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41. 发明授权

US5462943A Substituted acetic acid esters useful as pesticides per se and as intermediates for substitued acrylic esters pesticides 失效
标题翻译：用作农药本身的取代的乙酸酯和作为取代的丙烯酸酯类农药的中间体
公开(公告)号：US5462943A
公开(公告)日：1995-10-31
申请号：US89870
申请日：1993-07-09
申请人： Thomas Seitz , Alexander Klausener , Dieter Berg , Ulrike Wachendorff-Neumann , Christoph Erdelen , Gerd Hanssler , Wilhelm Brandes , Stefan Dutzmann
发明人： Thomas Seitz , Alexander Klausener , Dieter Berg , Ulrike Wachendorff-Neumann , Christoph Erdelen , Gerd Hanssler , Wilhelm Brandes , Stefan Dutzmann
IPC分类号： A01N43/54 , C07D403/04 , A61K31/505 , C07D403/10
CPC分类号： C07D403/04 , A01N43/54
摘要： Substituted acetic acid esters of the formula ##STR1## in which R.sup.1 Represents alkyl, or represents optionally substituted aralkyl,R.sup.2 Represents dialkylamino, alkoxy or alkylthio, or represents in each case optionally substituted aralkyloxy or arylalkylthio,R.sup.3 and R.sup.4 in each case independently of one another represent hydrogen, cyano, halogen or alkyl,R.sup.5, R.sup.6 and R.sup.8 represent hydrogen or other radicals, andR.sup.7 represents optionally substituted pyrimidinyl. The compounds are pesticidially active and also used as intermediates for other acetic acid compounds.
摘要翻译：取代的式“IMAGE”的乙酸酯，其中R 1表示烷基，或表示任选取代的芳烷基，R 2表示二烷基氨基，烷氧基或烷硫基，或在各种情况下表示任选取代的芳烷氧基或芳烷硫基，R 3和R 4各自独立地为一另一个代表氢，氰基，卤素或烷基，R 5，R 6和R 8表示氢或其它基团，并且R 7表示任选取代的嘧啶基。该化合物具有杀虫活性，也用作其它乙酸化合物的中间体。

42. 发明授权

US5420284A Process for the preparation of 2-substituted 5-alkyl-pyridines 失效
标题翻译：制备2-取代的5-烷基 - 吡啶的方法
公开(公告)号：US5420284A
公开(公告)日：1995-05-30
申请号：US133729
申请日：1993-10-07
申请人： Helmut Kraus , Alexander Klausener , Hauke Furstenwerth
发明人： Helmut Kraus , Alexander Klausener , Hauke Furstenwerth
IPC分类号： C07D213/61 , C07D213/64 , C07D213/73
CPC分类号： C07D213/64 , C07D213/61 , C07D213/73
摘要： The title compounds of the formula ##STR1## can be prepared by cyclization of aminomethylenated 2-pentenoic acid derivatives of the formula ##STR2## where R, X, R.sup.1, R.sup.2 and Z have the meaning given in the description,in the presence of acids or ammonia. Preferably, aminomethylenated pentenoic acid derivatives are employed which can be prepared from pentenoic acid derivatives of the formulaR--CH.sub.2 --CH.sub.2 --CH.dbd.CH--Z (III)orR--CH.sub.2 --CH.dbd.CH--CH.sub.2 --Z (IV)with ortho-amides of the formula ##STR3## The meanings of A and B are also given in the description.
摘要翻译：式（I）的标题化合物可以通过使式（II）的氨基亚甲基化2-戊烯酸衍生物环化来制备，其中R，X，R 1，R 2和Z具有在说明书中给出的含义，在酸或氨的存在下。优选使用氨基亚甲基化的戊烯酸衍生物，其可以由式R-CH 2 -CH 2 -CH = CH-Z（III）或R-CH 2 -CH = CH-CH 2 -Z（IV）的戊烯酸衍生物与邻位式（A）的酰胺（V）A和B的含义也在说明书中给出。

43. 发明授权

US5391767A Process for the preparation of alkylene carbonates 失效
标题翻译：制备碳酸亚烷基酯的方法
公开(公告)号：US5391767A
公开(公告)日：1995-02-21
申请号：US976877
申请日：1992-11-16
申请人： Franz-Josef Mais , Hans-Josef Buysch , Christine Mendoza-Frohn , Alexander Klausener
发明人： Franz-Josef Mais , Hans-Josef Buysch , Christine Mendoza-Frohn , Alexander Klausener
IPC分类号： B01J27/08 , C07B61/00 , C07D317/36 , C07D317/38 , C07D317/44 , C07D317/46 , C07D317/18
CPC分类号： C07D317/38
摘要： Alkylene carbonates can be prepared by catalytic reaction of alkylene oxides with carbon dioxide, catalysts which can be regenerated of the formulaa[MX]/b[ZnY.sub.2 ] (III)whereinM denotes an alkali metal,X and Y independently of one another denote chlorine, bromine or iodine anda and b denote fractions or integers in a range from 0.001 to 2being employed.The catalysts (III) can be regenerated by treating with a halogen compound. The halogen compounds which can be used for this purpose belong to the group comprising hydrogen halides, inorganic and organic acid halides, interhalogen compounds and organic halides with mobile halogen.
摘要翻译：碳酸亚烷基酯可以通过烯化氧与二氧化碳的催化反应制备，催化剂可以再生成式[MX] / b [ZnY 2]（III），其中M表示碱金属，X和Y彼此独立地表示氯，溴或碘，a和b表示使用0.001至2范围内的分数或整数。催化剂（III）可以通过用卤素化合物处理再生。可以用于此目的的卤素化合物属于包含卤化氢，无机和有机酰卤，卤间化合物和具有可移动卤素的有机卤化物的基团。

44. 发明授权

US5250533A Fungicidal pyridinylpyrimidines 失效
公开(公告)号：US5250533A
公开(公告)日：1993-10-05
申请号：US844808
申请日：1992-03-02
申请人： Ulrich Heinemann , Alexander Klausener , Dieter Berg , Stefan Dutzmann , Wilhelm Brandes
发明人： Ulrich Heinemann , Alexander Klausener , Dieter Berg , Stefan Dutzmann , Wilhelm Brandes
IPC分类号： A01N43/54 , C07D401/04 , C07D405/14 , C07D413/14 , C07D401/14
CPC分类号： C07D401/04 , A01N43/54
摘要： Fungicidal pyridinylpyrimidines of the formula ##STR1## in which R.sup.1 represents hydrogen, halogen, alkoxy, alkylthio, halogenoalkyl, amino or dialkylamino, where, in the case of dialkylamino, the two radicals may, together with the nitrogen to which they are bonded, form a 5- to 7-membered, saturated or unsaturated ring which optionally contains a further hetero atom and which is optionally substituted by 1 or 2 alkyl groups; orR.sup.1 represents in each case optionally substituted aryloxy, arylthio, aralkyloxy or aralkylthio,R.sup.2 and R.sup.3 are independent of one another and are identical or different and in each case represent hydrogen, halogen, alkyl, halogenoalkyl, alkoxy, alkylthio or alkoxycarbonyl,orR.sup.2 and R.sup.3 together represent anaylene chain having 3 to 6 carbon atoms which are linked via the ring positions 3 and 4 or 4 and 5,R.sup.4 represents hydrogen, halogen, alkyl, halogenoalkyl, hydroxyl, alkoxy, mercapto, alkylthio, amino or (di)alkylamino, where, in the case of dialkylamino, the two radicals may, together with the nitrogen atom to which they are bonded, form a 5- to 7-membered, 4-phenyl-2-(2-pyridyl)-pyrimidine and 4-chloro-6-phenyl-2-(2-pyridyl)-pyrimidine (disclosed in J. Org. Chem. 32 (5), 1591-6 (1967)).Furthermore, it has been found that the new pyridinylpyrimidine derivatives of the formula (I) ##STR2## in which R.sup.1 represents hydrogen, halogen, alkoxy, alkylthio, halogenoalkyl, amino or dialkylamino, where, in the case of dialkylamino, the two radicals may, together with the nitrogen atom to which they are bonded, form a 5- to 7-membered, saturated or unsaturated ring which optionally contains a further hetero atom and which is optionally substituted by 1 or 2 alkyl groups;in which furthermoreR.sup.1 represents in each case optionally substituted aryloxy, arylthio, aralkyloxy or aralkylthio,R.sup.2 and R.sup.3 are independent of one another and are identical or different and in each case represent hydrogen, halogen, alkyl, halogenoalkyl, alkoxy, alkylthio or alkoxycarbonyl,orR.sup.2 and R.sup.3 together represent an alkylene chain having 3 to 6 carbon atoms which are linked via the ring positionsorR.sup.2 and R.sup.3 together represent an alkylene chain having 3 to 6 carbon atoms which are linked via the ring positions 3 and 4 or 4 and 5,R.sup.5 represents hydrogen or alkyl andAr represents unsubstituted or substituted aryl,

45. 发明授权

US5189063A Pesticidal substituted acrylic esters 失效
标题翻译：杀虫剂替代丙烯酸酯
公开(公告)号：US5189063A
公开(公告)日：1993-02-23
申请号：US570099
申请日：1990-08-17
申请人： Alexander Klausener , Herbert Gayer , Wolfgang Kramer , Dieter Berg , Wilhelm Brandes , Gerd Hanssler , Ulrike Wachendorff-Neumann
发明人： Alexander Klausener , Herbert Gayer , Wolfgang Kramer , Dieter Berg , Wilhelm Brandes , Gerd Hanssler , Ulrike Wachendorff-Neumann
IPC分类号： C07D317/60 , A01N37/06 , A01N37/36 , A01N37/38 , A01N37/44 , A01N37/48 , A01N43/16 , A01N43/18 , A01N43/30 , A01N43/40 , A01N43/74 , A01N43/80 , C07C67/31 , C07C69/73 , C07C69/732 , C07C69/734 , C07C229/32 , C07C229/44 , C07C251/42 , C07C251/52 , C07C251/60 , C07C323/55 , C07C323/56 , C07C323/57 , C07D211/70 , C07D213/55 , C07D213/61 , C07D213/64 , C07D261/08 , C07D263/32 , C07D277/20 , C07D277/24 , C07D277/30 , C07D307/54 , C07D309/20 , C07D309/22 , C07D317/54 , C07D333/24 , C07D335/02 , C07D401/06 , C07D401/12 , C07D403/06 , C07D403/12 , C07D405/06 , C07D409/06 , C07D413/06 , C07D417/06 , C07D521/00
CPC分类号： A01N43/74 , A01N37/36 , A01N37/38 , A01N37/44 , A01N37/48 , A01N43/30 , A01N43/40 , A01N43/80 , C07C229/44 , C07C323/56 , C07C69/734 , C07D213/61 , C07D261/08 , C07D263/32 , C07D277/24 , C07D309/22 , C07D317/54 , C07D335/02
摘要： Pesticidal substituted acrylic esters of the formula ##STR1## in which R.sup.1 represents alkyl, or represents unsubstituted or substituted aralkyl,R.sup.2 represents dialkylamino, or represents a radical --Z--R.sup.3,R.sup.3 represents alkyl, or represents unsubstituted or substituted aralkyl,Z represents oxygen or sulphur,A represents ##STR2## where n represents a number from 0 to 6,R.sup.4 and R.sup.5 in each case independently of one another represent alkyl, or together represent an alkylene chain having 2 to 7 carbon atoms, andR.sup.6 represents alkyl, or represents a radical ##STR3## where R.sup.7 represents alkyl, alkoxy or dialkylamino,B represents the group CH--R.sup.8 or, whereR.sup.9 represents unsubstituted or substituted alkyl, alkenyl, alkynyl, aralkyl, aryl or hetaryl, and R and Q independently of one another represent hydrogen, alkyl, halogenoalkyl or alkoxy.
摘要翻译：式（I）的杀虫取代的丙烯酸酯，其中R 1表示烷基，或表示未取代或取代的芳烷基，R 2表示二烷基氨基，或表示基团-Z-R 3，R 3表示烷基，或表示未取代或取代的芳烷基， Z表示氧或硫，A表示其中n表示0至6的数，R4和R5各自独立地表示烷基，或一起表示具有2至7个碳原子的亚烷基链，R6表示烷基，或表示基团，其中R 7表示烷基，烷氧基或二烷基氨基，B表示基团CH-R 8，或其中R 9表示未取代或取代的烷基，烯基，炔基，芳烷基，芳基或杂芳基，R和Q独立地彼此表示氢，烷基，卤代烷基或烷氧基。

46. 发明授权

US5114959A Fungicidal substituted acrylic esters 失效
标题翻译：杀菌剂替代丙烯酸酯
公开(公告)号：US5114959A
公开(公告)日：1992-05-19
申请号：US478119
申请日：1990-02-09
申请人： Alexander Klausener , Gerd Kleefeld , Wilhelm Brandes , Stefan Dutzmann , Gerd Hanssler
发明人： Alexander Klausener , Gerd Kleefeld , Wilhelm Brandes , Stefan Dutzmann , Gerd Hanssler
IPC分类号： C07D277/20 , A01N43/74 , A01N43/76 , A01N43/78 , C07D263/34 , C07D263/38 , C07D263/46 , C07D263/48 , C07D277/32 , C07D277/34 , C07D277/36 , C07D277/38 , C07D277/42 , C07D277/56 , C07D413/04 , C07D417/04
CPC分类号： C07D277/56 , A01N43/74 , C07D277/42
摘要： Fungicidal substituted acrylic esters of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl or alkenyl, or represents in each case optionally substitued aralkyl, aralkenyl, aryl or heteroaryl,R.sup.2 represents halogen, cyano, nitro, formyl, halogenoalkyl, alkoxyalkyl or alkylthioalkyl, or represents hydroximinoalkyl, alkoximinoalkyl, N-alkyliminoalkyl, N-aryliminoalkyl or N,N-dialkylhydrazonoalkyl, or represents alkoxy, alkylthio, halogenoalkoxy or halogenoalkylthio, or represents aryloxy or arylthio, or represents alkanoyl, alkoxycarbonyl, N,N-dialkylcarbamoyl or heterocyclylcarbonyl,R.sup.3 represents alkyl, or represents optionally substituted aralkyl,R.sup.4 represents dialkylamino or represents a radical --Z--R.sup.5,X represents oxygen or sulphur andY represents oxygen or sulphur or represents a radical ##STR2## where R.sup.5 represents alkyl or represents optionally substituted aralkyl,R.sup.6 represents hydrogen, alkyl or alkanoyl, or represents in each case optionally substituted aralkyl or aryl, andZ represents oxygen or sulphur.
摘要翻译：式（I）的杀真菌取代的丙烯酸酯，其中R 1表示氢，烷基或烯基，或在每种情况下表示任选取代的芳烷基，芳烯基，芳基或杂芳基，R 2表示卤素，氰基，硝基，甲酰基，卤代烷基，烷氧基烷基或烷硫基烷基，或代表肟基烷基，烷肟基烷基，N-烷基亚氨基烷基，N-芳基亚氨基烷基或N，N-二烷基肼基烷基，或代表烷氧基，烷硫基，卤代烷氧基或卤代烷硫基，或代表芳氧基或芳硫基，或代表烷酰基，烷氧羰基，N，二烷基氨基甲酰基或杂环基羰基，R3代表烷基，或代表任意取代的芳烷基，R4代表二烷基氨基或代表基团-Z-R5，X代表氧或硫，Y代表氧或硫，或代表基团，其中R5代表烷基或代表任选取代的芳烷基，R 6表示氢，烷基或烷酰基，或在各种情况下表示任选取代的芳烷基或芳基，Z表示氧或硫。

47. 发明授权

US4861878A 1H-pyrido-(2,3-b) (1,4)-thiazines 失效
标题翻译： 1H-吡啶并（2,3-b）（1,4） - 噻嗪
公开(公告)号：US4861878A
公开(公告)日：1989-08-29
申请号：US927909
申请日：1986-11-06
申请人： Gerd Fengler , Alexander Klausener , Hans-Josef Buysch , Mithat Mardin , Bernhard Pelster
发明人： Gerd Fengler , Alexander Klausener , Hans-Josef Buysch , Mithat Mardin , Bernhard Pelster
IPC分类号： A61K31/54 , A61P11/00 , A61P29/00 , A61P37/08 , C07D513/04
CPC分类号： C07D513/04
摘要： New potent lipoxygenase inhibitors which are 1H-pyrido-[2,3-b][1,4] thiazines are disclosed. The new thiazines are of the formula ##STR1## in which R.sup.1 denotes hydrogen, halogen, optionally substituted alkyl or alkoxy or the group ##STR2## in which R.sup.5 and R.sup.6 are identical or different and denote hydrogen, optionally substituted alkyl or aryl, or can be linked to form a 5- or 6-membered heterocyclic ring,R.sup.2 and R.sup.3 are identical or different and denote hydrogen or optionally substituted alkyl or alkoxy andR.sup.4 denotes hydroxyl, the group ##STR3## in which R.sup.5 and R.sup.6 have the abovementioned meaning, or, in the case where R.sup.3 denotes hydrogen or optionally substituted alkoxy, also denotes optionally substituted alkoxy.
摘要翻译：公开了新的有效的脂氧合酶抑制剂，它们是1H-吡啶并[2,3-b] [1,4]噻嗪。新的噻嗪类具有式“IMAGE”，其中R 1表示氢，卤素，任选取代的烷基或烷氧基或其中R 5和R 6相同或不同并表示氢，任选取代的烷基或芳基或可以连接形成5-或6-元杂环，R2和R3相同或不同，表示氢或任选取代的烷基或烷氧基，R4表示羟基，其中R5和R6具有上述含义的基团或者在R3表示氢或任选取代的烷氧基的情况下，也表示任选取代的烷氧基。

48. 发明授权

US07671217B2 Method for the decarboxylation of dicarboxylic acids 失效
标题翻译：二羧酸脱羧的方法
公开(公告)号：US07671217B2
公开(公告)日：2010-03-02
申请号：US10538995
申请日：2003-12-04
申请人： Sigurd Buchholz , Alexander Klausener , Reinhard Langer , Leslaw Mleczko , Günter Rauchschwalbe
发明人： Sigurd Buchholz , Alexander Klausener , Reinhard Langer , Leslaw Mleczko , Günter Rauchschwalbe
IPC分类号： C07D495/02
CPC分类号： C07D495/04 , C07D333/38 , Y02P20/582
摘要： The invention relates to a method for the thermal decarboxylation of dicarboxylic acids, in particular to 3,4-ethylene dioxythiophene-2,5-dicarboxylic acid as an educt. According to said method the educt is used in solid form and/or the reaction is carried out in the presence of a plurality of fluidised bed bodies. No solvents are used in the reaction and the decarboxylation product that is formed during the reaction is carried away from the reaction zone in gaseous form.
摘要翻译：本发明涉及一种二羧酸热脱羧的方法，特别涉及作为溶出物的3,4-亚乙基二氧噻吩-2,5-二羧酸的热脱羧方法。根据所述方法，溶出物以固体形式使用和/或反应在多个流化床体的存在下进行。在反应中没有使用溶剂，并且在反应期间形成的脱羧产物以气态形式从反应区带走。

49. 发明授权

US07074941B2 Process for preparing 2-alkyl-3-aryl- and -heteroaryloxaziridines and novel 2-alkyl-3-aryloxaziridines 失效
标题翻译： 2-烷基-3-芳基和 - 杂芳基氮杂环丁烷的制备方法和新的2-烷基-3-芳氧基氮杂
公开(公告)号：US07074941B2
公开(公告)日：2006-07-11
申请号：US10830622
申请日：2004-04-23
申请人： Alexander Klausener , Reinhard Langer , Stephan Ratsch , Michael Dockner
发明人： Alexander Klausener , Reinhard Langer , Stephan Ratsch , Michael Dockner
IPC分类号： C07D273/01
CPC分类号： C07D273/00
摘要： 2-Alkyl-3-aryl- or -heteroaryloxaziridines are prepared in a particularly advantageous manner by oxidizing corresponding N-alkyl-aryl- or -heteroarylaldimines with an aromatic percarboxylic acid or a salt thereof in the presence of water, a water-soluble base, and a water-miscible solvent, at temperatures below 30° C. Using this method, it is also possible to obtain novel 2-alkyl-3-aryloxaziridines.
摘要翻译：通过在水，水溶性碱的存在下，用芳族过羧酸或其盐氧化相应的N-烷基 - 芳基 - 或 - 杂芳基醛亚胺，以特别有利的方式制备2-烷基-3-芳基 - 或 - 杂芳基氧氮丙啶，和水混溶性溶剂，温度低于30℃。使用这种方法，也可以获得新的2-烷基-3-芳氧基氮杂。

50. 发明授权

US06822095B1 Method for producing 4,6-dichloropyrimidine 失效
标题翻译：制备4,6-二氯嘧啶的方法
公开(公告)号：US06822095B1
公开(公告)日：2004-11-23
申请号：US10019093
申请日：2001-12-19
申请人： Franz-Josef Mais , Günther Cramm , Alexander Klausener , Guido Steffan
发明人： Franz-Josef Mais , Günther Cramm , Alexander Klausener , Guido Steffan
IPC分类号： C07D23930
CPC分类号： C07D239/30
摘要： The present invention relates to a process for preparing 4,6-dichloropyrimidine by reaction of 4-chloro-6-hydroxypyrimidine with an acid chloride.
摘要翻译：本发明涉及通过4-氯-6-羟基嘧啶与酰氯反应制备4,6-二氯嘧啶的方法。

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