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81. 发明专利

SG178115A1 ENANTIO- AND STEREO-SPECIFIC SYNTHESES OF ß-AMINO-a- HYDROXY AMIDES 未知
公开(公告)号：SG178115A1
公开(公告)日：2012-03-29
申请号：SG2012005658
申请日：2010-07-27
申请人： SCHERING CORP
发明人： TRAVERSE JOHN , LEONG WILLIAM W , MILLER STEVEN P , ALBANEZE-WALKER JENNIFER , HUNTER THOMAS J , WANG LIJUN , LIAO HONGBIAO , ARASAPPAN ASHOK , TRZASKA SCOTT T , SMITH RANDI M , LEKHAL AZZEDDINE , BOGEN STEPHANE L , KONG JIANSHE , BENNETT FRANK , NJOROGE F GEORGE , POIRIER MARC , KUO SHEN-CHUN , CHEN YONGGANG , MATTHEWS KENNETH S , DEMONCHAUX PATRICE , FERREIRA AMADEO
摘要： Processes useful for the preparation of a Compound of Formula I: Formula (I). Intermediates useful for the preparation of the compound of Formula I, and processes useful for preparing said intermediates are disclosed.

82. 发明专利

AU2010276490A1 Enantio- and stereo-specific syntheses of beta-amino-alpha- hydroxy amides 未知
公开(公告)号：AU2010276490A1
公开(公告)日：2012-03-08
申请号：AU2010276490
申请日：2010-07-27
申请人： SCHERING CORP
发明人： TRAVERSE JOHN , LEONG WILLIAM W , MILLER STEVEN P , ALBANEZE-WALKER JENNIFER , HUNTER THOMAS J , WANG LIJUN , LIAO HONGBIAO , ARASAPPAN ASHOK , TRZASKA SCOTT T , SMITH RANDI M , LEKHAL AZZEDDINE , BOGEN STEPHANE L , KONG JIANSHE , BENNETT FRANK , NJOROGE F GEORGE , POIRIER MARC , KUO SHEN-CHUN , CHEN YONGGANG , MATTHEWS KENNETH S , DEMONCHAUX PATRICE , FERREIRA AMADEO
IPC分类号： C07C315/00 , C07C237/02 , C07D209/52 , C07K5/06
摘要： Processes useful for the preparation of a Compound of Formula I: Formula (I). Intermediates useful for the preparation of the compound of Formula I, and processes useful for preparing said intermediates are disclosed.

83. 发明专利

SI2206697T1 EKSO- IN DIASTEREO-SELEKTIVNE SINTEZE HIMBACINSKIH ANALOGOV 未知
公开(公告)号：SI2206697T1
公开(公告)日：2012-02-29
申请号：SI200631234
申请日：2006-01-12
申请人： SCHERING CORP
发明人： WU GEORGE G , SUDHAKAR ANANTHA , WANG TAO , XIE JI , CHEN FRANK XING , POIRIER MARC , HUANG MINGSHENG , SABESEN VIJAY , KWOK DAW-LONG , CUI JIAN , YANG XIAOJING , THIRUVENGADAM TIRUVETTIPURAM K , LIAO JING
IPC分类号： C07C205/00 , C07C309/00

84. 发明专利

ES2374705T3 ALQUILACINO ENENTIOSELECTIVA DE COMPUESTOS TRICICLICOS. 未知
公开(公告)号：ES2374705T3
公开(公告)日：2012-02-21
申请号：ES10001106
申请日：2003-10-01
申请人： SCHERING CORP
发明人： CHEN FRANK X , WONG YEE-SHING , ECKERT JEFFREY M , ZOU NANFEI , LIANG FENG , KIM-MEADE AGNES S , POIRIER MARC , THIRUVENGADAM TIRUVETTIPURAM K , WU GEORGE G
IPC分类号： C07D221/16 , C07D401/14
摘要： Un procedimiento para la preparación de un compuesto representado por la fórmula I que comprende poner en contacto un compuesto representado por la fórmula VI con una cantidad eficaz de cianato sódico (NaOCN) y una cantidad eficaz de carbonato sódico (Na2CO3) en un disolvente orgánico miscible en agua, que comprende una cantidad eficaz de agua para formar el compuesto representado por la fórmula I.

85. 发明专利

ES2374379T3 SINTESIS EXO Y DIASTEREOSELECTIVA DE ANALOGOS DE HIMBACINA. 未知
公开(公告)号：ES2374379T3
公开(公告)日：2012-02-16
申请号：ES10001844
申请日：2006-01-12
申请人： SCHERING CORP
发明人： WU GEORGE G , SUDHAKAR ANANTHA , WANG TAO , XIE JI , CHEN FRANK XING , POIRIER MARC , HUANG MINGSHENG , SABESEN VIJAY , KWOK DAW-LONG , CUI JIAN , YANG XIAOJING , THIRUVENGADAM TIRUVETTIPURAM K , LIAO JING
IPC分类号： C07C205/55 , C07C205/44 , C07C309/08
摘要： Un compuesto seleccionado entre el grupo que consiste en:

86. 发明专利

PT2206697E SÍNTESES EXO- E DIASTEREOSSELECTIVAS DE ANÁLOGOS DA HIMBACINA 未知
公开(公告)号：PT2206697E
公开(公告)日：2012-01-10
申请号：PT10001844
申请日：2006-01-12
申请人： SCHERING CORP
发明人： CHEN FRANK XING , WU GEORGE G , THIRUVENGADAM TIRUVETTIPURAM K , SUDHAKAR ANANTHA , WANG TAO , XIE JI , POIRIER MARC , HUANG MINGSHENG , KWOK DAW-LONG , CUI JIAN , YANG XIAOJING , LIAO JING , SABESEN VIJAY
IPC分类号： C07C205/55 , C07C205/44 , C07C309/08

89. 发明专利

AT461921T 未知
公开(公告)号：AT461921T
公开(公告)日：2010-04-15
申请号：AT07002950
申请日：2003-10-01
申请人： SCHERING CORP
发明人： CHEN FRANK X , WONG YEE-SHING , ECKERT JEFFREY M , ZOU NANFEI , LIANG FENG , KIM-MEADE AGNES S , POIRIER MARC , THIRUVENGADAM TIRUVETTIPURAM K , WU GEORGE G
IPC分类号： C07D221/16 , C07D401/14
摘要： A process for the preparation of a compound represented by formula I is disclosed.

90. 发明专利

CA2406384C SYNTHESIS OF INTERMEDIATES USEFUL IN PREPARING ANTIHISTAMINE TRICYCLIC COMPOUNDS 未知
公开(公告)号：CA2406384C
公开(公告)日：2010-02-09
申请号：CA2406384
申请日：2001-04-17
申请人： SCHERING CORP
发明人： POIRIER MARC , WONG YEE-SHING , WU GEORGE G
IPC分类号： C07D221/16 , C07B61/00 , C07D213/79
摘要： A process is provided for preparing a compound having the formula (I) comprising (a) reacting a compound having the formula (II) with an isocyanate having the formula R1NCO to produce a compound having the formula (III), (b) optionally hydrolyzing the compound of formula (III) to form an amide having the formula (IV), (c) reacting the compound of formula (III) or the amide of formula (IV) with a compound having the formula (V) in the presence of a strong base to produce a compound having the formula (VI), and (d) cyclizing the compound of formula (VI) to obtain the compound of formula (I), wherein R is H or Cl, M is selected from the group consisting of Li, Na, K, MgX, ZnR A, and Al(R A)2, R A is alkyl, X is halo, R1 is selected from the group consisting of alkyl, aryl, aralkyl, heteroaryl, heteroaralkyl, cycloalkyl, cycloalkylalkyl, heterocycloalkyl, and heterocycloalkylalkyl, and L is a leaving group. Also provided is a process for preparing a compound having the formula (VIII) comprising reacting a compound having the formula (II) with CO2 and a protonating agent to obtain the compound of formula (VIII), wherein M is selected from the group consisting of Li, Na, K, MgX, ZnR A, and Al(R A)2, wherein R A is alkyl and X is halo.

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