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41. 发明授权

US4507141A Triazolylalkyl-thioether plant growth regulators and fungicides 失效
标题翻译：三唑基烷基 - 硫醚植物生长调节剂和杀真菌剂
公开(公告)号：US4507141A
公开(公告)日：1985-03-26
申请号：US354122
申请日：1982-03-02
申请人： Erik Regel , Karl H. Buchel , Klaus Lurssen , Paul-Ernst Frohberger
发明人： Erik Regel , Karl H. Buchel , Klaus Lurssen , Paul-Ernst Frohberger
IPC分类号： A01N43/653 , C07D249/08 , C07D521/00 , A01N43/64
CPC分类号： C07D231/12 , A01N43/653 , C07D233/56 , C07D249/08
摘要： Triazolylalkyl-thioether plant growth regulators and fungicides of the formula ##STR1## in which A represents the keto group or the CH(OH) group,R.sup.1 represents alkyl, alkenyl, alkynyl, optionally substituted cycloalkyl, alkylaminoalkyl, alkoxycarbonylalkyl, optionally substituted phenyl or optionally substituted phenylalkyl,R.sup.2 represents alkyl,R.sup.3 represents alkyl or halogenoalkyl,R.sup.4 represents alkyl, halogenoalkyl, alkoxy, alkoxymethyl, alkylthio, alkylthiomethyl, optionally substituted phenyl, optionally substituted benzyl, optionally substituted phenoxy, optionally substituted phenoxymethyl, optionally substituted phenylthio, optionally substituted phenylthiomethyl, alkenyl, alkoxycarbonyl or cyano, orR.sup.3 and R.sup.4, conjointly with the carbon atom to which they are bonded, represent optionally substituted cycloalkyl andX.sup.1, X.sup.2, X.sup.3, X.sup.4 and X.sup.5 are selected independently and each represent hydrogen, hologen, alkyl, halogenoalkyl, halogenoalkoxy, alkoxy, alkylthio, halogenoalkylthio, alkylamino, dialkylamino, nitro, cyano, hydroxyl, alkoxycarbonyl, optionally substituted phenyl, optionally substituted phenoxy or optionally substituted benzyloxy,or an acid addition salt or metal salt complex thereof.
摘要翻译：三唑基烷基 - 硫醚植物生长调节剂和式“IMAGE”的杀真菌剂，其中A代表酮基或CH（OH）基团，R1代表烷基，烯基，炔基，任选取代的环烷基，烷基氨基烷基，烷氧基羰基烷基，任选取代的苯基或任选地取代的苯基烷基，R 2表示烷基，R 3表示烷基或卤代烷基，R 4表示烷基，卤代烷基，烷氧基，烷氧基甲基，烷硫基，烷硫基甲基，任选取代的苯基，任选取代的苄基，任选取代的苯氧基，任选取代的苯氧基甲基，任选取代的苯硫基，任选取代的苯硫基甲基，烯基，烷氧基羰基或氰基，或者R 3和R 4与它们所键合的碳原子结合，表示任选取代的环烷基，且X 1，X 2，X 3，X 4和X 5独立选择，各自表示氢，氢原子，烷基，卤代烷基，卤代烷氧基，烷氧基，烷硫基，卤代烷硫基，烷基硝基，氰基，羟基，烷氧基羰基，任选取代的苯基，任意取代的苯氧基或任意取代的苄氧基，或其酸加成盐或金属盐络合物。

42. 发明授权

US4457938A Antimycotic agent, in the form of sticks, with a high release of active compound 失效
标题翻译：具有高释放活性化合物的棒状形式的抗真菌剂
公开(公告)号：US4457938A
公开(公告)日：1984-07-03
申请号：US346479
申请日：1982-02-05
申请人： Miklos von Bittera , Karl H. Buchel , Manfred Plempel , Erik Regel
发明人： Miklos von Bittera , Karl H. Buchel , Manfred Plempel , Erik Regel
IPC分类号： A61K9/00 , A61K9/06 , A61K31/415 , A61K47/10 , A61K47/12 , A61K47/14 , A61P31/04 , A61P31/10
CPC分类号： A61K47/10 , A61K31/415 , A61K47/12 , A61K47/14 , A61K9/0014 , Y10S424/05
摘要： The invention relates to stick formulations of antimycotic azole derivatives containing, in addition to the antimycotic azole derivatives, 3 to 5% by weight relative to the formulation, of benzyl alcohol, 2.5 to 10% by weight, relative to the formulation of spreading agent and one or more auxiliaries.
摘要翻译：本发明涉及抗真菌唑衍生物的粘性制剂，除了抗真菌唑衍生物之外，相对于制剂，除了抗真菌唑类衍生物之外，相对于铺展剂的制剂，苄基醇为2.5〜10重量％一种或多种助剂。

43. 发明授权

US4243670A .alpha.-(4-Biphenylyl)-benzyl-azolium salts and their use for combating micro-organisms 失效
标题翻译： α-（4-联苯基） - 苄基 - 唑烷鎓盐及其用于抗微生物的用途
公开(公告)号：US4243670A
公开(公告)日：1981-01-06
申请号：US14783
申请日：1979-02-23
申请人： Erik Regel , Wilfried Draber , Karl H. Buchel , Manfred Plempel
发明人： Erik Regel , Wilfried Draber , Karl H. Buchel , Manfred Plempel
IPC分类号： C08G69/48 , A61K31/41 , A61K31/415 , A61P31/04 , A61P31/10 , C07D233/56 , C07D233/58 , C07D233/60 , C07D249/08 , C07D521/00 , C08G69/00 , A01N43/26 , A01N43/28
CPC分类号： C07D231/12 , C07D233/56 , C07D249/08
摘要： The present invention relates to novel .alpha.-(4-biphenylyl)-benzyl-azolium salts of the general formula ##STR1## in which A represents the CH group or a N atomR.sup.1 and R.sup.2 are identical or different and each represents hydrogen, alkyl or optionally substituted phenyl,R.sup.3 represents hydrogen, alkyl, or an optionally substituted phenyl, phenylalkyl, phenylcarbonyl or phenylcarbonylalkyl group,X represents halogen, alkyl, halogenoalkyl, alkoxy, alkylthio, nitro or cyano,Y represents X or optionally substituted phenyl,m and n each represents 0 or an integer from1 to 5 andZ represents the anion of an inorganic or organic acid.The invention also includes processes for the preparation of the compounds and, in addition includes compositions containing the compounds and methods for their use. The compounds of the invention exhibit antimicrobial activity and sporicidal activity.
摘要翻译：本发明涉及其中A表示CH基团或N原子R1和R2相同或不同并且各自表示氢的通式为“IMA”（I）的新型α-（4-联苯基） - 苄基 - ，烷基或任选取代的苯基，R 3表示氢，烷基或任选取代的苯基，苯基烷基，苯基羰基或苯基羰基烷基，X表示卤素，烷基，卤代烷基，烷氧基，烷硫基，硝基或氰基，Y表示X或任选取代的苯基， m和n各自表示0或1至5的整数，Z表示无机或有机酸的阴离子。本发明还包括制备化合物的方法，并且还包括含有这些化合物的组合物及其使用方法。本发明的化合物显示出抗微生物活性和杀孢子活性。

44. 发明授权

US4911750A Synergistic compositions for inhibiting plant growth 失效
标题翻译：用于抑制植物生长的协同组合物
公开(公告)号：US4911750A
公开(公告)日：1990-03-27
申请号：US578233
申请日：1984-02-08
申请人： Klaus Lurssen , Graham Holmwood , Wolfgang Kramer , Erik Regel , Wolf Reiser , Rolf Schroder
发明人： Klaus Lurssen , Graham Holmwood , Wolfgang Kramer , Erik Regel , Wolf Reiser , Rolf Schroder
IPC分类号： A01N43/54 , A01N43/653 , A01N53/00 , A01N53/12 , A01N57/20 , C07D233/60 , C07D239/26 , C07D249/08 , C07D303/22 , C07D521/00
CPC分类号： C07D239/26 , A01N53/00 , A01N57/20 , C07D231/12 , C07D233/56 , C07D249/08 , C07D303/22
摘要： A plant growth-inhibiting composition comprising ##STR1## wherein the various radicals are as defined.

45. 发明授权

US4499281A Substituted triazolylmethyl-oxiranes and their use as intermediates for fungicides 失效
标题翻译：取代的三唑基甲基 - 环氧乙烷及其作为杀真菌剂的中间体
公开(公告)号：US4499281A
公开(公告)日：1985-02-12
申请号：US352689
申请日：1982-02-26
申请人： Graham Holmwood , Erik Regel
发明人： Graham Holmwood , Erik Regel
IPC分类号： C07D405/06 , A01N43/653 , C07D249/08 , C07D521/00 , A01N43/64
CPC分类号： C07D231/12 , C07D233/56 , C07D249/08
摘要： A substituted triazolylmethyl-oxirane of the formula ##STR1## in which R is optionally substituted alkyl, aryl or cycloalkyl is prepared by reacting a triazolyl-ketone of the formula ##STR2## with (a) dimethyloxosulphonium methylide of the formula ##STR3## or (b) trimethylsulphonium methylsulphate of the formula[(CH.sub.3).sub.3 S].sup..sym. CH.sub.3 SO.sub.4.sup..crclbar.in the presence of a diluent.The end product can then be reacted with a phenol of the formulaR"--OHto produce known fungicidally active compounds of the formula ##STR4## in which R" is optionally substituted phenyl.
摘要翻译：其中R为任选取代的烷基，芳基或环烷基的取代三唑基甲基 - 环氧乙烷通过使式（IMAGE）的三唑基酮与（a）式（IMAGE）的二甲基氧基锍甲基化物或（ b）在稀释剂存在下，式[（CH3）3S]（+）CH3SO4（ - ）的三甲基锍甲基硫酸盐。然后可以使最终产物与式R“-OH的酚反应以产生已知的具有式”IMAGE“的杀真菌活性化合物，其中R”为任选取代的苯基。

46. 发明授权

US4452625A Synergistic compositions for inhibiting plant growth 失效
标题翻译：用于抑制植物生长的协同组合物
公开(公告)号：US4452625A
公开(公告)日：1984-06-05
申请号：US337648
申请日：1982-01-07
申请人： Klaus Lurssen , Graham Holmwood , Wolfgang Kramer , Erik Regel , Wolf Reiser , Rolf Schroder
发明人： Klaus Lurssen , Graham Holmwood , Wolfgang Kramer , Erik Regel , Wolf Reiser , Rolf Schroder
IPC分类号： A01N43/54 , A01N43/653 , A01N53/00 , A01N53/12 , A01N57/20 , C07D233/60 , C07D239/26 , C07D249/08 , C07D303/22 , C07D521/00 , A01N43/64 , A01N37/00
CPC分类号： C07D239/26 , A01N53/00 , A01N57/20 , C07D231/12 , C07D233/56 , C07D249/08 , C07D303/22
摘要： A plant growth-inhibiting composition comprising ##STR1## wherein the various radicals are as defined.
摘要翻译：（VI）和（2）所示的植物生长抑制组合物，其包含（I））（VII）或（IMA）（VIII）其中各种基团如所定义。

47. 发明授权

US4174398A Combating fungi with 1-alkyl-1-(1,3,4-thiadiazol-2-yl)-3-phenyl-ureas 失效
标题翻译：抗真菌与1-烷基-1-（1,3,4-噻二唑-2-基）-3-苯基脲
公开(公告)号：US4174398A
公开(公告)日：1979-11-13
申请号：US882833
申请日：1978-03-02
申请人： Erik Regel , Paul-Ernst Frohberger , Volker Paul
发明人： Erik Regel , Paul-Ernst Frohberger , Volker Paul
IPC分类号： A01N47/36 , C07D285/12 , C07D285/135 , A01N9/12
CPC分类号： C07D285/135 , A01N47/36
摘要： 1-Alkyl-1-(1,3,4-thiadiazol-2-yl)-3-phenyl-ureas of the formula ##STR1## in which R.sup.1 is alkyl,R.sup.2 is phenyl or substituted phenyl, andX is hydrogen or halogen,which possess fungicidal properties.
摘要翻译：其中R1是烷基，R2是苯基或取代的苯基，X是氢或卤素的1-烷基-1-（1,3,4-噻二唑-2-基）-3-苯基脲，其中R1是烷基，，具有杀菌性。

48. 发明授权

US4062959A N-methyl-imidazole derivatives for treating mycotic infections 失效
标题翻译：用于治疗真菌感染的N-甲基 - 咪唑衍生物
公开(公告)号：US4062959A
公开(公告)日：1977-12-13
申请号：US554009
申请日：1975-02-28
申请人： Wilfried Draber , Karl Heinz Buchel , Erik Regel , Manfred Plempel
发明人： Wilfried Draber , Karl Heinz Buchel , Erik Regel , Manfred Plempel
IPC分类号： A61K31/495 , A61K31/505 , C07D241/12 , C07D403/06
CPC分类号： C07D403/06 , A61K31/495 , A61K31/505 , C07D241/12
摘要： N-methyl-imidazole derivatives of the formula: ##STR1## or a pharmaceutically acceptable non-toxic salt thereof, wherein X is an unsubstituted or substituted 6-membered heteroaromatic moiety having two nitro heteroatoms,Y is an unsubstituted or substituted aliphatic moiety, an unsubstituted or substituted cycloaliphatic moiety, an unsubstituted or substituted aralkyl moiety or an unsubstituted or substituted aryl moiety, andZ is an unsubstituted or substituted aliphatic moiety, an unsubstituted or substituted cycloaliphatic moiety, an unsubstituted or substituted aralkyl moiety, an unsubstituted or substituted aryl moiety, an unsubstituted or substituted pyridyl moiety or an alkoxycarbonyl moiety,Are useful as antimycotic agents.
摘要翻译：式（I）的N-甲基 - 咪唑衍生物或其药学上可接受的无毒盐，其中X是具有两个硝基杂原子的未取代或取代的6元杂芳族部分，Y是未取代或取代的脂族未取代或取代的脂环族部分，未取代或取代的芳烷基部分或未取代或取代的芳基部分，Z为未取代或取代的脂族部分，未取代或取代的脂环族部分，未取代或取代的芳烷基部分，未取代或取代的芳烷基部分，取代的芳基部分，未取代或取代的吡啶基部分或烷氧基羰基部分，可用作抗生药剂。

49. 发明授权

US4073636A Azolylamidine compounds and herbicidal compositions 失效
标题翻译：唑基脒化合物和除草组合物
公开(公告)号：US4073636A
公开(公告)日：1978-02-14
申请号：US607986
申请日：1975-08-26
申请人： Erik Regel , Ludwig Eue , Robert R. Schmidt
发明人： Erik Regel , Ludwig Eue , Robert R. Schmidt
IPC分类号： C07D207/34 , C07D231/12 , C07D231/56 , C07D233/68 , C07D233/92 , C07D249/04 , C07D249/08 , C07D249/10 , A01N9/22
CPC分类号： C07D249/08 , C07D207/34 , C07D231/12 , C07D231/56 , C07D233/68 , C07D233/92 , C07D249/04
摘要： New azolylamidines of the formula ##STR1## WHEREIN N IS AN INTEGER FROM 0 TO 5,R.sup.1 is halogen, alkyl, alkoxy, alkylthio, haloalkoxy, haloalkylthio, halophenoxy or haloalkyl;R.sup.2 and R.sup.3, independently of one another, are each hydrogen, alkyl, alkoxyalkyl, cycloalkyl, alkoxy or alkoxycarbonylalkyl, of, preferably not more than 7 carbon atoms; or taken together, represent a lower alkylene bridge which can be interrupted by one or more hetero-atoms; andAz represents an azolyl radical selected from imidazol-1-yl, pyrrol-1-yl, pyrazol-1-yl,1,2,4-triazol-1-yl, 1,2,4-triazol-4-yl or 1,2,3-triazol-1-yl,And their salts are outstandingly effective herbicides showing particularly selective action.
摘要翻译：式（I）的新的吡唑基脒，其中N为0至5的整数，R 1为卤素，烷基，烷氧基，烷硫基，卤代烷氧基，卤代烷硫基，卤代苯氧基或卤代烷基; R 2和R 3彼此独立地为氢，烷基，烷氧基烷基，环烷基，烷氧基或烷氧基羰基烷基，优选不超过7个碳原子; 或一起代表可被一个或多个杂原子中断的低级亚烷基桥; 并且Az表示选自咪唑-1-基，吡咯-1-基，吡唑-1-基，1,2,4-三唑-1-基，1,2,4-三唑-4-基或 1,2,3-三唑-1-基，它们的盐是非常有效的除草剂，显示出特别的选择性作用。

50. 发明授权

US3993469A Azolylamidine compounds and herbicidal compositions 失效
标题翻译：唑基脒化合物和除草组合物
公开(公告)号：US3993469A
公开(公告)日：1976-11-23
申请号：US459156
申请日：1974-04-08
申请人： Erik Regel , Ludwig Eue , Robert R. Schmidt
发明人： Erik Regel , Ludwig Eue , Robert R. Schmidt
IPC分类号： A01N37/52 , A01N43/52 , A01N43/647 , A01N57/00 , A01P13/00 , C07C275/70 , C07D207/327 , C07D207/34 , C07D231/12 , C07D231/56 , C07D233/56 , C07D233/61 , C07D233/68 , C07D233/92 , C07D233/95 , C07D235/06 , C07D235/08 , C07D249/04 , C07D249/08 , C07D249/10 , C07D521/00 , C07D233/90
CPC分类号： C07D249/08 , C07C275/70 , C07D207/34 , C07D231/12 , C07D231/56 , C07D233/56 , C07D233/68 , C07D233/92 , C07D235/06 , C07D249/04
摘要： New azolylamidines of the formula ##SPC1##Whereinn is an integer from 0 to 5,R.sup.1 is halogen, alkyl, alkoxy, alkylthio, haloalkoxy, haloalkylthio, halophenoxy or haloalkyl;R.sup.2 and R.sup.3, independently of one another, are each hydrogen, alkyl, alkoxyalkyl, cycloalkyl, alkoxy or alkoxycarbonylalkyl, of, preferably not more than 7 carbon atoms; or taken together, represent a lower alkylene bridge which can be interrupted by one or more hetero-atoms; andAz represents an azolyl radical selected from imidazol-1-yl, pyrrol-1-yl, pyrazol-1-yl, 1,2,4-triazol-1-yl, 1,2,4-triazol-4-yl or 1,2,3-triazol-1-yl,And their salts are outstandingly effective herbicides showing particularly selective action.
摘要翻译：新的具有下式的氮杂脒基，其中N为0至5的整数，R 1为卤素，烷基，烷氧基，烷硫基，卤代烷氧基，卤代烷硫基，卤代苯氧基或卤代烷基; R2和R3彼此独立地为氢，烷基，烷氧基烷基，环烷基，烷氧基或烷氧基羰基烷基，优选不超过7个碳原子; 或一起代表可被一个或多个杂原子中断的低级亚烷基桥; 并且Az表示选自咪唑-1-基，吡咯-1-基，吡唑-1-基，1,2,4-三唑-1-基，1,2,4-三唑-4-基或 1,2,3-三唑-1-基，它们的盐是非常有效的除草剂，显示出特别的选择性作用。

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