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81. 发明申请

WO1994029291A1 ANILINE DERIVATIVES 审中-公开
标题翻译：苯胺衍生物
公开(公告)号：WO1994029291A1
公开(公告)日：1994-12-22
申请号：PCT/EP1994001808
申请日：1994-06-03
申请人： ZENECA LIMITED , ZENECA-PHARMA S.A. , EDWARDS, Philip, Neil
发明人： ZENECA LIMITED , ZENECA-PHARMA S.A.
IPC分类号： C07D309/10
CPC分类号： C07D405/12 , C07D309/10
摘要： The invention concerns an aniline derivative of formula (I) wherein R includes hydrogen and (1-4C)alkyl; R includes hydrogen and (1-4C)alkyl; R is hydrogen or (1-4C)alkyl; X includes a group of the formula CR R wherein R is hydrogen or (1-4C)alkyl and R is hydrogen or (1-4C)alkyl; A includes a direct link to X ; X includes thio and sulphonyl; Ar includes phenylene, which may be optionally substituted; R includes hydrogen and (1-4C)alkyl; and R and R together form a ring having 5 to 6 ring atoms including one oxygen atom, and which ring may bear one, two or three substituents, including methyl alpha to the oxygen atom; or a pharmaceutically acceptable salt thereof; processes for their preparation; pharmaceutical compositions containing them and their use as 5-lipoxygenase inhibitors.
摘要翻译：本发明涉及式（I）的苯胺衍生物，其中R 4包括氢和（1-4C）烷基; R 5包括氢和（1-4C）烷基; R 6是氢或（1-4C）烷基; X 3包括式CR 7 R 8的基团，其中R 7是氢或（1-4C）烷基，R 8是氢或（1-4C）烷基; A <1>包括与X <1>的直接链接; X 1包括硫代和磺酰基; Ar包括可以任选取代的亚苯基; R 1包括氢和（1-4C）烷基; 并且R 2和R 3一起形成具有5至6个环原子的环，包括一个氧原子，并且该环可以带有一个，两个或三个取代基，包括氧原子的甲基α; 或其药学上可接受的盐; 其准备过程; 含有它们的药物组合物及其作为5-脂肪氧合酶抑制剂的用途。

82. 发明申请

WO1994028166A1 FLUORESCENCE ENERGY TRANSFER SUBSTRATES 审中-公开
标题翻译：荧光能量转移基板
公开(公告)号：WO1994028166A1
公开(公告)日：1994-12-08
申请号：PCT/GB1994001153
申请日：1994-05-27
申请人： ZENECA LIMITED , GARMAN, Andrew, John
发明人： ZENECA LIMITED
IPC分类号： C12Q01/37
CPC分类号： G01N33/533 , C12Q1/37 , Y10S435/968
摘要： A method for the preparation of a fluorescence resonance energy transfer (FRET) substrate having donor and acceptor species on opposite sides of a proteolytic cleavage site and wherein the donor and/or acceptor species are attached via the side chain(s) of amino acid(s) therein. The method comprises contacting a reactive donor or acceptor species with a polypeptide substrate having the side chain(s) of amino acid(s) therein adapted for reaction with the reactive species and then contacting the substrate so obtained with a corresponding reactive donor or acceptor species. Novel FRET substrates so prepared and their use in assays to identify modulators of protease activity.
摘要翻译：一种用于制备在蛋白水解切割位点的相对侧具有供体和受体物质的荧光共振能量转移（FRET）底物的方法，其中供体和/或受体物质通过氨基酸的侧链（ s）。该方法包括使反应性供体或受体物质与其中具有适于与反应物质反应的氨基酸侧链的多肽底物接触，然后将如此获得的底物与相应的反应性供体或受体物质。新型FRET底物如此制备，并在测定中用于鉴定蛋白酶活性的调节剂。

83. 发明申请

WO1994028061A1 POLYESTER COMPOSITION 审中-公开
标题翻译：聚酯组合物
公开(公告)号：WO1994028061A1
公开(公告)日：1994-12-08
申请号：PCT/GB1994001184
申请日：1994-06-01
申请人： ZENECA LIMITED , HAMMOND, Timothy , LIGGAT, John, Jamieson , MONTADOR, James, Henry , WEBB, Andrew
发明人： ZENECA LIMITED
IPC分类号： C08K05/00
CPC分类号： C08K5/0016 , C08L67/02 , C08L67/04 , C08L2666/02
摘要： Polyester composition comprising a biodegradable polyester and a plasticising quantity of at least one plasticiser selected from the group: high-boiling esters of polybasic acids; phosphoric acid drivatives; phosphorous acid derivatives; phosphonic acid derivatives; substituted fatty acids; high-boiling glycols, polyglycols, polyoxyalkylenes and glycerol each optionally substituted and optionally terminally esterified; pentaerythritols and derivatives; sulphonic acid derivatives; epoxy derivatives; chlorinated paraffins; polymeric esters; Wolflex-But3; provided that citrates does not include doubly esterified hydroxycarboxylic acids having at least 3 ester groups in its molecule and further provided that glycerols do not include glycerol triacetate and glycerol diacetate.
摘要翻译：包含可生物降解的聚酯和增塑量的至少一种增塑剂的聚酯组合物，其选自多元酸的高沸点酯; 磷酸驱动剂; 亚磷酸衍生物; 膦酸衍生物; 取代脂肪酸; 高沸点二醇，聚二醇，聚氧化烯和甘油，各自任选被取代并任选地被酯化; 季戊四醇及其衍生物; 磺酸衍生物; 环氧衍生物; 氯化石蜡; 聚合酯; Wolflex-But3; 条件是柠檬酸盐不包括其分子中具有至少3个酯基的双酯化羟基羧酸，并且进一步提供甘油不包括甘油三乙酸酯和甘油二乙酸酯。

84. 发明申请

WO1994028048A1 PROCESSING OF POLYESTERS 审中-公开
标题翻译：聚酯加工
公开(公告)号：WO1994028048A1
公开(公告)日：1994-12-08
申请号：PCT/GB1994001182
申请日：1994-06-01
申请人： ZENECA LIMITED , LIGGAT, John, Jamieson , O'BRIEN, Gregory
发明人： ZENECA LIMITED
IPC分类号： C08G63/88
CPC分类号： B29C71/02 , B29K2067/00 , C08G63/88
摘要： A process for improving mechanical properties of an aged polyester composition comprising at least one polyhydroxyalkanoate (PHA) and at least one plasticiser thereof, which comprises heating at a temperature whereby (i) the polyester is restored to its original non-aged properties, and (ii) subsequent ageing of the polyester is retarded as indicated by substantial improvement of at least one measurement indicative of ageing compared to non heat treated polyester of the same age. The invention includes a polyester composition and shaped articles which have been subjected to the process and in which ageing is retarded.
摘要翻译：一种用于改善包含至少一种聚羟基链烷酸酯（PHA）和至少一种增塑剂的老化聚酯组合物的机械性能的方法，其包括在以下温度下进行加热，由此（i）所述聚酯恢复到其原始的非老化性能，和 ii）聚酯的随后老化被延迟，如相对于相同年龄的非热处理的聚酯相比，表明老化的至少一个测量值的显着改善所表明的。本发明包括经过该方法并延迟老化的聚酯组合物和成型制品。

85. 发明申请

WO1994027999A1 BICYCLIC ETHER DERIVATIVES AND THEIR USE AS 5-LIPOXYGENASE INHIBITORS 审中-公开
标题翻译：双相醚衍生物及其作为5-LIPOXYGENASE抑制剂的用途
公开(公告)号：WO1994027999A1
公开(公告)日：1994-12-08
申请号：PCT/EP1994001805
申请日：1994-06-03
申请人： ZENECA LIMITED , ZENECA-PHARMA S.A. , EDWARDS, Philip, Neil
发明人： ZENECA LIMITED , ZENECA-PHARMA S.A.
IPC分类号： C07D493/08
CPC分类号： C07D495/08
摘要： The invention concerns a bicyclic ether derivative of formula (I), wherein Ar is phenyl or naphthyl, or a 10-membered bicyclic heterocyclic moiety containing one or two nitrogen heteroatoms and optionally containing a further heteroatom selected from nitrogen, oxygen and sulphur; A is a direct link to the group X or A is (1-4C)alkylene; X is oxy, thio, sulphinyl or sulphonyl; Ar is phenylene, pyridinediyl, pyrimidinediyl, thiophendiyl, furandiyl or thiazolediyl; and R is (1-4C)alkyl, (3-4C)alkenyl or (3-4C)alkynyl; or a pharmaceutically-acceptable salt thereof; processes for their preparation; pharmaceutical compositions containing them and their use as 5-lipoxygenase inhibitors.
摘要翻译：本发明涉及式（I）的双环醚衍生物，其中Ar 1是苯基或萘基，或含有一个或两个氮杂原子并任选地含有另外选自氮，氧和硫的杂原子的10元双环杂环部分 ; A是直接连接到X基团或A是（1-4C）亚烷基; X是氧基，硫基，亚磺酰基或磺酰基; Ar 2是亚苯基，吡啶二基，嘧啶二基，噻吩二基，呋喃二基或噻唑二基; 并且R 1是（1-4C）烷基，（3-4C）烯基或（3-4C）炔基; 或其药学上可接受的盐; 其准备过程; 含有它们的药物组合物及其作为5-脂肪氧合酶抑制剂的用途。

86. 发明申请

WO1994023344A1 COMPOSITION AND USE 审中-公开
标题翻译：组成和使用
公开(公告)号：WO1994023344A1
公开(公告)日：1994-10-13
申请号：PCT/GB1994000654
申请日：1994-03-29
申请人： ZENECA LIMITED , CAMPBELL, James, Stanley , GREGORY, Peter
发明人： ZENECA LIMITED
IPC分类号： G03G09/097
CPC分类号： G03G9/09783
摘要： A toner resin composition comprising a toner resin and a negative charging charge control agent (CCA) which is a di- or trivalent metal salt of a naphthalene oxy-carboxylic acid wherein the hydroxy group and carboxylic acid group are attached to adjacent carbon atoms of an aromatic ring. The CCA is preferably the zinc, aluminium or iron salt of 3-hydroxy-2-naphthoic acid.
摘要翻译：一种调色剂树脂组合物，其包含调色剂树脂和作为萘氧基羧酸的二价或三价金属盐的负带电电荷控制剂（CCA），其中羟基和羧酸基团连接到相邻的碳原子上芳香环。 CCA优选为3-羟基-2-萘甲酸的锌，铝或铁盐。

87. 发明申请

WO1994021606A1 PENTAFLUOROSULPHANYLPHENYL AND PENTAFLUOROSULPHANYLPYRIDIL SUBSTITUTED HETEROAROMATIC COMPOUNDS WITH INSECTICIDAL OR ACARICIDAL ACTIVITY 审中-公开
标题翻译：卟啉二苯醚和P UL UL ANY IL IL IL IL ITY ITY ITY ITY ITY ITY ITY ITY ITY ITY ITY ITY ITY ITY ITY ITY ITY
公开(公告)号：WO1994021606A1
公开(公告)日：1994-09-29
申请号：PCT/GB1994000612
申请日：1994-03-24
申请人： ZENECA LIMITED , SALMON, Roger , PEARSON, David, Philip, John , PARRY, David, Rees , KOZAKIEWICZ, Anthony, Marian
发明人： ZENECA LIMITED
IPC分类号： C07D207/36
CPC分类号： C07D213/64 , A01N43/36 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/56 , A01N47/02 , C07C381/00 , C07D207/36 , C07D231/12 , C07D231/28 , C07D231/38 , C07D233/56 , C07D233/64 , C07D233/84 , C07D233/88 , C07D239/36 , C07D249/08
摘要： Compounds with insecticidal or acaricidal activity have formula (IA) or (IB), wherein Ra represents hydrogen or from 1 to 4 optional substituents and Rb represents from 1 to 3 optional substituents and wherein A represents an optionally substituted N-linked nitrogen-containing five or six membered aromatic heterocyclic ring, for example imidazole, pyrrole, pyrazole, pyrimidinone and pyridone.
摘要翻译：具有杀虫或杀螨活性的化合物具有式（IA）或（IB），其中R a表示氢或1至4个任选的取代基，R b表示1至3个任选的取代基，并且其中A表示任选取代的N-连接的含氮五或六元芳族杂环，例如咪唑，吡咯，吡唑，嘧啶酮和吡啶酮。

88. 发明申请

WO1994020479A1 N-(BETA-BRANCHED ALKYL)-1,2-BENZISOTHIAZOLIN-3-ONES, THEIR PREPARATION AND USE AS INDUSTRIAL BIOCIDES 审中-公开
标题翻译： N-（β-分支烷基）-1,2-BENZISOTHIAZOLIN-3-ONES，其制备和用作工业生物
公开(公告)号：WO1994020479A1
公开(公告)日：1994-09-15
申请号：PCT/GB1994000320
申请日：1994-02-17
申请人： ZENECA LIMITED , AUSTIN, Peter, William
发明人： ZENECA LIMITED
IPC分类号： C07D275/04
CPC分类号： C07D275/04 , A01N43/80 , Y10S528/935
摘要： The invention relates to N-( beta -branched alkyl)-1,2-benzisothiazolin-3-ones having two or more carbon atoms in the alkyl side chain such as N-(2-ethylhexyl)-1,2-benzisothiazolin-3-one. The compounds are suitable as paint film fungicides.
摘要翻译：本发明涉及在烷基侧链中具有两个或更多个碳原子的N-（β-支链烷基）-1,2-苯并异噻唑啉-3-酮，例如N-（2-乙基己基）-1,2-苯并异噻唑啉-3 -一。该化合物适合作为漆膜杀真菌剂。

89. 发明申请

WO1994020204A1 PRODUCTION OF PARTICULATE MATERIALS 审中-公开
标题翻译：颗粒材料的生产
公开(公告)号：WO1994020204A1
公开(公告)日：1994-09-15
申请号：PCT/GB1993002554
申请日：1993-12-15
申请人： ZENECA LIMITED , IMPERIAL CHEMICAL INDUSTRIES PLC , OLIVER, Raymond , FAIRCLOUGH, Anthony, Rupert, Nigel , ANTONINI, Alejandro, Martin , MUNRO, Robert, James , LIPSCOMBE, Lynn, Wilfred
发明人： ZENECA LIMITED , IMPERIAL CHEMICAL INDUSTRIES PLC
IPC分类号： B01J02/04
CPC分类号： B01D1/18 , B01J2/04 , B05B7/0861
摘要： A process for producing solid particles by drying a spray of liquid droplets. The droplets are formed by projecting a liquid formulation as a plurality of jets (J) (Figure 6) in such a way that each jet breaks up into droplets of narrow size distribution. Prior to the onset of coalescence the droplets are contacted with a gas flow (G) which is arranged to reduce coalescence by disrupting slip streaming of the droplets and/or accelerating the droplets.
摘要翻译：通过干燥液滴喷雾来生产固体颗粒的方法。通过将液体制剂投影为多个喷嘴（J）（图6），使得每个射流分解成窄尺寸分布的液滴的方式形成液滴。在聚结开始之前，液滴与气流（G）接触，气流被设置为通过破坏液滴的滑动流动和/或加速液滴来减少聚结。

90. 发明申请

WO1994017062A1 SUBSTITUTED FUSED PYRAZOLO COMPOUNDS AND THEIR USE AS HERBICIDES 审中-公开
标题翻译：取代的FUSED PYRAZOLO化合物及其作为除草剂的用途
公开(公告)号：WO1994017062A1
公开(公告)日：1994-08-04
申请号：PCT/GB1994000067
申请日：1994-01-13
申请人： ZENECA LIMITED
发明人： ZENECA LIMITED , MICHAELY, William, James , CURTIS, Jeff, Kimo , KNUDSEN, Christopher, Glade
IPC分类号： C07D471/04
CPC分类号： C07D471/04 , A01N43/90 , C07D487/04
摘要： Novel substituted pyrazolo-rings fused to nitrogen containing heterocyclic rings having formula (I) in which at least one of Y, Z or W is N or N-O and the remainder of Y, Z or W is C-R wherein R is hydrogen; halogen; nitro; cyano; alkyl; alkoxymethyl; acetoxymethyl; hydroxymethyl; haloalkyl; formyl; alkylcarbonyl; carboxy and its salts; COO alkyl; azido (N3); amino; substituted amino wherein the substituents are alkyl, alkoxy, hydroxy, formyl, alkylcarbonyl, alkoxycarbonylalkyloxy, alkoxycarbonylalkylthio, alkoxycarbonylalkylidenecarbonyl, hydroxycarbonylalkoxy, hydroxycarbonylthio, cyanoalkoxy, hydroxycarbonylalkyledinecarbonyl, alkylsufonyl, haloalkylsulfonyl, aminocarbonyl, (di)alkylaminocarbonyl, alkoxycarbonyl, alkoxyalkyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, and amino; carboxyamido; substituted carboxyamido wherein said substituents can be selected from alkyl, alkylsulfonyl, and haloalkylsulfonyl; sulfonamido wherein the N is substituted with hydrogen and/or alkyl; YR wherein Y is O and S(O)m and R is selected from the group hydrogen, alkyl, haloalkyl, cyanolalkyl, alkoxycarbonylalkyl, hydroxycarbonylalkyl and aminocarbonylalkyl wherein the N is substituted with hydrogen and/or alkyl; m is 0 to 2; R is hydrogen and halogen; R is hydrogen, nitro, halogen, cyano, alkylthio, alkylsulfinyl, alkylsulfonyl, and alkoxy; R is halogen, haloalkyl, cyano, alkylthio, alkylsulfinyl, and alkylsulfonyl; R is hydrogen and halogen; X is N or C-R ; wherein R is hydrogen, haloalkyl, halogen, cyano, nitro, alkylthio, alkylsulfinyl, alkylsulfonyl, and alkoxy; and agriculturally acceptable salts thereof.
摘要翻译：与式（I）的含氮杂环稠合的新型取代的吡唑并环，其中Y，Z或W中的至少一个为N或N-O，Y，Z或W的其余部分为C-R，其中R为氢; 卤素; 硝基; 氰基; 烷基; 烷氧基; 乙酰氧基; 羟甲基; 卤代; 甲酰基; 羰基; 羧基及其盐; COO烷基; 叠氮（N 3）; 氨基; 取代的氨基，其中取代基是烷基，烷氧基，羟基，甲酰基，烷基羰基，烷氧基羰基烷氧基，烷氧基羰基烷硫基，烷氧基羰基亚烷基羰基，羟基羰基烷氧基，羟基羰基硫基，氰基烷氧基，羟基羰基烷基羰基，烷基磺酰基，卤代烷基磺酰基，氨基羰基，（二）烷基氨基羰基，烷氧基羰基，烷氧基烷基，羟基羰基烷基，烷氧基羰基烷基和氨基; 羧酰胺; 取代的羧酰胺基，其中所述取代基可以选自烷基，烷基磺酰基和卤代烷基磺酰基; 其中N被氢和/或烷基取代; YR 6其中Y是O且S（O）m和R 6选自氢，烷基，卤代烷基，环烷醇烷基，烷氧基羰基烷基，羟基羰基烷基和氨基羰基烷基，其中N被氢和/或烷基取代; m为0〜2; R 1是氢和卤素; R 2是氢，硝基，卤素，氰基，烷硫基，烷基亚磺酰基，烷基磺酰基和烷氧基; R 3是卤素，卤代烷基，氰基，烷硫基，烷基亚磺酰基和烷基磺酰基; R 4是氢和卤素; X是N或C-R 5; 其中R 5是氢，卤代烷基，卤素，氰基，硝基，烷硫基，烷基亚磺酰基，烷基磺酰基和烷氧基; 和其农业上可接受的盐。

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