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71. 发明申请

US20070142379A1 CYCLOHEXYL DERIVATIVES AS SELECTIVE ESTROGEN RECEPTOR MODULATORS 审中-公开
标题翻译： CYCLOHEXYL衍生物作为选择性雌激素受体调节剂
公开(公告)号：US20070142379A1
公开(公告)日：2007-06-21
申请号：US11624808
申请日：2007-01-19
申请人： Nareshkumar Jain , Mark Mecielag , William Murray , Raymond Ng , Zhihua Sui
发明人： Nareshkumar Jain , Mark Mecielag , William Murray , Raymond Ng , Zhihua Sui
IPC分类号： A61K31/5375 , A61K31/445 , A61K31/40 , C07C69/76 , C07D265/30 , C07D211/32 , C07D207/04
CPC分类号： C07D295/088 , C07C29/12 , C07C29/60 , C07C37/055 , C07C39/17 , C07C39/23 , C07C41/18 , C07C41/20 , C07C41/22 , C07C41/26 , C07C41/30 , C07C43/215 , C07C43/23 , C07C45/69 , C07C69/757 , C07C217/18 , C07C2601/14 , C07C2601/16 , C07C2602/08 , C07C2602/10 , C07D209/04 , C07C49/683 , C07C47/47 , C07C43/225 , C07C33/38
摘要： The present invention is directed to novel cyclohexyl derivatives, pharmaceutical compositions containing them and their use in the treatment of disorders and diseases mediated by an estrogen receptor.
摘要翻译：本发明涉及新颖的环己基衍生物，含有它们的药物组合物及其在治疗由雌激素受体介导的病症和疾病中的用途。

72. 发明授权

US07183445B2 Cyclohexyl derivatives as selective estrogen receptor modulators 失效
标题翻译：环己基衍生物作为选择性雌激素受体调节剂
公开(公告)号：US07183445B2
公开(公告)日：2007-02-27
申请号：US10858435
申请日：2004-06-01
申请人： Nareshkumar F. Jain , Mark J. Macielag , William V. Murray , Raymond A. Ng , Zhihua Sui
发明人： Nareshkumar F. Jain , Mark J. Macielag , William V. Murray , Raymond A. Ng , Zhihua Sui
IPC分类号： C07C39/06 , C07C39/23 , C07D295/027 , C07D265/30
CPC分类号： C07D295/088 , C07C29/12 , C07C29/60 , C07C37/055 , C07C39/17 , C07C39/23 , C07C41/18 , C07C41/20 , C07C41/22 , C07C41/26 , C07C41/30 , C07C43/215 , C07C43/23 , C07C45/69 , C07C69/757 , C07C217/18 , C07C2601/14 , C07C2601/16 , C07C2602/08 , C07C2602/10 , C07D209/04 , C07C49/683 , C07C47/47 , C07C43/225 , C07C33/38
摘要： The present invention is directed to novel cyclohexyl derivatives, pharmaceutical compositions containing them and their use in the treatment of disorders and diseases mediated by an estrogen receptor.
摘要翻译：本发明涉及新颖的环己基衍生物，含有它们的药物组合物及其在治疗由雌激素受体介导的病症和疾病中的用途。

73. 发明授权

US07183309B2 Indole derivatives useful as progesterone receptor modulators 有权
标题翻译：吲哚衍生物可用作孕激素受体调节剂
公开(公告)号：US07183309B2
公开(公告)日：2007-02-27
申请号：US11255444
申请日：2005-10-21
申请人： Weiqin Jiang , James J. Fiordeliso , Zhihua Sui
发明人： Weiqin Jiang , James J. Fiordeliso , Zhihua Sui
IPC分类号： A61K31/404 , C07D209/04
CPC分类号： C07D209/30
摘要： The present invention is directed to novel indole derivatives, pharmaceutical compositions containing them and their use in the treatment or prevention of disorders and diseases mediated by agonists and antagonists of the progesterone receptor. The clinical uses of these compounds are related to contraception, the treatment and/or prevention of secondary amenorrhea, dysfunctional bleeding, uterine leiomyomata, endometriosis; polycystic ovary syndrome, carcinomas and adenocarcinomas of the endometrium, ovary, breast, colon, prostate, or minication of side effects of cyclid menstrual bleeding. Additional uses of the invention include stimulation of food intake.
摘要翻译：本发明涉及新颖的吲哚衍生物，含有它们的药物组合物及其用于治疗或预防由孕酮受体的激动剂和拮抗剂介导的病症和疾病。这些化合物的临床应用与避孕，继发性闭经，功能障碍性出血，子宫平滑肌瘤，子宫内膜异位症的治疗和/或预防有关; 多囊卵巢综合征，子宫内膜癌，卵巢癌，乳腺癌，结肠癌，前列腺癌，腺瘤，子宫内膜异位症，副周围性月经出血副作用。本发明的额外用途包括刺激食物摄取。

74. 发明申请

US20070037877A1 Novel coumarin derivatives as ion channel openers 有权
标题翻译：新型香豆素衍生物作为离子通道开放剂
公开(公告)号：US20070037877A1
公开(公告)日：2007-02-15
申请号：US11334679
申请日：2006-01-18
申请人： Nareshkumar Jain , Zhihua Sui
发明人： Nareshkumar Jain , Zhihua Sui
IPC分类号： A61K31/366 , C07D311/02
CPC分类号： C07D311/16 , C07D311/18 , C07D493/04
摘要： The present invention is directed to novel coumarin derivatives, pharmaceutical compositions containing them and their use in the treatment of disorders related to ion channels such as potassium channels
摘要翻译：本发明涉及新颖的香豆素衍生物，含有它们的药物组合物及其用于治疗与离子通道相关的疾病如钾通道

75. 发明申请

US20060111402A1 Novel benzimidazole derivatives useful as selective androgen receptor modulators (SARMS) 有权
标题翻译：用作选择性雄激素受体调节剂（SARMS）的新型苯并咪唑衍生物
公开(公告)号：US20060111402A1
公开(公告)日：2006-05-25
申请号：US11235581
申请日：2005-09-26
申请人： Raymond Ng , Zhihua Sui , Jihua Guan , James Lanter , Vernon Alford
发明人： Raymond Ng , Zhihua Sui , Jihua Guan , James Lanter , Vernon Alford
IPC分类号： A61K31/4439 , A61K31/4184 , C07D403/02
CPC分类号： C07D405/06 , C07D235/10 , C07D235/12 , C07D235/14 , C07D235/16 , C07D401/06 , C07D403/10 , C07D409/06 , C07D409/14 , C07D413/06 , C07D417/10
摘要： The present invention is directed to novel benzimidazole derivatives, pharmaceutical compositions containing them and their use in the treatment of disorders and conditions modulated by the androgen receptor.
摘要翻译：本发明涉及新的苯并咪唑衍生物，含有它们的药物组合物及其在治疗由雄激素受体调节的病症和状况中的用途。

76. 发明申请

US20060040917A1 Benzoxazepine derivatives as selective estrogen receptor modulators 审中-公开
标题翻译：苯并西泮衍生物作为选择性雌激素受体调节剂
公开(公告)号：US20060040917A1
公开(公告)日：2006-02-23
申请号：US11191499
申请日：2005-07-28
申请人： James Lanter , Zhihua Sui , James Fiordeliso
发明人： James Lanter , Zhihua Sui , James Fiordeliso
IPC分类号： A61K31/553 , C07D267/02
CPC分类号： C07D267/10 , C07D267/14
摘要： The present invention is directed to novel benzoxazepine derivatives, pharmaceutical compositions containing them and their use in the treatment of disorders and diseases mediated by an estrogen receptor.
摘要翻译：本发明涉及新的苯并氧氮杂衍生物，含有它们的药物组合物及其在治疗由雌激素受体介导的病症和疾病中的用途。

77. 发明申请

US20050113402A1 Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors 审中-公开
标题翻译：用作磷酸二酯酶抑制剂的取代的吡咯并吡喃酮衍生物
公开(公告)号：US20050113402A1
公开(公告)日：2005-05-26
申请号：US10971476
申请日：2004-10-22
申请人： Zhihua Sui , Mark Macielag , Jihua Guan , Weigin Jiang , James Lanter
发明人： Zhihua Sui , Mark Macielag , Jihua Guan , Weigin Jiang , James Lanter
IPC分类号： A61K31/437 , A61K31/4709 , A61K31/496 , A61K31/506 , A61K31/5377 , A61P3/10 , A61P7/02 , A61P9/00 , A61P9/04 , A61P9/10 , A61P9/12 , A61P11/06 , A61P15/00 , A61P15/02 , A61P15/06 , A61P15/08 , A61P15/10 , A61P43/00 , C07D471/04 , A61K31/4745 , C07D471/02
CPC分类号： C07D471/04
摘要： The invention relates to novel pyrrolopyridinone derivatives of the formula (I) or (II): pharmaceutical compositions containing the compounds and their use for the treatment of sexual dysfunction.
摘要翻译：本发明涉及式（I）或（II）的新型吡咯并吡喃酮衍生物：含有化合物的药物组合物及其用于治疗性功能障碍的用途。

78. 发明授权

US07968580B2 Imidazolidin-2-one derivatives as selective androgen receptor modulators (SARMS) 有权
标题翻译：咪唑啉-2-酮衍生物作为选择性雄激素受体调节剂（SARMS）
公开(公告)号：US07968580B2
公开(公告)日：2011-06-28
申请号：US12413873
申请日：2009-03-30
申请人： James C. Lanter , Zhihua Sui
发明人： James C. Lanter , Zhihua Sui
IPC分类号： A61K31/4166 , C07D233/30
CPC分类号： C07D233/34
摘要： The present invention is directed to novel imidazolidin-2-one derivatives having a structure according to Formula I wherein a, b, R1, R2, R3, and R4 are as defined above, pharmaceutical compositions containing them and their use in the treatment of disorders and conditions modulated by the androgen receptor.
摘要翻译：本发明涉及具有式I结构的新的咪唑烷-2-酮衍生物，其中a，b，R1，R2，R3和R4如上定义，含有它们的药物组合物及其在治疗疾病中的用途和由雄激素受体调节的条件。

79. 发明授权

US07932399B2 2-substituted benzimidazoles as selective androgen receptor modulators (SARMS) 有权
标题翻译： 2-取代苯并咪唑作为选择性雄激素受体调节剂（SARMS）
公开(公告)号：US07932399B2
公开(公告)日：2011-04-26
申请号：US11626030
申请日：2007-01-23
申请人： Vernon C. Alford, Jr. , James C. Lanter , Raymond A. Ng , Zhihua Sui
发明人： Vernon C. Alford, Jr. , James C. Lanter , Raymond A. Ng , Zhihua Sui
IPC分类号： A61K31/4184 , C07D235/10
CPC分类号： C07F7/1804 , A61K31/4184 , C07D235/12 , C07D235/16 , C07D403/04 , C07D405/04 , C07D405/14 , C07D413/04
摘要： The present invention is directed to a novel 2-substituted benzimidazole derivatives, pharmaceutical compositions containing them and their use in the treatment of disorders and conditions modulated by the androgen receptor.
摘要翻译：本发明涉及一种新的2-取代苯并咪唑衍生物，含有它们的药物组合物及其用于治疗由雄激素受体调节的病症和状况。

80. 发明申请

US20100298383A1 NOVEL BENZIMIDAZOLE DERIVATIVES USEFUL AS SELECTIVE ANDROGEN RECEPTOR MODULATORS (SARMS) 审中-公开
标题翻译：新型苯并咪唑衍生物作为选择性受体调节剂（SARMS）有用
公开(公告)号：US20100298383A1
公开(公告)日：2010-11-25
申请号：US12849378
申请日：2010-08-03
申请人： Raymond Ng , Zhihua Sui , Jihua Guan , James C. Lanter , Vernon C. Alford, JR.
发明人： Raymond Ng , Zhihua Sui , Jihua Guan , James C. Lanter , Vernon C. Alford, JR.
IPC分类号： A61K31/4439 , A61K31/4184 , A61K31/422 , A61K31/433 , A61P43/00 , A61P35/00 , A61P3/04 , A61P17/14 , A61P31/18 , A61P15/16 , A61P15/00 , A61P17/10
CPC分类号： C07D405/06 , C07D235/10 , C07D235/12 , C07D235/14 , C07D235/16 , C07D401/06 , C07D403/10 , C07D409/06 , C07D409/14 , C07D413/06 , C07D417/10
摘要： The present invention is directed to novel benzimidazole derivatives, pharmaceutical compositions containing them and their use in the treatment of disorders and conditions modulated by the androgen receptor.
摘要翻译：本发明涉及新的苯并咪唑衍生物，含有它们的药物组合物及其在治疗由雄激素受体调节的病症和状况中的用途。

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