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61. 发明授权

US07312179B2 Cyclopropyl-thienyl-carboxamide as fungicides 失效
公开(公告)号：US07312179B2
公开(公告)日：2007-12-25
申请号：US10532847
申请日：2003-10-24
申请人： Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： A01N43/36 , C07D409/00
CPC分类号： C07D409/12 , C07D333/36 , C07D411/12 , C07D417/12
摘要： A fungicidally active compound of formula (I): where X is (X1), (X2) or (X3); Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, provided that the ring is not 1,2,3-triazole, the ring being substituted by groups R4, R5 and R6; R1 and R2 are each, independently, hydrogen, halo or methyl; R3 is optionally substituted C2-12 alkyl, optionally substituted C2-12 alkenyl, optionally substituted C2-12 alkynyl, optionally substituted C3−12 cycloalkyl, optionally substituted phenyl or optionally substituted heterocyclyl; R4, R5 and R6 are each, independently, selected from hydrogen, halo, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkylene and C 1-4 haloalkoxy(C1-4)alkylene, provided that at least one of R4, R5 and R6 is not hydrogen; and R7 and R8 are each, independently, hydrogen, halogen, C1-4 alkyl or Clue haloalkyl; the invention also relates to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to the preparation of intermediates, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi

62. 发明申请

US20060287328A1 Silicon compounds with microbiocidal activity 失效
公开(公告)号：US20060287328A1
公开(公告)日：2006-12-21
申请号：US10569343
申请日：2004-09-08
申请人： Josef Ehrenfreund , Clemens Lamberth , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Clemens Lamberth , Hans Tobler , Harald Walter
IPC分类号： C07D417/02 , C07D413/02 , C07D409/02 , C07D403/02 , A01N43/54 , A01N43/80 , A01N43/76 , A01N43/64
CPC分类号： C07F7/0812 , A01N55/00
摘要： Fungicidal compounds of formula (1): where X is O or S; RING is phenyl or thienyl; Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by one to four groups R4; R1 is hydrogen, optionally substituted (C1-4)alkyl, formyl, optionally substituted (C1-4)alkylC(═O), optionally substituted (C1-4)alkylC(═O)O, optionally substituted (C1-4)alkoxy(C1-4)alkyl, optionally substituted allyl, optionally substituted propargyl or optionally substituted allenyl; each R2 is, independently, halogen, optionally substituted (C1-4)alkyl, optionally substituted (C1-4)alkoxy or optionally substituted (C1-4)alkoxy(C1-4)alkyl; R3 is (CRaRb)m-Cy-(CRcRd)n—Y; each R4 is, independently, selected from halogen, C1-3 alkyl, C1-3 haloalkyl, C1-3alkoxy(C1-3)alkyl and cyano; Ra, Rb, Rc and Rd are each, independently, hydrogen or optionally substituted (C1-4)alkyl; Cy is an optionally substituted carbocyclic or heterocyclic 3-7 membered ring which may be saturated, unsaturated or aromatic and which optionally contains a silicon atom as a ring member; (CRaRb)m and (CRcRd), may be bound either to the same carbon or silicon atom of Cy or to different atoms separated by 1, 2 or 3 ring members; Y is Si(OpZ1)(OqZ2)(O5Z) and provided that Cy contains a silicon atom as a ring member then Y may also be hydrogen; Z is C1-4 alkyl or C2-4 alkenyl (each of which is optionally interrupted by one heteroatom selected from O, S and N and is optionally substituted by one to three independently selected halogen atoms); Z1 and Z2 are, independently, methyl or ethyl; in and n are each, independently, 0, 1, 2 or 3; p, q and s are each, independently, 0 or 1; and r is 0, 1 or 2; or an N-oxide thereof; novel intermediates used in the preparation of these compounds, agrochemical compositions which comprise at least one of the novel compounds as active ingredient and the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.

63. 发明申请

US20060030567A1 Cyclopropyl-thienyl-carboxamide as fungicides 失效
公开(公告)号：US20060030567A1
公开(公告)日：2006-02-09
申请号：US10532847
申请日：2003-10-24
申请人： Josef Ehrenfreund , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Hans Tobler , Harald Walter
IPC分类号： C07D409/02 , A01N43/64 , A01N43/54
CPC分类号： C07D409/12 , C07D333/36 , C07D411/12 , C07D417/12
摘要： A fungicidally active compound of formula (I): where X is (X1), (X2) or (X3); Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, provided that the ring is not 1,2,3-triazole, the ring being substituted by groups R4, R5 and R6; R1 and R2 are each, independently, hydrogen, halo or methyl; R3 is optionally substituted C2-12 alkyl, optionally substituted C2-12 alkenyl, optionally substituted C2-12 alkynyl, optionally substituted C3−12 cycloalkyl, optionally substituted phenyl or optionally substituted heterocyclyl; R4, R5 and R6 are each, independently, selected from hydrogen, halo, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkylene and C1-4 haloalkoxy(C1-4)alkylene, provided that at least one of R4, R5 and R6 is not hydrogen; and R7 and R8 are each, independently, hydrogen, halogen, C1-4 alkyl or Clue haloalkyl; the invention also relates to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to the preparation of intermediates, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.

64. 发明申请

US20050182107A1 Siliconated phenyl amides derivatives useful as microbiocide 失效
公开(公告)号：US20050182107A1
公开(公告)日：2005-08-18
申请号：US10509607
申请日：2003-03-21
申请人： Josef Ehrenfreund , Pierre Joseph Jung , Hans Tobler , Harald Walter
发明人： Josef Ehrenfreund , Pierre Joseph Jung , Hans Tobler , Harald Walter
IPC分类号： A01N55/00 , A01N55/10 , C07F7/08 , C07F7/10 , C07D213/46 , A01N43/36 , A01N43/40
CPC分类号： C07F7/0812 , A01N55/00
摘要： A fungicidal compound of formula (1): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by groups R7, R8 and R9; R1 is hydrogen, optionally substituted (C1-4)alkylC(═O), optionally substituted (C1-4)alkylC(═O)O, optionally substituted (C1-4)alkoxy(C1-4)alkyl, optionally substituted allyl, optionally substituted propargyl or optionally substituted allenyl; R2, R3, R4 and R5 are each, independently, hydrogen, halogen, optionally substituted (C1-4)alkoxy(C1-4)alkoxy or optionally substituted (C1-4)alkoxy(C1)alkyl; R6 is an organic group containing three to thirteen carbon atoms and at least one silicon atom and, optionally, one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, and is optionally substituted by one to four independently selected halogen atoms; R7, R8 and R9 are each, independently, hydrogen, halogen, C1-3alkyl, C1-3haloalkyl, C1-3alkoxy(C1-3)alkyl or cyano, where at least one of R7, R8 and R9 is not hydrogen; and X is O or S; or an N-oxide thereof; and when present, each optional substituent on alkyl moieties, allyl, propargyl and allenyl is, independently, selected from halogen, hydroxy, cyano, methoxycarbonyl, ethoxycarbonyl, methoxy, ethoxy, methylsulfonyl, ethylsulfonyl, diflouromethoxy, trifluoromethoxy and trifluorothiomethoxy.

65. 发明申请

US20110224241A1 ISOTHIAZOLE AND PYRAZOLE DERIVATIVES AS FUNGICIDES 失效
标题翻译：异噻唑和吡唑衍生物作为杀真菌剂
公开(公告)号：US20110224241A1
公开(公告)日：2011-09-15
申请号：US12668435
申请日：2008-07-09
申请人： Peter Ackermann , Carla Bobbio , Camilla Corsi , Josef Ehrenfreund , Ann Monica McGinley , Andreas Verras , Ruud Titulaer
发明人： Peter Ackermann , Carla Bobbio , Camilla Corsi , Josef Ehrenfreund , Ann Monica McGinley , Andreas Verras , Ruud Titulaer
IPC分类号： A61K31/506 , C07D417/06 , A61K31/4439 , A01N43/80 , A61P31/10 , A01P3/00 , C07D401/06 , A01N43/56
CPC分类号： C07D417/06 , A01N43/56 , A01N43/80 , C07D401/06 , C07D417/14
摘要： The present invention relates to compounds of Formula (I) wherein R1, R2, R3 or R4 are as defined in claim 1 or a salt or N-oxide thereof and their use in methods for the control and/or prevention of fungal infection, particularly in plants. The compounds claimed are isothiazole and pyrazole derivatives.
摘要翻译：本发明涉及其中R 1，R 2，R 3或R 4如权利要求1所定义的式（I）化合物或其盐或N-氧化物及其在控制和/或预防真菌感染的方法中的用途，特别是在植物中。所要求的化合物是异噻唑和吡唑衍生物。

66. 发明申请

US20100292258A1 SUBSTITUTED AROMATIC HETEROCYCLIC COMPOUNDS AS FUNGICIDES 审中-公开
标题翻译：取代的芳香杂环化合物作为防腐剂
公开(公告)号：US20100292258A1
公开(公告)日：2010-11-18
申请号：US12601317
申请日：2008-06-16
申请人： Peter Ackermann , Carla Bobbio , Camilla Corsi , Josef Ehrenfreund , Ann Monica McGinley
发明人： Peter Ackermann , Carla Bobbio , Camilla Corsi , Josef Ehrenfreund , Ann Monica McGinley
IPC分类号： A61K31/506 , C07D401/06 , C07D403/06 , A61K31/444 , A61K31/4439 , A01N43/54 , A01N43/40 , A01P3/00 , A61P31/10
CPC分类号： C07D401/06 , C07D403/06 , C07D405/14 , C07D409/14
摘要： The present invention relates to compounds of formula (I) wherein R1, R2, R3, R4, R5 and R6 are as defined in claim 1 or a salt or N-oxide thereof and their use in methods for the control and/or prevention of fungal infection, particularly in plants.
摘要翻译：本发明涉及其中R 1，R 2，R 3，R 4，R 5和R 6如权利要求1中所定义的式（I）化合物或其盐或N-氧化物及其在控制和/或预防真菌感染，特别是在植物中。

67. 发明授权

US08377953B2 Isothiazole and pyrazole derivatives as fungicides 失效
标题翻译：异噻唑和吡唑衍生物作为杀真菌剂
公开(公告)号：US08377953B2
公开(公告)日：2013-02-19
申请号：US12668435
申请日：2008-07-09
申请人： Peter Ackermann , Carla Bobbio , Camilla Corsi , Ann Monica McGinley , Andreas Verras , Ruud Titulaeu , Josef Ehrenfreund
发明人： Peter Ackermann , Carla Bobbio , Camilla Corsi , Ann Monica McGinley , Andreas Verras , Ruud Titulaeu , Josef Ehrenfreund
IPC分类号： A61K31/506 , A61K31/4439 , A01N43/56 , A01N43/80 , A01P3/00 , A61P31/10 , C07D401/06 , C07D417/06
CPC分类号： C07D417/06 , A01N43/56 , A01N43/80 , C07D401/06 , C07D417/14
摘要： The present invention relates to compounds of Formula (I) wherein R1, R2, R3 or R4 are as defined in claim 1 or a salt or N-oxide thereof and their use in methods for the control and/or prevention of fungal infection, particularly in plants. The compounds claimed are isothiazole and pyrazole derivatives.
摘要翻译：本发明涉及其中R 1，R 2，R 3或R 4如权利要求1所定义的式（I）化合物或其盐或N-氧化物及其在控制和/或预防真菌感染的方法中的用途，特别是在植物中。所要求的化合物是异噻唑和吡唑衍生物。

68. 发明授权

US06953811B2 N-substituted tetrahydropyridines and their use as pesticides 失效
标题翻译： N-取代四氢吡啶类及其作为农药的用途
公开(公告)号：US06953811B2
公开(公告)日：2005-10-11
申请号：US10470790
申请日：2002-02-04
申请人： Stephan Trah , Josef Ehrenfreund , Peter Maienfisch , André Jeanguenat , Saleem Farooq
发明人： Stephan Trah , Josef Ehrenfreund , Peter Maienfisch , André Jeanguenat , Saleem Farooq
IPC分类号： A01N43/40 , C07D211/70 , C07D211/94 , C07D401/06
CPC分类号： C07D401/06 , C07D211/70 , C07D211/94
摘要： A description is given of compounds of the formula in which R1 and R2 independently of one another are halogen, C1-C6alkyl, halo-C1-C6alkyl, C1-C6alkoxy, halo-C1-C6alkoxy, or SF5, R3 is hydrogen, OH, halogen, C1-C6alkoxy or —O—C(═O)—C1-C6alkyl, R4 is for example hydrogen, halogen, C1-C6alkyl, halo-C1-C6alkyl, C1-C6alkoxy, halo-C1-C6alkoxy or SCN; R5 and R6 independently of one another are for example hydrogen, C1-C12alkyl, halo-C1-C12alkyl, C2-C12alkenyl, halo-C2-C12alkenyl or C2-C12alkynyl; and q is 0 or 1; and, where appropriate, E/Z isomers, E/Z isomer mixtures and/or tautomers, each in free form or in salt form; a process for the preparation of these compounds and their use, pesticide compositions whose active ingredient is selected from these compounds, or an agrochemically useable salt thereof, a process for preparing these compositions, and their use, plant propagation material treated with these compositions, and a method of combating pests.
摘要翻译：给出下式的化合物，其中R 1和R 2彼此独立地是卤素，C 1 -C 3 C 6 -C 6烷基，卤代C 1 -C 6烷基，C 1 -C 6烷基，C 1 -C 6烷基，C 1 -C 6烷基，烷氧基，卤代-C 1 -C 6烷氧基或SF 5，R 3是氢，OH，卤素，C 1 -C 6烷氧基或-OC（-O）-C 1 -C 6 -C 6烷基 R 4是例如氢，卤素，C 1 -C 6烷基，卤代C 1 -C 4烷基， C 1 -C 6烷基，C 1 -C 6烷氧基，卤代C 1 -C 6烷基，C 1 -C 6烷氧基，C 1 -C 6烷基，烷氧基或SCN; R 5和R 6彼此独立地是例如氢，C 1 -C 12 - 烷基，卤代 C 1 -C 12烷基，C 2 -C 12链烯基，卤代-C 2烷基，C 1 -C 12烷基，C 2 -C 12 - C 12 -C 12链烯基或C 2 -C 12 - 炔基; q为0或1; 和/或互变异构体，各自为游离形式或盐形式的E / Z异构体，E / Z异构体混合物和/或互变异构体; 制备这些化合物及其用途的方法，其活性成分选自这些化合物的农药组合物或其农业上可用的盐，这些组合物的制备方法及其用途，用这些组合物处理的植物繁殖材料，以及一种防治害虫的方法。

69. 发明授权

US5457095A Substituted propane-phosponous acid compounds 失效
标题翻译：取代的丙烷 - 磷酸化合物
公开(公告)号：US5457095A
公开(公告)日：1995-10-10
申请号：US255308
申请日：1994-06-07
申请人： John G. Dingwall , Josef Ehrenfreund , Roger G. Hall , James Jack
发明人： John G. Dingwall , Josef Ehrenfreund , Roger G. Hall , James Jack
IPC分类号： C07F9/32 , C07F9/48 , A61K31/185 , A61K31/66
CPC分类号： C07F9/48 , C07F9/3211 , C07F9/4816
摘要： The compounds of the formula ##STR1## in which one of the groups R.sup.1, R.sup.2 and R.sup.3 represents hydrogen, C.sub.1-8 -alkyl, C.sub.3-6 -cycloalkyl, phenyl optionally substituted by halogeno, C.sub.1-4 -alkyl, C.sub.1-4 -alkoxy and/or trifluoromethyl, or C.sub.7-10 -phenylalkyl optionally substituted in the phenyl moiety by halogeno, C.sub.1-4 -alkyl, C.sub.1-4 -alkoxy and/or trifluormethyl, and the other two are hydrogen, or salts thereof.These compounds have valuable pharmaceutical properties.
摘要翻译：其中R 1，R 2和R 3中的一个代表氢，C 1-8 - 烷基，C 3-6 - 环烷基，任选被卤素取代的苯基，C 1-4 - 烷基，C 1-4 - 烷氧基和/或三氟甲基，或在苯基部分任选被卤代，C 1-4 - 烷基，C 1-4 - 烷氧基和/或三氟甲基取代的C 7-10 - 苯基烷基，另外两个是氢或其盐。这些化合物具有有价值的药物性质。

70. 发明授权

US5243062A Substituted propane-phosphonous acid compounds 失效
标题翻译：取代的丙烷 - 膦酸化合物
公开(公告)号：US5243062A
公开(公告)日：1993-09-07
申请号：US855130
申请日：1992-03-18
申请人： John Gray Dingwall , Josef Ehrenfreund , Roger Graham Hall , James Jack
发明人： John Gray Dingwall , Josef Ehrenfreund , Roger Graham Hall , James Jack
IPC分类号： C07F9/32 , C07F9/48
CPC分类号： C07F9/48 , C07F9/3211 , C07F9/4816
摘要： The compounds of the formula ##STR1## in which one of the groups R.sup.1, R.sup.2 and R.sup.3 represents hydrogen, C.sub.1 -.sub.8 -alkyl, C.sub.3 -.sub.6 -cycloalkyl, phenyl optionally substituted by halogeno, C.sub.1 -.sub.4 -alkyl, C.sub.1 -.sub.4 -alkoxy and/or trifluoromethyl, or C.sub.7 -.sub.10 -phenylalkyl optionally substituted in the phenyl moiety by halogeno, C.sub.1 -.sub.4 -alkyl, C.sub.1 -.sub.4 -alkoxy and/or trifluormethyl, and the other two are hydrogen, or salts thereof.These compounds have valuable pharmaceutical properties.
摘要翻译：其中R 1，R 2和R 3中的一个代表氢，C 1-8 - 烷基，C 3-6 - 环烷基，任选被卤代取代的苯基，C 1-4 - 烷基，C 1-4 - 烷氧基和/或三氟甲基，或在苯基部分任选被卤代，C 1-4 - 烷基，C 1-4 - 烷氧基和/或三氟甲基取代的C 7-10 - 苯基烷基，另外两个是氢或其盐。这些化合物具有有价值的药物性质。

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