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131. 发明申请

US20100160166A1 Inhibitors of a 9-cis epoxycarotenoid dioxygenase 有权
标题翻译： 9-顺式环氧类胡萝卜素双加氧酶抑制剂
公开(公告)号：US20100160166A1
公开(公告)日：2010-06-24
申请号：US12458781
申请日：2009-07-22
申请人： Suzanne R. Abrams , Michele C. Loewen , Jason Boyd , Adrian John Cutler , Yuanzhu Gai , Kenneth M. Nelson
发明人： Suzanne R. Abrams , Michele C. Loewen , Jason Boyd , Adrian John Cutler , Yuanzhu Gai , Kenneth M. Nelson
IPC分类号： A01N43/10 , C07D493/08 , C07C321/10 , C07D333/38 , C07D303/00 , A01N43/08 , A01N37/44 , A01N41/12
CPC分类号： C07D333/38 , A01N31/06 , A01N35/06 , A01N43/10 , A01N43/20 , C07C323/15 , C07C323/22 , C07C2601/14 , C07D493/08 , Y02P20/55
摘要： A compound of formula (I): wherein: R1 is —SR10, —O—C(O)—R11, —NR12R13, where R10 is a C1-8-alkyl group or a phenyl group unsubstituted or substituted by a C1-4-alkyl group, R11 is a thiophenenyl, furanyl or pyrrolyl group, R12 is H or a C1-4-alkyl group and R13 is a C1-8-alkyl group or a phenyl group unsubstituted or substituted by a C1-4-alkyl group; R2 is H or a C1-4-alkyl group; R3 and R4 are independently H or C1-4-alkyl groups; R5 and R6 are independently H, OH or OR14, or taken together are ═O, where R14 is a protecting group; R7 is H or a C1-4-alkyl group; and, R8 is H, R9 is OH and R15 is H, or R15 is H and R8 and R9 taken together are —O—, or R9 is OH and R8 and R15 taken together form a bond; and, R18 and R19 are both H, or R18 and R19 taken together form a bond, or a plant physiologically acceptable salt thereof is useful for inhibiting 9-cis-epoxycarotenoid dioxygenase (NCED) in a plant or seed and is therefore useful for regulating ABA biosynthesis in the plant or seed.
摘要翻译：式（I）的化合物：其中：R 1是-SR 10，-O-C（O）-R 11，-NR 12 R 13，其中R 10是C 1-8 - 烷基或未被取代或被C 1-4取代的苯基 - 烷基，R 11是噻吩基，呋喃基或吡咯基，R12是H或C1-4烷基，R13是C1-8 - 烷基或未被取代或被C1-4 - 烷基取代的苯基 ; R2是H或C1-4烷基; R3和R4独立地为H或C1-4烷基; R5和R6独立地为H，OH或OR14，或者一起为= O，其中R14为保护基; R 7为H或C 1-4 - 烷基; 并且，R 8为H，R 9为OH，R 15为H，R 15为H，R 8和R 9一起为-O-，或R 9为OH，R 8和R 15为一个键。 R18和R19均为H或R18和R19一起形成键，或其植物生理学上可接受的盐可用于抑制植物或种子中的9-顺式 - 环氧类胡萝卜素双加氧酶（NCED），因此可用于调节 ABA生物合成植物或种子。

132. 发明申请

US20100144785A1 FUNGICIDE N-6-MEMBERED FUSED (HETERO) ARYL-METHYLENE-N-CYCLOALKYL CARBOXAMIDE DERIVATIVES 有权
标题翻译：杀真菌剂N-6成分融合（异星）芳基 - 甲基-N-环烷基羧酰胺衍生物
公开(公告)号：US20100144785A1
公开(公告)日：2010-06-10
申请号：US12452921
申请日：2008-07-31
申请人： Philippe Desbordes , Stephanie Gary , Marie-Claire Grosjean-Cournoyer , Benoit Hartmann , Philippe Rinolfi , Arounarith Tuch
发明人： Philippe Desbordes , Stephanie Gary , Marie-Claire Grosjean-Cournoyer , Benoit Hartmann , Philippe Rinolfi , Arounarith Tuch
IPC分类号： A01N43/42 , C07D231/14 , C07D231/20 , A01N43/56 , C07D207/34 , A01N43/36 , C07D333/38 , A01N43/10 , C07D307/68 , A01N43/08 , C07D217/14 , C07D215/12 , A01P3/00
CPC分类号： C07D401/12 , C07D207/34 , C07D207/416 , C07D231/14 , C07D231/16 , C07D231/20 , C07D307/56 , C07D333/38 , C07D403/12 , C07D405/12 , C07D409/12 , C07D417/12
摘要： The present invention relates N-(aromatic, 6-membered, fused, (hetero)aryl-methylene)-N-cycloalkyl carboxamide derivatives, their thiocarboxamide or N-substituted carboximidamide analogues, all of formula (I) wherein A represents a carbo-linked 5-membered heterocyclyl group; T represents O, S, N—Rc, N—ORd, N—NRcRd or N—CN; Z1 to Z3 and B represents an aromatic, 6-membered, fused, (hetero)aryl; their process of preparation; their use as fungicide active agents, particularly in the form of fungicide compositions and methods for the control of phytopathogenic fungi, notably of plants, using these compounds or compositions.
摘要翻译：本发明涉及所有式（I）的N-（芳族，6元，稠合，（杂）芳基 - 亚甲基）-N-环烷基甲酰胺衍生物，它们的硫代甲酰胺或N-取代的肟基亚胺酰胺类似物，其中A表示碳 - 连接的5元杂环基; T表示O，S，N-Rc，N-ORd，N-NRcRd或N-CN; Z 1至Z 3，B表示芳族，6元稠合的（杂）芳基; 他们的准备过程; 它们用作杀真菌活性剂，特别是以杀真菌剂组合物的形式和用于使用这些化合物或组合物来控制植物病原真菌，特别是植物的方法。

133. 发明授权

US07714023B2 Treatment or prophylaxis of migraine or headache disorders using citalopram, escitalopram or citalopram metabolites 有权
标题翻译：使用西酞普兰，依他普仑或西酞普兰代谢物治疗或预防偏头痛或头痛
公开(公告)号：US07714023B2
公开(公告)日：2010-05-11
申请号：US11060067
申请日：2005-02-17
申请人： Timothy J. Barberich
发明人： Timothy J. Barberich
IPC分类号： A01N43/08 , A61K31/34 , A61K31/40 , A01N43/38 , A01N33/02 , A61K31/135 , C07D307/87
CPC分类号： A61K31/343
摘要： Methods for prophylaxis of or treating or preventing migraine or migraine headaches, or other headache disorders include administering to a subject in need of treatment a therapeutically effective amount of citalopram, escitalopram, or a racemic or optically pure citalopram metabolite, or pharmaceutically acceptable salts, solvates, polymorphs, or hydrates thereof.
摘要翻译：用于预防或治疗或预防偏头痛或偏头痛或其他头痛障碍的方法包括向需要治疗的受试者施用治疗有效量的西酞普兰，依他普仑或外消旋或光学纯的西酞普兰代谢物或其药学上可接受的盐溶剂化物，多晶型物或其水合物。

134. 发明申请

US20100048696A1 AGRICULTURAL DISEASE CONTROL AGENT 审中-公开
标题翻译：农业疾病控制代理
公开(公告)号：US20100048696A1
公开(公告)日：2010-02-25
申请号：US12522760
申请日：2008-01-11
申请人： Kazuo Sumi , Kazuyoshi Koike , Shinji Ito
发明人： Kazuo Sumi , Kazuyoshi Koike , Shinji Ito
IPC分类号： A01N43/08 , C07C57/145 , C07D307/36 , A01N37/06 , A01P1/00
CPC分类号： A01N37/06
摘要： The present invention provides a disinfectant comprising as an active ingredient maleic acid and/or maleic anhydride.
摘要翻译：本发明提供了包含马来酸和/或马来酸酐作为活性成分的消毒剂。

135. 发明申请

US20090215623A1 Insecticidal 3-acylaminobenzanilides 失效
标题翻译：杀虫剂3-酰氨基苯甲酰苯胺
公开(公告)号：US20090215623A1
公开(公告)日：2009-08-27
申请号：US11989485
申请日：2006-07-21
申请人： Akihiko Yanagi , Yukiyoshi Watanabe , Katsuaki Wada , Tetsuya Murata , Jun Mihara , Katsuhiko Shibuya , Eiichi Shimojo , Akira Emoto
发明人： Akihiko Yanagi , Yukiyoshi Watanabe , Katsuaki Wada , Tetsuya Murata , Jun Mihara , Katsuhiko Shibuya , Eiichi Shimojo , Akira Emoto
IPC分类号： A01N25/26 , C07D213/56 , C07C237/00 , C07D333/02 , C07D307/02 , C07D231/10 , C07D285/06 , A01N43/40 , A01N37/18 , A01N43/10 , A01N43/08 , A01N43/56 , A01N43/828 , A01P7/04
CPC分类号： C07C237/42 , A01N37/22 , A01N41/10 , A01N43/08 , A01N43/10 , A01N43/40 , A01N43/56 , A01N43/80 , A01N43/82 , C07D213/61 , C07D213/78 , C07D231/14 , C07D261/18 , C07D285/06 , C07D307/68 , C07D333/28 , C07D333/38
摘要： Novel 3-acylaminobenzanilides of the formula (I) wherein R1 represents phenyl which may be substituted or a 5-member or 6-member heterocyclic ring group, which may be substituted, containing at least one hetero-atom selected from the group consisting of N, O, and S; R2 represents halogen, C1-6 alkyl, or C1-6 haloalkyl; R3 represents C1-6 haloalkyl, C1-6 haloalkoxy, C1-6 haloalkylthio, C1-6 haloalkylsulfinyl, or C1-6 haloalkylsulfonyl; R4 represents halogen, C1-6 alkyl, or C1-6 haloalkyl; X represents halogen, C1-6 alkyl, or C1-6 haloalkyl; and n represents 0 or 1 and the compounds are used as insecticides, and a use of the new compounds as insecticides.
摘要翻译：式（I）的新型3-酰基氨基-N-苯甲酰苯胺，其中R 1表示可被取代的苯基或可以被取代的5-元件或6-元杂环基，其含有至少一个选自N ，O和S; R 2表示卤素，C 1-6烷基或C 1-6卤代烷基; R 3表示C 1-6卤代烷基，C 1-6卤代烷氧基，C 1-6卤代烷硫基，C 1-6卤代烷基亚磺酰基或C 1-6卤代烷基磺酰基; R 4表示卤素，C 1-6烷基或C 1-6卤代烷基; X表示卤素，C 1-6烷基或C 1-6卤代烷基; 并且n表示0或1，并且该化合物用作杀虫剂，并且使用新化合物作为杀虫剂。

136. 发明授权

US07569603B2 Ester compound and its use in pest control 失效
标题翻译：酯类化合物及其在病虫害防治中的应用
公开(公告)号：US07569603B2
公开(公告)日：2009-08-04
申请号：US11751306
申请日：2007-05-21
申请人： Tatsuya Mori
发明人： Tatsuya Mori
IPC分类号： A01N43/08 , C07D307/46
CPC分类号： C07D307/42 , A01N53/00
摘要： An ester compound represented by the formula (I): has excellent pest controlling activity and is useful as an active ingredient for a pest controlling agent.
摘要翻译：由式（I）表示的酯化合物：具有优异的害虫控制活性，可用作害虫控制剂的有效成分。

137. 发明申请

US20090163585A1 Carbosulfane-Based Pesticidal Compositions, Process for Preparing Same, Process for Controlling Insects/Mites/Nematodes, and Use of Said Compositions 审中-公开
标题翻译：基于碳硼烷的杀虫组合物，其制备方法，控制昆虫/螨虫/线虫的方法和所述组合物的用途
公开(公告)号：US20090163585A1
公开(公告)日：2009-06-25
申请号：US11817815
申请日：2006-03-09
申请人： Jair Sunega
发明人： Jair Sunega
IPC分类号： A01N43/08 , A01P5/00 , A01P7/02 , A01P7/04
CPC分类号： A01N47/24 , A01N2300/00
摘要： The present invention relates to pesticidal compositions comprising 2,3-dihydro-2,2-dimethylbenzofuran-7-yl(dibutylaminothio)methylcarbamate, namely benzofuranyl methylcarbamate, commonly known as carbosulfane, of structural formula (I). The present invention deals more particularly with compositions comprising this active compound at a high concentration, which makes it the most economical product for sale, more stable during storage and more effective in small quantities, and it may be further combined with one or more inerts. The present invention further discloses a process for preparing said compositions and a process for controlling insects/mites/nematode. The applications for these formulations include the treatment of seeds and leaves. In the latter case, in addition to the diluting agent, a mixture of anionic and non-ionic surfactants have been included in the formulation, so that the solution will become self-emulsifying upon being added to water.
摘要翻译：本发明涉及包含结构式（I）的2,3-二氢-2,2-二甲基苯并呋喃-7-基（二丁基氨基硫代）甲基氨基甲酸酯，即苯并呋喃基甲基氨基甲酸酯（通常称为碳硫烷）的农药组合物。本发明更具体地涉及包含这种高浓度活性化合物的组合物，其使其成为销售中最经济的产品，在储存期间更稳定并且更有效地少量，并且可以进一步与一种或多种惰性组合。本发明还公开了一种制备所述组合物的方法和一种防治昆虫/螨虫/线虫的方法。这些制剂的应用包括种子和叶子的处理。在后一种情况下，除了稀释剂之外，制剂中还包括阴离子和非离子表面活性剂的混合物，使得溶液在加入水中时将自乳化。

138. 发明申请

US20090118219A1 FLEA GABA RECEPTOR SUBUNIT NUCLEIC ACID MOLECULES 有权
标题翻译： FLEA GABA受体亚基核酸分子
公开(公告)号：US20090118219A1
公开(公告)日：2009-05-07
申请号：US12352535
申请日：2009-01-12
申请人： Nancy Wisnewski , Kevin S. Brandt
发明人： Nancy Wisnewski , Kevin S. Brandt
IPC分类号： A01N43/08 , C07H21/04 , C12N7/00 , A01P7/04 , C12N5/06
CPC分类号： C07K14/705 , A61K38/00 , G01N2500/04
摘要： The present invention relates to flea GABA receptor subunit nucleic acid molecules; to flea GABA receptor subunit proteins encoded by such nucleic acid molecules; to antibodies raised against such proteins; and to compounds that inhibit the activity of such proteins. The present invention also includes methods to obtain such proteins, nucleic acid molecules, antibodies, and inhibitory compounds. The present invention also includes therapeutic compositions comprising such proteins, nucleic acid molecules, antibodies and inhibitory compounds, particularly those that specifically inhibit flea GABA receptor subunit activity, as well as the use of such therapeutic compositions to treat animals.
摘要翻译：本发明涉及跳蚤GABA受体亚基核酸分子; 由这种核酸分子编码的跳蚤GABA受体亚基蛋白; 针对这种蛋白质产生的抗体; 以及抑制这些蛋白质活性的化合物。本发明还包括获得这些蛋白质，核酸分子，抗体和抑制性化合物的方法。本发明还包括包含这些蛋白质，核酸分子，抗体和抑制性化合物，特别是那些特异性抑制跳蚤GABA受体亚基活性的化合物的治疗组合物，以及这些治疗组合物用于治疗动物的治疗组合物。

139. 发明授权

US07488752B2 Thrombin receptor antagonists 有权
标题翻译：凝血酶受体拮抗剂
公开(公告)号：US07488752B2
公开(公告)日：2009-02-10
申请号：US11243708
申请日：2005-10-05
申请人： Samuel Chackalamannil , Mariappan V. Chelliah , Yan Xia , Keith A. Eagen
发明人： Samuel Chackalamannil , Mariappan V. Chelliah , Yan Xia , Keith A. Eagen
IPC分类号： A01N43/08 , A61K31/34 , C07D307/00 , C07D307/93 , C07D407/00
CPC分类号： C07D405/06 , C07D405/14 , C07D409/14 , C07D413/14 , C07D491/10
摘要： Heterocyclic-substituted tricyclics of the formula or a pharmaceutically acceptable salt or solvate of said compound, isomer or racemic mixture wherein z,1 represents an optional double bond, the dotted line is optionally a bond or no bond, resulting in a double bond or a single bond, as permitted by the valency requirement and wherein A, B, G, M, X, J, n, Het, R3, R10, R11, R32 and R33 are herein defined and the remaining substituents are as defined in the specification, are disclosed, as well as pharmaceutical compositions containing them and a method of treating diseases associated with thrombosis, atherosclerosis, restenosis, hypertension, angina pectoris, arrhythmia, heart failure, and cancer by administering said compounds. Combination therapy with other cardiovascular agents is also claimed.
摘要翻译：具有下式的杂环取代的三环或所述化合物，异构体或外消旋混合物的药学上可接受的盐或溶剂化物，其中z 1表示任选的双键，虚线任选是键或无键，得到双键或单价，如价格要求所允许的，其中A，B，G，M，X，J，n，Het，R 3，R 10，R 11，R 32和R 33在本文中定义，其余取代基如说明书中所定义，以及含有它们的药物组合物以及通过施用所述化合物治疗与血栓形成，动脉粥样硬化，再狭窄，高血压，心绞痛，心律失常，心力衰竭和癌症相关的疾病的方法。还要求与其它心血管药物联合治疗。

140. 发明申请

US20080319015A1 Insect Repellent Mixture 审中-公开
标题翻译：防虫混合物
公开(公告)号：US20080319015A1
公开(公告)日：2008-12-25
申请号：US12158355
申请日：2006-11-24
申请人： Hans-Werner Gruenewald , Alexandra Axt
发明人： Hans-Werner Gruenewald , Alexandra Axt
IPC分类号： A01N43/40 , A01N37/18 , A01N43/08 , A01N37/00 , A01P17/00
CPC分类号： A01N37/18 , A01N43/40 , A01N2300/00
摘要： The present invention relates to the use of an insect repellent, preferably selected from the group 2-(2-hydroxyethyl)-1-methylpropyl 1-piperidinecarboxylate, N,N-diethyl-3-methylbenzamide, dimethyl phthalate, butopyronoxyl, 2,3,4,5-bis(2-butylene)-tetrahydro-2-furaldehyde, N,N-diethylcaprylamide, N,N-diethylbenzamide, o-chloro-N,N-diethylbenzamide, dimethyl carbate, di-n-propyl isocinchomeronate, 2-ethylhexane-1,3-diol, N-octylbicycloheptenedicarboximide or piperonyl butoxide, particularly preferably 2-(2-hydroxyethyl)-1-methylpropyl 1-piperidinecarboxylate, as action enhancer for a second insect repellent, to corresponding compositions, and to the preparation thereof.
摘要翻译：本发明涉及驱虫剂的用途，优选选自1-（2-羟基乙基）-1-哌啶羧酸2-甲基丙酯，N，N-二乙基-3-甲基苯甲酰胺，邻苯二甲酸二甲酯，叠氮氧基，2,3 ，4,5-双（2-丁烯） - 四氢-2-糠醛，N，N-二乙基己酰胺，N，N-二乙基苯甲酰胺，邻氯-N，N-二乙基苯甲酰胺，碳酸二甲酯，异辛基二正丙基酯， 2-乙基己烷-1,3-二醇，N-辛基双环加二甲酰亚胺或胡椒基丁醚，特别优选2-（2-羟乙基）-1-甲基丙基1-哌啶羧酸酯作为第二驱虫剂的作用增强剂，相应的组合物，以及的制备。

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