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21. 发明公开

EP2531491A1 PYRIDAZINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS FUNGICIDES 审中-公开
标题翻译：哒嗪衍生物，它们的制备方法以及它们作为杀真菌剂的用途
公开(公告)号：EP2531491A1
公开(公告)日：2012-12-12
申请号：EP11701669.1
申请日：2011-02-01
申请人： Syngenta Participations AG
发明人： TRAH, Stephan , LAMBERTH, Clemens
IPC分类号： C07D237/12 , C07D237/14 , C07D307/58 , C07D307/60 , C07C69/612 , C07C69/734 , A01N43/58
CPC分类号： C07D237/12 , A01N43/58 , C07D237/14 , C07D307/58 , C07D307/60
摘要： The present invention relates to novel pyridazine derivatives of formula (I) wherein R
1 is methyl or ethyl; R
2 is H or chloro; R
3 is fluoro or chloro; R
4 is fluoro or methoxy; and R
5 is chloro or methoxy or an agrochemically usable salt from thereof, as active ingredients which have microbiodidal activity, in particular fungicidal activity.

22. 发明公开

EP2406231A1 IMIDAZOLE DERIVATIVES 审中-公开
标题翻译： IMIDAZOLDERIVATE
公开(公告)号：EP2406231A1
公开(公告)日：2012-01-18
申请号：EP10702325.1
申请日：2010-02-08
申请人： Syngenta Participations AG
发明人： DUMEUNIER, Raphael , LAMBERTH, Clemens , TRAH, Stephan
IPC分类号： C07D233/88 , A01N43/50
CPC分类号： C07D233/88
摘要： The present invention relates to novel imidazole derivatives of formula (I) having microbiocidal, in particular fungicidal, activity, to processes for their preparation and intermediates used in their preparation, to agrochemical compositions comprising them and to the use in agriculture or horticulture for controlling or preventing infestation of plants, harvested food crops, seeds or non-living materials by phytopathogenic microorganisms, preferably fungi.

23. 发明公开

EP2201000A1 NOVEL IMIDAZOLE DERIVATIVES 有权
标题翻译：新型咪唑衍生物
公开(公告)号：EP2201000A1
公开(公告)日：2010-06-30
申请号：EP08841505.4
申请日：2008-10-24
申请人： Syngenta Participations AG
发明人： DUMEUNIER, Raphael , LAMBERTH, Clemens , TRAH, Stephan , WENDEBORN, Sebastian
IPC分类号： C07D401/04 , C07D401/14 , C07D409/04 , C07D409/14 , A01N43/50 , A61P35/00 , A61K31/4439
CPC分类号： C07D233/54 , C07D233/61 , C07D233/68 , C07D401/04 , C07D409/04 , C07D409/14
摘要： The present invention relates to novel imidazole derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is halogen, C1-C4alkyl or C1-C4haloalkyl; R2 is an optionally substituted aryl or heteroaryl; R3 is halogen; R4 is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy or cyano; R5 is halogen; X is N or C(R); and R is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy or cyano; or an agrochemically usable salt form thereof; provided that when X is C(R), R2 cannot be an optionally substituted aryl.
摘要翻译：本发明涉及式（I）的新型咪唑衍生物作为活性成分，其具有杀微生物活性，特别是杀真菌活性：其中R 1为卤素，C 1 -C 4烷基或C 1 -C 4卤代烷基; R2是任选取代的芳基或杂芳基; R3是卤素; R4为氢，卤素，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或氰基; R5是卤素; X是N或C（R）; 和R为氢，卤素，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷氧基或氰基; 或其农业化学可用的盐形式; 条件是当X是C（R）时，R2不能是任选取代的芳基。

24. 发明公开

EP2046124A2 FUNGICIDAL COMPOUNDS AND COMPOSITIONS 审中-公开
标题翻译：杀真菌化合物和组合物
公开(公告)号：EP2046124A2
公开(公告)日：2009-04-15
申请号：EP07786424.7
申请日：2007-07-30
申请人： Syngenta Participations AG
发明人： GODWIN, Jeremy, R. , TRAH, Stephan , LAMBERTH, Clemens , WENDEBORN, Sebastian, Volker
IPC分类号： A01N43/58 , C07D237/12
CPC分类号： C07D237/12 , A01N43/58
摘要： The present invention relates, inter alia, to a compound having the formula (I):-wherein (R)n is selected from the group consisting of 4-Br, 4-OCH2CH3, 4-OCH2CF3, 2-CH3-4-C1, 2-CH3-4-OCH3, 2-CH3-4-OCF3, 2-F-4-Br, 2-F-4-CF3, 3-CH3-4-Br, 3-F-4-C1, 3-F-4-CH3, 3-F-4-Br, 3-F-4-OCH3 and 3-F-4-F. The present invention further relates to a fungicidal composition comprising a compound having the formula (I) - and also to fungicidal compositions comprising compounds having the formula (II) and/or (III):Furthermore, the present invention relates to methods for controlling pathogenic organisms using the compositions.

25. 发明公开

EP2041113A1 NOVEL PYRIDAZINE DERIVATIVES 审中-公开
标题翻译：新的哒嗪衍生物
公开(公告)号：EP2041113A1
公开(公告)日：2009-04-01
申请号：EP07801428.9
申请日：2007-07-16
申请人： Syngenta Participations AG
发明人： TRAH, Stephan , LAMBERTH, Clemens , WENDEBORN, Sebastian Volker
IPC分类号： C07D401/04 , C07D403/04 , C07D405/04 , C07D407/04 , C07D409/04 , C07D413/04 , C07D417/04 , A01N43/58
CPC分类号： C07D401/04 , A01N43/58 , A01N43/60 , A01N43/78 , A01N43/80 , A01N43/82 , C07D403/04 , C07D405/04 , C07D407/04 , C07D409/04 , C07D413/04 , C07D417/04
摘要： The present invention relates to novel pyridazine derivatives of formula I as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is hydrogen, C1-C6alkyl, C1-C6haloalkyl or C3-C6cycloalkyl; R2 is an optionally substituted heteroaryl; R3 is an optionally substituted aryl; and R4 is hydrogen, halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy, (VCehaloalkoxy, hydroxy or cyano; or an agrochemically usable salt form thereof.
摘要翻译：本发明涉及作为活性成分的式I的新型哒嗪衍生物，其具有杀微生物活性，特别是杀真菌活性：其中R 1为氢，C 1 -C 6烷基，C 1 -C 6卤代烷基或C 3 -C 6环烷基; R2是任选取代的杂芳基; R3是任选取代的芳基; 并且R 4是氢，卤素，C 1 -C 6烷基，C 1 -C 6卤代烷基，C 1 -C 6烷氧基，（C 1-6卤代烷氧基，羟基或氰基;或其农业化学上可用的盐形式。

26. 发明授权

EP1575922B1 BIPHENYL DERIVATIVES AND THEIR USE AS FUNGICIDES 有权
标题翻译： BENHENYLDERIVATE UND DEREN VERWENDUNG ALS FUNGIZIDE
公开(公告)号：EP1575922B1
公开(公告)日：2008-05-14
申请号：EP03813891.3
申请日：2003-12-15
申请人： Syngenta Participations AG
发明人： EHRENFREUND, Josef , LAMBERTH, Clemens , TOBLER, Hans , WALTER, Harald
IPC分类号： C07D231/14 , C07D231/16 , C07D207/34 , C07D277/56 , C07D263/34 , C07D333/38 , C07D307/68 , C07D309/28 , C07D327/06 , C07D213/82 , C07D239/28 , C07D239/30 , C07D237/24 , C07C233/03 , C07C211/45
CPC分类号： C07D213/82 , A01N43/06 , A01N43/14 , A01N43/32 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/74 , A01N43/80 , C07C25/24 , C07C211/45 , C07C211/52 , C07C217/76 , C07C219/32 , C07C233/03 , C07C2601/02 , C07C2601/08 , C07D207/34 , C07D231/14 , C07D231/16 , C07D237/24 , C07D239/28 , C07D239/30 , C07D263/34 , C07D277/56 , C07D307/68 , C07D309/28 , C07D327/06 , C07D333/38 , C07F7/0812
摘要： A fungicidally active compound of formula (I): where Het is a substituted 5- or 6-membered heterocyclic ring; R1 is hydrogen, formyl, CO-C1-4 alkyl, COO-C1-4 alkyl, C1-4 alkoxy(C1-4)alkylene, CO-C1-4 alkylenoxy(C1-4)alkyl, propargyl or allenyl; R2, R3, R4 and R5 are each, independently, hydrogen, halogen, methyl or CF3; each R6 is, independently, halogen, methyl or CF3; R7 is (Z)mC=C(Y1), (Z)mC(Y1)=C(Y2)(Y3) or tri(C1-4)alkylsilyl; X is O or S; Y1, Y2 and Y3 are each, independently, hydrogen, halogen, C1-6 alkyl [optionally substituted by one or more substituents each independently selected from halogen, hydroxy, C1-4 alkoxy, C1-4 haloalkoxy, C1-4 alkylthio, C1-4 haloalkylthio, C1-4 alkylamino, di(C1-4)alkylamino, C1-4 alkoxycarbonyl, C1-4 alkylcarbonyloxy and tri(C1-4)alkylsilyl], C2-4 alkenyl [optionally substituted by one or more substituents each independently selected from halogen], C2-4 alkynyl [optionally substituted by one or more substituents each independently selected from halogen], C3-7 cycloalkyl [optionally substituted by one or more substituents each independently selected from halogen, C1-4 alkyl and C1-4 haloalkyl] or tri(C14)alkylsilyl; Z is C1-4 alkylene [optionally substituted by one or more substituents each independently selected from hydroxy, cyano, C1-4 alkoxy, halogen, C1-4 haloalkyl, C1-4 haloalkoxy, C1-4 alkylthio, COOH and COO-C1-4 alkyl]; m is 0 or 1; and n is 0, 1 or 2; the invention also relates to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.
摘要翻译：杀真菌活性的式（1）化合物：其中Het是取代的5或6元杂环; R 1是氢，甲酰基，CO-C 1-4烷基，COO-C 1-4烷基，C 1〜 4个C 1-4烷氧基（C 1-4-4）亚烷基，CO-C 1-4亚烷基氧基（C 1-4-4烷基）烷基，炔丙基或二烯丙基; R 2，R 3，R 4和R 5各自独立地为氢，卤素，甲基或 CF _{3 ; 每个R 6独立地是卤素，甲基或CF 3; （Z）C（Y 1），（Z）m C（Y [任选被一个或多个各自独立地选自卤素的取代基取代的]烯基，任选被一个或多个各自独立地选自卤素的取代基取代的C 2-4 - 炔基，C 1-3 - 7个环烷基[任意被一个或多个取代基取代，各自独立地选自卤素，C 1-4烷基和C 1-4卤代烷基]或三（C _{1-4 ）烷基甲硅烷基; Z是任选被一个或多个各自独立地选自羟基，氰基，C 1-4烷氧基，卤素，C 1 -C 4烷基的取代基取代的C 1-4亚烷基 -4个卤代烷基，C 1-4卤代烷氧基，C 1-4烷基硫基，COOH和COO-C 1-4烷基 ]。 m为0或1; 并且n为0,1或2; 本发明还涉及用于制备这些化合物的新型中间体，包含至少一种新化合物作为活性成分的农用化学组合物以及农业或园艺中的活性成分或组合物用于控制或预防植物通过植物病原微生物，优选真菌。}}

27. 发明授权

EP1135369B1 ALPHA-SULFIN- AND ALPHA-SULFONAMINO ACID AMIDES 有权
标题翻译： α-Sulfin-和αSulFonAMino酸酰胺
公开(公告)号：EP1135369B1
公开(公告)日：2004-02-25
申请号：EP99968337.8
申请日：1999-12-01
申请人： Syngenta Participations AG
发明人： ZELLER, Martin , JEANGUENAT, André , LAMBERTH, Clemens
IPC分类号： C07C311/06 , C07C311/07 , C07C311/11 , C07C307/06 , A01N41/06
CPC分类号： A01N41/06 , C07C307/06 , C07C311/06 , C07C311/07 , C07C311/11
摘要： The invention relates to alpha -sulfin- and alpha -sulfonamimo acid amides of general formula(I) including the optical isomers thereof and mixtures of such isomers, wherein n is a number zero or one; R1 is C1-C12alkyl, C1-C12alkyl substituted with C1-C4alkoxy, C1-C4alkylthio, C1-C4alkylsulfonyl, C3-C8cycloalkyl, cyano, C1-C6alkoxycarbonyl, C3-C6alkenyloxycarbonyl or C3-C6alkynyloxycarbonyl; C3-C8cycloalkyl; C2-C12alkenyl; C2-C12alkynyl; C1-C12haloalkyl; or a group NR12R13 wherein R12 and R13 are each independently of the other hydrogen or C1-C6-alkyl, or together are tetra- or penta-methylene; R2 and R3 are each independently hydrogen; C1-C8alkyl; C1-C8alkyl substituted with hydroxy, mercapto, C1-C4alkoxy or C1-C4alkylthio; C3-C8alkenyl; C3-C8alkynyl; C3-C8cycloalkyl; C3-C8cycloalkyl-C1-C4alkyl; or the two groups R2 and R3 together with the carbon atom to which they are bonded form a three- to eight-membered hydrocarbon ring; R4, R5, R6 and R7 are each independently hydrogen or C1-C4alkyl; R8 is C1-C6alkyl, C3-C6alkenyl or C3-C6alkynyl; R9, R10, R14, R15, R16 and R17 are each independently hydrogen or C1-C4alkyl; A is optionally substituted phenyl, and to the preparation of those substances and to agrochemical compositions comprising at least one of those compounds as active ingredient. The invention relates also to the preparation of the said compositions and to the use of the compounds or of the compositions in controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.
摘要翻译：本发明涉及通式（I）的α-亚磺酰 - 和α-亚磺酰氨基酰胺，包括其光学异构体和这些异构体的混合物，其中n是数字0或1; R1为C1-C12烷基，C1-C4烷氧基，C1-C4烷硫基，C1-C4烷基磺酰基，C3-C8环烷基，氰基，C1-C6烷氧基羰基，C3- C3-C8环烷基; C2--C 12烯; C2-C12alkynyl; C1-C12haloalkyl; 或基团NR 12 R 13，其中R 12和R 13各自独立地为氢或C 1 -C 6烷基，或一起为四 - 或五 - 亚甲基; R2和R3各自独立地为氢; C1-C8烷基; 被羟基，巯基，C1-C4烷氧基或C1-C4烷硫基取代的C1-C8烷基; C3-C8烯基; C3-C8炔; C3-C8环烷基; C3-C8环烷基-C1-C4烷基; 或者两个基团R2和R3与它们所键合的碳原子一起形成三至八元烃环; R 4，R 5，R 6和R 7各自独立地为氢或C 1 -C 4烷基; R 8是C 1 -C 6烷基，C 3 -C 6烯基或C 3 -C 6炔基; R9，R10，R14，R15，R16和R17各自独立地为氢或C1-C4烷基; A是任选取代的苯基，并涉及这些物质的制备以及包含至少一种这些化合物作为活性成分的农业化学组合物。本发明还涉及所述组合物的制备以及化合物或组合物在控制或预防植物病原微生物特别是真菌侵染植物中的用途。

28. 发明公开

EP1272461A1 ALPHA-SULFIN- AND ALPHA-SULFONAMINO ACID AMIDE DERIVATIVES 审中-公开
标题翻译： α-Sulfin-和α-磺酰氨基酸衍生物
公开(公告)号：EP1272461A1
公开(公告)日：2003-01-08
申请号：EP01938109.4
申请日：2001-04-11
申请人： Syngenta Participations AG
发明人： ZELLER, Martin , LAMBERTH, Clemens , SZCZEPANSKI, Henry , DE MESMAEKER, Alain
IPC分类号： C07C307/06 , C07C311/06 , C07C313/06
CPC分类号： C07C307/06 , A01N41/06 , C07C311/06 , C07C313/06 , C07C2601/02
摘要： The invention relates to novel pesticidally active α-sulfin and α-sulfonamino acid amides of the general formula (I) including the optical isomers thereof and mixtures of such isomers, wherein n is a number zero or one; R1, R2, R3, R4, R5, R6 and R7 have the meanings given in the specification, and R8 is either hydrogen, (a), (b), (c), (d) or (e) wherein R11, R12, R13, R15 and R17 are each independently hydrogen or C1-C4 alkyl, R13 is C4-C12 alkyl, C1-C12 halogenalkyl; C3-C8 cycloalkyl; optionally substituted aryl or optionally substituted heteroaryl, R16 is optionally substituted aryl or optionally substituted heteroaryl; and Z is oxygen, sulfur -CR18R19- or -NR20-, wherein R18, R19 and R20 independently of each other are hydrogen or C1-C4 alkyl. The novel compounds possess plant-protecting properties and are suitable for protecting plants against infestation by phytopathogenic microorganisms.
摘要翻译：本发明涉及通式（I）的新型农药活性α-亚磺酰和α-磺酰氨基酸酰胺，包括其光学异构体和这些异构体的混合物，其中n是数字0或1; （a），（b），（c），（d）或（e）其中R 11，R 12和R 7具有本说明书中给出的含义， R 13，R 15和R 17各自独立地为氢或C 1 -C 4烷基，R 13为C 4 -C 12烷基，C 1 -C 12卤代烷基; C3-C8环烷基; 任选取代的芳基或任选取代的杂芳基，R 16为任选取代的芳基或任选取代的杂芳基; 和Z是氧，硫-CR 18 R 19 - 或-NR 20 - ，其中R 18，R 19和R 20彼此独立地是氢或C 1 -C 4烷基。这些新化合物具有植物保护特性，并且适用于保护植物免受植物病原微生物侵染。

29. 发明公开

EP1272460A1 NOVEL ALPHA-SULFIN- AND ALPHA-SULFONAMINO ACID AMIDE DERIVATIVES 审中-公开
标题翻译：新的Alpha和α-亚SULFONAMIDOSÄUREAMID衍生物
公开(公告)号：EP1272460A1
公开(公告)日：2003-01-08
申请号：EP01919450.5
申请日：2001-04-11
申请人： Syngenta Participations AG
发明人： ZELLER, Martin , LAMBERTH, Clemens , SZCZEPANSKI, Henry , DE MESMAEKER, Alain
IPC分类号： C07C307/06 , C07C311/06 , C07C313/06
CPC分类号： A01N41/06 , C07C307/06 , C07C311/06 , C07C313/06
摘要： The invention relates to novel pesticidally active α-sulfin- and α-sulfonamino acid amides of the general formula (I) including the optical isomers thereof and mixtures of such isomers, wherein n is a number zero or one, R1 - R7 have the meanings given in the specification. R8 is either hydrogen, (a), (b), (c), (d) or (e) wherein R11, R12, R14, R15 and R17 are each independently hydrogen or C1-C4alkyl, R13 is C4-C12alkyl; C1-C12 halogenalkyl; C3-C8 cycloalkyl; optionally substituted aryl or optionally substituted heteroaryl, R16 is optionally substituted aryl or optionally substituted heteroaryl; and Z is oxygen, sulfur -CR18R19- or -NR20-, wherein R18, R19, R20 independently of each other are hydrogen or C1-C4alkyl. The novel compounds possess plant-protecting properties and are suitable for protecting plants against infestation by phytopathogenic microorganisms.

30. 发明公开

EP1135369A2 ALPHA-SULFIN- AND ALPHA-SULFONAMINO ACID AMIDES 有权
标题翻译： α-Sulfin-和αSulFonAMino酸酰胺
公开(公告)号：EP1135369A2
公开(公告)日：2001-09-26
申请号：EP99968337.8
申请日：1999-12-01
申请人： Syngenta Participations AG
发明人： ZELLER, Martin , JEANGUENAT, André , LAMBERTH, Clemens
IPC分类号： C07C311/06 , C07C311/07 , C07C311/11 , C07C307/06 , A01N41/06
CPC分类号： A01N41/06 , C07C307/06 , C07C311/06 , C07C311/07 , C07C311/11
摘要： The invention relates to α-sulfin- and α-sulfonamimo acid amides of general formula(I) including the optical isomers thereof and mixtures of such isomers, wherein n is a number zero or one; R1 is C1-C12alkyl, C1-C12alkyl substituted with C1-C4alkoxy, C1-C4alkylthio, C1-C4alkylsulfonyl, C3-C8cycloalkyl, cyano, C1-C6alkoxycarbonyl, C3-C6alkenyloxycarbonyl or C3-C6alkynyloxycarbonyl; C3-C8cycloalkyl; C2-C12alkenyl; C2-C12alkynyl; C1-C12haloalkyl; or a group NR12R13 wherein R12 and R13 are each independently of the other hydrogen or C1-C6-alkyl, or together are tetra- or penta-methylene; R2 and R3 are each independently hydrogen; C1-C8alkyl; C1-C8alkyl substituted with hydroxy, mercapto, C1-C4alkoxy or C1-C4alkylthio; C3-C8alkenyl; C3-C8alkynyl; C3-C8cycloalkyl; C3-C8cycloalkyl-C1-C4alkyl; or the two groups R2 and R3 together with the carbon atom to which they are bonded form a three- to eight-membered hydrocarbon ring; R4, R5, R6 and R7 are each independently hydrogen or C1-C4alkyl; R8 is C1-C6alkyl, C3-C6alkenyl or C3-C6alkynyl; R9, R10, R14, R15, R16 and R17 are each independently hydrogen or C1-C4alkyl; A is optionally substituted phenyl, and to the preparation of those substances and to agrochemical compositions comprising at least one of those compounds as active ingredient. The invention relates also to the preparation of the said compositions and to the use of the compounds or of the compositions in controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.
摘要翻译：本发明涉及通式（I）的α-亚磺酰 - 和α-亚磺酰氨基酰胺，包括其光学异构体和这样的异构体的混合物，其中n是数字0或1; R1为C1-C12烷基，C1-C4烷氧基，C1-C4烷硫基，C1-C4烷基磺酰基，C3-C8环烷基，氰基，C1-C6烷氧基羰基，C3- C3-C8环烷基; C2--C 12烯; C2-C12alkynyl; C1-C12haloalkyl; 或基团NR 12 R 13，其中R 12和R 13各自独立地为氢或C 1 -C 6烷基，或一起为四 - 或五 - 亚甲基; R2和R3各自独立地为氢; C1-C8烷基; 被羟基，巯基，C1-C4烷氧基或C1-C4烷硫基取代的C1-C8烷基; C3-C8烯基; C3-C8炔; C3-C8环烷基; C3-C8环烷基-C1-C4烷基; 或者两个基团R2和R3与它们所键合的碳原子一起形成三至八元烃环; R 4，R 5，R 6和R 7各自独立地为氢或C 1 -C 4烷基; R 8是C 1 -C 6烷基，C 3 -C 6烯基或C 3 -C 6炔基; R9，R10，R14，R15，R16和R17各自独立地为氢或C1-C4烷基; A是任选取代的苯基，并涉及这些物质的制备以及包含至少一种这些化合物作为活性成分的农业化学组合物。本发明还涉及所述组合物的制备以及化合物或组合物在控制或预防植物病原微生物特别是真菌侵染植物中的用途。

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