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1. 发明授权

EP2668154B1 FORMULATION COMPONENT 有权
公开(公告)号：EP2668154B1
公开(公告)日：2018-03-21
申请号：EP11793390.3
申请日：2011-11-29
申请人： Syngenta Limited
发明人： BELL, Gordon, Alastair , PERRY, Richard , RAMSAY, Julia, Lynne , STOCK, David , TAYLOR, Philip
IPC分类号： C07C233/65 , C07C233/69 , A01N25/00 , A01N41/06 , A01N47/36 , A01N41/10 , A01N43/90
CPC分类号： A01N25/00 , A01N37/18 , A01N37/20 , A01N41/06 , A01N41/10 , A01N43/54 , A01N43/90 , A01N47/36 , C07C233/65 , C07C233/69 , A01N2300/00
摘要： The present invention relates to agrochemical compositions comprising certain benzamide compounds and to the use of those benzamide compounds as adjuvants, especially in formulations,in particular in agrochemical formulations and in environmentally friendly formulations. The invention further extends to certain novel benzamide compounds and a process to prepare such novel compounds.

3. 发明公开

EP2891489A4 ENDOPARASITE CONTROL AGENT AND USE THEREOF 有权
标题翻译：禁止对其进行内分泌控制和使用
公开(公告)号：EP2891489A4
公开(公告)日：2016-01-27
申请号：EP13832194
申请日：2013-08-29
申请人： UNIV TOKYO , NIHON NOHYAKU CO LTD
发明人： KITA KIYOSHI , SUWA AKIYUKI , ODA MASATSUGU , TANAKA KOJI
IPC分类号： A61K31/166 , A61K31/415 , A61K31/44 , A61P33/00 , C07C235/60 , C07C317/32 , C07C323/62 , C07D213/61 , C07D213/64 , C07D213/643 , C07D213/74 , C07D231/12 , C07D231/16 , C07D231/18 , C07D231/20 , C07D401/04
CPC分类号： C07D401/04 , A61K31/166 , A61K31/415 , A61K31/44 , C07C233/69 , C07C235/46 , C07C235/60 , C07C317/32 , C07C323/42 , C07C323/62 , C07D213/56 , C07D213/61 , C07D213/643 , C07D213/74 , C07D231/12 , C07D231/16 , C07D231/18 , C07D231/20
摘要： An object of the present invention is to provide a novel endoparasite control agent as a parasiticide, an antiprotozoal or the like. Provided is an endoparasite control agent comprising a carboxamide derivative represented by the general formula (I): or a salt thereof as an active ingredient.

4. 发明授权

EP1481965B1 AROMATIC AMINO ACID DERIVATIVES AND MEDICINAL COMPOSITIONS 有权
标题翻译：芳香族氨基酸衍生物及医药组合物
公开(公告)号：EP1481965B1
公开(公告)日：2015-07-29
申请号：EP03703151.5
申请日：2003-02-03
申请人： Endo, Hitoshi
发明人： ENDO, Hitoshi , KANAI, Yoshikatsu , TSUJIHARA, Kenji , SAITO, Kunio
IPC分类号： C07C229/36 , C07C255/54 , C07D207/333
CPC分类号： C07D207/325 , C07C229/36 , C07C233/47 , C07C233/69 , C07C255/54 , C07C271/10 , C07C2602/10 , C07D209/08 , C07D213/30 , C07D213/74 , C07D215/14 , C07D235/18 , C07D239/42 , C07D263/32 , C07D263/56 , C07D265/36 , C07D277/24 , C07D277/66 , C07D307/79 , C07D307/82 , C07D307/83 , C07D307/91 , C07D311/30 , C07D401/04 , C07D413/04 , C07D417/04 , C07D471/06 , Y02P20/55

5. 发明公开

EP2891489A1 ENDOPARASITE CONTROL AGENT AND USE THEREOF 有权
标题翻译：内毒素控制剂及其用途
公开(公告)号：EP2891489A1
公开(公告)日：2015-07-08
申请号：EP13832194.8
申请日：2013-08-29
申请人： The University of Tokyo , Nihon Nohyaku Co., Ltd.
发明人： KITA, Kiyoshi , SUWA, Akiyuki , ODA, Masatsugu , TANAKA, Koji
IPC分类号： A61K31/166 , A61K31/415 , A61K31/44 , A61P33/00
CPC分类号： C07D401/04 , A61K31/166 , A61K31/415 , A61K31/44 , C07C233/69 , C07C235/46 , C07C235/60 , C07C317/32 , C07C323/42 , C07C323/62 , C07D213/56 , C07D213/61 , C07D213/643 , C07D213/74 , C07D231/12 , C07D231/16 , C07D231/18 , C07D231/20
摘要： An object of the present invention is to provide a novel endoparasite control agent as a parasiticide, an antiprotozoal or the like. Provided is an endoparasite control agent comprising a carboxamide derivative represented by the general formula (I):

or
a salt thereof as an active ingredient.
摘要翻译：本发明的一个目的是提供一种新的内寄生虫防治剂作为杀寄生虫剂，抗原生动物剂等。提供了一种内寄生物防治剂，其包含由通式（I）表示的甲酰胺衍生物或其盐作为活性成分。

6. 发明授权

EP2403824B1 PROCESS FOR PREPARING CARBOXYLIC ACID AMIDES USEFUL IN THE TREATMENT OF MUSCULAR DISORDERS 有权
标题翻译：工艺制备用于肌肉疾病的处理的合适羧酸酰胺
公开(公告)号：EP2403824B1
公开(公告)日：2013-05-15
申请号：EP10707335.5
申请日：2010-03-03
申请人： UCL Business Plc.
发明人： SELWOOD, David
IPC分类号： C07C231/02 , C07C233/68 , C07C231/12
CPC分类号： C07C231/02 , C07C231/12 , C07C233/69

7. 发明公开

EP2196451A4 ACYLATION REACTION OF HYDROXYL GROUP 审中-公开
标题翻译：酰化反应羟基
公开(公告)号：EP2196451A4
公开(公告)日：2011-03-30
申请号：EP08838350
申请日：2008-10-10
申请人： TAKASAGO PERFUMERY CO LTD
发明人： MASHIMA KAZUSHI , OHSHIMA TAKASHI , IWASAKI TAKANORI , SAYO NOBORU
IPC分类号： C07C67/03 , C07B61/00 , C07C69/24 , C07C69/612 , C07C69/618 , C07C69/78 , C07C213/06 , C07C219/14 , C07C219/22 , C07C219/24 , C07C253/30 , C07C255/57
CPC分类号： C07D213/55 , C07C67/03 , C07C67/08 , C07C213/06 , C07C231/02 , C07C253/30 , C07C2601/14 , C07C2602/08 , C07C2602/10 , C07D211/34 , C07D295/195 , C07C69/618 , C07C69/24 , C07C69/612 , C07C69/76 , C07C69/78 , C07C219/14 , C07C219/18 , C07C219/22 , C07C233/69 , C07C233/73 , C07C255/57
摘要： Disclosed is a selective ester production process of an alcoholic hydroxyl group, which proceeds under chemically mild conditions, while having adequate environmental suitability, operability and economical efficiency. Specifically disclosed is a process for producing an ester compound, which is characterized in that an alcohol and a carboxylic acid ester compound are reacted in the presence of a compound containing zinc element, thereby selectively acylating a hydroxyl group of the alcohol.

8. 发明公开

EP2059499A4 PROCESSES OF PREPARING ASYMMETRIC DINITROBENZAMIDE MUSTARD COMPOUNDS, INTERMEDIATE COMPOUNDS USEFUL THEREIN AND PRODUCTS OBTAINED THEREFROM 审中-公开
标题翻译：用于生产不对称DINITROBENZAMIDSENFVERBINDUNGEN，BETWEEN和物品获得的产品从来没有有用的链接
公开(公告)号：EP2059499A4
公开(公告)日：2011-02-09
申请号：EP07834856
申请日：2007-09-04
申请人： AUCKLAND UNISERVICES LTD
发明人： ATWELL GRAHAM JOHN , DENNY WILLIAM ALEXANDER , YANG SHANGJIN
IPC分类号： C07C309/66 , C07C227/04 , C07C229/60 , C07C231/12 , C07C233/69 , C07C237/30 , C07C303/28 , C07D203/10 , C07F9/09 , C07H15/18
CPC分类号： C07D203/10 , C07C227/06 , C07C231/12 , C07C303/28 , C07C309/66 , C07C309/67 , C07D307/20 , C07F9/091 , C07C229/56 , C07C233/69

9. 发明公开

EP2196451A1 ACYLATION REACTION OF HYDROXYL GROUP 审中-公开
标题翻译： ACYLIERUNGSREAKING EINER HYDROXYLGRUPPE
公开(公告)号：EP2196451A1
公开(公告)日：2010-06-16
申请号：EP08838350.0
申请日：2008-10-10
申请人： Takasago International Corporation
发明人： MASHIMA, Kazushi , OHSHIMA, Takashi , IWASAKI, Takanori , SAYO, Noboru
IPC分类号： C07C67/03 , C07C69/24 , C07C69/612 , C07C69/618 , C07C69/78 , C07C213/06 , C07C219/14 , C07C219/22 , C07C219/24 , C07C253/30 , C07C255/57 , C07B61/00
CPC分类号： C07D213/55 , C07C67/03 , C07C67/08 , C07C213/06 , C07C231/02 , C07C253/30 , C07C2601/14 , C07C2602/08 , C07C2602/10 , C07D211/34 , C07D295/195 , C07C69/618 , C07C69/24 , C07C69/612 , C07C69/76 , C07C69/78 , C07C219/14 , C07C219/18 , C07C219/22 , C07C233/69 , C07C233/73 , C07C255/57
摘要： Disclosed is a selective ester production process of an alcoholic hydroxyl group, which proceeds under chemically mild conditions, while having adequate environmental suitability, operability and economical efficiency. Specifically disclosed is a process for producing an ester compound, which is characterized in that an alcohol and a carboxylic acid ester compound are reacted in the presence of a compound containing zinc element, thereby selectively acylating a hydroxyl group of the alcohol.
摘要翻译：公开了在化学温和条件下进行的醇羟基的选择性酯生产方法，同时具有足够的环境适应性，可操作性和经济效率。具体公开了一种酯化合物的制造方法，其特征在于，在含有锌元素的化合物的存在下使醇和羧酸酯化合物反应，从而选择性地酰化醇的羟基。

10. 发明公开

EP2177503A1 MODULATORS OF CANNABINOID RECEPTORS 有权
标题翻译：大麻素受体的调节因子
公开(公告)号：EP2177503A1
公开(公告)日：2010-04-21
申请号：EP09012361.3
申请日：2005-02-21
申请人： UCL Business PLC
发明人： Okuyama, Masahiro , Baker, David , Pryce, Gareth , Selwood, David , Visintin, Cristina
IPC分类号： C07C233/68 , C07C233/77 , C07C63/04 , C07C69/78 , A61K31/167 , A61K31/192 , A61K31/216 , A61K31/235
CPC分类号： C07C235/42 , A61K31/165 , C07C69/76 , C07C69/78 , C07C233/11 , C07C233/65 , C07C233/66 , C07C233/69 , C07C235/34 , C07C235/78 , C07C235/84 , C07C237/32 , C07C237/38 , C07C237/42 , C07C255/41 , C07C255/44
摘要： The present invention relates to a compound of formula I, or a pharmaceutically acceptable salt thereof,

wherein Z is OR 1 or NR 1 R 2 wherein each of R 1 and R 2 is independently H, or a hydrocarbyl group;X is an alkylene, alkenylene, or alkynylene group, each of which may be optionally substituted by one or more substituents selected from alkyl, COOH, CO 2 -alkyl, alkenyl, CN, NH 2 , hydroxy, halo, alkoxy, CF 3 and nitro;
Y is a polar functional group selected from OH, NO 2 CN, COR 3 , COOR 3 , NR 3 R 4 , CONR 3 R 4 , SO 3 H, SO 2 -R 3 , SO 2 NR 3 R 4 and CF 3 , where each of R 3 and R 4 is independently H or a hydrocarbyl group;
A is an aryl or heteroaryl group, each of which may be optionally substituted; and
B is (CH 2 ) n where n is 0, 1, 2, 3, 4 or 5;

with the proviso that:
(i) when A is phenyl, n is 0, and Z is OH, X-Y is other than meta -C≡C-(CH 2 ) 2 CO 2 H, meta -C≡C-(CH 2 ) 2 OH, meta -C≡C-(CH 2 ) 2 CO 2 Me, meta- (CH 2 ) 4 CO 2 H, ortho -CH 2 CO 2 H, ortho -(CH 2 ) 2 CO 2 H and ortho -(CH 2 ) 4 CO 2 H; and
(ii) when A is phenyl, n is 0, and Z is OMe, X-Y is other than meta -C≡C-(CH 2 ) 4 OH.
Further aspects of the invention relate to the use of such compounds in the preparation of a medicament for the treatment of a muscular disorder, a gastrointestinal disorder, or for controlling spasticity or tremors.
摘要翻译：本发明涉及式I化合物或其药学上可接受的盐，其中Z为OR1或NR1R2，其中R1和R2各自独立地为H或烃基; X为亚烷基，亚烯基或亚炔基，其各自可任选被一个或多个选自烷基，COOH，CO 2 - 烷基，烯基，CN，NH 2，羟基，卤素，烷氧基，CF 3和硝基的取代基取代; Y是选自OH，NO 2 CN，COR 3，COOR 3，NR 3 R 4，CONR 3 R 4，SO 3 H，SO 2 -R 3，SO 2 NR 3 R 4和CF 3的极性官能团，其中R 3和R 4各自独立地为H或烃基; A是芳基或杂芳基，它们中的每一个可以任选被取代; 并且B是（CH 2）n，其中n是0,1,2,3,4或5; 条件是：（i）当A为苯基，n为0且Z为OH时，XY不是间位C≡C-（CH 2）2 CO 2 H，间位C≡C-（CH 2）2 OH， C≡C-（CH2）2CO2Me，间 - （CH2）4CO2H，邻CH2CO2H，邻 - （CH2）2CO2H和邻 - （CH2）4CO2H; 和（ii）当A是苯基时，n是0，并且Z是OMe，X-Y不同于间位C≡C-（CH 2）4 OH。本发明的其他方面涉及这些化合物在制备用于治疗肌肉疾病，胃肠疾病或用于控制痉挛状态或震颤的药物中的用途。

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