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71. 发明授权

US06169200A Method for producing &agr;-hydroxy-&bgr;-aminocarboxylic acids 失效
标题翻译： α-羟基-β-氨基羧酸的制备方法
公开(公告)号：US06169200A
公开(公告)日：2001-01-02
申请号：US09186272
申请日：1998-11-05
申请人： Takayuki Suzuki , Yutaka Honda , Kunisuke Izawa
发明人： Takayuki Suzuki , Yutaka Honda , Kunisuke Izawa
IPC分类号： C07C31728
CPC分类号： C07C323/29 , C07C317/28 , C07C327/30
摘要： The present invention provides a simple and inexpensive method for producing &agr;-hydroxy-&bgr;-aminocarboxylic acids and their esters. An ester of an N-protected &agr;-amino acid ester is converted into a &bgr;-ketosulfoxide, which is then processed with an acid to give an &agr;-ketohemimercaptal. Next, this is acylated and then processed with a base to obtain an N-protected &agr;-acyloxy-&bgr;-amino-thioester, which is then saponified to obtain an intended compound. According to the method of the present invention, it is possible to produce &agr;-hydroxy-&bgr;-aminocarboxylic acid derivatives, which are intermediates in producing various HIV protease inhibitors, renin inhibitors and carcinostatics, from a-amino acids. The method comprises reduced reaction steps, the selectivity in the method to give the intended product is high, and the yield of the product obtained is high.
摘要翻译：本发明提供了用于生产α-羟基-β-氨基羧酸及其酯的简单和便宜的方法。将N-保护的α-氨基酸酯的酯转化为β-氧亚砜，然后用酸处理给予α-酮基咪唑。接下来，将其进行酰化，然后用碱处理，得到N-保护的α-酰氧基-β-氨基 - 硫代酯，然后皂化，得到目的化合物。根据本发明的方法，可以生产α-羟基-β-氨基羧酸衍生物，它们是从α-氨基酸生产各种HIV蛋白酶抑制剂，肾素抑制剂和制癌剂的中间体。该方法包括减少反应步骤，得到所需产物的方法中的选择性高，所得产物的产率高。

72. 发明授权

US6028217A Optically active salts of 2-hydroxymethyl-3-phenylpropionic acid with cis-1-amino-2-indanol, .alpha.-methylbenzylamine, or 3-methyl-2-phenyl-1-butylamine 失效
标题翻译： 2-羟甲基-3-苯基丙酸与顺式-1-氨基-2-茚满醇，α-甲基苄胺或3-甲基-2-苯基-1-丁胺的光学活性盐
公开(公告)号：US6028217A
公开(公告)日：2000-02-22
申请号：US166124
申请日：1998-10-05
申请人： Hiroyuki Nohira , Takayuki Suzuki , Takayuki Hamada , Kunisuke Izawa
发明人： Hiroyuki Nohira , Takayuki Suzuki , Takayuki Hamada , Kunisuke Izawa
IPC分类号： C07B57/00 , C07C51/487 , C07C59/48 , C07C211/27 , C07C215/44 , C07B55/00
CPC分类号： C07C215/44 , C07C211/27 , C07C51/487 , C07C59/48
摘要： A compound selected from the group consisting of(a) optically active 2-hydroxymethyl-3-phenylpropionic acid cis-1-amino-2-indanol salt,(b) optically active 2-hydroxymethyl-3-phenylpropionic acid .alpha.-methylbenzylamine salt,(c) optically active 2-hydroxymethyl-3-phenylpropionic acid 3-methyl-2-phenyl-1-butylamine salt,(d) a salt of (S)-2-hydroxymethyl-3-phenylpropionic acid with (1R, 2S)-(+)-cis-1-amino-2-indanol,(e) a salt of (R)-2-hydroxymethyl-3-phenylpropionic acid with (1S, 2R)-(-)-cis-1-amino-2-indanol,(f) a salt of (R)-2-hydroxymethyl-3-phenylpropionic acid with (S)-(-)-.alpha.-methylbenzylamine,(g) a salt of (S)-2-hydroxymethyl-3-phenylpropionic acid with (R)-(+)-.alpha.-methylbenzylamine,(h) a salt of (S)-2-hydroxymethyl-3-phenylpropionic acid with (S)-(-)-3-methyl-2-phenyl-1-butylamine, and(i) a salt of (R)-2-hydroxymethyl-3-phenylpropionic acid with (R)-(+)-3-methyl-2-phenyl-1-butylamine.
摘要翻译：选自（a）光学活性2-羟甲基-3-苯基丙酸顺式-1-氨基-2-二氢化茚醇盐，（b）光学活性2-羟甲基-3-苯基丙酸α-甲基苄基胺盐的化合物，（c）光学活性的2-羟甲基-3-苯基丙酸3-甲基-2-苯基-1-丁胺盐，（d）（S）-2-羟甲基-3-苯基丙酸与（1R，2S）（±） - 顺式-1-氨基-2-茚满醇，（e）（R）-2-羟甲基-3-苯基丙酸与（1S，2R） - （ - ） - 顺式-1-氨基-2- （R）-2-羟甲基-3-苯基丙酸与（S） - （ - ） - α-甲基苄胺的盐，（g）（S）-2-羟甲基-3 （（R） - （+） - α-甲基苄基胺，（h）（S）-2-羟甲基-3-苯基丙酸与（S） - （ - ） - 3-甲基-2-苯基 -1-丁胺，和（i）（R）-2-羟甲基-3-苯基丙酸与（R） - （+） - 3-甲基-2-苯基-1-丁基胺的盐。

73. 发明授权

US5979966A Cowling brace of motorcycle 失效
标题翻译：摩托车的大括号
公开(公告)号：US5979966A
公开(公告)日：1999-11-09
申请号：US50178
申请日：1998-03-30
申请人： Takayuki Suzuki
发明人： Takayuki Suzuki
IPC分类号： B62J17/00 , B62K19/48
CPC分类号： B62K19/48 , B62J17/00
摘要： A motorcycle is provided with a cowling brace having a sub-frame structure for attaching a cowling and a cowling peripheral part to a front head portion of a body frame of a motorcycle. The cowling brace is composed of a front brace member integrally formed of a synthetic resin material, a rear brace member assembled by using a metal material to be combined with the front brace member, a front fixture member formed integrally with the front brace member and adapted to fix the cowling and the cowling peripheral part, and a rear fixture member formed to rear brace member and adapted to fix the rear brace member to the body frame of the motorcycle.
摘要翻译：摩托车设置有具有子框架结构的整流罩支架，用于将整流罩和整流罩周边部分附接到摩托车的车身框架的前头部。整流罩支架由由合成树脂材料一体形成的前支撑构件，通过使用与前支撑构件组合的金属材料组装的后支撑构件构成，前固定构件与前支撑构件一体地形成并适应固定整流罩和整流罩周边部分，以及形成在后支撑构件上并适于将后支撑构件固定到摩托车的车体框架上的后固定构件。

74. 发明授权

US5744037A Method of treating foul water 失效
标题翻译：污水处理方法
公开(公告)号：US5744037A
公开(公告)日：1998-04-28
申请号：US758249
申请日：1996-11-27
申请人： Hiroyuki Fujimura , Takayuki Suzuki , Norio Yamada , Yoshiyuki Ichiki
发明人： Hiroyuki Fujimura , Takayuki Suzuki , Norio Yamada , Yoshiyuki Ichiki
IPC分类号： C02F3/12 , C02F3/28 , C02F11/06 , F23G7/00 , B01D37/00
CPC分类号： C02F3/286 , C02F11/06 , C02F3/12 , C02F3/28 , C02F3/2846 , F23G7/001 , Y02E50/343 , Y02W10/15 , Y02W10/37 , Y02W10/40 , Y10S210/903
摘要： In an improved method of treating foul water, the solids that are produced during the process of treatment of foul water such as wastewater or liquid sludges are treated with a heat treatment apparatus and the resulting thermal energy and/or gas is utilized in the treatment of said foul water. The foul water may be subjected, directly and/or after a treatment, to a filtration step using a filter packed with nonflammable particulate matter such as sand, and the trapped solids are fed into a fluidized-bed heat treatment apparatus such as a fluidized-bed incinerator or gasification furnace and, thereafter, the nonflammable particulate matter in the heat treatment apparatus is returned to the filtration step. The foul water can be treated with effective utilization of the energy of the organic matter in the foul water or the solids that are produced during the process of its treatment.
摘要翻译：在处理污水的改进方法中，在处理污水如废水或液体污泥的过程中产生的固体用热处理装置处理，并且所得热能和/或气体用于处理说脏水。可以使用装有不可燃颗粒物质如沙子的过滤器将污水直接和/或处理后进行过滤步骤，并且将捕获的固体进料到流化床热处理装置如流化床处理装置中，床焚烧炉或气化炉，然后将热处理设备中的不可燃颗粒物质返回到过滤步骤。可以有效利用污水中的有机物质的能量或其处理过程中产生的固体来处理污水。

75. 外观设计

USD391013S Gas lighter 失效
公开(公告)号：USD391013S
公开(公告)日：1998-02-17
申请号：US63018
申请日：1996-11-21
申请人： Isao Inoue , Takayuki Suzuki
设计人： Isao Inoue , Takayuki Suzuki

76. 发明授权

US5521180A Morpholine derivative 失效
标题翻译：吗啉衍生物
公开(公告)号：US5521180A
公开(公告)日：1996-05-28
申请号：US495619
申请日：1995-08-03
申请人： Mitsuo Fujii , Takayuki Suzuki , Satoshi Hayashibe , Shin-ichi Tsukamoto , Shin-ichi Yatsugi , Tokio Yamaguchi
发明人： Mitsuo Fujii , Takayuki Suzuki , Satoshi Hayashibe , Shin-ichi Tsukamoto , Shin-ichi Yatsugi , Tokio Yamaguchi
IPC分类号： C07D265/30 , A61K31/535
CPC分类号： C07D265/30
摘要： A morpholine derivative represented by formula (I) or a pharmaceutically acceptable salt thereof: ##STR1## wherein R.sup.1 and R.sup.3, which may be the same or different, each represent a hydrogen atom or a lower alkyl group; R.sup.2 represents a halogen atom; and the dotted line indicates an optional double bond. These compounds exhibit a selective 5-HT reuptake inhibitory activity and a selective 5-HT.sub.2 receptor antagonistic activity and useful as a therapeutic agent for depression, anxiety, etc. with reduced side effects.
摘要翻译： PCT No.PCT / JP94 / 00186 Sec。 371日期：1995年8月3日 102（e）日期1995年8月3日PCT 1994年2月8日PCT PCT。公开号WO94 / 18182 日本美国专利申请公开说明书（公告）日本公开一般公开说明书（公开号）（Ⅰ）所示的吗啉衍生物或其药学上可接受的盐：其中R 1和R 3可以相同或不同，各自表示氢原子或低级烷基; R2表示卤原子; 虚线表示可选的双键。这些化合物表现出选择性的5-HT再摄取抑制活性和选择性的5-HT2受体拮抗活性，并且可用作抑制，焦虑等的治疗剂，副作用降低。

77. 发明授权

US5430466A Thermal transfer recording method 失效
标题翻译：热转印记录法
公开(公告)号：US5430466A
公开(公告)日：1995-07-04
申请号：US721872
申请日：1991-06-26
申请人： Takayuki Suzuki
发明人： Takayuki Suzuki
IPC分类号： B41M5/395 , B41J2/325 , B41M5/26 , B41M5/30 , B41M5/392 , G01D9/00 , G01D15/10
CPC分类号： B41M5/395 , Y10S428/913
摘要： A thermal transfer recording method involving providing a thermal transfer medium having a support and ink layer thereon, the binder being chosen so as to have a melt viscosity which falls within a range that is temperature dependent, contacting the thermal transfer medium with a recording medium, applying energy with a recording head to transfer an image to the recording medium, and moving, in a unit period of time, the thermal transfer material through a distance relative to the recording head that is smaller than the distance through which the recording medium moves in that time.
摘要翻译：一种热转印记录方法，包括提供其上具有支撑和油墨层的热转印介质，所述粘合剂选择为具有落入温度依赖性的范围内的熔融粘度，使所述热转印介质与记录介质接触，用记录头施加能量以将图像转印到记录介质上，并且在单位时间内将热转印材料相对于记录头移动一定距离，该距离小于记录介质移动的距离那时。

78. 发明授权

US5389429A Thermal transfer material and thermal transfer recording method 失效
标题翻译：热转印材料和热转印记录方法
公开(公告)号：US5389429A
公开(公告)日：1995-02-14
申请号：US115105
申请日：1993-09-02
申请人： Yoshihisa Takizawa , Naoki Kushida , Takayuki Suzuki , Tetsuo Hasegawa
发明人： Yoshihisa Takizawa , Naoki Kushida , Takayuki Suzuki , Tetsuo Hasegawa
IPC分类号： B41M5/00 , B41M5/26 , B41M5/395
CPC分类号： B41M5/395 , Y10S428/913 , Y10S428/914 , Y10T428/31935
摘要： A thermal transfer material including a support and a heat-transferable ink layer disposed thereon, wherein the heat-transferable ink layer has a storage elasticity modulus E' satisfying a relationship of: 1.times.10.sup.7 .ltoreq.E'.ltoreq.1.times.10.sup.9 N/m.sup.2 at 30.degree. C.; and the temperature providing a thermal differential value of dynamic energy loss angle (tan .delta.) satisfying a relationship of d(tan .delta.)/dT=1.times.10.sup.-2 is in the range of 40.degree. to 60.degree. C.
摘要翻译：一种热转印材料，其包括支撑体和设置在其上的可热转印的油墨层，其中所述可转印油墨层具有满足以下关系的储能弹性模量E'：1×107

79. 发明授权

US5269865A Thermal transfer material and thermal transfer recording method 失效
标题翻译：热转印材料和热转印记录方法
公开(公告)号：US5269865A
公开(公告)日：1993-12-14
申请号：US931407
申请日：1992-08-24
申请人： Naoki Kushida , Yasuyuki Tamura , Takayuki Suzuki , Koichi Tohma , Masanobu Asaoka
发明人： Naoki Kushida , Yasuyuki Tamura , Takayuki Suzuki , Koichi Tohma , Masanobu Asaoka
IPC分类号： B41J2/325 , B41J17/00 , B44C1/17 , B32B31/00 , B41J2/45
CPC分类号： B44C1/1712 , B41J17/00 , B41J2/325 , Y10S428/913
摘要： There are provided a "self-correctable" thermal transfer material and a thermal transfer recording method using the transfer material. The thermal transfer material comprises a support, a first ink layer, a second ink layer and a third ink layer disposed in this order on the support, wherein the first ink layer is a substantially non-transferable layer, the second ink layer is capable of causing separation from the first ink layer on heating; and the third ink layer comprising a thermoplastic resin and a colorant. A recorded image formed by the above-mentioned transfer material can be removed through lift-off correction, by causing the transfer material to adhere to the recorded image under heating, and separating the transfer material from the recording medium without causing separation of the second ink layer.
摘要翻译：提供了使用转印材料的“自校正”热转印材料和热转印记录方法。热转印材料包括在支撑体上依次设置的支撑体，第一油墨层，第二油墨层和第三油墨层，其中第一油墨层是基本不可转移的层，第二油墨层能够导致在加热时与第一油墨层分离; 并且第三油墨层包含热塑性树脂和着色剂。由上述转印材料形成的记录图像可以通过剥离校正，通过使转印材料在加热下粘附到记录图像上，并将转印材料从记录介质上分离而不会导致第二墨水分离层。

80. 发明授权

US5268704A Thermal transfer recording method reducing ground staining and improving ink transferability 失效
标题翻译：热转印记录方法减少地面染色和改善油墨转移性
公开(公告)号：US5268704A
公开(公告)日：1993-12-07
申请号：US905527
申请日：1992-06-29
申请人： Tetsuo Hasegawa , Takayuki Suzuki , Naoki Kushida , Yoshihisa Takizawa
发明人： Tetsuo Hasegawa , Takayuki Suzuki , Naoki Kushida , Yoshihisa Takizawa
IPC分类号： B41J2/32 , B41J31/00 , B41M5/395
CPC分类号： B41M5/395
摘要： Thermal transfer recording is improved by a recording method involving providing a thermal transfer material having a support and an ink layer disposed thereon and which in turn includes a binder and a colorant. The binder includes 45-70 wt. % of an ethylene-vinyl acetate copolymer, 25-50 wt. % of a wax, and 7-12 wt. % of a tackifier based on a total weight of the binder. The ink layer has a breakdown strength of 30-80 kg/cm.sup.2 at 25.degree. C. The method also involves contacting an ink layer side of the thermal transfer material with a recording medium, supplying a pattern of energy from a recording head to the thermal transfer material, and separating the thermal transfer material from the recording medium to leave a transferred image on the recording medium. The thermal transfer material moves in a unit period of time by a first distance relative to the recording head which is smaller than a second distance through which the recording medium moves relative to the recording head in the same unit period of time.
摘要翻译：通过提供具有支撑体的热转印材料和设置在其上的油墨层并且还包括粘合剂和着色剂的热转印材料的记录方法来改进热转印记录。粘合剂包括45-70wt。％的乙烯 - 乙酸乙烯酯共聚物，25-50wt。％的蜡，和7-12wt。基于粘合剂的总重量的增粘剂的％。油墨层在25℃下的击穿强度为30-80kg / cm2。该方法还包括使热转印材料的油墨层与记录介质接触，将记录头的能量图案提供给热转印材料，并将热转印材料与记录介质分离，以将转印图像留在记录介质上。热转印材料在单位时间内相对于记录头移动第一距离，该距离小于记录介质在相同的单位时间内相对于记录头移动的第二距离。

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