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91. 发明申请

US20140371065A1 Fungicidal Pyrimidine Compounds 有权
标题翻译：杀真菌嘧啶化合物
公开(公告)号：US20140371065A1
公开(公告)日：2014-12-18
申请号：US14375240
申请日：2013-01-30
申请人： Wassilios Grammenos , Ian Robert Craig , Nadege Boudet , Bernd Mueller , Jochen Dietz , Erica May Wilson Lauterwasser , Jan Klaas Lohmann , Jurith Montag
发明人： Wassilios Grammenos , Ian Robert Craig , Nadege Boudet , Bernd Mueller , Jochen Dietz , Erica May Wilson Lauterwasser , Jan Klaas Lohmann , Jurith Montag
IPC分类号： A01N43/90 , A01N43/54 , C07D487/04 , C07D401/12
CPC分类号： A01N43/90 , A01N43/54 , C07D401/12 , C07D487/04 , C07D491/04
摘要： The present invention relates to fungicidal pyrimidine compounds I, to their use and to methods for combating phytopathogenic fungi. The present invention also relates to seeds treated with at least one such compound. Furthermore the invention relates to processes for preparing compounds of formula I.
摘要翻译：本发明涉及杀真菌嘧啶化合物I，其用途和用于防治植物病原真菌的方法。本发明还涉及用至少一种这样的化合物处理的种子。此外，本发明涉及制备式I化合物的方法。

92. 发明申请

US20140045689A1 3,4-disubstituted pyrrole 2,5-diones and their use as fungicides 审中-公开
标题翻译： 3,4-二取代吡咯2,5-二酮及其作为杀真菌剂的用途
公开(公告)号：US20140045689A1
公开(公告)日：2014-02-13
申请号：US14112616
申请日：2012-04-19
申请人： Richard Riggs , Jochen Dietz , Wassilios Grammenos , Bernd Mueller , Jan Klaas Lohmann , Nadege Boudet , Ian Robert Craig , Egon Haden , Jurith Montag
发明人： Richard Riggs , Jochen Dietz , Wassilios Grammenos , Bernd Mueller , Jan Klaas Lohmann , Nadege Boudet , Ian Robert Craig , Egon Haden , Jurith Montag
IPC分类号： A01N43/36
CPC分类号： A01N43/36 , A01N37/32 , A01N37/34 , A01N37/36 , A01N37/38 , A01N37/44 , C07D207/456
摘要： The present invention relates to the use of 3,4-disubstituted pyrrole 2,5-diones of the formula I as defined in the description for controlling phytopathogenic fungi. Further the invention relates to novel compounds of the formula I.
摘要翻译：本发明涉及用于控制植物病原真菌的描述中所定义的式I的3,4-二取代吡咯2,5-二酮的用途。本发明还涉及新的式I化合物。

93. 发明申请

US20140031208A1 Use of substituted dithiine-tetracarboximides for combating phytopathogenic fungi 有权
标题翻译：使用取代的二硫代四羧酰亚胺对抗植物病原性真菌
公开(公告)号：US20140031208A1
公开(公告)日：2014-01-30
申请号：US14111270
申请日：2012-04-10
申请人： Bernd Mueller , Nadege Boudet , Jochen Dietz , Wassilios Grammenos , Jan Klaas Lohmann , Richard Riggs , Ian Robert Craig , Jurith Montag , Egon Haden
发明人： Bernd Mueller , Nadege Boudet , Jochen Dietz , Wassilios Grammenos , Jan Klaas Lohmann , Richard Riggs , Ian Robert Craig , Jurith Montag , Egon Haden
IPC分类号： A01N43/36
CPC分类号： A01N43/36 , A01N43/90
摘要： The present invention relates to the use of dithiine-tetracarboximide compounds of formula I as defined in the description, and the N-oxides, and salts thereof for combating harmful fungi and seed coated with at least one such compound. The invention also relates to novel dithiine-tetracarboximides, processes and intermediates for preparing these compounds and also to compositions comprising at least one such compound.
摘要翻译：本发明涉及描述中所定义的式I的二硫代 - 四甲酰亚胺化合物及其N-氧化物及其盐用于防治有害真菌和用至少一种这样的化合物包被的种子。本发明还涉及用于制备这些化合物的新型二硫代 - 四酰亚胺化物，方法和中间体以及包含至少一种这样的化合物的组合物。

94. 发明申请

US20080262000A1 5-Alkoxyalkyl-6-alkyl-7-Aminoazolopyrimidines, Process for Their Preparation, Their Use for Controlling Harmful Fungi, and Compositions Comprising Them 审中-公开
标题翻译： 5-烷氧基烷基-6-烷基-7-氨基偶氮嘧啶，其制备方法，它们用于控制有害真菌的用途，以及包含它们的组合物
公开(公告)号：US20080262000A1
公开(公告)日：2008-10-23
申请号：US11884412
申请日：2006-02-14
申请人： Peter Schafer , Udo Hunger , Maria Scherer , Harald Kohle , Helmut Schiffer , Thomas Grote , Jochen Dietz , Wassilios Grammenos , Jan Klaas Lohmann , Bernd Muller , Joachim Rheinheimer , Frank Schieweck , Anja Schwogler
发明人： Peter Schafer , Udo Hunger , Maria Scherer , Harald Kohle , Helmut Schiffer , Thomas Grote , Jochen Dietz , Wassilios Grammenos , Jan Klaas Lohmann , Bernd Muller , Joachim Rheinheimer , Frank Schieweck , Anja Schwogler
IPC分类号： A01N43/90 , C07D487/04 , A01P3/00
CPC分类号： C07D487/04
摘要： 5-Alkoxyalkyl-6-alkyl-7-aminoazolopyrimidines of the formula I in which the substituents are defined as follows: R1 is alkyl, cycloalkyl, alkenyl, alkynyl, alkoxyalkyl, cyanoalkyl, and benzyloxyalkyl, where the groups in the aliphatic or aromatic moiety may be unsubstituted or may have substitution by from one to three groups Ra: Ra is halogen, cyano, nitro, hydroxy, cycloalkyl, alkoxy, alkylthio, and NRARB; RA, RB are hydrogen and alkyl; R2 is alkoxyalkyl, phenoxyalkyl, alkylthioalkyl, and phenylthioalkyl, which groups may have no substitution or may have substitution according to the description; R3 is hydrogen and alkyl; A is N and C—RA; processes for preparation of these compounds, compositions comprising them, and their use for controlling phytopathogenic harmful fungi.
摘要翻译：式I的5-烷氧基烷基-6-烷基-7-氨基偶氮嘧啶，其中取代基定义如下：R 1是烷基，环烷基，烯基，炔基，烷氧基烷基，氰基烷基和苄氧基烷基，其中脂族或芳族部分中的基团可以是未取代的或可以具有一至三个基团的取代基：R a是卤素，氰基，硝基，羟基，环烷基，烷氧基，烷硫基和NR A R B， R A，B B是氢和烷基; R 2是烷氧基烷基，苯氧基烷基，烷硫基烷基和苯硫基烷基，该基团可以不具有取代基或可以根据描述进行取代; R 3是氢和烷基; A是N和C-R A; 制备这些化合物的方法，包含它们的组合物及其用于控制植物病原性有害真菌的用途。

95. 发明申请

US20100130359A1 Fungicidal Pyridazines, Processes for Their Preparation and Their Use for Controlling Harmful Fungi, and Compositions Comprising Them 审中-公开
标题翻译：杀真菌哒嗪，其制备方法及其用于控制有害真菌的组合物及其组合物
公开(公告)号：US20100130359A1
公开(公告)日：2010-05-27
申请号：US12597972
申请日：2008-04-25
申请人： Jochen Dietz , Marianna Vrettou , Bernd Mueller , Jens Renner , Sarah Ulmscheneider , Jan Klaas Lohmann
发明人： Jochen Dietz , Marianna Vrettou , Bernd Mueller , Jens Renner , Sarah Ulmscheneider , Jan Klaas Lohmann
IPC分类号： A01C1/06 , C07D401/04 , A61K31/50 , A01N43/58 , C07D237/02
CPC分类号： C07D237/12 , C07D237/16
摘要： Pyridazines of the formula I in which the substituents are defined according to the description, processes and intermediates for preparing these compounds, compositions comprising them and also their use for controlling phytopathogenic harmful fungi, and also the use of the pyridazines for preparing a medicament for treating cancer.
摘要翻译：其中取代基根据描述，制备这些化合物的方法和中间体，包含它们的组合物以及它们用于控制植物病原性有害真菌的用途，以及使用哒嗪制备用于治疗的药物的式I的哒嗪癌症。

96. 发明申请

US20090036305A1 PYRAZOLECARBOXAMIDES 失效
标题翻译：吡咯烷氧基胺
公开(公告)号：US20090036305A1
公开(公告)日：2009-02-05
申请号：US11919588
申请日：2006-05-10
申请人： Markus Gewehr , Jochen Dietz , Thomas Grote , Wassilios Gremmenos , Udo Hunger , Bernd Muller , Frank Schieweck , Anja Schwogler , Jan Klaas Lohmann , Joachim Rheinheimer , Jens Renner , Peter Schafer
发明人： Markus Gewehr , Jochen Dietz , Thomas Grote , Wassilios Gremmenos , Udo Hunger , Bernd Muller , Frank Schieweck , Anja Schwogler , Jan Klaas Lohmann , Joachim Rheinheimer , Jens Renner , Peter Schafer
IPC分类号： A01N43/56 , C07D231/14 , A01P3/00
CPC分类号： A01N43/56 , C07D231/14
摘要： The present invention relates to pyrazolecarboxamides of the formula I in which the variables are as defined below: X is trifluoromethyl; R1 is F, Cl, Br, C1-C4-alkyl or C1-C4-haloalkyl; R2 is hydrogen, halogen or C1-C4-alkyl; R3 is hydrogen, C1-C4-alkyl, C1-C4-haloalkyl, C2-C4-alkenyl, C2-C4-alkynyl or C3-C6-cycloalkyl; W is O or S; with the proviso that, if R3 is hydrogen and W is oxygen, a) R1 and R2 are not simultaneously methyl and F, respectively; b) R1 and R2 are not simultaneously trifluoromethyl and hydrogen or fluorine, respectively. to processes for preparing these compounds, to seeds and compositions comprising them and to methods for controlling harmful fungi.
摘要翻译：本发明涉及式I的吡唑酰胺，其中变量如下所定义：X是三氟甲基; R1是F，Cl，Br，C1-C4-烷基或C1-C4卤代烷基; R2是氢，卤素或C1-C4-烷基; R 3是氢，C 1 -C 4 - 烷基，C 1 -C 4卤代烷基，C 2 -C 4 - 烯基，C 2 -C 4 - 炔基或C 3 -C 6 - 环烷基; W为O或S; 条件是，如果R3是氢并且W是氧，则a）R1和R2分别不同时为甲基和F; b）R1和R2分别不同时为三氟甲基和氢或氟。制备这些化合物的方法，包括它们的种子和组合物以及用于控制有害真菌的方法。

97. 发明申请

US20140121103A1 COMPOSITIONS COMPRISING FUNGICIDAL SUBSTITUTED DITHIINES AND FURTHER ACTIVES 审中-公开
标题翻译：包含杀真菌剂替代物和其他活性的组合物
公开(公告)号：US20140121103A1
公开(公告)日：2014-05-01
申请号：US14126644
申请日：2012-06-15
申请人： Nadege Boudet , Wassilios Grammenos , Jochen Dietz , Egon Haden , Richard Riggs , Bernd Müller , Jan Klaas Lohmann , Jurith Montag , Ian Robert Craig
发明人： Nadege Boudet , Wassilios Grammenos , Jochen Dietz , Egon Haden , Richard Riggs , Bernd Müller , Jan Klaas Lohmann , Jurith Montag , Ian Robert Craig
IPC分类号： A01N43/32 , A01N43/52 , A01N43/90 , A01N43/653 , A01N43/78 , A01N43/40 , A01N43/56 , A01N37/34
CPC分类号： A01N43/32 , A01N37/34 , A01N43/40 , A01N43/52 , A01N43/56 , A01N43/653 , A01N43/78 , A01N43/90 , A01N2300/00 , A01N37/24 , A01N37/46 , A01N43/50 , A01N43/54 , A01N47/12 , A01N47/18 , A01N47/24 , A01N47/38
摘要： The present invention relates to synergistic mixtures comprising at least one compound I and at least one active compound II as defined herein and to the use of these mixtures for combating phytopathogenic fungi, and to seeds coated with at least one such mixture. The invention also relates methods for combating harmful fungi using such mixtures.
摘要翻译：本发明涉及包含至少一种化合物I和本文定义的至少一种活性化合物II以及这些混合物用于防治植物病原性真菌的用途的协同混合物，以及用至少一种这样的混合物涂覆的种子。本发明还涉及使用这种混合物对抗有害真菌的方法。

98. 发明申请

US20100184994A1 Method for Producing Difluoromethyl-Substituted Pyrazole Compounds 有权
标题翻译：二氟甲基取代吡唑化合物的制备方法
公开(公告)号：US20100184994A1
公开(公告)日：2010-07-22
申请号：US12664448
申请日：2008-06-13
申请人： Markus Nett , Thomas Grote , Jan Klaas Lohmann , Jochen Dietz , Sebastian Peer Smidt , Michael Rack , Thomas Zierke
发明人： Markus Nett , Thomas Grote , Jan Klaas Lohmann , Jochen Dietz , Sebastian Peer Smidt , Michael Rack , Thomas Zierke
IPC分类号： C07D231/14 , C07C229/06
CPC分类号： C07D231/12 , C07D231/14
摘要： The present invention relates to a process for preparing 3-difluoromethyl-substituted pyrazole compounds of the formula (I) in which R1 is H, halogen, nitro, C1-C8-alkyl, C1-C8-haloalkyl, C3-C8-cycloalkyl, phenyl, naphthyl, hetaryl, cyano, —C(═O)—OR1a, —C(═O)—NR1bR1c, —C(═O)—SR1d or —C(═S)—SR1e; R2 is H, C1-C4-alkyl, benzyl or phenyl; R3 is H, halogen, C1-C8-alkoxy, C1-C8-haloalkoxy, C3-C8-cycloalkoxy, C2-C8-alkenyloxy, C1-C8-alkylthio, C1-C8-haloalkylthio, C3-C8-cyclo-alkylthio or C2-C8-alkenylthio; compounds of the formula (II.a) or (II.b), in which R1 and R3 each have one of the definitions given above; R4 is halogen, —OR4a, —SR4a, —O—SO2—R4a or an —NR4bR4c group; R5 and R6 are each C1-C8-alkyl, C1-C8-haloalkyl, C3-C8-cycloalkyl, benzyl or phenyl, or, together with the nitrogen atom to which they are bonded, are a 3- to 8-membered heterocycle; Lewis acid adducts of compounds of the formula (II.b); the use of compounds of the formula (II.a) or (II.b) and of the Lewis acid adducts for preparing compounds of the formula (I) or (VI); and to a process for converting such compounds to the corresponding 3-difluoro-pyrazol-4-ylcarboxylic acids.
摘要翻译：本发明涉及制备式（I）的3-二氟甲基取代的吡唑化合物的方法，其中R 1是H，卤素，硝基，C 1 -C 8 - 烷基，C 1 -C 8 - 卤代烷基，C 3 -C 8 - 环烷基，苯基，萘基，杂芳基，氰基，-C（= O）-OR1a，-C（= O）-NR1bR1c，-C（= O）-SR1d或-C（= S）-SR1e; R2是H，C1-C4-烷基，苄基或苯基; R 3是H，卤素，C 1 -C 8 - 烷氧基，C 1 -C 8 - 卤代烷氧基，C 3 -C 8 - 环烷氧基，C 2 -C 8 - 烯氧基，C 1 -C 8 - 烷硫基，C 1 -C 8 - 卤代烷硫基，C 3 -C 8环 - C 2 -C 8 - 烯硫基; 式（II.a）或（II.b）化合物，其中R 1和R 3各自具有上述定义之一; R4是卤素，-OR4a，-SR4a，-O-SO2-R4a或-NR4bR4c基团; R 5和R 6各自为C 1 -C 8 - 烷基，C 1 -C 8 - 卤代烷基，C 3 -C 8 - 环烷基，苄基或苯基，或与它们所键合的氮原子一起为3-至8-元杂环; 式（II.b）化合物的路易斯酸加合物; 使用式（II.a）或（II.b）化合物和路易斯酸加成物制备式（I）或（VI）化合物的方法; 以及将这些化合物转化为相应的3-二氟 - 吡唑-4-基羧酸的方法。

99. 发明授权

US08115012B2 Process for preparing difluoromethylpyrazolyl carboxylates 失效
标题翻译：制备二氟甲基吡唑羧酸酯的方法
公开(公告)号：US08115012B2
公开(公告)日：2012-02-14
申请号：US12513003
申请日：2007-11-02
申请人： Martin Sukopp , Michael Rack , Sebastian Peer Smidt , Sandra Löhr , Michael Keil , Jochen Dietz , Joachim Rheinheimer , Thomas Grote , Thomas Zierke , Jan Klaas Lohmann
发明人： Martin Sukopp , Michael Rack , Sebastian Peer Smidt , Sandra Löhr , Michael Keil , Jochen Dietz , Joachim Rheinheimer , Thomas Grote , Thomas Zierke , Jan Klaas Lohmann
IPC分类号： C07D231/10 , C07F7/08
CPC分类号： C07D231/14
摘要： The present invention relates to a process for preparing difluoromethyl-substituted pyrazol-4-ylcarboxylates of the formula I in which R1 is C1-C8-alkyl, C3-C8-cycloalkyl, C1-C4-alkoxy-C1-C4-alkyl, etc.; and R2 is hydrogen, C1-C4-alkyl, benzyl or phenyl, wherein a) a compound of the general formula II in which X is fluorine, chlorine or bromine, R1 has one of the meanings given above and R4 is C1-C8-alkyl, C3-C8-cycloalkyl, C2-C8-alkenyl, benzyl or phenyl, is reacted with a silane compound of the general formula R3nSiCl(4-n) in which n is 1, 2 or 3 and the substituents R3 are independently of one another selected from the group consisting of C1-C8-alkyl and phenyl and with a metal selected from the metals of groups 1, 2, 3, 4 and 12 of the Periodic Table of the Elements having a redox potential of less than −0.7 V, based on a normal hydrogen electrode (at 25° C. and 101.325 kPa); and b) the reaction mixture from step a) is reacted with a compound of the general formula III R2HN—NH2 (III) in which R2 has one of the meanings given above.
摘要翻译：本发明涉及制备式Ⅰ的二氟甲基取代的吡唑-4-基羧酸酯的方法，其中R 1是C 1 -C 8烷基，C 3 -C 8环烷基，C 1 -C 4烷氧基-C 1 -C 4烷基等。 R 2是氢，C 1 -C 4 - 烷基，苄基或苯基，其中a）通式II的化合物，其中X是氟，氯或溴，R 1具有上面给出的含义之一，R 4是C 1 -C 8 - 烷基，C 3 -C 8 - 环烷基，C 2 -C 8 - 烯基，苄基或苯基与通式R 3 n SiCl（4-n）的硅烷化合物反应，其中n为1,2或3，取代基R 3独立地为选自由C 1 -C 8 - 烷基和苯基组成的组中的一种，以及选自元素周期表第1,2,3,4和12族金属的金属，其氧化还原电位小于-0.7 V，基于正常的氢电极（在25℃和101.325kPa）; 和b）将来自步骤a）的反应混合物与通式III的化合物R2HN-NH2（III）反应，其中R2具有上述含义之一。

100. 发明申请

US20100069646A1 Process for preparing difluoromethylpyrazolyl carboxylates 失效
标题翻译：制备二氟甲基吡唑羧酸酯的方法
公开(公告)号：US20100069646A1
公开(公告)日：2010-03-18
申请号：US12513003
申请日：2007-11-02
申请人： Martin Sukopp , Michael Rack , Sebastian Peer Smidt , Sandra Löhr , Michael Keil , Jochen Dietz , Joachim Rheinheimer , Thomas Grote , Thomas Zierke , Jan Klaas Lohmann
发明人： Martin Sukopp , Michael Rack , Sebastian Peer Smidt , Sandra Löhr , Michael Keil , Jochen Dietz , Joachim Rheinheimer , Thomas Grote , Thomas Zierke , Jan Klaas Lohmann
IPC分类号： C07D231/10 , C07F7/08
CPC分类号： C07D231/14
摘要： The present invention relates to a process for preparing difluoromethyl-substituted pyrazol-4-ylcarboxylates of the formula I in which R1 is C1-C8-alkyl, C3-C8-cycloalkyl, C1-C4-alkoxy-C1-C4-alkyl, etc.; and R2 is hydrogen, C1-C4-alkyl, benzyl or phenyl, wherein a) a compound of the general formula II in which X is fluorine, chlorine or bromine, R1 has one of the meanings given above and R4 is C1-C8-alkyl, C3-C8-cycloalkyl, C2-C8-alkenyl, benzyl or phenyl, is reacted with a silane compound of the general formula R3nSiCl(4-n) in which n is 1, 2 or 3 and the substituents R3 are independently of one another selected from the group consisting of C1-C8-alkyl and phenyl and with a metal selected from the metals of groups 1, 2, 3, 4 and 12 of the Periodic Table of the Elements having a redox potential of less than −0.7 V, based on a normal hydrogen electrode (at 25° C. and 101.325 kPa); and b) the reaction mixture from step a) is reacted with a compound of the general formula III R2HN—NH2 (III) in which R2 has one of the meanings given above.
摘要翻译：本发明涉及制备式Ⅰ的二氟甲基取代的吡唑-4-基羧酸酯的方法，其中R 1是C 1 -C 8烷基，C 3 -C 8环烷基，C 1 -C 4烷氧基-C 1 -C 4烷基等。并且R 2是氢，C 1 -C 4 - 烷基，苄基或苯基，其中a）通式II的化合物，其中X是氟，氯或溴，R 1具有上面给出的含义之一，R 4是C 1 -C 8 - 烷基，C 3 -C 8 - 环烷基，C 2 -C 8 - 烯基，苄基或苯基与通式R 3 n SiCl（4-n）的硅烷化合物反应，其中n为1,2或3，取代基R 3独立地为选自由C 1 -C 8 - 烷基和苯基组成的组中的一种，以及选自元素周期表第1,2,3,4和12族金属的金属，其氧化还原电位小于-0.7 V，基于正常的氢电极（在25℃和101.325kPa）; 和b）将来自步骤a）的反应混合物与通式III的化合物R2HN-NH2（III）反应，其中R2具有上述含义之一。

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