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1. 发明专利

JP2020117528A ジフェニルメタン誘導体の製造方法审中-公开
公开(公告)号：JP2020117528A
公开(公告)日：2020-08-06
申请号：JP2020068458
申请日：2020-04-06
申请人： DAE WOONG PHARMA , GREEN CROSS CORP
发明人： YOON HEE-KYOON , PARK SE-HWAN , YOON JI-SUNG , CHOI SOONGYU , SEO HEE JEONG , PARK EUN-JUNG , KONG YOUNGGYU , SONG KWANG-SEOP , KIM MIN JU , PARK SO OK
IPC分类号： C07D407/04
摘要：【課題】ナトリウム依存性グルコース共輸送体(SGLT)阻害剤として有効なジフェニルメタン誘導体の結晶形の提供。【解決手段】下記式で示される化合物の結晶形。上記結晶形が、Cu-Kα光源を用いて照射した場合に、6.2°±0.2°、7.2°±0.2°、8.8°±0.2°、17.6°±0.2°、19.0°±0.2°、22.5°±0.2°、および25.1°±0.2°の回折角(2θ)におけるピークを含むX線回折(XRD)スペクトルを有し、優れた物理化学的特性から、医薬品製造などの分野で有効に利用することができる。【選択図】なし

2. 发明公开

EP3244895A4 NOVEL PHARMACEUTICAL COMPOSITION 有权
公开(公告)号：EP3244895A4
公开(公告)日：2018-07-25
申请号：EP16737566
申请日：2016-01-14
申请人： DAE WOONG PHARMA , BIO SYNECTICS INC
发明人： KIM SANGHEE , CHANG HEE CHUL , JUNG JI HOON
IPC分类号： A61K9/48 , A61K31/5377 , A61P1/08 , A61P25/00
CPC分类号： A61K9/4858 , A61K9/10 , A61K9/1617 , A61K9/4808 , A61K9/4866 , A61K31/5377
摘要： Disclosed herein a pharmaceutical composition comprising aprepitant a pharmaceutically acceptable salt thereof; at least one hydrocarbon derivative selected from among a fatty acid of 14 to 18 carbon atoms, and a fatty alcohol of 14 to 18 carbon atoms; and at least one selected from among polyoxyethyelene-type nonionic surfactant, sucrose fatty acid ester, and Macrogol 15 hydroxystearate. The pharmaceutical composition of the present disclosure can release aprepitant or a pharmaceutically acceptable salt thereof to effectively exert the pharmaceutical efficacy, and can be dissolved in a fasted state simulated gastrointestinal fluid so that it can be useful for study on the in vivo pharmacokinetic behavior of aprepitant.

3. 发明公开

EP3082776A4 FILM COATED TABLET CONTAINING CHOLINE ALFOSCERATE AND PROCESS FOR PREPARING THE SAME 有权
标题翻译： FILMTABLETTE MIT CHOLIN-ALFOSCERAT UND VERFAHREN ZUR HERSTELLUNG DAVON
公开(公告)号：EP3082776A4
公开(公告)日：2017-07-26
申请号：EP14871661
申请日：2014-12-15
申请人： DAE WOONG PHARMA
发明人： PARK SANG-HAN , CHANG HEE-CHUL
IPC分类号： A61K9/28 , A61K9/20
CPC分类号： A61K9/2866 , A61K9/124 , A61K9/2095 , A61K9/282 , A61K9/284 , A61K31/661 , A61K33/12
摘要： The present invention provides a film coated tablet comprising a first film coating layer comprising hydroxypropyl methylcellulose and a second film coating layer comprising polyvinyl alcohol, on a tablet containing choline alfoscerate as an active ingredient and magnesium aluminometasilicate as an additive; and a process for preparing the same.
摘要翻译：本发明提供了一种薄膜包衣片剂，其包含含有羟丙基甲基纤维素的第一薄膜包衣层和包含聚乙烯醇的第二薄膜包衣层，所述片剂含有作为活性成分的甘磷酸胆碱和作为添加剂的硅酸铝镁; 及其制备方法。

4. 发明公开

EP3060549A4 NOVEL ANTIFUNGAL OXODIHYDROPYRIDINECARBOHYDRAZIDE DERIVATIVE 有权
标题翻译：杀菌剂杀真菌剂
公开(公告)号：EP3060549A4
公开(公告)日：2017-06-21
申请号：EP14856658
申请日：2014-10-21
申请人： DAE WOONG PHARMA
发明人： PARK JOON SEOK , YOON YOUN JUNG , PARK CHANG MIN , NA YUN SOO , CHO MIN JAE , LEE HO BIN , HAN MI RYEONG , PARK YEON JUNG , KIM JI DUCK
IPC分类号： C07D213/63 , A61K31/4412 , A61P31/04 , C07D213/82 , C07D401/04 , C07D401/06 , C07D401/12 , C07D417/06 , C07D471/04 , C07D487/08 , C07D498/08
CPC分类号： C07D213/82 , C07D213/63 , C07D401/04 , C07D401/06 , C07D401/12 , C07D417/06 , C07D471/04 , C07D487/04 , C07D498/08
摘要： The present invention relates to novel oxodihydropyridinecarbohydrazide derivatives with excellent antifungal activities, an antifungal composition containing the same, and its use for the prevention and treatment of fungal infectious diseases. The oxodihydropyridinecarbohydrazide derivatives of the present invention have excellent antifungal and fungicidal activities, and thus will be useful for the prevention and treatment of various fungal infections by Candida spp., Aspergillus spp., Cryptococcus neoformans and Trichophyton spp., etc. Additionally, the oxodihydropyridinecarbohydrazide derivatives of the present invention, unlike other fungicidal preparations, can be orally administered.
摘要翻译：本发明涉及具有优异抗真菌活性的新型氧代二氢吡啶碳酰肼衍生物，含有其的抗真菌组合物，及其用于预防和治疗真菌感染性疾病的用途。本发明的氧代二氢吡啶碳酰肼衍生物具有优异的抗真菌和杀真菌活性，因此可用于预防和治疗假丝酵母属，曲霉属，新隐球菌属和毛癣菌属等各种真菌感染。此外，氧代二氢吡啶碳酰肼不像其他杀真菌制剂，本发明的衍生物可以口服给药。

5. 发明公开

EP2627652A4 NOVEL PYRIDYL BENZOXAZINE DERIVATIVES, PHARMACEUTICAL COMPOSITION COMPRISING THE SAME, AND USE THEREOF 有权
标题翻译：新PYRIDYLBENZOXAZINDERIVATE，药物组合物适当地使用该
公开(公告)号：EP2627652A4
公开(公告)日：2014-10-01
申请号：EP11832767
申请日：2011-10-13
申请人： DAE WOONG PHARMA
发明人： KIM JI DUCK , YOON HONG CHUL , KIM IN WOO , CHO MIN JAE , LEE IN YOUNG , LEE SANG HO , PARK EUN KYUNG , LIM KWON JO , NAM SANG HYUN
IPC分类号： C07D413/14 , A61K31/538 , A61P25/04
CPC分类号： C07D413/14

6. 发明公开

EP2411392A4 NOVEL CRYSTAL FORMS OF ADEFOVIR DIPIVOXIL AND PROCESSES FOR PREPARING THE SAME 有权
标题翻译：新的ADEFOVIRIPIVOXIL晶体形式及其生产方法
公开(公告)号：EP2411392A4
公开(公告)日：2012-10-10
申请号：EP10756377
申请日：2010-03-26
申请人： DAE WOONG PHARMA , DAEWOONG BIO INC
发明人： CHOI SOO JIN , LEE BYUNG GOO , OH SEONG SOO , KIM YONG TAE , KIM KWANG JOO , KIM HYE JIN
IPC分类号： C07D473/34 , C07F9/28
CPC分类号： C07D473/34 , C07F9/65616

7. 发明公开

EP1986664A4 COMPOSITION FOR TREATING CANCER COMPRISING OLIGONUCLEOTIDE AND NON-TOXIC LPS 审中-公开
标题翻译：组合物技术癌的寡核苷酸和无毒的LPS的治疗
公开(公告)号：EP1986664A4
公开(公告)日：2009-07-22
申请号：EP06715813
申请日：2006-02-01
申请人： EYEGENE INC , DAE WOONG PHARMA
发明人： AHN BO-YOUNG , CHO YANG-JE , YOO WON-IL , LEE NA-GYONG , KIM DOO-SIK
IPC分类号： A61K31/7088 , A61K31/739 , A61P35/00
CPC分类号： A61K31/7088 , A61K31/739 , A61K2300/00
摘要： Disclosed is a composition for treating cancer including oligodeoxynucleotides and LPS-derived non-toxic lipopolysaccharides as effective components.

8. 发明公开

EP1322315A4 FORMULATIONS FOR REDUCING OR ELIMINATING TOXICITY OF ENVIRONMENTAL HORMONES CONTAINING URSODEOXYCHOLIC ACID 有权
标题翻译：制剂用于减少或消除环境激素熊去氧胆酸的毒性
公开(公告)号：EP1322315A4
公开(公告)日：2004-05-26
申请号：EP01972783
申请日：2001-09-28
申请人： DAE WOONG PHARMA
发明人： YEON JAE-DUCK , BAIK KYONG-UP , JUNG KYU-HYUCK , PARK SEUNG-KOOK
IPC分类号： C07D319/24 , A61K31/575 , A61P3/00 , A61P3/10 , A61P15/08 , A61P35/00 , A61P37/04 , C07J9/00
CPC分类号： A61K31/575
摘要： The present invention relates to formulations for reducing or eliminating toxicity of environmental hormone containing as detoxifying agent ursodeoxycholic acid, or pharmaceutically acceptable salts or esters thereof.

9. 发明公开

EP3197867A4 NOVEL 4-METHOXY PYRROLE DERIVATIVES OR SALTS THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME 有权
标题翻译： NEUARTIGE 4-METHOXYRROLDERIVATE ODER SALZE DAVON UND PHARMAZEUTISCHE ZUSAMMENSETZUNG DAMIT
公开(公告)号：EP3197867A4
公开(公告)日：2017-09-06
申请号：EP16786741
申请日：2016-04-27
申请人： DAE WOONG PHARMA
发明人： LEE CHUN HO , LEE SEUNG CHUL , LEE YEON IM , EOM DEOK KI , HAN MI RYEONG , KOH EUN JI
IPC分类号： C07D207/48 , A61K31/095 , A61K31/40 , C07D207/30 , C07D207/335 , C07D207/36
CPC分类号： C07D207/48
摘要： The present invention provides a 4-methoxy pyrrole derivative or a pharmaceutically acceptable salt thereof, a preparation method thereof, and a pharmaceutical composition containing the same. The 4-methoxy pyrrole derivatives or pharmaceutically acceptable salts thereof according to the present invention have not only excellent proton pump inhibitory activity, gastric damage-inhibiting activity and defensive factor-enhancing effects, but also excellent eradication activity against H. pylori. Therefore, the 4-methoxy pyrrole derivatives or pharmaceutically acceptable salts thereof can be effectively used for the prevention and treatment of gastrointestinal damage due to gastrointestinal tract ulcer, gastritis, reflux esophagitis or H. pylori. Moreover, the 4-methoxy pyrrole derivatives or pharmaceutically acceptable salts thereof, have inhibitory activities against GPCR and thus can be effectively used for the prevention and treatment of 5-HT receptor-mediated or muscarinic acetylcholine receptor-mediated diseases.
摘要翻译：本发明提供4-甲氧基吡咯衍生物或其药学上可接受的盐，其制备方法和含有其的药物组合物。根据本发明的4-甲氧基吡咯衍生物或其药学上可接受的盐不仅具有优异的质子泵抑制活性，胃损伤抑制活性和防御因子增强作用，而且还具有优良的抗幽门螺杆菌根除活性。因此，4-甲氧基吡咯衍生物或其药学上可接受的盐可以有效地用于预防和治疗胃肠道溃疡，胃炎，反流性食管炎或幽门螺杆菌引起的胃肠道损伤。此外，4-甲氧基吡咯衍生物或其药学上可接受的盐具有对GPCR的抑制活性，因此可有效用于预防和治疗5-HT受体介导的或毒蕈碱乙酰胆碱受体介导的疾病。

10. 发明公开

EP3052484A4 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME 有权
标题翻译： SULFONYLINDOLDERIVATE和方法及其生产
公开(公告)号：EP3052484A4
公开(公告)日：2017-03-01
申请号：EP14850178
申请日：2014-10-02
申请人： DAE WOONG PHARMA
发明人： YU KYUNG A , YOON JI SUNG , EOM DEOK KI , LEE YEON IM , SHIN HYE RYUN , LEE JUN HEE , SEO HA NEE , KIM JI DUCK , LEE SANG HO , LEE CHUN HO
IPC分类号： A61K31/4439 , A61K31/4045 , A61K31/437 , A61K31/444 , A61P1/04 , C07D209/30 , C07D401/12 , C07D401/14 , C07D405/14 , C07D471/04
CPC分类号： C07D209/30 , C07D209/14 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/04 , C07D403/12 , C07D405/14 , C07D471/04
摘要： Disclosed are a sulfonylindole derivative useful for the prevention or treatment of peptic ulcer, gastritis or reflux esophagitis, a method of preparing the same, and a pharmaceutical composition containing the same.

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