请日：2012-07-30
申请人： Yoichi Takahashi , Nobumasa Awai , Hidenori Akatsuka , Takayuki Kawaguchi , Toru Iljima
发明人： Yoichi Takahashi , Nobumasa Awai , Hidenori Akatsuka , Takayuki Kawaguchi , Toru Iljima
IPC分类号： C07D265/00
CPC分类号： C07D265/16 , C07D311/20 , C07D311/58 , C07D311/96 , C07D405/14 , C07D413/04
摘要： Fused bicyclic compound having an affinity to mineral corticoid receptor (MR), of formula [I]: wherein ring A is benzene having a substituent R1, fused to an adjacent 6-membered heterocyclic ring and further optionally having a substituent(s) other than R1, R1 is alkylsulfonylamino, etc., R2 and R3 are (a) the same of different and are hydrogen, alkyl, or optionally substituted aryl, or (b) combined with each other to form an oxo group or (c) combined with each other at its terminal together with the adjacent carbon atom to form cycloalkyl, X is ═N—, ═C(R4)— or —CH(R4)—, R4 is (a) hydrogen, (b) cyano, (c) halogen, (d) alkyl, (e) alkenyl, (f) cycloalkyl, (g) alkanoyl, (h) carbamoyl, or (i) cycloalkenyl, Ar is an optionally substituted aromatic cyclic group and a dotted line means presence or absence of a double bond, or a pharmaceutically acceptable salt thereof, useful e.g. as an antihypertensive agent.
摘要翻译：具有式[I]的矿物质类皮质激素受体（MR）的亲和性的稠合双环化合物：其中环A是具有取代基R 1的苯，与相邻的6元杂环稠合，并且进一步任选具有除 R 1，R 1是烷基磺酰基氨基等，R 2和R 3是（a）不同的并且是氢，烷基或任选取代的芳基，或（b）彼此结合形成氧代基或（c）与 X是= N - ， - C（R4） - 或-CH（R4） - ，R4是（a）氢，（b）氰基，（c）卤素，（d）烷基，（e）烯基，（f）环烷基，（g）烷酰基，（h）氨基甲酰基或（i）环烯基，Ar是任选取代的芳族环状基团，虚线表示存在或不存在双键或其药学上可接受的盐，例如，作为抗高血压药。

13. 发明授权

US08258131B2 Fused bicyclic compound 有权
标题翻译：稠合双环化合物
公开(公告)号：US08258131B2
公开(公告)日：2012-09-04
申请号：US12671479
申请日：2008-07-21
申请人： Yoichi Takahashi , Nobumasa Awai , Hidenori Akatsuka , Takayuki Kawaguchi , Toru Iijima
发明人： Yoichi Takahashi , Nobumasa Awai , Hidenori Akatsuka , Takayuki Kawaguchi , Toru Iijima
IPC分类号： C07D265/16 , A61K31/352 , A61K31/353
CPC分类号： C07D265/16 , C07D311/20 , C07D311/58 , C07D311/96 , C07D405/14 , C07D413/04
摘要： The present invention provides a novel fused bicyclic compound having an affinity to a receptor of mineral corticoid (MR), shown by the formula [I]: wherein the ring A is a benzene ring having a substituent R1, fused to an adjacent 6-membered heterocyclic ring and further optionally having a substituent(s) other than R1, R1 is an alkylsulfonylamino group etc., R2 and R3 are (a) the same of different and a hydrogen atom, an alkyl group or a substituted or unsubstituted aryl group, (b) combined each other to form an oxo group or (c) combined each other at its terminal together with the adjacent carbon atom to form a cycloalkyl group, X is a group of ═N—, ═C(R4)— or —CH(R4)—, R4 is (a) a hydrogen atom, (b) a cyano group, (c) a halogen atom, (d) an alkyl group, (e) an alkenyl group, (f) a cycloalkyl group (g) an alkanoyl group, (h) a carbamoyl group or (i) a cycloalkenyl group, Ar is an optionally substituted aromatic cyclic group and a dotted line means presence or absence of a double bond, or a pharmaceutically acceptable salt thereof, which is useful as an antihypertensive agent etc.
摘要翻译：本发明提供了对式[I]所示的对矿物质类皮质激素（MR）的受体具有亲和性的新的稠合双环化合物：其中环A是具有取代基R 1的苯环，与相邻的6元杂环，并且还可任选地具有除R1以外的取代基，R 1是烷基磺酰基氨基等，R 2和R 3是（a）不同的，和氢原子，烷基或取代或未取代的芳基，（b）彼此组合以形成氧代基团，或（c）在其末端与相邻的碳原子一起相互结合形成环烷基，X是一个= N - ， - C（R 4） - 或 - CH（R4） - ，R4是（a）氢原子，（b）氰基，（c）卤原子，（d）烷基，（e）烯基，（f）环烷基 g）烷酰基，（h）氨基甲酰基或（i）环烯基，Ar是任选取代的芳环基，虚线表示存在或不存在双键或其药学上可接受的盐，其可用作抗高血压剂等。

14. 发明申请

US20120079266A1 COMMUNICATION SYSTEM, COMMUNICATION DEVICE, AND COMMUNICATION METHOD 有权
标题翻译：通信系统，通信设备和通信方法
公开(公告)号：US20120079266A1
公开(公告)日：2012-03-29
申请号：US13077528
申请日：2011-03-31
申请人： Hideaki Ogata , Yoichi Takahashi
发明人： Hideaki Ogata , Yoichi Takahashi
IPC分类号： H04L9/28 , G06F21/00
CPC分类号： H04L63/0428 , G06F21/608 , H04L9/16 , H04L63/20
摘要： A first communication device includes a security policy storing unit that store a security policy and a default policy applied to communication to which the security policy is not applied, a communication unit that performs communication, and a communication control unit that performs an encryption process and a decryption process according to the default policy when the communication does not correspond to the target of the policy. A second communication device includes an input and output receiving processing unit that receives an input of an encryption key of the default policy of the first communication device, a communication control unit that generates a policy including an encryption method of the default policy and the input encryption key and performs an encryption process and a decryption process in communication with the first communication device according to the policy, and a communication unit that performs communication of a communication packet.
摘要翻译：第一通信设备包括存储安全策略和应用于不应用安全策略的通信的默认策略的安全策略存储单元，执行通信的通信单元和执行加密处理的通信控制单元解密过程根据默认策略，当通信不符合策略的目标时。第二通信设备包括输入和输出接收处理单元，其接收第一通信设备的默认策略的加密密钥的输入，生成包括默认策略的加密方法和输入加密的策略的通信控制单元密钥，并且执行根据策略与第一通信设备通信的加密处理和解密处理，以及执行通信分组的通信的通信单元。

15. 发明授权

US07778764B2 Fuel injection control apparatus and method for a multi-fuel engine, and engine incorporating same 有权
标题翻译：用于多燃料发动机的燃料喷射控制装置和方法，以及包含其的发动机
公开(公告)号：US07778764B2
公开(公告)日：2010-08-17
申请号：US12378686
申请日：2009-02-18
申请人： Atsushi Ito , Yoichi Takahashi
发明人： Atsushi Ito , Yoichi Takahashi
IPC分类号： F02D41/30
CPC分类号： F02D41/0025 , F02D19/061 , F02D19/084 , F02D19/088 , F02D41/1454 , F02D2200/023 , F02D2200/0404 , Y02T10/36
摘要： A fuel injection control apparatus for a multi-fuel engine can optimize a fuel injection quantity, using only one basic injection map, irrespective of alcohol concentration of a fuel. An E-concentration determining apparatus determines alcohol concentration of a fuel, based on a measured oxygen amount in exhaust. Basic injection quantities are stored in a basic injection map. E-concentration coefficients are stored in an E-concentration coefficient table for a plurality of alcohol concentrations in the fuel. A basic injection quantity, corresponding to a current rotary engine speed and a throttle opening, is selected from the basic injection map. A concentration coefficient, corresponding to the alcohol concentration and the basic injection quantity, is selected from the E-concentration coefficient table. A fuel injection quantity calculator determines an applied fuel injection quantity by multiplying the basic injection quantity by the concentration coefficient. Further adjustments using a number of additional correction coefficients may be made, as needed.
摘要翻译：不管燃料的酒精浓度如何，用于多燃料发动机的燃料喷射控制装置可以仅使用一个基本喷射图来优化燃料喷射量。电离浓度测定装置基于排气中测定的氧量来确定燃料的醇浓度。基本注射量存储在基本注射图中。 E浓度系数存储在燃料中的多个醇浓度的E浓度系数表中。从基本注入图中选择对应于当前旋转发动机转速和节气门开度的基本喷射量。从E浓度系数表中选出与酒精浓度和碱性喷射量对应的浓度系数。燃料喷射量计算器通过将基本喷射量乘以浓度系数来确定施加的燃料喷射量。可以根据需要进行使用多个附加校正系数的进一步调整。

16. 外观设计

USD537434S1 Combined radio tuner and amplifier 有权
标题翻译：组合无线电调谐器和放大器
公开(公告)号：USD537434S1
公开(公告)日：2007-02-27
申请号：US29227989
申请日：2005-04-18
申请人： Yoichi Takahashi , Yohei Tanaka , Shinji Makino
设计人： Yoichi Takahashi , Yohei Tanaka , Shinji Makino

17. 发明申请

US20060082485A1 Semiconductor device with A/D converter 有权
标题翻译：具有A / D转换器的半导体器件
公开(公告)号：US20060082485A1
公开(公告)日：2006-04-20
申请号：US11248158
申请日：2005-10-13
申请人： Keiko Kobayashi , Yoichi Takahashi , Tomotake Ooba , Fujio Higuchi , Keiichi Iwazumi , Akira Saitou
发明人： Keiko Kobayashi , Yoichi Takahashi , Tomotake Ooba , Fujio Higuchi , Keiichi Iwazumi , Akira Saitou
IPC分类号： H03M1/12
CPC分类号： B60C23/0433 , G01L9/065
摘要： A semiconductor device includes a reference voltage generating section configured to generate a first reference voltage and a second reference voltage based on a voltage supplied from an external power supply; and an AD (analog/digital) conversion circuit operating based on the first reference voltage to generate an AD conversion signal corresponding to an output signal supplied from an external device through AD conversion. The second reference voltage is supplied to the external device, and a ratio of the first reference voltage and the second reference voltage is kept to a constant value regardless of a temperature of the semiconductor device.
摘要翻译：一种半导体器件，包括：参考电压产生部，被配置为基于从外部电源提供的电压产生第一参考电压和第二参考电压; 以及基于第一参考电压工作的AD（模拟/数字）转换电路，以产生对应于通过AD转换从外部设备提供的输出信号的AD转换信号。第二参考电压被提供给外部设备，并且第一参考电压和第二参考电压的比率被保持为恒定值，而与半导体器件的温度无关。

18. 发明申请

US20060077048A1 Variation detection device, data communication apparatus, and method of detecting variation 失效
公开(公告)号：US20060077048A1
公开(公告)日：2006-04-13
申请号：US11257651
申请日：2005-10-13
申请人： Akira Saitou , Yoichi Takahashi , Tomotake Ooba , Keiichi Iwazumi , Fujio Higuchi , Keiko Kobayashi
发明人： Akira Saitou , Yoichi Takahashi , Tomotake Ooba , Keiichi Iwazumi , Fujio Higuchi , Keiko Kobayashi
IPC分类号： B60R25/10
CPC分类号： B60C23/0408
摘要： A variation detection device has a processor, an AD converter converting a signal voltage output from a sensor to generate an AD converted value and outputting the AD converted value to the processor, a temperature sensor detecting a temperature of the sensor, and a memory storing a table which indicates a relationship between temperatures and initial values. When receiving the AD converted value, the processor identifies a temperature of the sensor based on an output of the temperature sensor, reads out an initial value corresponding to the identified temperature from the table, and calculates a variation between the initial value and the AD converted value.

19. 发明授权

US06592511B2 Incubator 有权
公开(公告)号：US06592511B2
公开(公告)日：2003-07-15
申请号：US09902794
申请日：2001-07-11
申请人： Naoki Honma , Yoichi Takahashi , Tatsuhiko Seki , Kazuo Matubara
发明人： Naoki Honma , Yoichi Takahashi , Tatsuhiko Seki , Kazuo Matubara
IPC分类号： A61G1100
CPC分类号： A61G11/009 , A61G11/00 , A61G11/005 , A61G11/006 , Y10T292/28
摘要： In this incubator, the door rotation restricting means in the operating state restrains the rotation of the door in the opening direction beyond the operating angle. Thus, in the case that the door rotation restricting means is in the operating state, even if the door is pushed by the accommodated baby from the inside of the hood under the state wherein the door is not fixed by the door fixing means in a closing state, the door does not rotate in the opening direction beyond the operating angle and the angle of the door does not exceed the operating angle. Therefore, even if opening and closing operation of the nursing window is not securely performed, at least the environment inside the hood hardly deviates from the physiological environment appropriate for the accommodated baby.

20. 发明授权

US4894518A Toaster oven with initial temperature compensation and sensor check 失效
标题翻译：烤箱烤箱具有初始温度补偿和传感器检查
公开(公告)号：US4894518A
公开(公告)日：1990-01-16
申请号：US294994
申请日：1989-01-06
申请人： Kazuhiko Ishikawa , Yoichi Takahashi
发明人： Kazuhiko Ishikawa , Yoichi Takahashi
IPC分类号： A47J37/06 , A47J37/08 , G05D23/19
CPC分类号： A47J37/0635 , A47J37/0842 , G05D23/1951
摘要： An electric oven such as a toaster oven according to this invention includes in addition to a heating chamber, a heater for the heating chamber and a temperature detector for measuring the temperature therein, a control device serving to automatically determine a target temperature on the basis of the initial temperature inside the heating chamber so that a desired degree of heating can be effected independently of the initial temperature inside the heating chamber by switching off the power supply when the detected temperature reaches the target temperature thus set. According to another embodiment of the present invention, minimum and maximum heating times are set such that the control device will additionally serve to continue the heating independently of the measured temperature if the preset minimum heating time has not elapsed from the beginning of the heating and to shut off the power supply independently of the measured temperature if the preset maximum heating time has elapsed, so that the heating can be effected safely and dependably even if the temperature detector malfunctions.
摘要翻译：根据本发明的电烤箱如烤箱烤箱除了加热室以外，还包括用于加热室的加热器和用于测量其中的温度的温度检测器，用于基于以下方式自动确定目标温度的控制装置加热室内的初始温度，使得当检测到的温度达到如此设定的目标温度时，通过切断电源，可以独立于加热室内的初始温度来实现所需的加热程度。根据本发明的另一个实施例，设定最小加热时间和最大加热时间，使得控制装置另外用于独立于测量温度继续加热，如果预设的最小加热时间从加热开始还没有经过，并且如果预设的最大加热时间已经过去，则独立于测量的温度关闭电源，使得即使温度检测器发生故障，也可以安全可靠地进行加热。

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