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61. 发明专利

ES8306372A1 "PROCEDIMIENTO PARA LA PREPARACION DE N-(2-(((5-DIMETILAMINO)-METIL-2-FURANIL)-METIL)-TIO)-ETIL)-N'-(3,4-METILENDIOXIBENCIL)-2-NITRO-1,1-ETENDIAMINA". 未知
公开(公告)号：ES8306372A1
公开(公告)日：1983-06-01
申请号：ES515068
申请日：1982-08-17
申请人： AUSONIA FARMA SRL
IPC分类号： A61K31/34 , A61P1/04 , A61P35/00 , C07D307/52 , C07D317/58 , C07D407/12 , A61K31/36
摘要： PROCEDIMIENTO PARA LA OBTENCION DE N-(2-(((5-DIMETILAMINO)-METIL-2-FURANIL)-METIL)-TIO)-ETIL)-N C-(3,4- METILENDIOXIBENCIL)-2-NITRO-1,1-ETENDIAMINA Y DE SUS SALES DE ADICION DE ACIDOS FISIOLOGICAMENTE COMPATIBLES; QUE TIENEN APLICACIONES FARMACOLOGICAS POR SU ACTIVIDAD ANTIULCEROSA. CONSISTE EN LA REACCION DE 2-((2-AMINOETIL)-TIO-METIL)-5-(DIMETILAMINOMETIL)-FURANO CON 1-NITRO-2-METILTIO-2-(3,4-METILENDIOXIBENCILAMINO)-ETANO. LA REACCION SE LLEVA A CABO EN DISOLVENTES APROTICOS, TALES COMO CLOROHIDROCARBUROS, A UNA TEMPERATURA COMPRENDIDA ENTRE 30 C Y 120 C.

62. 发明专利

ZA824414B A COMPOUND WITH ANALGESIC, ANTIINFLAMMATORY AND ANTIPYRETIC ACTIVITY, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS THEREFROM 未知
公开(公告)号：ZA824414B
公开(公告)日：1983-04-27
申请号：ZA824414
申请日：1982-06-22
申请人： AUSONIA FARMA SRL
发明人： DE VINCENTIIS L
IPC分类号： C07C67/14 , A61K31/23 , A61P25/04 , A61P29/00 , C07C69/92 , C07C , A61K , C07D

63. 发明专利

GB2049690B DERIVATIVES OF METHYL-SUBSTITUTED OR METHOXY-SUBSTITUTED 2-HYDROXYBENZOIC ACIDS A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL FORMULATIONS CONTAINING THEM 未知
公开(公告)号：GB2049690B
公开(公告)日：1983-04-27
申请号：GB8011654
申请日：1980-04-09
申请人： AUSONIA FARMA SRL
IPC分类号： A61K31/215 , A61K31/60 , A61P25/04 , A61P29/00 , C07C69/618 , A61P31/04 , C07C69/90 , C07C69/86 , A61K31/19 , A61K31/235 , C07C69/88
摘要： The invention relates to methyl- or methoxy-substituted 2-cynnamoyloxy-benzoic acids or to cynnamylesters of methyl- or methoxy-substituted 2-hydroxybenzoic acids, endowed with an interesting antiinflammatory, analgesic and antibacterial activity; and to a process for preparing said compounds.

64. 发明专利

AR228589A1 未知
公开(公告)号：AR228589A1
公开(公告)日：1983-03-30
申请号：AR28424381
申请日：1981-02-09
申请人： AUSONIA FARMA SRL
IPC分类号： C07C69/003 , A61K31/215 , A61K31/38 , A61K31/381 , A61K31/40 , A61K31/403 , A61K31/4035 , A61P25/04 , A61P29/00 , C07D209/44 , C07D209/46 , C07D333/22 , C07D333/24 , C08G65/332 , C08G65/333 , C07C69/612 , C08G65/00
摘要： The present invention concerns diesters of polyethylene glycols (with n ranging between 4 approximately and 100 approximately) with 2-arylpropionic acids (known as anti-inflammatory agents). These esters, while possessing all the characteristics of low toxicity and gastric injuring effects shown by the related acids, differ advantageously from the latter because their anti-inflammatory activity is much more prolonged, and their bio-availability markedly better.

65. 发明专利

ES8304060A1 "PROCEDIMIENTO PARA LA PREPARACION DE 3,4,5-TRIMETOXIBENZOATO DE 2-(4-ISOBUTILFENIL)PROPANOL-1". 未知
公开(公告)号：ES8304060A1
公开(公告)日：1983-03-01
申请号：ES513331
申请日：1982-06-22
申请人： AUSONIA FARMA SRL
IPC分类号： C07C67/14 , A61K31/23 , A61P25/04 , A61P29/00 , C07C69/92 , C07C65/24 , A61K31/235
摘要： PROCEDIMIENTO PARA LA OBTENCION DE 3,4,5-TRIMETOXIBENZOATO DE 2-(4-ISOBUTILFENIL)-PROPANOL-1, QUE TIENE APLICACIONES FARMACOLOGICAS POR SU ACTIVIDAD ANALGESICA, ANTIINFLAMATORIA Y ANTIPIRETICA. CONSISTE EN LA REACCION DEL CLORURO DEL ACIDO 3,4,5-TRIMETOXIBENZOICO CON 2-(4-ISOBUTILFENIL)PROPANOL-1. LA REACCION SE LLEVA A CABO EN UN DISOLVENTE APROTICO, EN PRESENCIA DE ACEPTORES DE ACIDO, TALES COMO PIRIDINA O TRIETILAMINA, A UNA TEMPERATURA COMPRENDIDA ENTRE 20 C Y 100 C.

66. 发明专利

ES513331A0 未知
公开(公告)号：ES513331A0
公开(公告)日：1983-03-01
申请号：ES513331
申请日：1982-06-22
申请人： AUSONIA FARMA SRL
IPC分类号： C07C67/14 , A61K31/23 , A61P25/04 , A61P29/00 , C07C69/92 , C07C65/24 , A61K31/235

67. 发明专利

BE894802A VERBINDING MET ANTIVIRUS-ACTIVITEIT EN WERKWIJZE VOOR DE BEREIDING DAARVAN 未知
公开(公告)号：BE894802A
公开(公告)日：1983-02-14
申请号：BE2059880
申请日：1982-10-26
申请人： AUSONIA FARMA SRL
IPC分类号： A61K31/66 , A61P31/12 , A61P31/22 , C07C67/00 , C07C231/00 , C07C231/12 , C07C235/14 , C07F9/38 , C07F9/40 , C07F , A61K

68. 发明专利

LU84284A1 未知
公开(公告)号：LU84284A1
公开(公告)日：1983-02-07
申请号：LU84284
申请日：1982-07-20
申请人： AUSONIA FARMA SRL
发明人： VINCENTIIS LEONARDO DE
IPC分类号： A61K31/435 , A61P7/02 , A61P9/00 , C07D461/00 , C07D , A61K
摘要： 13a-ethyl-2,3,5,6,13a,13b-hexahydro-1H-indolo (3,2,1-de)pyrido (3,2,1-ij) (1,5) naphthiridin-12-phthalidile carboxylate, having the formula given below, and a procedure for its preparation, are described. The compound lends itself to the prevention and treatment of cerebrovascular affections and organic and functional syndromes caused by a deterioration of cerebral circulation.

69. 发明专利

PT75822A PROCESS FOR PREPARING N-(2,6-DICHLOROPHENYL)-ACETAMIDINE AND OF PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME 未知
公开(公告)号：PT75822A
公开(公告)日：1982-12-01
申请号：PT7582282
申请日：1982-11-10
申请人： AUSONIA FARMA SRL
发明人： VINCENTIIS LEONARDO DE
IPC分类号： A61K31/155 , A61K20060101 , A61K31/165 , A61K31/275 , A61P9/08 , C07C20060101 , C07C67/00 , C07C239/00 , C07C249/02 , C07C257/14 , C07D20060101 , C07F13/00 , C07C , A61K
摘要： The compound N-(2,6-dichlorophenyl)acetamidine (I) and its addition salts with pharmaceutically compatible inorganic and organic acids, exhibit a fast, strong vasodilator and antihypertensive action, which is of prolonged duration.

70. 发明专利

ES503933A0 未知
公开(公告)号：ES503933A0
公开(公告)日：1982-11-01
申请号：ES503933
申请日：1981-07-14
申请人： AUSONIA FARMA SRL
IPC分类号： A61K31/43 , A61K31/545 , A61K31/546 , A61P31/04 , C07D499/00 , C07D499/76 , C07D501/20 , C07D501/24 , C07D501/26 , C07D501/34 , C07D501/38 , C07D501/46 , C07D501/57
摘要： New derivatives of 1,3-thiazolidin-4-yl carboxylic acid of the general formula I (I) wherein R represents hydrogen, (C1-4)alkyl, aralkyl, phenyl, phenyl substituted by a halogen atom or a methoxy group, formyl, acyl, trimethylsilyl; R' represents hydrogen, a pharmaceutically acceptable inorganic or organic cation, (C1-4)alkyl, 2,2,2-trichloroethyl, acetonyl, benzyl, benzyl substituted by nitro or methoxy, phenyl, nitrophenyl, benzhydryl or trimethylsilyl; R' may also represent a radical capable of providing metabolic activation in vivo selected from acetoxymethyl, pivaloyloxymethyl, phthalidyl, benzoyloxymethyl, 5-indanyl, a group of formula or a group of formula in which R'' stands for (C1-4)alkyl, (C5-6)cycloalkyl or aryl; A represents hydrogen, halogen, N3, OH, NH2; or a quaternary N-atom, particularly (and in this case R' is a negative charge; or a O-CO-NH2 group; or a group of the formula OR'''; O-COR''', NH-CO-R''' or SR''', where R''' is (C1-C4)alkyl, aryl, substituted aryl or a heterocyclic group which can carry lower alkyls; n may be zero or 1. The compounds possess antibacterial utility against microbial infections in man, animals and plants.

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